UB Paderborn / Katalog / Suche / in CDI

1 – 25 von 31

Sortiert nach

Identification of a Chemical Probe for Bromo and Extra C‑Terminal Bromodomain Inhibition through Optimization of a Fragment-Derived Hit

Journal of medicinal chemistry, 2012-11, Vol.55 (22), p.9831-9837

2012

Link zum Volltext

Verfügbarkeit prüfen

Communications and High-Precision Positioning (CHP2): Hardware Architecture, Implementation, and Validation

Sensors (Basel, Switzerland), 2023-01, Vol.23 (3), p.1343

2023

Link zum Volltext

Verfügbarkeit prüfen

Discovery of Potent and Orally Available Bicyclo[1.1.1]pentane-Derived Indoleamine-2,3-dioxygenase 1 (IDO1) Inhibitors

ACS medicinal chemistry letters, 2020-08, Vol.11 (8), p.1548-1554

2020

Link zum Volltext

Verfügbarkeit prüfen

The NLRP3 inflammasome mediates DSS-induced intestinal inflammation in Nod2 knockout mice

Innate immunity (London, England), 2019-02, Vol.25 (2), p.132-143

2019

Link zum Volltext

Verfügbarkeit prüfen

Discovery of Amino-cyclobutarene-derived Indoleamine-2,3-dioxygenase 1 (IDO1) Inhibitors for Cancer Immunotherapy

ACS medicinal chemistry letters, 2019-11, Vol.10 (11), p.1530-1536

2019

Link zum Volltext

Verfügbarkeit prüfen

Strategic Incorporation of Polarity in Heme-Displacing Inhibitors of Indoleamine-2,3-dioxygenase‑1 (IDO1)

ACS medicinal chemistry letters, 2020-04, Vol.11 (4), p.550-557

2020

Link zum Volltext

Verfügbarkeit prüfen

Decarboxylative biaryl synthesis in a continuous flow reactor

Chemical communications (Cambridge, England), 2011-01, Vol.47 (12), p.3628-3630

2011

Link zum Volltext

Verfügbarkeit prüfen

Continuous Flow Enables Metallaphotoredox Catalysis in a Medicinal Chemistry Setting: Accelerated Optimization and Library Execution of a Reductive Coupling between Benzylic Chlorides and Aryl Bromides

Organic letters, 2020-01, Vol.22 (2), p.410-416

2020

Link zum Volltext

Verfügbarkeit prüfen

Photoredox Ni-catalyzed peptide C(sp)-O cross-coupling: from intermolecular reactions to side chain-to-tail macrocyclization

Chemical science (Cambridge), 2019-05, Vol.1 (19), p.573-578

2019

Link zum Volltext

Verfügbarkeit prüfen

Synthesis of Cyclic Peptidomimetics via a Pd-Catalyzed Macroamination Reaction

Organic letters, 2016-08, Vol.18 (16), p.4072-4075

2016

Link zum Volltext

Verfügbarkeit prüfen

Photoredox Ni-catalyzed peptide C(sp2)–O cross-coupling: from intermolecular reactions to side chain-to-tail macrocyclization† †Electronic supplementary information (ESI) available. See DOI: 10.1039/c9sc00694j

Chemical science (Cambridge), 2019-04, Vol.10 (19), p.5073-5078

2019

Link zum Volltext

Verfügbarkeit prüfen

Synthesis of Bridged Bicyclic Amines by Intramolecular Amination of Remote C–H Bonds: Synergistic Activation by Light and Heat

Organic letters, 2020-08, Vol.22 (16), p.6578-6583

2020

Link zum Volltext

Verfügbarkeit prüfen

Discovery of IDO1 inhibitors containing a decahydroquinoline, decahydro-1,6-naphthyridine, or octahydro-1H-pyrrolo[3,2-c]pyridine scaffold

Bioorganic & medicinal chemistry letters, 2021-10, Vol.49, p.128314-128314, Article 128314

2021

Link zum Volltext

Verfügbarkeit prüfen

Development of a Platform To Enable Efficient Permeability Evaluation of Novel Organo-Peptide Macrocycles

ACS medicinal chemistry letters, 2019-06, Vol.10 (6), p.874-879

2019

Link zum Volltext

Verfügbarkeit prüfen

SAR towards indoline and 3-azaindoline classes of IDO1 inhibitors

Bioorganic & medicinal chemistry letters, 2021-09, Vol.47, p.128214-128214, Article 128214

2021

Link zum Volltext

Verfügbarkeit prüfen

Informing the Selection of Screening Hit Series with in Silico Absorption, Distribution, Metabolism, Excretion, and Toxicity Profiles

Journal of medicinal chemistry, 2017-08, Vol.60 (16), p.6771

2017

Link zum Volltext

Verfügbarkeit prüfen

The NLRP3 inflammasome mediates DSS-induced intestinal inflammation in knockout mice

Innate immunity (London, England), 2019-02, Vol.25

2019

Link zum Volltext

Verfügbarkeit prüfen

Carbamate and N‑Pyrimidine Mitigate Amide Hydrolysis: Structure-Based Drug Design of Tetrahydroquinoline IDO1 Inhibitors

ACS medicinal chemistry letters, 2021-03, Vol.12 (3), p.389-396

2021

Link zum Volltext

Verfügbarkeit prüfen

Discovery of N‑(Indazol-3-yl)piperidine-4-carboxylic Acids as RORγt Allosteric Inhibitors for Autoimmune Diseases

ACS medicinal chemistry letters, 2020-02, Vol.11 (2), p.114-119

2020

Link zum Volltext

Verfügbarkeit prüfen

Diminishing GSH-Adduct Formation of Tricyclic Diazepine-based Mutant IDH1 Inhibitors

ACS medicinal chemistry letters, 2022-04, Vol.13 (4), p.734-741

2022

Link zum Volltext

Verfügbarkeit prüfen

Informing the Selection of Screening Hit Series with in Silico Absorption, Distribution, Metabolism, Excretion, and Toxicity Profiles: Miniperspective

Journal of medicinal chemistry, 2017-08, Vol.60 (16), p.6771-6780

2017

Link zum Volltext

Verfügbarkeit prüfen

Aryloxypyrazines as highly selective antagonists of Oxytocin

Bioorganic & medicinal chemistry letters, 2009-05, Vol.19 (10), p.2634-2636

2009

Link zum Volltext

Verfügbarkeit prüfen

Joint Positioning-Communications System Design and Experimental Demonstration

2019 IEEE/AIAA 38th Digital Avionics Systems Conference (DASC), 2019, p.1-6

2019

Link zum Volltext
Volltext

PGVL Hub: An integrated desktop tool for medicinal chemists to streamline design and synthesis of chemical libraries and singleton compounds

Methods in molecular biology (Clifton, N.J.), 2011, Vol.685, p.295

2011

Link zum Volltext

Verfügbarkeit prüfen

1 – 25 von 31

Suche als RSS-Feed

Suchergebnisse filtern

Filter anzeigen

Nur zeigen

Geprüft (Peer-Review)
(25)
Mit Volltextzugriff
(30)

Publikationsform

Sprache

Englisch
(31)
Japanisch
(5)

Erscheinungsjahr

n.n

Thema

Science & Technology
(22)
Life Sciences & Biomedicine
(14)
Chemistry
(12)
Chemistry, Medicinal
(12)
Pharmacology & Pharmacy
(12)
Physical Sciences
(11)
Chemistry, Organic
(8)
Letter
(7)
Humans
(6)
Drug Discovery
(5)
Animals
(4)
Ido1
(4)
Structure-Activity Relationship
(4)
Biochemistry
(3)
Biochemistry & Molecular Biology
(3)
Indoleamine-Pyrrole 2,3,-Dioxygenase - Metabolism
(3)
Molecular Structure
(3)
Organic Chemistry
(3)
Autonomous Vehicles
(2)
Cancer Immunotherapy
(2)

15 weitere anzeigen...

Weniger anzeigen...

Zeitschrift / Serie

5 weitere anzeigen...

Weniger anzeigen...

Menü

Weitere Dienste

Einstellungen

Identification of a Chemical Probe for Bromo and Extra C‑Terminal Bromodomain Inhibition through Optimization of a Fragment-Derived Hit

Communications and High-Precision Positioning (CHP2): Hardware Architecture, Implementation, and Validation

Discovery of Potent and Orally Available Bicyclo[1.1.1]pentane-Derived Indoleamine-2,3-dioxygenase 1 (IDO1) Inhibitors

The NLRP3 inflammasome mediates DSS-induced intestinal inflammation in Nod2 knockout mice

Discovery of Amino-cyclobutarene-derived Indoleamine-2,3-dioxygenase 1 (IDO1) Inhibitors for Cancer Immunotherapy

Strategic Incorporation of Polarity in Heme-Displacing Inhibitors of Indoleamine-2,3-dioxygenase‑1 (IDO1)

Decarboxylative biaryl synthesis in a continuous flow reactor

Continuous Flow Enables Metallaphotoredox Catalysis in a Medicinal Chemistry Setting: Accelerated Optimization and Library Execution of a Reductive Coupling between Benzylic Chlorides and Aryl Bromides

Photoredox Ni-catalyzed peptide C(sp)-O cross-coupling: from intermolecular reactions to side chain-to-tail macrocyclization

Synthesis of Cyclic Peptidomimetics via a Pd-Catalyzed Macroamination Reaction

Photoredox Ni-catalyzed peptide C(sp2)–O cross-coupling: from intermolecular reactions to side chain-to-tail macrocyclization† †Electronic supplementary information (ESI) available. See DOI: 10.1039/c9sc00694j

Synthesis of Bridged Bicyclic Amines by Intramolecular Amination of Remote C–H Bonds: Synergistic Activation by Light and Heat

Discovery of IDO1 inhibitors containing a decahydroquinoline, decahydro-1,6-naphthyridine, or octahydro-1H-pyrrolo[3,2-c]pyridine scaffold

Oxetane Promise Delivered: Discovery of Long-Acting IDO1 Inhibitors Suitable for Q3W Oral or Parenteral Dosing

Development of a Platform To Enable Efficient Permeability Evaluation of Novel Organo-Peptide Macrocycles

SAR towards indoline and 3-azaindoline classes of IDO1 inhibitors

Informing the Selection of Screening Hit Series with in Silico Absorption, Distribution, Metabolism, Excretion, and Toxicity Profiles

The NLRP3 inflammasome mediates DSS-induced intestinal inflammation in knockout mice

Carbamate and N‑Pyrimidine Mitigate Amide Hydrolysis: Structure-Based Drug Design of Tetrahydroquinoline IDO1 Inhibitors

Discovery of N‑(Indazol-3-yl)piperidine-4-carboxylic Acids as RORγt Allosteric Inhibitors for Autoimmune Diseases

Diminishing GSH-Adduct Formation of Tricyclic Diazepine-based Mutant IDH1 Inhibitors

Informing the Selection of Screening Hit Series with in Silico Absorption, Distribution, Metabolism, Excretion, and Toxicity Profiles: Miniperspective

Aryloxypyrazines as highly selective antagonists of Oxytocin

Joint Positioning-Communications System Design and Experimental Demonstration

PGVL Hub: An integrated desktop tool for medicinal chemists to streamline design and synthesis of chemical libraries and singleton compounds

Suchergebnisse filtern