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Discovery of novel multifunctional ligands targeting GABA transporters, butyrylcholinesterase, β-secretase, and amyloid β aggregation as potential treatment of Alzheimer's disease

European journal of medicinal chemistry, 2023-12, Vol.261, p.115832-115832, Article 115832

2023

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Naturally Inspired Molecules for Neuropathic Pain Inhibition-Effect of Mirogabalin and Cebranopadol on Mechanical and Thermal Nociceptive Threshold in Mice

Molecules (Basel, Switzerland), 2023-11, Vol.28 (23), p.7862

2023

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Novel GPR18 Ligands in Rodent Pharmacological Tests: Effects on Mood, Pain, and Eating Disorders

International journal of molecular sciences, 2023-05, Vol.24 (10), p.9046

2023

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8-Hydroxyquinolylnitrones as multifunctional ligands for the therapy of neurodegenerative diseases

Acta pharmaceutica Sinica. B, 2023-05, Vol.13 (5), p.2152-2175

2023

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Discovery of new, highly potent and selective inhibitors of BuChE - design, synthesis, in vitro and in vivo evaluation and crystallography studies

European journal of medicinal chemistry, 2023-03, Vol.249, p.115135, Article 115135

2023

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KM-408, a novel phenoxyalkyl derivative as a potential anticonvulsant and analgesic compound for the treatment of neuropathic pain

Pharmacological reports, 2023-02, Vol.75 (1), p.128-165

2023

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Lipopolysaccharide-Induced Model of Neuroinflammation: Mechanisms of Action, Research Application and Future Directions for Its Use

Molecules (Basel, Switzerland), 2022-08, Vol.27 (17), p.5481

2022

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Phenylalanine-Based AMPA Receptor Antagonist as the Anticonvulsant Agent with Neuroprotective Activity-In Vitro and In Vivo Studies

Molecules (Basel, Switzerland), 2022-01, Vol.27 (3), p.875

2022

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Development and crystallography-aided SAR studies of multifunctional BuChE inhibitors and 5-HT6R antagonists with β-amyloid anti-aggregation properties

European journal of medicinal chemistry, 2021-12, Vol.225, p.113792-113792, Article 113792

2021

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Development and crystallography-aided SAR studies of multifunctional BuChE inhibitors and 5-HT 6 R antagonists with β-amyloid anti-aggregation properties

European journal of medicinal chemistry, 2021-12, Vol.225, p.113792

2021

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Development of tricyclic N-benzyl-4-hydroxybutanamide derivatives as inhibitors of GABA transporters mGAT1-4 with anticonvulsant, antinociceptive, and antidepressant activity

European journal of medicinal chemistry, 2021-10, Vol.221, p.113512-113512, Article 113512

2021

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Novel Functionalized Amino Acids as Inhibitors of GABA Transporters with Analgesic Activity

ACS chemical neuroscience, 2021-08, Vol.12 (16), p.3073-3100

2021

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Sex, Pramipexole and Tiagabine Affect Behavioral and Hormonal Response to Traumatic Stress in a Mouse Model of PTSD

Frontiers in pharmacology, 2021-06, Vol.12, p.691598-691598

2021

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The Microglial Activation Inhibitor Minocycline, Used Alone and in Combination with Duloxetine, Attenuates Pain Caused by Oxaliplatin in Mice

Molecules (Basel, Switzerland), 2021-06, Vol.26 (12), p.3577

2021

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Antiepileptic Drug Tiagabine Does Not Directly Target Key Cardiac Ion Channels Kv11.1, Nav1.5 and Cav1.2

Molecules (Basel, Switzerland), 2021-06, Vol.26 (12), p.3522

2021

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Serotonergic Neurotransmission System Modulator, Vortioxetine, and Dopaminergic D2/D3 Receptor Agonist, Ropinirole, Attenuate Fibromyalgia-Like Symptoms in Mice

Molecules (Basel, Switzerland), 2021-04, Vol.26 (8), p.2398

2021

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Serotonergic Neurotransmission System Modulator, Vortioxetine, and Dopaminergic D 2 /D 3 Receptor Agonist, Ropinirole, Attenuate Fibromyalgia-Like Symptoms in Mice

Molecules (Basel, Switzerland), 2021-04, Vol.26 (8)

2021

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Wide-Range Measurement of Thermal Preference-A Novel Method for Detecting Analgesics Reducing Thermally-Evoked Pain in Mice

Molecules (Basel, Switzerland), 2021-01, Vol.26 (3), p.612

2021

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The Inclusion of Tolfenamic Acid into Cyclodextrins Stimulated by Microenvironmental pH Modification as a Way to Increase the Anti-Migraine Effect

Journal of pain research, 2021-01, Vol.14, p.981-992

2021

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Synthesis, anticonvulsant, and antinociceptive activity of new 3‐(3‐methyl‐2,5‐dioxo‐3‐phenylpyrrolidin‐1‐yl)propanamides and 3‐phenyl‐butanamides

Archiv der Pharmazie (Weinheim), 2021-01, Vol.354 (1), p.e2000225-n/a

2021

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Structure-activity relationship study of tryptophan-based butyrylcholinesterase inhibitors

European journal of medicinal chemistry, 2020-12, Vol.208, p.112766-112766, Article 112766

2020

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KM-416, a novel phenoxyalkylaminoalkanol derivative with anticonvulsant properties exerts analgesic, local anesthetic, and antidepressant-like activities. Pharmacodynamic, pharmacokinetic, and forced degradation studies

European journal of pharmacology, 2020-11, Vol.886, p.173540, Article 173540

2020

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Anticonvulsant and analgesic in neuropathic pain activity in a group of new aminoalkanol derivatives

Bioorganic & medicinal chemistry letters, 2020-08, Vol.30 (16), p.127325, Article 127325

2020

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Chemotherapy-induced peripheral neuropathy—part 2: focus on the prevention of oxaliplatin-induced neurotoxicity

Pharmacological reports, 2020-06, Vol.72 (3), p.508-527

Sałat, Kinga

2020

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Chemotherapy-induced peripheral neuropathy: part 1—current state of knowledge and perspectives for pharmacotherapy

Pharmacological reports, 2020-06, Vol.72 (3), p.486-507

Sałat, Kinga

2020

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Discovery of novel multifunctional ligands targeting GABA transporters, butyrylcholinesterase, β-secretase, and amyloid β aggregation as potential treatment of Alzheimer's disease

Naturally Inspired Molecules for Neuropathic Pain Inhibition-Effect of Mirogabalin and Cebranopadol on Mechanical and Thermal Nociceptive Threshold in Mice

Novel GPR18 Ligands in Rodent Pharmacological Tests: Effects on Mood, Pain, and Eating Disorders

8-Hydroxyquinolylnitrones as multifunctional ligands for the therapy of neurodegenerative diseases

Discovery of new, highly potent and selective inhibitors of BuChE - design, synthesis, in vitro and in vivo evaluation and crystallography studies

KM-408, a novel phenoxyalkyl derivative as a potential anticonvulsant and analgesic compound for the treatment of neuropathic pain

Lipopolysaccharide-Induced Model of Neuroinflammation: Mechanisms of Action, Research Application and Future Directions for Its Use

Phenylalanine-Based AMPA Receptor Antagonist as the Anticonvulsant Agent with Neuroprotective Activity-In Vitro and In Vivo Studies

Development and crystallography-aided SAR studies of multifunctional BuChE inhibitors and 5-HT6R antagonists with β-amyloid anti-aggregation properties

Development and crystallography-aided SAR studies of multifunctional BuChE inhibitors and 5-HT 6 R antagonists with β-amyloid anti-aggregation properties

Development of tricyclic N-benzyl-4-hydroxybutanamide derivatives as inhibitors of GABA transporters mGAT1-4 with anticonvulsant, antinociceptive, and antidepressant activity

Novel Functionalized Amino Acids as Inhibitors of GABA Transporters with Analgesic Activity

Sex, Pramipexole and Tiagabine Affect Behavioral and Hormonal Response to Traumatic Stress in a Mouse Model of PTSD

The Microglial Activation Inhibitor Minocycline, Used Alone and in Combination with Duloxetine, Attenuates Pain Caused by Oxaliplatin in Mice

Antiepileptic Drug Tiagabine Does Not Directly Target Key Cardiac Ion Channels Kv11.1, Nav1.5 and Cav1.2

Serotonergic Neurotransmission System Modulator, Vortioxetine, and Dopaminergic D2/D3 Receptor Agonist, Ropinirole, Attenuate Fibromyalgia-Like Symptoms in Mice

Serotonergic Neurotransmission System Modulator, Vortioxetine, and Dopaminergic D 2 /D 3 Receptor Agonist, Ropinirole, Attenuate Fibromyalgia-Like Symptoms in Mice

Wide-Range Measurement of Thermal Preference-A Novel Method for Detecting Analgesics Reducing Thermally-Evoked Pain in Mice

The Inclusion of Tolfenamic Acid into Cyclodextrins Stimulated by Microenvironmental pH Modification as a Way to Increase the Anti-Migraine Effect

Synthesis, anticonvulsant, and antinociceptive activity of new 3‐(3‐methyl‐2,5‐dioxo‐3‐phenylpyrrolidin‐1‐yl)propanamides and 3‐phenyl‐butanamides

Structure-activity relationship study of tryptophan-based butyrylcholinesterase inhibitors

KM-416, a novel phenoxyalkylaminoalkanol derivative with anticonvulsant properties exerts analgesic, local anesthetic, and antidepressant-like activities. Pharmacodynamic, pharmacokinetic, and forced degradation studies

Anticonvulsant and analgesic in neuropathic pain activity in a group of new aminoalkanol derivatives

Chemotherapy-induced peripheral neuropathy—part 2: focus on the prevention of oxaliplatin-induced neurotoxicity

Chemotherapy-induced peripheral neuropathy: part 1—current state of knowledge and perspectives for pharmacotherapy

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