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Discovery of 2‑Aminopyrimidines as Potent Agonists for the Bitter Taste Receptor TAS2R14

Journal of medicinal chemistry, 2023-03, Vol.66 (5), p.3499-3521

2023

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Rational design of agonists for bitter taste receptor TAS2R14: from modeling to bench and back

Cellular and molecular life sciences : CMLS, 2020-02, Vol.77 (3), p.531-542

2020

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Structure-based development of caged dopamine D2/D3 receptor antagonists

Scientific reports, 2020-01, Vol.10 (1), p.829-829, Article 829

2020

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The Bitter Taste Receptor TAS2R14 as a Drug Target

Chimia, 2022-05, Vol.76 (5), p.418

2022

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Presynaptic vesicular accumulation is required for antipsychotic efficacy in psychotic-like rats

Journal of psychopharmacology (Oxford), 2021-01, Vol.35 (1), p.65-77

2021

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Bioisosteric Replacement Leading to Biologically Active [2.2]Paracyclophanes with Altered Binding Profiles for Aminergic G-Protein-Coupled Receptors

Journal of medicinal chemistry, 2010-10, Vol.53 (19), p.7219-7228

2010

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A Chimeric Ligand Approach Leading to Potent Antiprion Active Acridine Derivatives: Design, Synthesis, and Biological Investigations

Journal of medicinal chemistry, 2006-11, Vol.49 (22), p.6591-6595

2006

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Discovery of dopamine D4 receptor antagonists with planar chirality

Bioorganic & medicinal chemistry, 2013-04, Vol.21 (7), p.1680-1684

2013

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Novel azulene derivatives for the treatment of erectile dysfunction

Bioorganic & medicinal chemistry letters, 2012-12, Vol.22 (23), p.7151-7154

2012

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Tricyclic antidepressants, quinacrine and a novel, synthetic chimera thereof clear prions by destabilizing detergent‐resistant membrane compartments

Journal of neurochemistry, 2006-08, Vol.98 (3), p.748-759

2006

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Synthesis, Radiofluorination, and In Vitro Evaluation of Pyrazolo[1,5-a]pyridine-Based Dopamine D4 Receptor Ligands: Discovery of an Inverse Agonist Radioligand for PET

Journal of medicinal chemistry, 2008-03, Vol.51 (6), p.1800-1810

2008

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Recent advances in the search for D3 - and D4 -selective drugs: probes, models and candidates

Trends in pharmacological sciences (Regular ed.), 2011-03, Vol.32 (3), p.148-157

2011

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Click chemistry on solid support: synthesis of a new REM resin and application for the preparation of tertiary amines

Tetrahedron, 2004-09, Vol.60 (39), p.8699-8702

2004

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Bivalent molecular probes for dopamine D2-like receptors

Bioorganic & medicinal chemistry, 2012-01, Vol.20 (1), p.455-466

2012

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GPCR crystal structures: Medicinal chemistry in the pocket

Bioorganic & medicinal chemistry, 2015-07, Vol.23 (14), p.3880-3906

2015

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Quinpramine ameliorates rat experimental autoimmune neuritis and redistributes MHC class II molecules

PloS one, 2011-06, Vol.6 (6), p.e21223-e21223

2011

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Structure-based discovery of opioid analgesics with reduced side effects

Nature (London), 2016-09, Vol.537 (7619), p.185-190

2016

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Recent advances in the search for D 3- and D 4-selective drugs: probes, models and candidates

Trends in pharmacological sciences (Regular ed.), 2011-03, Vol.32 (3), p.148-157

2011

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Inhibiting a promiscuous GPCR: iterative discovery of bitter taste receptor ligands

Cellular and molecular life sciences : CMLS, 2023-04, Vol.80 (4), p.114-114, Article 114

2023

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Elucidating structural determinants of biased signaling at the 5-HT1A G protein-coupled receptor through molecular dynamics simulations

Biophysical journal, 2024-02, Vol.123 (3), p.481a-482a

2024

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Synthesis and radioiodination of selective ligands for the dopamine D3 receptor subtype

Bioorganic & medicinal chemistry letters, 2004-08, Vol.14 (15), p.3963-3966

2004

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Derivatization of common antidepressant drugs increases inhibition of acid sphingomyelinase and reduces induction of phospholipidosis

Journal of Neural Transmission, 2018-12, Vol.125 (12), p.1837-1845

2018

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Synthesis and binding profile of haloperidol-based bivalent ligands targeting dopamine D2-like receptors

Bioorganic & medicinal chemistry letters, 2014-08, Vol.24 (16), p.3753-3756

2014

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T215. THE ANTIPSYCHOTIC ACTION OF HALOPERIDOL IN PSYCHOTIC-LIKE RATS REQUIRES PRESYNAPTIC VESICULAR ACCUMULATION

Schizophrenia bulletin, 2020-05, Vol.46 (Supplement_1), p.S314-S314

2020

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18F-Labeled FAUC 346 and BP 897 Derivatives as Subtype-Selective Potential PET Radioligands for the Dopamine D3 Receptor

ChemMedChem, 2008-05, Vol.3 (5), p.788-793

2008

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Discovery of 2‑Aminopyrimidines as Potent Agonists for the Bitter Taste Receptor TAS2R14

Rational design of agonists for bitter taste receptor TAS2R14: from modeling to bench and back

Structure-based development of caged dopamine D2/D3 receptor antagonists

The Bitter Taste Receptor TAS2R14 as a Drug Target

Presynaptic vesicular accumulation is required for antipsychotic efficacy in psychotic-like rats

Bioisosteric Replacement Leading to Biologically Active [2.2]Paracyclophanes with Altered Binding Profiles for Aminergic G-Protein-Coupled Receptors

A Chimeric Ligand Approach Leading to Potent Antiprion Active Acridine Derivatives: Design, Synthesis, and Biological Investigations

Discovery of dopamine D4 receptor antagonists with planar chirality

Novel azulene derivatives for the treatment of erectile dysfunction

Tricyclic antidepressants, quinacrine and a novel, synthetic chimera thereof clear prions by destabilizing detergent‐resistant membrane compartments

Synthesis, Radiofluorination, and In Vitro Evaluation of Pyrazolo[1,5-a]pyridine-Based Dopamine D4 Receptor Ligands: Discovery of an Inverse Agonist Radioligand for PET

Recent advances in the search for D3 - and D4 -selective drugs: probes, models and candidates

Click chemistry on solid support: synthesis of a new REM resin and application for the preparation of tertiary amines

Bivalent molecular probes for dopamine D2-like receptors

GPCR crystal structures: Medicinal chemistry in the pocket

Quinpramine ameliorates rat experimental autoimmune neuritis and redistributes MHC class II molecules

Structure-based discovery of opioid analgesics with reduced side effects

Recent advances in the search for D 3- and D 4-selective drugs: probes, models and candidates

Inhibiting a promiscuous GPCR: iterative discovery of bitter taste receptor ligands

Elucidating structural determinants of biased signaling at the 5-HT1A G protein-coupled receptor through molecular dynamics simulations

Synthesis and radioiodination of selective ligands for the dopamine D3 receptor subtype

Derivatization of common antidepressant drugs increases inhibition of acid sphingomyelinase and reduces induction of phospholipidosis

Synthesis and binding profile of haloperidol-based bivalent ligands targeting dopamine D2-like receptors

T215. THE ANTIPSYCHOTIC ACTION OF HALOPERIDOL IN PSYCHOTIC-LIKE RATS REQUIRES PRESYNAPTIC VESICULAR ACCUMULATION

18F-Labeled FAUC 346 and BP 897 Derivatives as Subtype-Selective Potential PET Radioligands for the Dopamine D3 Receptor

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