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Antitumor activity of the glutaminase inhibitor CB-839 in triple-negative breast cancer

Molecular cancer therapeutics, 2014-04, Vol.13 (4), p.890-901

2014

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High-throughput electrophysiological assays for voltage gated ion channels using SyncroPatch 768PE

PloS one, 2017-07, Vol.12 (7), p.e0180154-e0180154

2017

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An impedance-based cell contraction assay using human primary smooth muscle cells and fibroblasts

Journal of pharmacological and toxicological methods, 2018-01, Vol.89, p.47-53

2018

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XP13512 [(+/-)-1-([(alpha-isobutanoyloxyethoxy)carbonyl] aminomethyl)-1-cyclohexane acetic acid], a novel gabapentin prodrug: I. Design, synthesis, enzymatic conversion to gabapentin, and transport by intestinal solute transporters

The Journal of pharmacology and experimental therapeutics, 2004-10, Vol.311 (1), p.315

2004

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Distinctive Drug Binding Sites and Gating Mechanisms of the Nociceptive Ion Channel TRPA1

Biophysical journal, 2018-02, Vol.114 (3), p.640a-640a

2018

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A Non-covalent Ligand Reveals Biased Agonism of the TRPA1 Ion Channel

Neuron (Cambridge, Mass.), 2021-01, Vol.109 (2), p.273-284.e4

2021

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High-Throughput Screening of Nav1.7 Sodium Channel Blockers in an Automated Patch Clamp Assay

Biophysical journal, 2017-02, Vol.112 (3), p.240a-240a

2017

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A TRPA1 inhibitor suppresses neurogenic inflammation and airway contraction for asthma treatment

The Journal of experimental medicine, 2021-04, Vol.218 (4)

2021

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TRPA1 modulation by piperidine carboxamides suggests an evolutionarily conserved binding site and gating mechanism

Proceedings of the National Academy of Sciences - PNAS, 2019-12, Vol.116 (51), p.26008-26019

2019

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Mechanism-specific assay design facilitates the discovery of Nav1.7-selective inhibitors

Proceedings of the National Academy of Sciences - PNAS, 2018-01, Vol.115 (4), p.E792-E801

2018

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Discovery of TRPA1 Antagonist GDC-6599: Derisking Preclinical Toxicity and Aldehyde Oxidase Metabolism with a Potential First-in-Class Therapy for Respiratory Disease

Journal of medicinal chemistry, 2024-03, Vol.67 (5), p.3287-3306

2024

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A Novel Membrane Potential Assay to Identify Nav1.7-Selective Blockers

Biophysical journal, 2017-02, Vol.112 (3), p.333a-333a

2017

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A Generic Method for the Production of Cell Lines Expressing High Levels of 7-Transmembrane Receptors

Analytical biochemistry, 1997-07, Vol.250 (1), p.51-60

1997

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Ligand binding kinetics of IL-2 and IL-15 to heteromers formed by extracellular domains of the three IL-2 receptor subunits

International immunology, 1995-11, Vol.7 (11), p.1839-1849

1995

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Discovery of a novel potent GABA(B) receptor agonist

Bioorganic & medicinal chemistry letters, 2011-11, Vol.21 (21), p.6582-6585

2011

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Abstract 1877: Anti-tumor activity of novel, potent, selective and orally-bioavailable glutaminase inhibitors

Cancer research (Chicago, Ill.), 2013-04, Vol.73 (8_Supplement), p.1877-1877

2013

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Abstract 5604: Preclinical antitumor activity of novel small molecule glutaminase inhibitors in triple-negative breast cancer

Cancer research (Chicago, Ill.), 2013-04, Vol.73 (8_Supplement), p.5604-5604

2013

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Discovery of a novel potent GABAB receptor agonist

Bioorganic & medicinal chemistry letters, 2011-11, Vol.21 (21), p.6582-6585

2011

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Discovery of a novel potent GABA sub(B receptor agonist)

Bioorganic & medicinal chemistry letters, 2011-11, Vol.21 (21), p.6582-6585

2011

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Discovery of a novel potent GABA B receptor agonist

Bioorganic & medicinal chemistry letters, 2011, Vol.21 (21), p.6582-6585

2011

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Generation of a water-soluble oligomeric ectodomain of the Rous sarcoma virus envelope glycoprotein

Journal of Virology, 1993-11, Vol.67 (11), p.6889-6892

1993

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Ligand binding kinetics of IL-2 and IL-5 to heteromers formed by extracellular domains of the three IL-2 receptor subunits

International immunology, 1995-11, Vol.7 (11), p.1839-1839

1995

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CHAPTER 13 - EFFECTS OF EICOSAPENTAENOIC ACID ON IMMUNE RESPONSES AND INFLAMMATION IN HUMANS

Health Effects of Polyunsaturated Fatty Acids in Seafoods, 1986, p.239-246

1986

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Antitumor activity of the glutaminase inhibitor CB-839 in triple-negative breast cancer

High-throughput electrophysiological assays for voltage gated ion channels using SyncroPatch 768PE

An impedance-based cell contraction assay using human primary smooth muscle cells and fibroblasts

XP13512 [(+/-)-1-([(alpha-isobutanoyloxyethoxy)carbonyl] aminomethyl)-1-cyclohexane acetic acid], a novel gabapentin prodrug: I. Design, synthesis, enzymatic conversion to gabapentin, and transport by intestinal solute transporters

Distinctive Drug Binding Sites and Gating Mechanisms of the Nociceptive Ion Channel TRPA1

A Non-covalent Ligand Reveals Biased Agonism of the TRPA1 Ion Channel

High-Throughput Screening of Nav1.7 Sodium Channel Blockers in an Automated Patch Clamp Assay

A TRPA1 inhibitor suppresses neurogenic inflammation and airway contraction for asthma treatment

TRPA1 modulation by piperidine carboxamides suggests an evolutionarily conserved binding site and gating mechanism

Mechanism-specific assay design facilitates the discovery of Nav1.7-selective inhibitors

Discovery of TRPA1 Antagonist GDC-6599: Derisking Preclinical Toxicity and Aldehyde Oxidase Metabolism with a Potential First-in-Class Therapy for Respiratory Disease

Structure- and Ligand-Based Discovery of Chromane Arylsulfonamide Nav1.7 Inhibitors for the Treatment of Chronic Pain

A Novel Membrane Potential Assay to Identify Nav1.7-Selective Blockers

A Generic Method for the Production of Cell Lines Expressing High Levels of 7-Transmembrane Receptors

Ligand binding kinetics of IL-2 and IL-15 to heteromers formed by extracellular domains of the three IL-2 receptor subunits

Structure- and Ligand-Based Discovery of Chromane Arylsulfonamide Na v 1.7 Inhibitors for the Treatment of Chronic Pain

Discovery of a novel potent GABA(B) receptor agonist

Abstract 1877: Anti-tumor activity of novel, potent, selective and orally-bioavailable glutaminase inhibitors

Abstract 5604: Preclinical antitumor activity of novel small molecule glutaminase inhibitors in triple-negative breast cancer

Discovery of a novel potent GABAB receptor agonist

Discovery of a novel potent GABA sub(B receptor agonist)

Discovery of a novel potent GABA B receptor agonist

Generation of a water-soluble oligomeric ectodomain of the Rous sarcoma virus envelope glycoprotein

Ligand binding kinetics of IL-2 and IL-5 to heteromers formed by extracellular domains of the three IL-2 receptor subunits

CHAPTER 13 - EFFECTS OF EICOSAPENTAENOIC ACID ON IMMUNE RESPONSES AND INFLAMMATION IN HUMANS

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