UB Paderborn / Katalog / Suche / in CDI

An RTK UAV-Based Method for Radial Velocity Validation of Weather Radar

Remote sensing (Basel, Switzerland), 2024-04, Vol.16 (7), p.1153

2024

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A Comparative Analysis of Aerosol Microphysical, Optical and Radiative Properties during the Spring Festival Holiday over Beijing and Surrounding Regions

Aerosol and Air Quality Research, 2018-07, Vol.18 (7), p.1774-1784

2018

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A New Method for Distinguishing Unactivated Particles in Cloud Condensation Nuclei Measurements: Implications for Aerosol Indirect Effect Evaluation

Geophysical research letters, 2019-12, Vol.46 (23), p.14185-14194

2019

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A Comprehensive Study of a Winter Haze Episode over the Area around Bohai Bay in Northeast China: Insights from Meteorological Elements Observations of Boundary Layer

Sustainability, 2022-05, Vol.14 (9), p.5424

2022

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Target-triggered entropy-driven amplification system-templated silver nanoclusters for multiplexed microRNA analysis

Biosensors & bioelectronics, 2021-01, Vol.172, p.112757-112757, Article 112757

2021

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First discovery of novel 3-hydroxy-quinazoline-2,4(1H,3H)-diones as specific anti-vaccinia and adenovirus agents via ‘privileged scaffold’ refining approach

Bioorganic & medicinal chemistry letters, 2016-11, Vol.26 (21), p.5182-5186

2016

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Inhibitors of Influenza Virus Polymerase Acidic (PA) Endonuclease: Contemporary Developments and Perspectives

Journal of medicinal chemistry, 2017-05, Vol.60 (9), p.3533-3551

2017

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Newly Emerging Strategies in Antiviral Drug Discovery: Dedicated to Prof. Dr. Erik De Clercq on Occasion of His 80th Anniversary

Molecules (Basel, Switzerland), 2022-01, Vol.27 (3), p.850

2022

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Discovery of non-peptide small molecular CXCR4 antagonists as anti-HIV agents: Recent advances and future opportunities

European journal of medicinal chemistry, 2016-05, Vol.114, p.65-78

2016

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A Highly Efficient and Linear Class-AB/F Power Amplifier for Multimode Operation

IEEE transactions on microwave theory and techniques, 2008-01, Vol.56 (1), p.77-87

2008

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Discovery of GluN2A subtype-selective N -methyl-d-aspartate (NMDA) receptor ligands

Acta pharmaceutica Sinica. B, 2024-05, Vol.14 (5), p.1987-2005

2024

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Design, Synthesis, and Evaluation of Thiophene[3,2‑d]pyrimidine Derivatives as HIV‑1 Non-nucleoside Reverse Transcriptase Inhibitors with Significantly Improved Drug Resistance Profiles

Journal of medicinal chemistry, 2016-09, Vol.59 (17), p.7991-8007

2016

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Exploiting the Tolerant Region I of the Non-Nucleoside Reverse Transcriptase Inhibitor (NNRTI) Binding Pocket: Discovery of Potent Diarylpyrimidine-Typed HIV‑1 NNRTIs against Wild-Type and E138K Mutant Virus with Significantly Improved Water Solubility and Favorable Safety Profiles

Journal of medicinal chemistry, 2019-02, Vol.62 (4), p.2083-2098

2019

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Structure-Based Optimization of Thiophene[3,2‑d]pyrimidine Derivatives as Potent HIV‑1 Non-nucleoside Reverse Transcriptase Inhibitors with Improved Potency against Resistance-Associated Variants

Journal of medicinal chemistry, 2017-05, Vol.60 (10), p.4424-4443

2017

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Exploring the hydrophobic channel of NNIBP leads to the discovery of novel piperidine-substituted thiophene[3,2-d]pyrimidine derivatives as potent HIV-1 NNRTIs

Acta pharmaceutica Sinica. B, 2020-05, Vol.10 (5), p.878-894

2020

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Targeting the entrance channel of NNIBP: Discovery of diarylnicotinamide 1,4-disubstituted 1,2,3-triazoles as novel HIV-1 NNRTIs with high potency against wild-type and E138K mutant virus

European journal of medicinal chemistry, 2018-05, Vol.151, p.339-350

2018

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An improved synthesis approach of the HIV-1 inhibitor RDEA427, a pyrrolo[2,3-d]pyrimidine derivative

ARKIVOC free online journal of organic chemistry, 2021, Vol.2016 (6), p.45-51

2021

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Design, synthesis, and biological evaluation of piperidinyl‐substituted [1,2,4]triazolo[1,5‐a]pyrimidine derivatives as potential anti‐HIV‐1 agents with reduced cytotoxicity

Chemical biology & drug design, 2021-01, Vol.97 (1), p.67-76

2021

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Feasibility of developing hospital preparation by semisolid extrusion 3D printing: personalized amlodipine besylate chewable tablets

Pharmaceutical development and technology, 2022-02, Vol.27 (2), p.164-174

2022

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Optimization of N‑Substituted Oseltamivir Derivatives as Potent Inhibitors of Group‑1 and -2 Influenza A Neuraminidases, Including a Drug-Resistant Variant

Journal of medicinal chemistry, 2018-07, Vol.61 (14), p.6379-6397

2018

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Structure-Based Design and Discovery of Pyridyl-Bearing Fused Bicyclic HIV‑1 Inhibitors: Synthesis, Biological Characterization, and Molecular Modeling Studies

Journal of medicinal chemistry, 2021-09, Vol.64 (18), p.13604-13621

2021

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Novel diarylpyrimidines and diaryltriazines as potent HIV-1 NNRTIs with dramatically improved solubility: a patent evaluation of US20140378443A1

Expert opinion on therapeutic patents, 2016-02, Vol.26 (2), p.281-289

2016

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Structure-Based Design and Development of Chemical Probes Targeting Putative MOR-CCR5 Heterodimers to Inhibit Opioid Exacerbated HIV‑1 Infectivity

Journal of medicinal chemistry, 2021-06, Vol.64 (11), p.7702-7723

2021

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Discovery of novel diarypyrimidine derivatives bearing six-membered non-aromatic heterocycles as potent HIV-1 NNRTIs with improved anti-resistance and drug-like profiles

European journal of medicinal chemistry, 2023-10, Vol.258, p.115605-115605, Article 115605

2023

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The development of an effective synthetic route of lesinurad (RDEA594)

BMC chemistry, 2017-09, Vol.11 (1), p.1

2017

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An RTK UAV-Based Method for Radial Velocity Validation of Weather Radar

A Comparative Analysis of Aerosol Microphysical, Optical and Radiative Properties during the Spring Festival Holiday over Beijing and Surrounding Regions

A New Method for Distinguishing Unactivated Particles in Cloud Condensation Nuclei Measurements: Implications for Aerosol Indirect Effect Evaluation

A Comprehensive Study of a Winter Haze Episode over the Area around Bohai Bay in Northeast China: Insights from Meteorological Elements Observations of Boundary Layer

Target-triggered entropy-driven amplification system-templated silver nanoclusters for multiplexed microRNA analysis

First discovery of novel 3-hydroxy-quinazoline-2,4(1H,3H)-diones as specific anti-vaccinia and adenovirus agents via ‘privileged scaffold’ refining approach

Inhibitors of Influenza Virus Polymerase Acidic (PA) Endonuclease: Contemporary Developments and Perspectives

Newly Emerging Strategies in Antiviral Drug Discovery: Dedicated to Prof. Dr. Erik De Clercq on Occasion of His 80th Anniversary

Discovery of non-peptide small molecular CXCR4 antagonists as anti-HIV agents: Recent advances and future opportunities

A Highly Efficient and Linear Class-AB/F Power Amplifier for Multimode Operation

Discovery of GluN2A subtype-selective N -methyl-d-aspartate (NMDA) receptor ligands

Design, Synthesis, and Evaluation of Thiophene[3,2‑d]pyrimidine Derivatives as HIV‑1 Non-nucleoside Reverse Transcriptase Inhibitors with Significantly Improved Drug Resistance Profiles

Exploiting the Tolerant Region I of the Non-Nucleoside Reverse Transcriptase Inhibitor (NNRTI) Binding Pocket: Discovery of Potent Diarylpyrimidine-Typed HIV‑1 NNRTIs against Wild-Type and E138K Mutant Virus with Significantly Improved Water Solubility and Favorable Safety Profiles

Structure-Based Optimization of Thiophene[3,2‑d]pyrimidine Derivatives as Potent HIV‑1 Non-nucleoside Reverse Transcriptase Inhibitors with Improved Potency against Resistance-Associated Variants

Exploring the hydrophobic channel of NNIBP leads to the discovery of novel piperidine-substituted thiophene[3,2-d]pyrimidine derivatives as potent HIV-1 NNRTIs

Targeting the entrance channel of NNIBP: Discovery of diarylnicotinamide 1,4-disubstituted 1,2,3-triazoles as novel HIV-1 NNRTIs with high potency against wild-type and E138K mutant virus

An improved synthesis approach of the HIV-1 inhibitor RDEA427, a pyrrolo[2,3-d]pyrimidine derivative

Design, synthesis, and biological evaluation of piperidinyl‐substituted [1,2,4]triazolo[1,5‐a]pyrimidine derivatives as potential anti‐HIV‐1 agents with reduced cytotoxicity

Feasibility of developing hospital preparation by semisolid extrusion 3D printing: personalized amlodipine besylate chewable tablets

Optimization of N‑Substituted Oseltamivir Derivatives as Potent Inhibitors of Group‑1 and -2 Influenza A Neuraminidases, Including a Drug-Resistant Variant

Structure-Based Design and Discovery of Pyridyl-Bearing Fused Bicyclic HIV‑1 Inhibitors: Synthesis, Biological Characterization, and Molecular Modeling Studies

Novel diarylpyrimidines and diaryltriazines as potent HIV-1 NNRTIs with dramatically improved solubility: a patent evaluation of US20140378443A1

Structure-Based Design and Development of Chemical Probes Targeting Putative MOR-CCR5 Heterodimers to Inhibit Opioid Exacerbated HIV‑1 Infectivity

Discovery of novel diarypyrimidine derivatives bearing six-membered non-aromatic heterocycles as potent HIV-1 NNRTIs with improved anti-resistance and drug-like profiles

The development of an effective synthetic route of lesinurad (RDEA594)

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