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Exploring the hydrophobic channel of NNIBP leads to the discovery of novel piperidine-substituted thiophene[3,2-d]pyrimidine derivatives as potent HIV-1 NNRTIs

Acta pharmaceutica Sinica. B, 2020-05, Vol.10 (5), p.878-894

2020

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Boronic acid-containing diarylpyrimidine derivatives as novel HIV-1 NNRTIs: Design, synthesis and biological evaluation

Chinese chemical letters, 2021-12, Vol.32 (12), p.4053-4057

2021

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Development of a practical synthesis of etravirine via a microwave-promoted amination

BMC chemistry, 2018-12, Vol.12 (1), p.1-6

2018

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Discovery of piperidine-substituted thiazolo[5,4-d]pyrimidine derivatives as potent and orally bioavailable HIV-1 non-nucleoside reverse transcriptase inhibitors

Communications chemistry, 2019-06, Vol.2 (1), Article 74

2019

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Structure-Based Bioisosterism Yields HIV‑1 NNRTIs with Improved Drug-Resistance Profiles and Favorable Pharmacokinetic Properties

Journal of medicinal chemistry, 2020-05, Vol.63 (9), p.4837-4848

2020

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Current medicinal chemistry strategies in the discovery of novel HIV-1 ribonuclease H inhibitors

European journal of medicinal chemistry, 2022-12, Vol.243, p.114760-114760, Article 114760

2022

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In situ click chemistry-based rapid discovery of novel HIV-1 NNRTIs by exploiting the hydrophobic channel and tolerant regions of NNIBP

European journal of medicinal chemistry, 2020-05, Vol.193, p.112237-112237, Article 112237

2020

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Discovery and Characterization of Fluorine-Substituted Diarylpyrimidine Derivatives as Novel HIV‑1 NNRTIs with Highly Improved Resistance Profiles and Low Activity for the hERG Ion Channel

Journal of medicinal chemistry, 2020-02, Vol.63 (3), p.1298-1312

2020

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Identification of Dihydrofuro[3,4‑d]pyrimidine Derivatives as Novel HIV‑1 Non-Nucleoside Reverse Transcriptase Inhibitors with Promising Antiviral Activities and Desirable Physicochemical Properties

Journal of medicinal chemistry, 2019-02, Vol.62 (3), p.1484-1501

2019

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Discovery, optimization, and target identification of novel coumarin derivatives as HIV-1 reverse transcriptase-associated ribonuclease H inhibitors

European journal of medicinal chemistry, 2021-12, Vol.225, p.113769-113769, Article 113769

2021

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Discovery and optimizing polycyclic pyridone compounds as anti-HBV agents

Expert opinion on therapeutic patents, 2020-09, Vol.30 (9), p.715-721

2020

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Design, synthesis, and biological evaluation of novel double-winged galloyl derivatives as HIV-1 RNase H inhibitors

European journal of medicinal chemistry, 2022-10, Vol.240, p.114563-114563, Article 114563

2022

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Discovery and Characterization of Fluorine-Substituted Diarylpyrimidines Derivatives as Novel HIV-1 NNRTIs with Highly Improved Resistance Profiles and Low Activity for the hERG Ion Channel

Journal of medicinal chemistry, 2020-01, Vol.63 (3), p.1298-1312

2020

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Structure–Activity Relationship Exploration of NNIBP Tolerant Region I Leads to Potent HIV‑1 NNRTIs

ACS infectious diseases, 2020-08, Vol.6 (8), p.2225-2234

2020

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HIV-1 and HBV RNase H as Metal-Chelating Inhibitors: Discovery and Medicinal Chemistry Strategies

Human Viruses: Diseases, Treatments and Vaccines, 2021, p.585-602

Ahmad, Shamim I

2021

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Recent Developments in Small Molecular HIV-1 and Hepatitis B Virus RNase H Inhibitors

Advances in Metallodrugs, 2020, p.273-292

2020

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The Medicinal Chemistry of Zika Virus

Human Viruses: Diseases, Treatments and Vaccines, 2021, p.233-295

Ahmad, Shamim I

2021

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MicroRNA-153/Nrf-2/GPx1 pathway regulates radiosensitivity and stemness of glioma stem cells via reactive oxygen species

Oncotarget, 2015-09, Vol.6 (26), p.22006-22027

2015

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Knockdown of miR-210 decreases hypoxic glioma stem cells stemness and radioresistance

Experimental cell research, 2014-08, Vol.326 (1), p.22-35

2014

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Downregulation of miR-210 expression inhibits proliferation, induces apoptosis and enhances radiosensitivity in hypoxic human hepatoma cells in vitro

Experimental cell research, 2012-05, Vol.318 (8), p.944-954

2012

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NAD+ depletion radiosensitizes 2-DG-treated glioma cells by abolishing metabolic adaptation

Free radical biology & medicine, 2021-01, Vol.162, p.514-522

2021

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FLASH X-ray spares intestinal crypts from pyroptosis initiated by cGAS-STING activation upon radioimmunotherapy

Proceedings of the National Academy of Sciences - PNAS, 2022-10, Vol.119 (43), p.e2208506119

2022

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Effects of knockdown of miR-210 in combination with ionizing radiation on human hepatoma xenograft in nude mice

Radiation oncology (London, England), 2013-04, Vol.8 (1), p.102-102, Article 102

2013

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Mechanisms underlying melatonin-mediated prevention of fenvalerate-induced behavioral and oxidative toxicity in zebrafish

Journal of Toxicology and Environmental Health, Part A, 2017-01, Vol.80 (23-24), p.1331-1341

2017

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EVI5 is a novel independent prognostic predictor in hepatocellular carcinoma after radical hepatectomy

Oncology reports, 2017-10, Vol.38 (4), p.2251-2258

2017

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Exploring the hydrophobic channel of NNIBP leads to the discovery of novel piperidine-substituted thiophene[3,2-d]pyrimidine derivatives as potent HIV-1 NNRTIs

Boronic acid-containing diarylpyrimidine derivatives as novel HIV-1 NNRTIs: Design, synthesis and biological evaluation

Development of a practical synthesis of etravirine via a microwave-promoted amination

Discovery of piperidine-substituted thiazolo[5,4-d]pyrimidine derivatives as potent and orally bioavailable HIV-1 non-nucleoside reverse transcriptase inhibitors

Structure-Based Bioisosterism Yields HIV‑1 NNRTIs with Improved Drug-Resistance Profiles and Favorable Pharmacokinetic Properties

Current medicinal chemistry strategies in the discovery of novel HIV-1 ribonuclease H inhibitors

In situ click chemistry-based rapid discovery of novel HIV-1 NNRTIs by exploiting the hydrophobic channel and tolerant regions of NNIBP

Discovery and Characterization of Fluorine-Substituted Diarylpyrimidine Derivatives as Novel HIV‑1 NNRTIs with Highly Improved Resistance Profiles and Low Activity for the hERG Ion Channel

Identification of Dihydrofuro[3,4‑d]pyrimidine Derivatives as Novel HIV‑1 Non-Nucleoside Reverse Transcriptase Inhibitors with Promising Antiviral Activities and Desirable Physicochemical Properties

Discovery, optimization, and target identification of novel coumarin derivatives as HIV-1 reverse transcriptase-associated ribonuclease H inhibitors

Discovery and optimizing polycyclic pyridone compounds as anti-HBV agents

Design, synthesis, and biological evaluation of novel double-winged galloyl derivatives as HIV-1 RNase H inhibitors

Discovery and Characterization of Fluorine-Substituted Diarylpyrimidines Derivatives as Novel HIV-1 NNRTIs with Highly Improved Resistance Profiles and Low Activity for the hERG Ion Channel

Structure–Activity Relationship Exploration of NNIBP Tolerant Region I Leads to Potent HIV‑1 NNRTIs

HIV-1 and HBV RNase H as Metal-Chelating Inhibitors: Discovery and Medicinal Chemistry Strategies

Recent Developments in Small Molecular HIV-1 and Hepatitis B Virus RNase H Inhibitors

The Medicinal Chemistry of Zika Virus

MicroRNA-153/Nrf-2/GPx1 pathway regulates radiosensitivity and stemness of glioma stem cells via reactive oxygen species

Knockdown of miR-210 decreases hypoxic glioma stem cells stemness and radioresistance

Downregulation of miR-210 expression inhibits proliferation, induces apoptosis and enhances radiosensitivity in hypoxic human hepatoma cells in vitro

NAD+ depletion radiosensitizes 2-DG-treated glioma cells by abolishing metabolic adaptation

FLASH X-ray spares intestinal crypts from pyroptosis initiated by cGAS-STING activation upon radioimmunotherapy

Effects of knockdown of miR-210 in combination with ionizing radiation on human hepatoma xenograft in nude mice

Mechanisms underlying melatonin-mediated prevention of fenvalerate-induced behavioral and oxidative toxicity in zebrafish

EVI5 is a novel independent prognostic predictor in hepatocellular carcinoma after radical hepatectomy

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