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Characterization of SB-705498, a potent and selective vanilloid receptor-1 (VR1/TRPV1) antagonist that inhibits the capsaicin-, acid-, and heat-mediated activation of the receptor

The Journal of pharmacology and experimental therapeutics, 2007-06, Vol.321 (3), p.1183

2007

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1,3-Biarylureas as selective non-peptide antagonists of the orexin-1 receptor

Bioorganic & medicinal chemistry letters, 2001-07, Vol.11 (14), p.1907-1910

2001

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Discovery of small molecule antagonists of TRPV1

Bioorganic & medicinal chemistry letters, 2004-07, Vol.14 (14), p.3631-3634

2004

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Old drugs with new skills: fenoprofen as an allosteric enhancer at melanocortin receptor 3

Cellular and molecular life sciences : CMLS, 2017-04, Vol.74 (7), p.1335-1345

2017

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Inhibition of C6 glioma cell proliferation by anandamide, 1-arachidonoylglycerol, and by a water soluble phosphate ester of anandamide: variability in response and involvement of arachidonic acid

Biochemical pharmacology, 2003-09, Vol.66 (5), p.757-767

2003

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The physiology and pharmacology of the orexins

Pharmacology & therapeutics (Oxford), 2002-04, Vol.94 (1), p.51-61

2002

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Discovery of SB-705498: A potent, selective and orally bioavailable TRPV1 antagonist suitable for clinical development

Bioorganic & medicinal chemistry letters, 2006-06, Vol.16 (12), p.3287-3291

2006

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Characterisation of the binding of [3H]‐SB‐674042, a novel nonpeptide antagonist, to the human orexin‐1 receptor

British journal of pharmacology, 2004-01, Vol.141 (2), p.340-346

2004

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A High-Throughput Electrophysiology Assay Identifies Inhibitors of the Inwardly Rectifying Potassium Channel Kir7.1

Journal of biomolecular screening, 2015-07, Vol.20 (6), p.739-747

2015

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Pharmacology of vanilloids at recombinant and endogenous rat vanilloid receptors

Biochemical pharmacology, 2003, Vol.65 (1), p.143-151

2003

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Design and synthesis of 6-phenylnicotinamide derivatives as antagonists of TRPV1

Bioorganic & medicinal chemistry, 2008-10, Vol.18 (20), p.5609-5613

2008

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Pharmacological characterisation of human 5-HT2 receptor subtypes

European journal of pharmacology, 2001-02, Vol.414 (1), p.23-30

2001

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Cannabinoid activation of recombinant and endogenous vanilloid receptors

European journal of pharmacology, 2001-07, Vol.424 (3), p.211-219

2001

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Characterisation using FLIPR of human vanilloid VR1 receptor pharmacology

European journal of pharmacology, 2001-04, Vol.417 (1), p.51-58

2001

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N-Tetrahydroquinolinyl, N-quinolinyl and N-isoquinolinyl biaryl carboxamides as antagonists of TRPV1

Bioorganic & medicinal chemistry letters, 2006-09, Vol.16 (17), p.4533-4536

2006

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Structure–activity analysis of truncated orexin-A analogues at the orexin-1 receptor

Bioorganic & medicinal chemistry letters, 2001-03, Vol.11 (5), p.737-740

2001

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Characterisation of an endogenous bombesin receptor in CHO/DG44 cells

European journal of pharmacology, 2000-12, Vol.409 (3), p.259-263

2000

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Characterization of the binding of [3H]‐SB‐204269, a radiolabelled form of the new anticonvulsant SB‐204269, to a novel binding site in rat brain membranes

British journal of pharmacology, 1997-08, Vol.121 (8), p.1687-1691

1997

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Synthesis of Novel trans-4-(Substituted-benzamido)-3,4-dihydro-2H-benzo[b]pyran-3-ol Derivatives as Potential Anticonvulsant Agents with a Distinctive Binding Profile

Journal of medicinal chemistry, 1996-11, Vol.39 (23), p.4537-4539

1996

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Low pH modulation of recombinant vanilloid receptors and perivascular capsaicin-sensitive sensory neurotransmission

Autonomic neuroscience, 2001-04, Vol.88 (1), p.36-44

2001

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Cellular Screening for 7TM Receptors Using Label-Free Detection

Label-Free Technologies For Drug Discovery, 2011, p.205-222

2011

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Identification of (-)-cis-6-acetyl-4S-(3-chloro-4-fluoro-benzoylamino)-3,4-dihydro-2,2-dimethyl-2H-benzo[b]pyran-3S-ol as a potential antimigraine agent

Bioorganic & medicinal chemistry letters, 1999-01, Vol.9 (2), p.285-290

1999

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Pharmacological characterisation of human 5-HT 2 receptor subtypes

European journal of pharmacology, 2001, Vol.414 (1), p.23-30

2001

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Identification of a series of 1,2,3,4-tetrahydroisoquinolinyl- benzamides with potential anticonvulsant activity

Bioorganic & medicinal chemistry letters, 1998-10, Vol.8 (20), p.2903-2906

1998

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Identification of (−)- cis-6-acetyl-4 S-(3-chloro-4-fluoro-benzoylamino)-3,4-dihydro-2,2-dimethyl-2 H-benzo[b]pyran-3 S-ol as a potential antimigraine agent

Bioorganic & medicinal chemistry letters, 1999, Vol.9 (2), p.285-290

1999

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Characterization of SB-705498, a potent and selective vanilloid receptor-1 (VR1/TRPV1) antagonist that inhibits the capsaicin-, acid-, and heat-mediated activation of the receptor

1,3-Biarylureas as selective non-peptide antagonists of the orexin-1 receptor

Discovery of small molecule antagonists of TRPV1

Old drugs with new skills: fenoprofen as an allosteric enhancer at melanocortin receptor 3

Inhibition of C6 glioma cell proliferation by anandamide, 1-arachidonoylglycerol, and by a water soluble phosphate ester of anandamide: variability in response and involvement of arachidonic acid

The physiology and pharmacology of the orexins

Discovery of SB-705498: A potent, selective and orally bioavailable TRPV1 antagonist suitable for clinical development

Characterisation of the binding of [3H]‐SB‐674042, a novel nonpeptide antagonist, to the human orexin‐1 receptor

A High-Throughput Electrophysiology Assay Identifies Inhibitors of the Inwardly Rectifying Potassium Channel Kir7.1

Pharmacology of vanilloids at recombinant and endogenous rat vanilloid receptors

Design and synthesis of 6-phenylnicotinamide derivatives as antagonists of TRPV1

Pharmacological characterisation of human 5-HT2 receptor subtypes

Cannabinoid activation of recombinant and endogenous vanilloid receptors

Characterisation using FLIPR of human vanilloid VR1 receptor pharmacology

N-Tetrahydroquinolinyl, N-quinolinyl and N-isoquinolinyl biaryl carboxamides as antagonists of TRPV1

Structure–activity analysis of truncated orexin-A analogues at the orexin-1 receptor

Characterisation of an endogenous bombesin receptor in CHO/DG44 cells

Characterization of the binding of [3H]‐SB‐204269, a radiolabelled form of the new anticonvulsant SB‐204269, to a novel binding site in rat brain membranes

Synthesis of Novel trans-4-(Substituted-benzamido)-3,4-dihydro-2H-benzo[b]pyran-3-ol Derivatives as Potential Anticonvulsant Agents with a Distinctive Binding Profile

Low pH modulation of recombinant vanilloid receptors and perivascular capsaicin-sensitive sensory neurotransmission

Cellular Screening for 7TM Receptors Using Label-Free Detection

Identification of (-)-cis-6-acetyl-4S-(3-chloro-4-fluoro-benzoylamino)-3,4-dihydro-2,2-dimethyl-2H-benzo[b]pyran-3S-ol as a potential antimigraine agent

Pharmacological characterisation of human 5-HT 2 receptor subtypes

Identification of a series of 1,2,3,4-tetrahydroisoquinolinyl- benzamides with potential anticonvulsant activity

Identification of (−)- cis-6-acetyl-4 S-(3-chloro-4-fluoro-benzoylamino)-3,4-dihydro-2,2-dimethyl-2 H-benzo[b]pyran-3 S-ol as a potential antimigraine agent

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