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Pyrrolidine in Drug Discovery: A Versatile Scaffold for Novel Biologically Active Compounds

Topics in current chemistry (2016), 2021-10, Vol.379 (5), p.34-34, Article 34

2021

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Insights into the Zinc-Dependent Deacetylase LpxC: Biochemical Properties and Inhibitor Design

Current topics in medicinal chemistry, 2016-09, Vol.16 (21), p.2379

2016

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Characterization of Histone Deacetylase 8 (HDAC8) Selective Inhibition Reveals Specific Active Site Structural and Functional Determinants

Journal of medicinal chemistry, 2018-11, Vol.61 (22), p.10000-10016

2018

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Structure and function of an irreversible agonist-β2 adrenoceptor complex

Nature (London), 2011-01, Vol.469 (7329), p.236-240

2011

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Editorial: Emerging heterocycles as bioactive compounds

Frontiers in chemistry, 2023-04, Vol.11, p.1202192-1202192

2023

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Synthesis and biological evaluation of flexible and conformationally constrained LpxC inhibitors

Organic & biomolecular chemistry, 2013-09, Vol.11 (36), p.6056-6070

2013

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Bioactive pyrrole-based compounds with target selectivity

European journal of medicinal chemistry, 2020-12, Vol.208, p.112783-112783, Article 112783

2020

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LpxC inhibitors: a patent review (2010-2016)

Expert opinion on therapeutic patents, 2017-11, Vol.27 (11), p.1227-1250

2017

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Design and stereoselective synthesis of a C-aryl furanoside as a conformationally constrained CHIR-090 analogue

Carbohydrate research, 2012-10, Vol.359, p.59-64

2012

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Chiral pool synthesis and biological evaluation of C-furanosidic and acyclic LpxC inhibitors

European journal of medicinal chemistry, 2016-03, Vol.110, p.340-375

2016

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Phenylethylene glycol-derived LpxC inhibitors with diverse Zn2+-binding groups

Tetrahedron, 2019-01, Vol.75 (4), p.486-509

2019

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Synthesis and biological evaluation of triazolyl-substituted benzyloxyacetohydroxamic acids as LpxC inhibitors

Bioorganic & medicinal chemistry, 2020-07, Vol.28 (13), p.115529-115529, Article 115529

2020

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Synthesis and biological evaluation of C-ethynyl furanosides as LpxC inhibitors

Tetrahedron, 2015-02, Vol.71 (6), p.956-966

2015

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Synthesis, biological evaluation, and molecular docking studies of deoxygenated C-glycosides as LpxC inhibitors

Bioorganic chemistry, 2021-12, Vol.117, p.105403-105403, Article 105403

2021

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Novel Potent Proline-Based Metalloproteinase Inhibitors: Design, (Radio)Synthesis, and First in Vivo Evaluation as Radiotracers for Positron Emission Tomography

Journal of medicinal chemistry, 2016-10, Vol.59 (20), p.9541-9559

2016

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Synthesis and biological evaluation of enantiomerically pure glyceric acid derivatives as LpxC inhibitors

Bioorganic & medicinal chemistry, 2016-03, Vol.24 (5), p.1032-1044

2016

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Antibacterial activity of xylose-derived LpxC inhibitors – Synthesis, biological evaluation and molecular docking studies

Bioorganic chemistry, 2021-02, Vol.107, p.104603-104603, Article 104603

2021

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Chiral Pool Synthesis, Biological Evaluation and Molecular Docking Studies of C‐Furanosidic LpxC Inhibitors

ChemMedChem, 2019-04, Vol.14 (8), p.871-886

2019

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Proline-based hydroxamates targeting the zinc-dependent deacetylase LpxC: Synthesis, antibacterial properties, and docking studies

Bioorganic & medicinal chemistry, 2019-05, Vol.27 (10), p.1997-2018

2019

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C-Triazolyl β-d-furanosides as LpxC inhibitors: stereoselective synthesis and biological evaluation

Tetrahedron, 2014-09, Vol.70 (37), p.6569-6577

2014

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Structure‐Based Design, Synthesis, and Biological Evaluation of Triazole‐Based smHDAC8 Inhibitors

ChemMedChem, 2020-04, Vol.15 (7), p.571-584

2020

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Front Cover: Structure‐Based Design, Synthesis, and Biological Evaluation of Triazole‐Based smHDAC8 Inhibitors (ChemMedChem 7/2020)

ChemMedChem, 2020-04, Vol.15 (7), p.559-559

2020

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Synthesis, biological evaluation and molecular docking studies of benzyloxyacetohydroxamic acids as LpxC inhibitors

Bioorganic & medicinal chemistry, 2014-02, Vol.22 (3), p.1016-1028

2014

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Synthesis, biological evaluation, and molecular docking studies of aldotetronic acid-based LpxC inhibitors

Bioorganic chemistry, 2023-02, Vol.131, p.106331-106331, Article 106331

2023

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Development of novel LpxC inhibitors: chiral-pool synthesis of C-triazolyl glycosides

Tetrahedron, 2013-11, Vol.69 (45), p.9434-9442

2013

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Pyrrolidine in Drug Discovery: A Versatile Scaffold for Novel Biologically Active Compounds

Insights into the Zinc-Dependent Deacetylase LpxC: Biochemical Properties and Inhibitor Design

Characterization of Histone Deacetylase 8 (HDAC8) Selective Inhibition Reveals Specific Active Site Structural and Functional Determinants

Structure and function of an irreversible agonist-β2 adrenoceptor complex

Editorial: Emerging heterocycles as bioactive compounds

Synthesis and biological evaluation of flexible and conformationally constrained LpxC inhibitors

Bioactive pyrrole-based compounds with target selectivity

LpxC inhibitors: a patent review (2010-2016)

Design and stereoselective synthesis of a C-aryl furanoside as a conformationally constrained CHIR-090 analogue

Chiral pool synthesis and biological evaluation of C-furanosidic and acyclic LpxC inhibitors

Phenylethylene glycol-derived LpxC inhibitors with diverse Zn2+-binding groups

Synthesis and biological evaluation of triazolyl-substituted benzyloxyacetohydroxamic acids as LpxC inhibitors

Synthesis and biological evaluation of C-ethynyl furanosides as LpxC inhibitors

Synthesis, biological evaluation, and molecular docking studies of deoxygenated C-glycosides as LpxC inhibitors

Novel Potent Proline-Based Metalloproteinase Inhibitors: Design, (Radio)Synthesis, and First in Vivo Evaluation as Radiotracers for Positron Emission Tomography

Synthesis and biological evaluation of enantiomerically pure glyceric acid derivatives as LpxC inhibitors

Antibacterial activity of xylose-derived LpxC inhibitors – Synthesis, biological evaluation and molecular docking studies

Chiral Pool Synthesis, Biological Evaluation and Molecular Docking Studies of C‐Furanosidic LpxC Inhibitors

Proline-based hydroxamates targeting the zinc-dependent deacetylase LpxC: Synthesis, antibacterial properties, and docking studies

C-Triazolyl β-d-furanosides as LpxC inhibitors: stereoselective synthesis and biological evaluation

Structure‐Based Design, Synthesis, and Biological Evaluation of Triazole‐Based smHDAC8 Inhibitors

Front Cover: Structure‐Based Design, Synthesis, and Biological Evaluation of Triazole‐Based smHDAC8 Inhibitors (ChemMedChem 7/2020)

Synthesis, biological evaluation and molecular docking studies of benzyloxyacetohydroxamic acids as LpxC inhibitors

Synthesis, biological evaluation, and molecular docking studies of aldotetronic acid-based LpxC inhibitors

Development of novel LpxC inhibitors: chiral-pool synthesis of C-triazolyl glycosides

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