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Discovery of Selective Irreversible Inhibitors for Bruton's Tyrosine Kinase

ChemMedChem, 2007-01, Vol.2 (1), p.58-61

2007

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CRA-024781: a novel synthetic inhibitor of histone deacetylase enzymes with antitumor activity in vitro and in vivo

Molecular cancer therapeutics, 2006-05, Vol.5 (5), p.1309-1317

2006

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Design and Synthesis of 4-Azaindoles as Inhibitors of p38 MAP Kinase

Journal of medicinal chemistry, 2003-10, Vol.46 (22), p.4702-4713

2003

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Identification and pre-clinical testing of a reversible cathepsin protease inhibitor reveals anti-tumor efficacy in a pancreatic cancer model

Biochimie, 2010-11, Vol.92 (11), p.1618-1624

2010

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Testosterone and IL-6 Requirements for Human C-Reactive Protein Gene Expression in Transgenic Mice

The Journal of immunology (1950), 1998-06, Vol.160 (11), p.5294-5299

1998

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Evaluation of antitumor properties of novel saframycin analogs in vitro and in vivo

Bioorganic & medicinal chemistry letters, 2006-09, Vol.16 (18), p.4884-4888

2006

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Embryonic Lethality, Liver Degeneration, and Impaired NF-κB Activation in IKK-β-Deficient Mice

Immunity (Cambridge, Mass.), 1999-04, Vol.10 (4), p.421-429

1999

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Discovery of 6-(2,4-Difluorophenoxy)-2-[3-hydroxy-1-(2-hydroxyethyl)propylamino]-8-methyl-8H-pyrido[2,3-d]pyrimidin-7-one (Pamapimod) and 6-(2,4-Difluorophenoxy)-8-methyl-2-(tetrahydro-2H-pyran-4-ylamino)pyrido[2,3-d]pyrimidin-7(8H)-one (R1487) as Orally Bioavailable and Highly Selective Inhibitors of p38α Mitogen-Activated Protein Kinase

Journal of medicinal chemistry, 2011-04, Vol.54 (7), p.2255-2265

2011

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p38 mitogen activated protein kinase as a therapeutic target for Alzheimer's disease

Journal of molecular neuroscience, 2002-12, Vol.19 (3), p.295-299

Dalrymple, Stacie A

2002

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A Small Molecule Ubiquitination Inhibitor Blocks NF-κB-dependent Cytokine Expression in Cells and Rats

The Journal of biological chemistry, 2002-06, Vol.277 (26), p.23573-23581

2002

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Targeting B cells for the treatment of rheumatoid arthritis

Arthritis research & therapy, 2003-01, Vol.5 Suppl 4 (Suppl 4), p.S7-11

2003

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The cytokine stew and innate resistance to L. monocytogenes

Immunological reviews, 1997-08, Vol.158 (1), p.107-114

1997

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Discovery of 6-(2,4-Difluorophenoxy)-2-[3-hydroxy-1-(2-hydroxyethyl)propylamino]-8-methyl-8 H -pyrido[2,3- d ]pyrimidin-7-one (Pamapimod) and 6-(2,4-Difluorophenoxy)-8-methyl-2-(tetrahydro-2 H -pyran-4-ylamino)pyrido[2,3- d ]pyrimidin-7(8 H )-one (R1487) as Orally Bioavailable and Highly Selective Inhibitors of p38α Mitogen-Activated Protein Kinase

Journal of medicinal chemistry, 2011-04, Vol.54 (7), p.2255-2265

2011

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Regulation of interleukin-6, osteoclastogenesis, and bone mass by androgens. The role of the androgen receptor

The Journal of clinical investigation, 1995-06, Vol.95 (6), p.2886-2895

1995

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Identification and preclinical testing of a reversible cathepsin protease inhibitor reveals anti-tumor efficacy in a pancreatic cancer model

Biochimie, 2010-05, Vol.92 (11)

2010

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Impaired resistance to the development of toxoplasmic encephalitis in interleukin-6-deficient mice

Infection and Immunity, 1997-06, Vol.65 (6), p.2339-2345

1997

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Subcutaneous Dosing of CRA-027483, a Small Molecule FVIIa Inhibitor, Prevents Arterial Thrombosis in a Baboon Model

Blood, 2005-11, Vol.106 (11), p.1867-1867

2005

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A Selective Small Molecule Factor VIIa Inhibitor, CRA-027483, Suppresses Acute Inflammation in Mice

Blood, 2005-11, Vol.106 (11), p.3089-3089

2005

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Models of Inflammation: Adjuvant‐Induced Arthritis in the Rat

Current Protocols in Pharmacology, 2001-08, Vol.13 (1), p.5.5.1-5.5.5

2001

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A Small Molecule Ubiquitination Inhibitor Blocks NF-ÎºB-dependent Cytokine Expression in Cells and Rats

The Journal of biological chemistry, 2002-06, Vol.277 (26), p.23573

2002

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Models of Inflammation: Carrageenan Air Pouch in the Rat

Current Protocols in Pharmacology, 1998-03 (1)

1998

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Models of inflammation: measuring gastrointestinal ulceration in the rat

Current Protocols in Pharmacology, 2001-05, Vol.Chapter 10 (1), p.Unit 10.2-Unit 10.2

2001

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BK virus T antigens induce kidney carcinomas and thymoproliferative disorders in transgenic mice

Journal of Virology, 1990-03, Vol.64 (3), p.1182-1191

1990

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A novel series of IKKβ inhibitors part I: Initial SAR studies of a HTS hit

Bioorganic & medicinal chemistry letters, 2011-01, Vol.21 (1), p.417-422

2011

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Discovery of Selective Irreversible Inhibitors for Bruton's Tyrosine Kinase

CRA-024781: a novel synthetic inhibitor of histone deacetylase enzymes with antitumor activity in vitro and in vivo

Design and Synthesis of 4-Azaindoles as Inhibitors of p38 MAP Kinase

Identification and pre-clinical testing of a reversible cathepsin protease inhibitor reveals anti-tumor efficacy in a pancreatic cancer model

Testosterone and IL-6 Requirements for Human C-Reactive Protein Gene Expression in Transgenic Mice

Evaluation of antitumor properties of novel saframycin analogs in vitro and in vivo

Embryonic Lethality, Liver Degeneration, and Impaired NF-κB Activation in IKK-β-Deficient Mice

Discovery of S-[5-Amino-1-(4-fluorophenyl)-1H-pyrazol-4-yl]-[3-(2,3-dihydroxypropoxy)phenyl]methanone (RO3201195), an Orally Bioavailable and Highly Selective Inhibitor of p38 Map Kinase

p38 mitogen activated protein kinase as a therapeutic target for Alzheimer's disease

A Small Molecule Ubiquitination Inhibitor Blocks NF-κB-dependent Cytokine Expression in Cells and Rats

Targeting B cells for the treatment of rheumatoid arthritis

The cytokine stew and innate resistance to L. monocytogenes

Regulation of interleukin-6, osteoclastogenesis, and bone mass by androgens. The role of the androgen receptor

Identification and preclinical testing of a reversible cathepsin protease inhibitor reveals anti-tumor efficacy in a pancreatic cancer model

Impaired resistance to the development of toxoplasmic encephalitis in interleukin-6-deficient mice

Subcutaneous Dosing of CRA-027483, a Small Molecule FVIIa Inhibitor, Prevents Arterial Thrombosis in a Baboon Model

A Selective Small Molecule Factor VIIa Inhibitor, CRA-027483, Suppresses Acute Inflammation in Mice

Models of Inflammation: Adjuvant‐Induced Arthritis in the Rat

A Small Molecule Ubiquitination Inhibitor Blocks NF-ÎºB-dependent Cytokine Expression in Cells and Rats

Models of Inflammation: Carrageenan Air Pouch in the Rat

Models of inflammation: measuring gastrointestinal ulceration in the rat

BK virus T antigens induce kidney carcinomas and thymoproliferative disorders in transgenic mice

A novel series of IKKβ inhibitors part I: Initial SAR studies of a HTS hit

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