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CCR1 blockade reduces tumor burden and osteolysis in vivo in a mouse model of myeloma bone disease

Blood, 2012-08, Vol.120 (7), p.1449-1457

2012

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Pharmacokinetic and Pharmacodynamic Evaluation of the Novel CCR1 Antagonist CCX354 in Healthy Human Subjects: Implications for Selection of Clinical Dose

Clinical pharmacology and therapeutics, 2011-05, Vol.89 (5), p.726-734

2011

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Discovery and initial SAR of inhibitors of interleukin-1 receptor-associated kinase-4

Bioorganic & medicinal chemistry letters, 2006-06, Vol.16 (11), p.2842-2845

2006

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OP0204 Characterization of the novel C5AR antagonist CCX168, a potential therapeutic for ANCA-vasculitis, rheumatoid arthritis, and other autoimmune disorders

Annals of the rheumatic diseases, 2013-06, Vol.71 (Suppl 3), p.124-124

2013

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Selective, Covalent Modification of β -Tubulin Residue Cys-239 by T138067, an Antitumor Agent with in vivo Efficacy against Multidrug-Resistant Tumors

Proceedings of the National Academy of Sciences - PNAS, 1999-05, Vol.96 (10), p.5686-5691

1999

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2-Amino-4H-3,1-benzoxazin-4-ones as Inhibitors of C1r Serine Protease

Journal of medicinal chemistry, 1998-03, Vol.41 (7), p.1060-1067

1998

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Novel halogenated sulfonamides inhibit the growth of multidrug resistant MCF-7/ADR cancer cells

Bioorganic & medicinal chemistry letters, 1999-07, Vol.9 (13), p.1843-1846

1999

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Secreted Site-1 Protease Cleaves Peptides Corresponding to Luminal Loop of Sterol Regulatory Element-binding Proteins

The Journal of biological chemistry, 1999-08, Vol.274 (32), p.22805-22812

1999

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Hydrophilic, Pro-Drug Analogues of T138067 Are Efficacious in Controlling Tumor Growth In Vivo and Show a Decreased Ability To Cross the Blood Brain Barrier

Journal of medicinal chemistry, 2001-10, Vol.44 (22), p.3599-3605

2001

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Novel antineoplastic agents with efficacy against multidrug resistant tumor cells

Bioorganic & medicinal chemistry letters, 1998-10, Vol.8 (19), p.2653-2656

1998

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Advances in the Discovery of C5a Receptor Antagonists

Annual Reports in Medicinal Chemistry, 2011, Vol.46, p.171-186

2011

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4-(1,2,5,6-Tetrahydro-1-alkyl-3-pyridinyl)-2-thiazolamines: a novel class of compounds with central dopamine agonist properties

Journal of medicinal chemistry, 1990-01, Vol.33 (1), p.311-317

1990

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Identification and characterization of m4 selective muscarinic antagonists

Bioorganic & medicinal chemistry letters, 1998-08, Vol.8 (15), p.1991-1996

1998

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Design and Synthesis of m1-Selective Muscarinic Agonists: (R)-(−)-(Z)-1-Azabicyclo[2.2.1]heptan-3-one, O-(3-(3‘-Methoxyphenyl)-2-propynyl)- oxime Maleate (CI-1017), a Functionally m1-Selective Muscarinic Agonist

Journal of medicinal chemistry, 1998-07, Vol.41 (14), p.2524-2536

1998

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Acetylcholinesterase inhibition by fused dihydroquinazoline compounds

Bioorganic & medicinal chemistry letters, 1996-03, Vol.6 (6), p.737-742

1996

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Aryl 1-But-3-ynyl-4-phenyl-1,2,3,6-tetrahydropyridines as Potential Antipsychotic Agents: Synthesis and Structure−Activity Relationships

Journal of medicinal chemistry, 1996-08, Vol.39 (16), p.3179-3187

1996

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Synthesis and evaluation of 2-aryl-4H-3,1-benzoxazin-4-ones as C1r serine protease inhibitors

Bioorganic & medicinal chemistry letters, 1996-03, Vol.6 (6), p.679-682

1996

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Kynurenic Acid Derivatives Inhibit the Binding of Nerve Growth Factor (NGF) to the Low-Affinity p75 NGF Receptor

Journal of medicinal chemistry, 1995-10, Vol.38 (22), p.4439-4445

1995

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Identification and Characterization of m1 Selective Muscarinic Receptor Antagonists

Journal of medicinal chemistry, 1999-02, Vol.42 (3), p.356-363

1999

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2-(1,3,5-Dithiazinan-5-yl)ethanol Heterocycles, Structure and Reactivity

Heterocycles, 2004-10, Vol.63 (10), p.2269

2004

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Evaluation of the effects of the enantiomers of reduced haloperidol, azaperol, and related 4-amino-1-arylbutanols on dopamine and .sigma. receptors

Journal of medicinal chemistry, 1993-11, Vol.36 (24), p.3929-3936

1993

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Identification of a 3-Hydroxylated Tacrine Metabolite in Rat and Man: Metabolic Profiling Implications and Pharmacology

Journal of medicinal chemistry, 1996-07, Vol.39 (15), p.3014-3018

1996

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The Discovery and Structure-Activity Relationships of 1,2,3,6-Tetrahydro-4-phenyl-1-[(arylcyclohexenyl)alkyl]pyridines. Dopamine Autoreceptor Agonists and Potential Antipsychotic Agents

Journal of medicinal chemistry, 1994-10, Vol.37 (21), p.3523-3533

1994

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Characterization of muscarinic agonists in recombinant cell lines

Life sciences (1973), 1993, Vol.52 (5), p.465-472

1993

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Dopamine autoreceptor agonists as potential antipsychotics. 2. (Aminoalkoxy)-4H-1-benzopyran-4-ones

Journal of medicinal chemistry, 1991-01, Vol.34 (1), p.248-256

1991

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CCR1 blockade reduces tumor burden and osteolysis in vivo in a mouse model of myeloma bone disease

Pharmacokinetic and Pharmacodynamic Evaluation of the Novel CCR1 Antagonist CCX354 in Healthy Human Subjects: Implications for Selection of Clinical Dose

Discovery and initial SAR of inhibitors of interleukin-1 receptor-associated kinase-4

OP0204 Characterization of the novel C5AR antagonist CCX168, a potential therapeutic for ANCA-vasculitis, rheumatoid arthritis, and other autoimmune disorders

Selective, Covalent Modification of β -Tubulin Residue Cys-239 by T138067, an Antitumor Agent with in vivo Efficacy against Multidrug-Resistant Tumors

2-Amino-4H-3,1-benzoxazin-4-ones as Inhibitors of C1r Serine Protease

Novel halogenated sulfonamides inhibit the growth of multidrug resistant MCF-7/ADR cancer cells

Secreted Site-1 Protease Cleaves Peptides Corresponding to Luminal Loop of Sterol Regulatory Element-binding Proteins

Hydrophilic, Pro-Drug Analogues of T138067 Are Efficacious in Controlling Tumor Growth In Vivo and Show a Decreased Ability To Cross the Blood Brain Barrier

Novel antineoplastic agents with efficacy against multidrug resistant tumor cells

Advances in the Discovery of C5a Receptor Antagonists

4-(1,2,5,6-Tetrahydro-1-alkyl-3-pyridinyl)-2-thiazolamines: a novel class of compounds with central dopamine agonist properties

Identification and characterization of m4 selective muscarinic antagonists

Design and Synthesis of m1-Selective Muscarinic Agonists: (R)-(−)-(Z)-1-Azabicyclo[2.2.1]heptan-3-one, O-(3-(3‘-Methoxyphenyl)-2-propynyl)- oxime Maleate (CI-1017), a Functionally m1-Selective Muscarinic Agonist

Acetylcholinesterase inhibition by fused dihydroquinazoline compounds

Aryl 1-But-3-ynyl-4-phenyl-1,2,3,6-tetrahydropyridines as Potential Antipsychotic Agents: Synthesis and Structure−Activity Relationships

Synthesis and evaluation of 2-aryl-4H-3,1-benzoxazin-4-ones as C1r serine protease inhibitors

Kynurenic Acid Derivatives Inhibit the Binding of Nerve Growth Factor (NGF) to the Low-Affinity p75 NGF Receptor

Identification and Characterization of m1 Selective Muscarinic Receptor Antagonists

2-(1,3,5-Dithiazinan-5-yl)ethanol Heterocycles, Structure and Reactivity

Evaluation of the effects of the enantiomers of reduced haloperidol, azaperol, and related 4-amino-1-arylbutanols on dopamine and .sigma. receptors

Identification of a 3-Hydroxylated Tacrine Metabolite in Rat and Man: Metabolic Profiling Implications and Pharmacology

The Discovery and Structure-Activity Relationships of 1,2,3,6-Tetrahydro-4-phenyl-1-[(arylcyclohexenyl)alkyl]pyridines. Dopamine Autoreceptor Agonists and Potential Antipsychotic Agents

Characterization of muscarinic agonists in recombinant cell lines

Dopamine autoreceptor agonists as potential antipsychotics. 2. (Aminoalkoxy)-4H-1-benzopyran-4-ones

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