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High-precision realization for sensing charged particles based on optomechanically induced two-color second-order sidebands

Journal of applied physics, 2023-12, Vol.134 (23)

2023

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Successful generation of structural information for fragment-based drug discovery

Drug discovery today, 2015-09, Vol.20 (9), p.1104-1111

2015

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Discovery of benzothiazole guanidines as novel inhibitors of thrombin and trypsin IV

Bioorganic & medicinal chemistry letters, 2012-07, Vol.22 (14), p.4839-4843

2012

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Structural Insights and Biological Effects of Glycogen Synthase Kinase 3-specific Inhibitor AR-A014418

The Journal of biological chemistry, 2003-11, Vol.278 (46), p.45937-45945

2003

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Discovery of Checkpoint Kinase Inhibitor (S)-5-(3-Fluorophenyl)-N-(piperidin-3-yl)-3-ureidothiophene-2-carboxamide (AZD7762) by Structure-Based Design and Optimization of Thiophenecarboxamide Ureas

Journal of medicinal chemistry, 2012-06, Vol.55 (11), p.5130-5142

2012

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Total Synthesis and Structural Confirmation of Chlorodysinosin A

Journal of the American Chemical Society, 2006-08, Vol.128 (32), p.10491-10495

2006

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Synthesis and structure-activity relationship of 4-(1,3-benzothiazol-2-yl)-thiophene-2-sulfonamides as cyclin-dependent kinase 5 (cdk5)/p25 inhibitors

Bioorganic & medicinal chemistry letters, 2012-09, Vol.22 (18), p.5919-5923

2012

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Exploitation of structural and regulatory diversity in glutamate racemases

Nature, 2007-06, Vol.447 (7146), p.817-822

2007

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Compounds Binding to the S2−S3 Pockets of Thrombin

Journal of medicinal chemistry, 2009-05, Vol.52 (9), p.2708-2715

2009

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Clavatadine A, A Natural Product with Selective Recognition and Irreversible Inhibition of Factor XIa

Journal of medicinal chemistry, 2008-06, Vol.51 (12), p.3583-3587

2008

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Design and synthesis of 2′-anilino-4,4′-bipyridines as selective inhibitors of c-Jun N-terminal kinase-3

Bioorganic & medicinal chemistry letters, 2006-03, Vol.16 (5), p.1397-1401

2006

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Experimental Study on Water Production Function for Waterlogging Stress on Corn

Procedia engineering, 2012, Vol.28, p.598-603

2012

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Discovery of the Fibrinolysis Inhibitor AZD6564, Acting via Interference of a Protein–Protein Interaction

ACS medicinal chemistry letters, 2014-05, Vol.5 (5), p.538-543

2014

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Structure-based organic synthesis of unnatural aeruginosin hybrids as potent inhibitors of thrombin

Bioorganic & medicinal chemistry letters, 2007-06, Vol.17 (12), p.3480-3485

2007

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Design and synthesis of 6-anilinoindazoles as selective inhibitors of c-Jun N-terminal kinase-3

Bioorganic & medicinal chemistry letters, 2005-11, Vol.15 (22), p.5095-5099

2005

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From natural products to achiral drug prototypes: Potent thrombin inhibitors based on P2/P3 dihydropyrid-2-one core motifs

Bioorganic & medicinal chemistry letters, 2009-09, Vol.19 (18), p.5429-5432

2009

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Hit-to-lead studies: the discovery of potent, orally active, thiophenecarboxamide IKK-2 inhibitors

Bioorganic & medicinal chemistry letters, 2004-06, Vol.14 (11), p.2817-2822

2004

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Structure-driven HtL: Design and synthesis of novel aminoindazole inhibitors of c-Jun N-terminal kinase activity

Bioorganic & medicinal chemistry letters, 2005-07, Vol.15 (14), p.3459-3462

2005

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Structure-based ligand design to overcome CYP inhibition in drug discovery projects

Drug discovery today, 2014-07, Vol.19 (7), p.905-911

2014

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Fragment Screening of RORγt Using Cocktail Crystallography: Identification of Simultaneous Binding of Multiple Fragments

ChemMedChem, 2016-09, Vol.11 (17), p.1881-1885

2016

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Crystal structure of spinach plastocyanin at 1.7 Å resolution

Protein science, 1998-10, Vol.7 (10), p.2099-2105

1998

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Phenolic P2/P3 core motif as thrombin inhibitors : Design, synthesis, and X-ray co-crystal structure

Bioorganic & medicinal chemistry letters, 2006-02, Vol.16 (4), p.1032-1036

2006

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A Strategically Positioned Cation Is Crucial for Efficient Catalysis by Chorismate Mutase

The Journal of biological chemistry, 2000-11, Vol.275 (47), p.36832-36838

2000

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Analysis of underground pressure in fully mechanized top coal caving mining face in greater inclined and weak coal seam

IOP conference series. Earth and environmental science, 2020-06, Vol.526 (1), p.12116

2020

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Fragment Screening of ROR[gamma]t Using Cocktail Crystallography: Identification of Simultaneous Binding of Multiple Fragments

ChemMedChem, 2016-09, Vol.11 (17), p.1881

2016

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High-precision realization for sensing charged particles based on optomechanically induced two-color second-order sidebands

Successful generation of structural information for fragment-based drug discovery

Discovery of benzothiazole guanidines as novel inhibitors of thrombin and trypsin IV

Structural Insights and Biological Effects of Glycogen Synthase Kinase 3-specific Inhibitor AR-A014418

Discovery of Checkpoint Kinase Inhibitor (S)-5-(3-Fluorophenyl)-N-(piperidin-3-yl)-3-ureidothiophene-2-carboxamide (AZD7762) by Structure-Based Design and Optimization of Thiophenecarboxamide Ureas

Total Synthesis and Structural Confirmation of Chlorodysinosin A

Synthesis and structure-activity relationship of 4-(1,3-benzothiazol-2-yl)-thiophene-2-sulfonamides as cyclin-dependent kinase 5 (cdk5)/p25 inhibitors

Exploitation of structural and regulatory diversity in glutamate racemases

Compounds Binding to the S2−S3 Pockets of Thrombin

Clavatadine A, A Natural Product with Selective Recognition and Irreversible Inhibition of Factor XIa

Design and synthesis of 2′-anilino-4,4′-bipyridines as selective inhibitors of c-Jun N-terminal kinase-3

Experimental Study on Water Production Function for Waterlogging Stress on Corn

Discovery of the Fibrinolysis Inhibitor AZD6564, Acting via Interference of a Protein–Protein Interaction

Structure-based organic synthesis of unnatural aeruginosin hybrids as potent inhibitors of thrombin

Design and synthesis of 6-anilinoindazoles as selective inhibitors of c-Jun N-terminal kinase-3

From natural products to achiral drug prototypes: Potent thrombin inhibitors based on P2/P3 dihydropyrid-2-one core motifs

Hit-to-lead studies: the discovery of potent, orally active, thiophenecarboxamide IKK-2 inhibitors

Structure-driven HtL: Design and synthesis of novel aminoindazole inhibitors of c-Jun N-terminal kinase activity

Structure-based ligand design to overcome CYP inhibition in drug discovery projects

Fragment Screening of RORγt Using Cocktail Crystallography: Identification of Simultaneous Binding of Multiple Fragments

Crystal structure of spinach plastocyanin at 1.7 Å resolution

Phenolic P2/P3 core motif as thrombin inhibitors : Design, synthesis, and X-ray co-crystal structure

A Strategically Positioned Cation Is Crucial for Efficient Catalysis by Chorismate Mutase

Analysis of underground pressure in fully mechanized top coal caving mining face in greater inclined and weak coal seam

Fragment Screening of ROR[gamma]t Using Cocktail Crystallography: Identification of Simultaneous Binding of Multiple Fragments

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