UB Paderborn / Katalog / Suche / in CDI

1 – 25 von 31

Sortiert nach

A road map to evaluate the proteome-wide selectivity of covalent kinase inhibitors

Nature chemical biology, 2014-09, Vol.10 (9), p.760

2014

Link zum Volltext

Verfügbarkeit prüfen

Comprehensive Peptidomimetic Libraries Targeting Protein–Protein Interactions

Accounts of chemical research, 2012-10, Vol.45 (10), p.1698-1709

2012

Link zum Volltext

Verfügbarkeit prüfen

Selective inhibitors of JAK1 targeting an isoform-restricted allosteric cysteine

Nature chemical biology, 2022-12, Vol.18 (12), p.1388

2022

Link zum Volltext

Verfügbarkeit prüfen

TLR4/MD-2 activation by a synthetic agonist with no similarity to LPS

Proceedings of the National Academy of Sciences - PNAS, 2016-02, Vol.113 (7), p.E884-E893

2016

Link zum Volltext

Verfügbarkeit prüfen

Metabolically Labile Fumarate Esters Impart Kinetic Selectivity to Irreversible Inhibitors

Journal of the American Chemical Society, 2016-12, Vol.138 (49), p.15841-15844

2016

Link zum Volltext

Verfügbarkeit prüfen

Development and Optimization of Piperidyl-1,2,3-Triazole Ureas as Selective Chemical Probes of Endocannabinoid Biosynthesis

Journal of medicinal chemistry, 2013-11, Vol.56 (21), p.8257-8269

2013

Link zum Volltext

Verfügbarkeit prüfen

Discovery and Optimization of Piperidyl-1,2,3-Triazole Ureas as Potent, Selective, and in Vivo-Active Inhibitors of α/β-Hydrolase Domain Containing 6 (ABHD6)

Journal of medicinal chemistry, 2013-11, Vol.56 (21), p.8270-8279

2013

Link zum Volltext

Verfügbarkeit prüfen

Design, Synthesis, and Validation of a β-Turn Mimetic Library Targeting Protein–Protein and Peptide–Receptor Interactions

Journal of the American Chemical Society, 2011-07, Vol.133 (26), p.10184-10194

2011

Link zum Volltext

Verfügbarkeit prüfen

Small-Molecule Fusion Inhibitors Bind the pH-Sensing Stable Signal Peptide-GP2 Subunit Interface of the Lassa Virus Envelope Glycoprotein

Journal of virology, 2016-08, Vol.90 (15), p.6799-6807

2016

Link zum Volltext

Verfügbarkeit prüfen

Quantitative Chemical Proteomic Profiling of the in Vivo Targets of Reactive Drug Metabolites

ACS chemical biology, 2017-08, Vol.12 (8), p.2040-2050

2017

Link zum Volltext

Verfügbarkeit prüfen

Design, Synthesis, and Evaluation of an α-Helix Mimetic Library Targeting Protein−Protein Interactions

Journal of the American Chemical Society, 2009-04, Vol.131 (15), p.5564-5572

2009

Link zum Volltext

Verfügbarkeit prüfen

Inhibition of adenovirus replication by a trisubstituted piperazin-2-one derivative

Antiviral research, 2014-08, Vol.108, p.65-73

2014

Link zum Volltext

Verfügbarkeit prüfen

SAR studies of 4-acyl-1,6-dialkylpiperazin-2-one arenavirus cell entry inhibitors

Bioorganic & medicinal chemistry letters, 2019-11, Vol.29 (22), p.126620-126620, Article 126620

2019

Link zum Volltext

Verfügbarkeit prüfen

Small molecule inhibitors of Myc/Max dimerization and Myc-induced cell transformation

Bioorganic & medicinal chemistry letters, 2009-11, Vol.19 (21), p.6038-6041

2009

Link zum Volltext

Verfügbarkeit prüfen

Small molecule inhibitors of the RNA-dependent protein kinase

Biochemical and biophysical research communications, 2003-08, Vol.308 (1), p.50-57

2003

Link zum Volltext

Verfügbarkeit prüfen

Discovery of HIV fusion inhibitors targeting gp41 using a comprehensive α-helix mimetic library

Bioorganic & medicinal chemistry letters, 2012-04, Vol.22 (8), p.2861-2865

2012

Link zum Volltext

Verfügbarkeit prüfen

NMR-assisted computational studies of peptidomimetic inhibitors bound in the hydrophobic pocket of HIV-1 glycoprotein 41

Journal of computer-aided molecular design, 2013-07, Vol.27 (7), p.569-582

2013

Link zum Volltext

Verfügbarkeit prüfen

Selective inhibitors and tailored activity probes for lipoprotein-associated phospholipase A2

Bioorganic & medicinal chemistry letters, 2013-02, Vol.23 (3), p.839-843

2013

Link zum Volltext

Verfügbarkeit prüfen

Selective inhibitors and tailored activity probes for lipoprotein-associated phospholipase A

Bioorganic & medicinal chemistry letters, 2013-02, Vol.23 (3), p.839-843

2013

Link zum Volltext

Verfügbarkeit prüfen

Controlling activation of the RNA-dependent protein kinase by siRNAs using site-specific chemical modification

Nucleic acids research, 2006-10, Vol.34 (17), p.4900

2006

Link zum Volltext

Verfügbarkeit prüfen

Identification of broad-based HIV-1 protease inhibitors from combinatorial libraries

Biochemical journal, 2010-08, Vol.429 (3), p.527-532

2010

Link zum Volltext

Verfügbarkeit prüfen

Small molecule peptidomimetic inhibitors of importin α/β mediated nuclear transport

Bioorganic & medicinal chemistry, 2010-11, Vol.18 (21), p.7611-7620

2010

Link zum Volltext

Verfügbarkeit prüfen

Characterization of lassa virus cell entry inhibitors: Determination of the active enantiomer by asymmetric synthesis

Bioorganic & medicinal chemistry letters, 2009-07, Vol.19 (14), p.3771-3774

2009

Link zum Volltext

Verfügbarkeit prüfen

Abstract 6411: Discovery of covalent ligands to novel E3 ligases enables bispecific degraders with highly differentiated protein degradation across a broad range of targets

Cancer research (Chicago, Ill.), 2020-08, Vol.80 (16_Supplement), p.6411-6411

2020

Link zum Volltext

Verfügbarkeit prüfen

1 – 25 von 31

Suche als RSS-Feed

Suchergebnisse filtern

Filter anzeigen

Nur zeigen

Geprüft (Peer-Review)
(31)
Mit Volltextzugriff
(28)

Publikationsform

Artikel
(31)

Sprache

Englisch
(31)
Japanisch
(6)

Erscheinungsjahr

n.n

Thema

15 weitere anzeigen...

Weniger anzeigen...

Menü

Weitere Dienste

Einstellungen

A road map to evaluate the proteome-wide selectivity of covalent kinase inhibitors

Comprehensive Peptidomimetic Libraries Targeting Protein–Protein Interactions

Selective inhibitors of JAK1 targeting an isoform-restricted allosteric cysteine

TLR4/MD-2 activation by a synthetic agonist with no similarity to LPS

Metabolically Labile Fumarate Esters Impart Kinetic Selectivity to Irreversible Inhibitors

Development and Optimization of Piperidyl-1,2,3-Triazole Ureas as Selective Chemical Probes of Endocannabinoid Biosynthesis

Discovery and Optimization of Piperidyl-1,2,3-Triazole Ureas as Potent, Selective, and in Vivo-Active Inhibitors of α/β-Hydrolase Domain Containing 6 (ABHD6)

Proteomic discovery of chemical probes that perturb protein complexes in human cells

Design, Synthesis, and Validation of a β-Turn Mimetic Library Targeting Protein–Protein and Peptide–Receptor Interactions

Small-Molecule Fusion Inhibitors Bind the pH-Sensing Stable Signal Peptide-GP2 Subunit Interface of the Lassa Virus Envelope Glycoprotein

Quantitative Chemical Proteomic Profiling of the in Vivo Targets of Reactive Drug Metabolites

Design, Synthesis, and Evaluation of an α-Helix Mimetic Library Targeting Protein−Protein Interactions

Inhibition of adenovirus replication by a trisubstituted piperazin-2-one derivative

SAR studies of 4-acyl-1,6-dialkylpiperazin-2-one arenavirus cell entry inhibitors

Small molecule inhibitors of Myc/Max dimerization and Myc-induced cell transformation

Small molecule inhibitors of the RNA-dependent protein kinase

Discovery of HIV fusion inhibitors targeting gp41 using a comprehensive α-helix mimetic library

NMR-assisted computational studies of peptidomimetic inhibitors bound in the hydrophobic pocket of HIV-1 glycoprotein 41

Selective inhibitors and tailored activity probes for lipoprotein-associated phospholipase A2

Selective inhibitors and tailored activity probes for lipoprotein-associated phospholipase A

Controlling activation of the RNA-dependent protein kinase by siRNAs using site-specific chemical modification

Identification of broad-based HIV-1 protease inhibitors from combinatorial libraries

Small molecule peptidomimetic inhibitors of importin α/β mediated nuclear transport

Characterization of lassa virus cell entry inhibitors: Determination of the active enantiomer by asymmetric synthesis

Abstract 6411: Discovery of covalent ligands to novel E3 ligases enables bispecific degraders with highly differentiated protein degradation across a broad range of targets

Suchergebnisse filtern