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Identification of Novel Inhibitors of the Transforming Growth Factor β1 (TGF-β1) Type 1 Receptor (ALK5)

Journal of medicinal chemistry, 2002-02, Vol.45 (5), p.999-1001

2002

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SB-431542 is a potent and specific inhibitor of transforming growth factor-beta superfamily type I activin receptor-like kinase (ALK) receptors ALK4, ALK5, and ALK7

Molecular pharmacology, 2002-07, Vol.62 (1), p.65-74

2002

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3,4-Dihydro-2H-benzoxazinones are 5-HT1A receptor antagonists with potent 5-HT reuptake inhibitory activity

Bioorganic & medicinal chemistry letters, 2005-02, Vol.15 (3), p.737-741

2005

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Serotonin 5-HT3 and 5-HT4 receptor antagonists

Medicinal research reviews, 1997-03, Vol.17 (2), p.163-214

1997

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8-piperazinyl-2,3-dihydropyrrolo[3,2-g]isoquinolines : Potent, selective, orally bioavailable 5-HT1 receptor ligands

Bioorganic & medicinal chemistry letters, 2005-10, Vol.15 (19), p.4370-4374

2005

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N-[(1-Butyl-4-piperidinyl)methyl]-3,4- dihydro-2H-[1,3]oxazino[3,2-a]indole- 10-carboxamide hydrochloride: the first potent and selective 5-HT4 receptor antagonist amide with oral activity

Journal of medicinal chemistry, 1995-11, Vol.38 (24), p.4760-4763

1995

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(.+-.)-3-Amino-6-carboxamido-1,2,3,4-tetrahydrocarbazole: a conformationally restricted analog of 5-carboxamidotryptamine with selectivity for the serotonin 5-HT1D receptor

Journal of medicinal chemistry, 1993-06, Vol.36 (13), p.1918-1919

1993

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(1-Butyl-4-piperidinyl)methyl 8-amino-7-chloro-1,4-benzodioxane-5-carboxylate hydrochloride: a highly potent and selective 5-HT4 receptor antagonist derived from metoclopramide

Journal of medicinal chemistry, 1993-12, Vol.36 (25), p.4121-4123

1993

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4-(6-Methoxy-2-naphthyl)butan-2-one and related analogs, a novel structural class of antiinflammatory compounds

Journal of medicinal chemistry, 1978-12, Vol.21 (12), p.1260-1264

1978

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Overview Central & Peripheral Nervous System: 5-HT4 receptor antagonists

Expert opinion on therapeutic patents, 1994-04, Vol.4 (4), p.323-332

1994

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Biarylcarbamoylindolines are novel and selective 5-HT(2C) receptor inverse agonists: identification of 5-methyl-1-[[2-[(2-methyl-3-pyridyl)oxy]- 5-pyridyl]carbamoyl]-6-trifluoromethylindoline (SB-243213) as a potential antidepressant/anxiolytic agent

Journal of medicinal chemistry, 2000-03, Vol.43 (6), p.1123-1134

2000

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Substituted 3-amino-1,1-diaryl-2-propanols as potential antidepressant agents

Journal of medicinal chemistry, 1979-11, Vol.22 (11), p.1373-1379

1979

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(.+-.)-3-Amino-6-carboxamido-1,2,3,4-tetrahydrocarbazole: A conformationally restricted analog of 5-carboxamidotryptamine with selectivity for the serotonin 5-HT1D receptor. [Erratum to document cited in CA119(11):117079z]

Journal of medicinal chemistry, 1993-10, Vol.36 (21), p.3218-3218

1993

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SB-236057, a selective 5-HT1B receptor inverse agonist, blocks the 5-HT human terminal autoreceptor

European journal of pharmacology, 1999-06, Vol.375 (1-3), p.359-365

1999

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3,4-Dihydro-2H-benzoxazinones are 5-HT(1A) receptor antagonists with potent 5-HT reuptake inhibitory activity

Bioorganic & medicinal chemistry letters, 2005-02, Vol.15 (3), p.737-741

2005

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3,4-Dihydro-2 H-benzoxazinones are 5-HT 1A receptor antagonists with potent 5-HT reuptake inhibitory activity

Bioorganic & medicinal chemistry letters, 2005, Vol.15 (3), p.737-741

2005

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8-Piperazinyl-2,3-dihydropyrrolo[3,2- g]isoquinolines: Potent, selective, orally bioavailable 5-HT 1 receptor ligands

Bioorganic & medicinal chemistry letters, 2005, Vol.15 (19), p.4370-4374

2005

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SB-431542 Is a Potent and Specific Inhibitor of Transforming Growth Factor-Î² Superfamily Type I Activin Receptor-Like Kinase (ALK) Receptors ALK4, ALK5, and ALK7

Molecular pharmacology, 2002-07, Vol.62 (1), p.65

2002

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Increased defaecation caused by 5-HT4 receptor activation in the mouse

European journal of pharmacology, 1996-07, Vol.308 (2), p.181-186

1996

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Identification of novel inhibitors of the transforming growth factor beta1 (TGF-beta1) type 1 receptor (ALK5)

Journal of medicinal chemistry, 2002-02, Vol.45 (5), p.999-1001

2002

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SB-236057, a selective 5-HT 1B receptor inverse agonist, blocks the 5-HT human terminal autoreceptor

European journal of pharmacology, 1999, Vol.375 (1), p.359-365

1999

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Overview Central & Peripheral Nervous System: 5-HT 4 receptor antagonists

Expert opinion on therapeutic patents, 1994-04, Vol.4 (4), p.323-332

1994

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Blockade of human atrial 5-HT4 receptors by SB 207710, a selective and high affinity 5-HT4 receptor antagonist

Naunyn-Schmiedeberg's archives of pharmacology, 1994-05, Vol.349 (5), p.546-548

1994

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Identification of Novel Inhibitors of the Transforming Growth Factor β1 (TGF-β1) Type 1 Receptor (ALK5)

SB-431542 is a potent and specific inhibitor of transforming growth factor-beta superfamily type I activin receptor-like kinase (ALK) receptors ALK4, ALK5, and ALK7

3,4-Dihydro-2H-benzoxazinones are 5-HT1A receptor antagonists with potent 5-HT reuptake inhibitory activity

Serotonin 5-HT3 and 5-HT4 receptor antagonists

Biarylcarbamoylindolines Are Novel and Selective 5-HT2C Receptor Inverse Agonists: Identification of 5-Methyl-1-[[2-[(2-methyl-3-pyridyl)oxy]- 5-pyridyl]carbamoyl]-6-trifluoromethylindoline (SB-243213) as a Potential Antidepressant/Anxiolytic Agent

8-piperazinyl-2,3-dihydropyrrolo[3,2-g]isoquinolines : Potent, selective, orally bioavailable 5-HT1 receptor ligands

N-[(1-Butyl-4-piperidinyl)methyl]-3,4- dihydro-2H-[1,3]oxazino[3,2-a]indole- 10-carboxamide hydrochloride: the first potent and selective 5-HT4 receptor antagonist amide with oral activity

(.+-.)-3-Amino-6-carboxamido-1,2,3,4-tetrahydrocarbazole: a conformationally restricted analog of 5-carboxamidotryptamine with selectivity for the serotonin 5-HT1D receptor

(1-Butyl-4-piperidinyl)methyl 8-amino-7-chloro-1,4-benzodioxane-5-carboxylate hydrochloride: a highly potent and selective 5-HT4 receptor antagonist derived from metoclopramide

4-(6-Methoxy-2-naphthyl)butan-2-one and related analogs, a novel structural class of antiinflammatory compounds

Overview Central & Peripheral Nervous System: 5-HT4 receptor antagonists

Biarylcarbamoylindolines are novel and selective 5-HT(2C) receptor inverse agonists: identification of 5-methyl-1-[[2-[(2-methyl-3-pyridyl)oxy]- 5-pyridyl]carbamoyl]-6-trifluoromethylindoline (SB-243213) as a potential antidepressant/anxiolytic agent

Substituted 3-amino-1,1-diaryl-2-propanols as potential antidepressant agents

(.+-.)-3-Amino-6-carboxamido-1,2,3,4-tetrahydrocarbazole: A conformationally restricted analog of 5-carboxamidotryptamine with selectivity for the serotonin 5-HT1D receptor. [Erratum to document cited in CA119(11):117079z]

SB-236057, a selective 5-HT1B receptor inverse agonist, blocks the 5-HT human terminal autoreceptor

3,4-Dihydro-2H-benzoxazinones are 5-HT(1A) receptor antagonists with potent 5-HT reuptake inhibitory activity

3,4-Dihydro-2 H-benzoxazinones are 5-HT 1A receptor antagonists with potent 5-HT reuptake inhibitory activity

8-Piperazinyl-2,3-dihydropyrrolo[3,2- g]isoquinolines: Potent, selective, orally bioavailable 5-HT 1 receptor ligands

SB-431542 Is a Potent and Specific Inhibitor of Transforming Growth Factor-Î² Superfamily Type I Activin Receptor-Like Kinase (ALK) Receptors ALK4, ALK5, and ALK7

Increased defaecation caused by 5-HT4 receptor activation in the mouse

Identification of novel inhibitors of the transforming growth factor beta1 (TGF-beta1) type 1 receptor (ALK5)

SB-236057, a selective 5-HT 1B receptor inverse agonist, blocks the 5-HT human terminal autoreceptor

Biarylcarbamoylindolines Are Novel and Selective 5-HT 2C Receptor Inverse Agonists: Identification of 5-Methyl-1-[[2-[(2-methyl-3-pyridyl)oxy]- 5-pyridyl]carbamoyl]-6-trifluoromethylindoline (SB-243213) as a Potential Antidepressant/Anxiolytic Agent

Overview Central & Peripheral Nervous System: 5-HT 4 receptor antagonists

Blockade of human atrial 5-HT4 receptors by SB 207710, a selective and high affinity 5-HT4 receptor antagonist

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