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Strategies for the Selective Regulation of Kinases with Allosteric Modulators: Exploiting Exclusive Structural Features

ACS chemical biology, 2013-01, Vol.8 (1), p.58-70

2013

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Natural-product-derived fragments for fragment-based ligand discovery

Nature chemistry, 2013-01, Vol.5 (1), p.21

2013

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Development of a Fluorescent-Tagged Kinase Assay System for the Detection and Characterization of Allosteric Kinase Inhibitors

Journal of the American Chemical Society, 2009-09, Vol.131 (37), p.13286-13296

2009

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Potent inhibition of HIV-1 by TRIM5-cyclophilin fusion proteins engineered from human components

The Journal of clinical investigation, 2009-10, Vol.119 (10), p.3035-3047

2009

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ALK Mutations Conferring Differential Resistance to Structurally Diverse ALK Inhibitors

Clinical cancer research, 2011-12, Vol.17 (23), p.7394-7401

2011

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Targeting Drug Resistance in EGFR with Covalent Inhibitors: A Structure-Based Design Approach

Journal of medicinal chemistry, 2015-09, Vol.58 (17), p.6844-6863

2015

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Selective Detection of Allosteric Phosphatase Inhibitors

Journal of the American Chemical Society, 2013-05, Vol.135 (18), p.6838-6841

2013

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Hybrid Compound Design To Overcome the Gatekeeper T338M Mutation in cSrc

Journal of medicinal chemistry, 2009-07, Vol.52 (13), p.3915-3926

2009

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Skepinone-L is a selective p38 mitogen-activated protein kinase inhibitor

Nature chemical biology, 2011-12, Vol.8 (2), p.141

2011

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Design, Synthesis, and Biological Evaluation of Novel Disubstituted Dibenzosuberones as Highly Potent and Selective Inhibitors of p38 Mitogen Activated Protein Kinase

Journal of medicinal chemistry, 2012-06, Vol.55 (12), p.5868-5877

2012

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Identification of Type II and III DDR2 Inhibitors

Journal of medicinal chemistry, 2014-05, Vol.57 (10), p.4252-4262

2014

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Structure of the PRYSPRY-domain: Implications for autoinflammatory diseases

FEBS letters, 2006-01, Vol.580 (1), p.99-106

2006

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An Invariant Surface Patch on the TRIM5α PRYSPRY Domain Is Required for Retroviral Restriction but Dispensable for Capsid Binding

Journal of Virology, 2009-04, Vol.83 (7), p.3365-3373

2009

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A new screening assay for allosteric inhibitors of cSrc

Nature chemical biology, 2009-06, Vol.5 (6), p.394-396

2009

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Fluorophore Labeling of the Glycine-Rich Loop as a Method of Identifying Inhibitors That Bind to Active and Inactive Kinase Conformations

Journal of the American Chemical Society, 2010-03, Vol.132 (12), p.4152-4160

2010

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cytokine-neutralizing antibody as a structural mimetic of 2 receptor interactions

Proceedings of the National Academy of Sciences - PNAS, 2008-12, Vol.105 (51), p.20251-20256

2008

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Dibenzosuberones as p38 Mitogen-Activated Protein Kinase Inhibitors with Low ATP Competitiveness and Outstanding Whole Blood Activity

Journal of medicinal chemistry, 2013-01, Vol.56 (1), p.241-253

2013

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Fluorophore labeled kinase detects ligands that bind within the MAPK insert of p38α kinase

PloS one, 2012-07, Vol.7 (7), p.e39713-e39713

2012

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Targeting Gain of Function and Resistance Mutations in Abl and KIT by Hybrid Compound Design

Journal of medicinal chemistry, 2013-07, Vol.56 (14), p.5757-5772

2013

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Displacement Assay for the Detection of Stabilizers of Inactive Kinase Conformations

Journal of medicinal chemistry, 2010-01, Vol.53 (1), p.357-367

2010

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Die Pilotkantone zur Einführung des Geodatenmodells der amtlichen Vermessung DMAV Version 1.0 sind bestimmt

Cadastre : Fachzeitschrift für das schweizerische Katasterwesen, 2023-12 (43), p.11

Grütter, Christian

2023

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Identification of Ustilago maydis Aurora Kinase As a Novel Antifungal Target

ACS chemical biology, 2011-09, Vol.6 (9), p.926-933

2011

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Neues Geodatenmodell der amtlichen Vermessung DMAV : Stand der Modelldokumentation

Cadastre : Fachzeitschrift für das schweizerische Katasterwesen, 2023-04 (41), p.4

Grütter, Christian

2023

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Documentation du nouveau modèle de géodonnées de la mensuration officielle DMAV : un état des lieux

Cadastre : revue spécialisée consacrée au cadastre suisse, 2023-04 (41), p.4

Grütter, Christian

2023

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Targeting GSK3 from Ustilago maydis: Type-II Kinase Inhibitors as Potential Antifungals

ACS chemical biology, 2012-07, Vol.7 (7), p.1257-1267

2012

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Strategies for the Selective Regulation of Kinases with Allosteric Modulators: Exploiting Exclusive Structural Features

Natural-product-derived fragments for fragment-based ligand discovery

Development of a Fluorescent-Tagged Kinase Assay System for the Detection and Characterization of Allosteric Kinase Inhibitors

Potent inhibition of HIV-1 by TRIM5-cyclophilin fusion proteins engineered from human components

ALK Mutations Conferring Differential Resistance to Structurally Diverse ALK Inhibitors

Targeting Drug Resistance in EGFR with Covalent Inhibitors: A Structure-Based Design Approach

Selective Detection of Allosteric Phosphatase Inhibitors

Hybrid Compound Design To Overcome the Gatekeeper T338M Mutation in cSrc

Skepinone-L is a selective p38 mitogen-activated protein kinase inhibitor

Design, Synthesis, and Biological Evaluation of Novel Disubstituted Dibenzosuberones as Highly Potent and Selective Inhibitors of p38 Mitogen Activated Protein Kinase

Identification of Type II and III DDR2 Inhibitors

Structure of the PRYSPRY-domain: Implications for autoinflammatory diseases

An Invariant Surface Patch on the TRIM5α PRYSPRY Domain Is Required for Retroviral Restriction but Dispensable for Capsid Binding

A new screening assay for allosteric inhibitors of cSrc

Fluorophore Labeling of the Glycine-Rich Loop as a Method of Identifying Inhibitors That Bind to Active and Inactive Kinase Conformations

cytokine-neutralizing antibody as a structural mimetic of 2 receptor interactions

Dibenzosuberones as p38 Mitogen-Activated Protein Kinase Inhibitors with Low ATP Competitiveness and Outstanding Whole Blood Activity

Fluorophore labeled kinase detects ligands that bind within the MAPK insert of p38α kinase

Targeting Gain of Function and Resistance Mutations in Abl and KIT by Hybrid Compound Design

Displacement Assay for the Detection of Stabilizers of Inactive Kinase Conformations

Die Pilotkantone zur Einführung des Geodatenmodells der amtlichen Vermessung DMAV Version 1.0 sind bestimmt

Identification of Ustilago maydis Aurora Kinase As a Novel Antifungal Target

Neues Geodatenmodell der amtlichen Vermessung DMAV : Stand der Modelldokumentation

Documentation du nouveau modèle de géodonnées de la mensuration officielle DMAV : un état des lieux

Targeting GSK3 from Ustilago maydis: Type-II Kinase Inhibitors as Potential Antifungals

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