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Discovery of N-(4-methoxy-7-methylbenzo[d]thiazol-2-yl)isonicatinamide, ML293, as a novel, selective and brain penetrant positive allosteric modulator of the muscarinic 4 (M4) receptor

Bioorganic & medicinal chemistry letters, 2012-08, Vol.22 (15), p.5084-5088

2012

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Identification of ML204, a Novel Potent Antagonist That Selectively Modulates Native TRPC4/C5 Ion Channels

The Journal of biological chemistry, 2011-09, Vol.286 (38), p.33436-33446

2011

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Discovery of Potent 2-Aryl-6,7-dihydro-5 H-pyrrolo[1,2- a]imidazoles as WDR5-WIN-Site Inhibitors Using Fragment-Based Methods and Structure-Based Design

Journal of medicinal chemistry, 2018-07, Vol.61 (13), p.5623-5642

2018

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Discovery of Potent 2‑Aryl-6,7-dihydro‑5H‑pyrrolo[1,2‑a]imidazoles as WDR5-WIN-Site Inhibitors Using Fragment-Based Methods and Structure-Based Design

Journal of medicinal chemistry, 2018-07, Vol.61 (13), p.5623-5642

2018

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Discovery of thiophene inhibitors of polo-like kinase

Bioorganic & medicinal chemistry letters, 2009-02, Vol.19 (3), p.1018-1021

2009

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The discovery of VU0486846: steep SAR from a series of M 1 PAMs based on a novel benzomorpholine core

Bioorganic & medicinal chemistry letters, 2018-07, Vol.28 (12), p.2175

2018

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The discovery of VU0486846: steep SAR from a series of M1 PAMs based on a novel benzomorpholine core

Bioorganic & medicinal chemistry letters, 2018-07, Vol.28 (12), p.2175-2179

2018

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Novel M4 positive allosteric modulators derived from questioning the role and impact of a presumed intramolecular hydrogen-bonding motif in β-amino carboxamide-harboring ligands

Bioorganic & medicinal chemistry letters, 2019-02, Vol.29 (3), p.362-366

2019

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Synthesis of 1,3-diarylsubstituted indazoles utilizing a Suzuki cross-coupling/deprotection/N-arylation sequence

Tetrahedron letters, 2010-07, Vol.51 (29), p.3796-3799

2010

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Discovery and characterization of a novel series of N-phenylsulfonyl-1H-pyrrole picolinamides as positive allosteric modulators of the metabotropic glutamate receptor 4 (mGlu4)

Bioorganic & medicinal chemistry letters, 2016-07, Vol.26 (13), p.2984-2987

2016

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Synthesis of 2,3-diarylsubstituted indazoles utilizing a Suzuki cross-coupling/deprotection/N-arylation sequence

Tetrahedron letters, 2010-07, Vol.51 (29), p.3796-3799

2010

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Synthesis and SAR of a novel metabotropic glutamate receptor 4 (mGlu₄) antagonist: Unexpected ‘molecular switch’ from a closely related mGlu₄ positive allosteric modulator

Bioorganic & medicinal chemistry letters, 2011-12, Vol.21 (23), p.6955-6959

2011

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Discovery and optimization of imidazo[1,2- a]pyridine inhibitors of insulin-like growth factor-1 receptor (IGF-1R)

Bioorganic & medicinal chemistry letters, 2009-02, Vol.19 (3), p.1004-1008

2009

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Novel M 4 positive allosteric modulators derived from questioning the role and impact of a presumed intramolecular hydrogen-bonding motif in β-amino carboxamide-harboring ligands

Bioorganic & medicinal chemistry letters, 2019-02, Vol.29 (3), p.362

2019

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Discovery of Potent 2-Aryl-6,7-dihydro-5 H-pyrrolo1,2- aimidazoles as WDR5-WIN-Site Inhibitors Using Fragment-Based Methods and Structure-Based Design

Journal of medicinal chemistry, 2018-07, Vol.61 (13), p.5623

2018

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Discovery and characterization of a novel series of N -phenylsulfonyl-1 H -pyrrole picolinamides as positive allosteric modulators of the metabotropic glutamate receptor 4 (mGlu 4 )

Bioorganic & medicinal chemistry letters, 2016-07, Vol.26 (13), p.2984-2987

2016

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Synthesis and SAR of a novel metabotropic glutamate receptor 4 (mGlu 4) antagonist: Unexpected ‘molecular switch’ from a closely related mGlu 4 positive allosteric modulator

Bioorganic & medicinal chemistry letters, 2011-12, Vol.21 (23), p.6955-6959

2011

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Regioselective synthesis of benzimidazole thiophene inhibitors of polo-like kinase 1

Tetrahedron letters, 2008-10, Vol.49 (44), p.6348-6351

2008

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Synthesis and SAR of a novel metabotropic glutamate receptor 4 (mGlu sub(4) antagonist: Unexpected &; lsquo; molecular switch" from a closely related mGlu) sub(4) positive allosteric modulator

Bioorganic & medicinal chemistry letters, 2011-12, Vol.21 (23), p.6955-6959

2011

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Stereoselective synthesis of a nonracemic hydronaphthalene subunit of kijanolide

Journal of organic chemistry, 1990-04, Vol.55 (8), p.2398-2403

1990

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Matrix metalloproteinase inhibitors containing a (carboxyalkyl)amino zinc ligand : modification of the P1 and P2' residues

Journal of medicinal chemistry, 1994-03, Vol.37 (5), p.674-688

1994

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ChemInform Abstract: Synthesis of 1,3-Diaryl-Substituted Indazoles Utilizing a Suzuki Cross-Coupling/Deprotection/N-Arylation Sequence

ChemInform, 2010-11, Vol.41 (45), p.no-no

2010

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ChemInform Abstract: Regioselective Synthesis of Benzimidazole Thiophene Inhibitors of Polo-Like Kinase 1

ChemInform, 2009-02, Vol.40 (7), p.no-no

2009

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Discovery of N-(4-methoxy-7-methylbenzo[d]thiazol-2-yl)isonicatinamide, ML293, as a novel, selective and brain penetrant positive allosteric modulator of the muscarinic 4 (M4) receptor

Identification of ML204, a Novel Potent Antagonist That Selectively Modulates Native TRPC4/C5 Ion Channels

Discovery of Potent 2-Aryl-6,7-dihydro-5 H-pyrrolo[1,2- a]imidazoles as WDR5-WIN-Site Inhibitors Using Fragment-Based Methods and Structure-Based Design

Discovery of Potent 2‑Aryl-6,7-dihydro‑5H‑pyrrolo[1,2‑a]imidazoles as WDR5-WIN-Site Inhibitors Using Fragment-Based Methods and Structure-Based Design

Discovery of thiophene inhibitors of polo-like kinase

The discovery of VU0486846: steep SAR from a series of M 1 PAMs based on a novel benzomorpholine core

The discovery of VU0486846: steep SAR from a series of M1 PAMs based on a novel benzomorpholine core

Novel M4 positive allosteric modulators derived from questioning the role and impact of a presumed intramolecular hydrogen-bonding motif in β-amino carboxamide-harboring ligands

Discovery, Synthesis, and Preclinical Characterization of N‑(3-Chloro-4-fluorophenyl)‑1H‑pyrazolo[4,3‑b]pyridin-3-amine (VU0418506), a Novel Positive Allosteric Modulator of the Metabotropic Glutamate Receptor 4 (mGlu4)

Synthesis of 1,3-diarylsubstituted indazoles utilizing a Suzuki cross-coupling/deprotection/N-arylation sequence

Discovery and characterization of a novel series of N-phenylsulfonyl-1H-pyrrole picolinamides as positive allosteric modulators of the metabotropic glutamate receptor 4 (mGlu4)

Synthesis of 2,3-diarylsubstituted indazoles utilizing a Suzuki cross-coupling/deprotection/N-arylation sequence

Synthesis and SAR of a novel metabotropic glutamate receptor 4 (mGlu₄) antagonist: Unexpected ‘molecular switch’ from a closely related mGlu₄ positive allosteric modulator

Discovery and optimization of imidazo[1,2- a]pyridine inhibitors of insulin-like growth factor-1 receptor (IGF-1R)

Novel M 4 positive allosteric modulators derived from questioning the role and impact of a presumed intramolecular hydrogen-bonding motif in β-amino carboxamide-harboring ligands

Discovery of Potent 2-Aryl-6,7-dihydro-5 H-pyrrolo1,2- aimidazoles as WDR5-WIN-Site Inhibitors Using Fragment-Based Methods and Structure-Based Design

Discovery and characterization of a novel series of N -phenylsulfonyl-1 H -pyrrole picolinamides as positive allosteric modulators of the metabotropic glutamate receptor 4 (mGlu 4 )

Synthesis and SAR of a novel metabotropic glutamate receptor 4 (mGlu 4) antagonist: Unexpected ‘molecular switch’ from a closely related mGlu 4 positive allosteric modulator

Regioselective synthesis of benzimidazole thiophene inhibitors of polo-like kinase 1

Discovery, Synthesis, and Preclinical Characterization of N -(3-Chloro-4-fluorophenyl)-1 H -pyrazolo[4,3- b ]pyridin-3-amine (VU0418506), a Novel Positive Allosteric Modulator of the Metabotropic Glutamate Receptor 4 (mGlu 4 )

Synthesis and SAR of a novel metabotropic glutamate receptor 4 (mGlu sub(4) antagonist: Unexpected &; lsquo; molecular switch" from a closely related mGlu) sub(4) positive allosteric modulator

Stereoselective synthesis of a nonracemic hydronaphthalene subunit of kijanolide

Matrix metalloproteinase inhibitors containing a (carboxyalkyl)amino zinc ligand : modification of the P1 and P2' residues

ChemInform Abstract: Synthesis of 1,3-Diaryl-Substituted Indazoles Utilizing a Suzuki Cross-Coupling/Deprotection/N-Arylation Sequence

ChemInform Abstract: Regioselective Synthesis of Benzimidazole Thiophene Inhibitors of Polo-Like Kinase 1

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