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Discovery of selective biaryl ethers as PDE10A inhibitors: Improvement in potency and mitigation of Pgp-mediated efflux

Bioorganic & medicinal chemistry letters, 2012-12, Vol.22 (24), p.7371-7375

2012

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Discovery of Highly Selective and Potent p38 Inhibitors Based on a Phthalazine Scaffold

Journal of medicinal chemistry, 2008-10, Vol.51 (20), p.6271-6279

2008

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Discovery and in Vivo Evaluation of (S)‑N‑(1-(7-Fluoro-2-(pyridin-2-yl)quinolin-3-yl)ethyl)‑9H‑purin-6-amine (AMG319) and Related PI3Kδ Inhibitors for Inflammation and Autoimmune Disease

Journal of medicinal chemistry, 2015-01, Vol.58 (1), p.480-511

2015

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Palladium-Catalyzed Chemoselective Monoarylation of Hydrazides for the Synthesis of [1,2,4]Triazolo[4,3-a]pyridines

Organic letters, 2010-02, Vol.12 (4), p.792-795

2010

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Isolation and Identification of Eukaryotic Initiation Factor 4A as a Molecular Target for the Marine Natural Product Pateamine A

Methods in Enzymology, 2007, Vol.431, p.303-324

2007

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Novel Vanilloid Receptor-1 Antagonists: 2. Structure−Activity Relationships of 4-Oxopyrimidines Leading to the Selection of a Clinical Candidate

Journal of medicinal chemistry, 2007-07, Vol.50 (15), p.3515-3527

2007

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Synthesis and preliminary biological evaluation of potent and selective 2-(3-alkoxy-1-azetidinyl) quinolines as novel PDE10A inhibitors with improved solubility

Bioorganic & medicinal chemistry, 2014-12, Vol.22 (23), p.6570-6585

2014

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Hetero Diels−Alder Reactions Catalyzed by the Metallocenium Complex [Cp2Ce][BPh4]

Journal of organic chemistry, 2000-02, Vol.65 (4), p.1215-1217

2000

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Discovery of 2-methylpyridine-based biaryl amides as γ-secretase modulators for the treatment of Alzheimer’s disease

Bioorganic & medicinal chemistry letters, 2013-12, Vol.23 (23), p.6447-6454

2013

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Novel Vanilloid Receptor-1 Antagonists: 1. Conformationally Restricted Analogues of trans-Cinnamides

Journal of medicinal chemistry, 2007-07, Vol.50 (15), p.3497-3514

2007

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Chromenones as potent bradykinin B1 antagonists

Bioorganic & medicinal chemistry letters, 2012-01, Vol.22 (1), p.619-622

2012

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Structure-activity relationships of 3,4-dihydro-1H-quinazolin-2-one derivatives as potential CDK5 inhibitors

Bioorganic & medicinal chemistry, 2007-10, Vol.15 (20), p.6574-6595

2007

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3-Amino-7-phthalazinylbenzoisoxazoles as a Novel Class of Potent, Selective, and Orally Available Inhibitors of p38α Mitogen-Activated Protein Kinase

Journal of medicinal chemistry, 2008-10, Vol.51 (20), p.6280-6292

2008

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Design and synthesis of 6-oxo-1,6-dihydropyridines as CDK5 inhibitors

Bioorganic & medicinal chemistry letters, 2009-12, Vol.19 (23), p.6591-6594

2009

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Total Synthesis and Immunosuppressive Activity of (−)-Pateamine A and Related Compounds: Implementation of a β-Lactam-Based Macrocyclization

Journal of the American Chemical Society, 1998-12, Vol.120 (47), p.12237-12254

1998

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Design and synthesis of quinolin-2(1 H)-one derivatives as potent CDK5 inhibitors

Bioorganic & medicinal chemistry letters, 2007-10, Vol.17 (19), p.5384-5389

2007

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Total Synthesis of the Novel, Immunosuppressive Agent (−)-Pateamine A from Mycale sp. Employing a β-Lactam-Based Macrocyclization

Journal of the American Chemical Society, 1998-01, Vol.120 (3), p.591-592

1998

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Discovery and in Vivo Evaluation of ( S )- N -(1-(7-Fluoro-2-(pyridin-2-yl)quinolin-3-yl)ethyl)-9 H -purin-6-amine (AMG319) and Related PI3Kδ Inhibitors for Inflammation and Autoimmune Disease

Journal of medicinal chemistry, 2015-01, Vol.58 (1), p.480-511

2015

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3-Amino-7-phthalazinylbenzoisoxazoles as a Novel Class of Potent, Selective, and Orally Available Inhibitors of p38a Mitogen-Activated Protein Kinase

Journal of medicinal chemistry, 2008, Vol.51 (20), p.6280-6292

2008

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Structure–activity relationships of 3,4-dihydro-1 H-quinazolin-2-one derivatives as potential CDK5 inhibitors

Bioorganic & medicinal chemistry, 2007, Vol.15 (20), p.6574-6595

2007

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Structural and Synthetic Studies of the Pateamines: Synthesis and Absolute Configuration of the Hydroxydienoate Fragment

Tetrahedron letters, 1995-07, Vol.36 (30), p.5307-5310

Rzasa, R

1995

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3-amino-7-phthalazinylbenzoisoxazoles as a novel class of potent, selective, and orally available inhibitors of p38alpha mitogen-activated protein kinase

Journal of medicinal chemistry, 2008-10, Vol.51 (20), p.6280

2008

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ChemInform Abstract: Palladium-Catalyzed Chemoselective Monoarylation of Hydrazides for the Synthesis of [1,2,4]Triazolo[4,3-a]pyridines

ChemInform, 2010-07, Vol.41 (27), p.no-no

2010

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ChemInform Abstract: Hetero Diels-Alder Reactions Catalyzed by the Metallocenium Complex [Cp2Ce][BPh4]

ChemInform, 2000-06, Vol.31 (24), p.no-no

2000

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ChemInform Abstract: Total Synthesis of Immunosuppressive Activity of (-)-Pateamine A and Related Compounds: Implementation of a β-Lactam-Based Macrocyclization

ChemInform, 1999-05, Vol.30 (18), p.no-no

1999

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Discovery of selective biaryl ethers as PDE10A inhibitors: Improvement in potency and mitigation of Pgp-mediated efflux

Discovery of Highly Selective and Potent p38 Inhibitors Based on a Phthalazine Scaffold

Discovery and in Vivo Evaluation of (S)‑N‑(1-(7-Fluoro-2-(pyridin-2-yl)quinolin-3-yl)ethyl)‑9H‑purin-6-amine (AMG319) and Related PI3Kδ Inhibitors for Inflammation and Autoimmune Disease

Palladium-Catalyzed Chemoselective Monoarylation of Hydrazides for the Synthesis of [1,2,4]Triazolo[4,3-a]pyridines

Isolation and Identification of Eukaryotic Initiation Factor 4A as a Molecular Target for the Marine Natural Product Pateamine A

Novel Vanilloid Receptor-1 Antagonists: 2. Structure−Activity Relationships of 4-Oxopyrimidines Leading to the Selection of a Clinical Candidate

Synthesis and preliminary biological evaluation of potent and selective 2-(3-alkoxy-1-azetidinyl) quinolines as novel PDE10A inhibitors with improved solubility

Hetero Diels−Alder Reactions Catalyzed by the Metallocenium Complex [Cp2Ce][BPh4]

Discovery of 2-methylpyridine-based biaryl amides as γ-secretase modulators for the treatment of Alzheimer’s disease

Novel Vanilloid Receptor-1 Antagonists: 1. Conformationally Restricted Analogues of trans-Cinnamides

Chromenones as potent bradykinin B1 antagonists

Structure-activity relationships of 3,4-dihydro-1H-quinazolin-2-one derivatives as potential CDK5 inhibitors

3-Amino-7-phthalazinylbenzoisoxazoles as a Novel Class of Potent, Selective, and Orally Available Inhibitors of p38α Mitogen-Activated Protein Kinase

Design and synthesis of 6-oxo-1,6-dihydropyridines as CDK5 inhibitors

Total Synthesis and Immunosuppressive Activity of (−)-Pateamine A and Related Compounds: Implementation of a β-Lactam-Based Macrocyclization

Design and synthesis of quinolin-2(1 H)-one derivatives as potent CDK5 inhibitors

Total Synthesis of the Novel, Immunosuppressive Agent (−)-Pateamine A from Mycale sp. Employing a β-Lactam-Based Macrocyclization

Discovery and in Vivo Evaluation of ( S )- N -(1-(7-Fluoro-2-(pyridin-2-yl)quinolin-3-yl)ethyl)-9 H -purin-6-amine (AMG319) and Related PI3Kδ Inhibitors for Inflammation and Autoimmune Disease

3-Amino-7-phthalazinylbenzoisoxazoles as a Novel Class of Potent, Selective, and Orally Available Inhibitors of p38a Mitogen-Activated Protein Kinase

Structure–activity relationships of 3,4-dihydro-1 H-quinazolin-2-one derivatives as potential CDK5 inhibitors

Structural and Synthetic Studies of the Pateamines: Synthesis and Absolute Configuration of the Hydroxydienoate Fragment

3-amino-7-phthalazinylbenzoisoxazoles as a novel class of potent, selective, and orally available inhibitors of p38alpha mitogen-activated protein kinase

ChemInform Abstract: Palladium-Catalyzed Chemoselective Monoarylation of Hydrazides for the Synthesis of [1,2,4]Triazolo[4,3-a]pyridines

ChemInform Abstract: Hetero Diels-Alder Reactions Catalyzed by the Metallocenium Complex [Cp2Ce][BPh4]

ChemInform Abstract: Total Synthesis of Immunosuppressive Activity of (-)-Pateamine A and Related Compounds: Implementation of a β-Lactam-Based Macrocyclization

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