UB Paderborn / Katalog / Suche / in CDI

Sortiert nach

Einfacher Volltextzugriff von (fast) überall

Installieren Sie die LibKey Nomad-Browsererweiterung und erhalten Sie von vielen Webseiten einfachen Zugriff auf lizenzierte Volltexte oder Open Access Publikationen. Mehr erfahren...

Identification and characterization of NVP-BKM120, an orally available pan-class I PI3-kinase inhibitor

Molecular cancer therapeutics, 2012-02, Vol.11 (2), p.317-328

2012

Volltextzugriff (PDF)

Identification and characterization of NVP-BEZ235, a new orally available dual phosphatidylinositol 3-kinase/mammalian target of rapamycin inhibitor with potent in vivo antitumor activity

Molecular cancer therapeutics, 2008-07, Vol.7 (7), p.1851-1863

2008

Volltextzugriff (PDF)

Genetic resistance to JAK2 enzymatic inhibitors is overcome by HSP90 inhibition

The Journal of experimental medicine, 2012-02, Vol.209 (2), p.259-273

2012

Volltextzugriff (PDF)

Tetra-substituted imidazoles as a new class of inhibitors of the p53–MDM2 interaction

Bioorganic & medicinal chemistry letters, 2014-05, Vol.24 (9), p.2110-2114

2014

Volltextzugriff (PDF)

Modulation of activation-loop phosphorylation by JAK inhibitors is binding mode dependent

Cancer discovery, 2012-06, Vol.2 (6), p.512-523

2012

Volltextzugriff (PDF)

2-Amino-aryl-7-aryl-benzoxazoles as potent, selective and orally available JAK2 inhibitors

Bioorganic & medicinal chemistry letters, 2010-03, Vol.20 (5), p.1724-1727

2010

Volltextzugriff (PDF)

Factors influencing the inhibition of protein kinases

Journal of enzyme inhibition and medicinal chemistry, 2012-04, Vol.27 (2), p.194-200

2012

Volltextzugriff (PDF)

Characterization of the novel and specific PI3Kα inhibitor NVP-BYL719 and development of the patient stratification strategy for clinical trials

Molecular cancer therapeutics, 2014-05, Vol.13 (5), p.1117-1129

2014

Volltextzugriff (PDF)

Effects of intestinal fatty acid-binding protein overexpression on fatty acid metabolism in Caco-2 cells

Journal of lipid research, 2000, Vol.41 (1), p.84-92

2000

Volltextzugriff (PDF)

The central valine concept provides an entry in a new class of non peptide inhibitors of the p53–MDM2 interaction

Bioorganic & medicinal chemistry letters, 2012-05, Vol.22 (10), p.3498-3502

2012

Volltextzugriff (PDF)

Study of the Selectivity of Insulin-Like Growth Factor-1 Receptor (IGF1R) Inhibitors

The open enzyme inhibition journal, 2010-07, Vol.3 (1), p.27-37

2010

Volltextzugriff (PDF)

Potent and selective inhibition of polycythemia by the quinoxaline JAK2 inhibitor NVP-BSK805

Molecular cancer therapeutics, 2010-07, Vol.9 (7), p.1945-1955

2010

Volltextzugriff (PDF)

Corrigendum to “Tetra-substituted imidazoles as a new class of inhibitors of the p53–MDM2 interaction” [Bioorg. Med. Chem. Lett. 24 (9) (2014) 2110–2114]

Bioorganic & medicinal chemistry letters, 2015-03, Vol.25 (6), p.1356-1356

2015

Volltextzugriff (PDF)

Leveraging the contribution of thermodynamics in drug discovery with the help of fluorescence-based thermal shift assays

Journal of biomolecular screening, 2011-06, Vol.16 (5), p.552-556

2011

Volltextzugriff (PDF)

Abstract 3748: NVP-BYL719, a novel PI3Kalpha selective inhibitor with all the characteristics required for clinical development as an anti-cancer agent

Cancer research (Chicago, Ill.), 2012-04, Vol.72 (8_Supplement), p.3748-3748

2012

Volltextzugriff (PDF)

Abstract 1922: 2-Aminothiazoles as potent and selective PI3Kalpha inhibitors: Discovery of NVP-BYL719 and structural basis for the isoform selectivity

Cancer research (Chicago, Ill.), 2012-04, Vol.72 (8_Supplement), p.1922-1922

2012

Volltextzugriff (PDF)

Genetic Resistance to JAK2 Enzymatic Inhibitors Is Overcome by HSP90 Inhibition

Blood, 2011-11, Vol.118 (21), p.62-62

2011

Volltextzugriff (PDF)

Simultaneous protein expression and modification: an efficient approach for production of unphosphorylated and biotinylated receptor tyrosine kinases by triple infection in the baculovirus expression system

Journal of biomolecular techniques, 2010-04, Vol.21 (1), p.9-17

2010

Volltextzugriff (PDF)

Novel, Potent and Selective JAK2 Inhibitors

Blood, 2009-11, Vol.114 (22), p.3777-3777

2009

Volltextzugriff (PDF)

Characterisation of Na/K-ATPase, its isoforms, and the inotropic response to ouabain in isolated failing human hearts

Cardiovascular research, 1993-12, Vol.27 (12), p.2229-2237

1993

Volltextzugriff (PDF)

Epidermal growth factor regulates fatty acid uptake and metabolism in Caco-2 cells

American journal of physiology: Gastrointestinal and liver physiology, 1999-03, Vol.276 (3), p.G606-G612

1999

Volltextzugriff (PDF)

Kinetic Study of Human Full-Length Wild-Type JAK2 and V617F Mutant Proteins

The open enzyme inhibition journal, 2009-01, Vol.1 (1), p.80-84

2009

Volltextzugriff (PDF)

Differential Regulation of Intestinal and Liver Fatty Acid-Binding Proteins in Human Intestinal Cell line (Caco-2): Role of Collagen

Experimental cell research, 1998-11, Vol.244 (2), p.441-447

1998

Volltextzugriff (PDF)

Epidermal growth factor regulates fatty acid uptake and metabolism in Caco-2 cells

American journal of physiology: Gastrointestinal and liver physiology, 1999-03, Vol.39 (3), p.G606-G612

1999

Volltextzugriff (PDF)

Epidermal growth factor regulates fatty acid uptake and metabolism in Caco-2 cells

American journal of physiology: Gastrointestinal and liver physiology, 1999-03, Vol.276 (3), p.G606

1999

Volltextzugriff (PDF)

1 – 25 von 33

Suche als RSS-Feed

Suchergebnisse filtern

Filter anzeigen

Nur zeigen

Geprüft (Peer-Review)
(31)
Mit Volltextzugriff
(33)

Publikationsform

Artikel
(33)

Sprache

Englisch
(33)

Erscheinungsjahr

n.n

Thema

Life Sciences & Biomedicine
(18)
Science & Technology
(18)
Humans
(14)
Animals
(13)
Cell Line, Tumor
(7)
Pharmacology & Pharmacy
(7)
Mice
(6)
Oncology
(6)
Biological And Medical Sciences
(5)
Models, Molecular
(5)
Rats
(5)
Chemistry
(4)
Chemistry, Medicinal
(4)
Guinea Pigs
(4)
Janus Kinase 2 - Antagonists & Inhibitors
(4)
Kinetics
(4)
Medical Sciences
(4)
Physical Sciences
(4)
Protein Binding
(4)
Protein Kinase Inhibitors - Pharmacology
(4)

15 weitere anzeigen...

Weniger anzeigen...

Menü

Weitere Dienste

Einstellungen

Identification and characterization of NVP-BKM120, an orally available pan-class I PI3-kinase inhibitor

Identification and characterization of NVP-BEZ235, a new orally available dual phosphatidylinositol 3-kinase/mammalian target of rapamycin inhibitor with potent in vivo antitumor activity

Genetic resistance to JAK2 enzymatic inhibitors is overcome by HSP90 inhibition

Tetra-substituted imidazoles as a new class of inhibitors of the p53–MDM2 interaction

Modulation of activation-loop phosphorylation by JAK inhibitors is binding mode dependent

2-Amino-aryl-7-aryl-benzoxazoles as potent, selective and orally available JAK2 inhibitors

Factors influencing the inhibition of protein kinases

Characterization of the novel and specific PI3Kα inhibitor NVP-BYL719 and development of the patient stratification strategy for clinical trials

Effects of intestinal fatty acid-binding protein overexpression on fatty acid metabolism in Caco-2 cells

The central valine concept provides an entry in a new class of non peptide inhibitors of the p53–MDM2 interaction

Study of the Selectivity of Insulin-Like Growth Factor-1 Receptor (IGF1R) Inhibitors

Potent and selective inhibition of polycythemia by the quinoxaline JAK2 inhibitor NVP-BSK805

Corrigendum to “Tetra-substituted imidazoles as a new class of inhibitors of the p53–MDM2 interaction” [Bioorg. Med. Chem. Lett. 24 (9) (2014) 2110–2114]

Leveraging the contribution of thermodynamics in drug discovery with the help of fluorescence-based thermal shift assays

Abstract 3748: NVP-BYL719, a novel PI3Kalpha selective inhibitor with all the characteristics required for clinical development as an anti-cancer agent

Abstract 1922: 2-Aminothiazoles as potent and selective PI3Kalpha inhibitors: Discovery of NVP-BYL719 and structural basis for the isoform selectivity

Genetic Resistance to JAK2 Enzymatic Inhibitors Is Overcome by HSP90 Inhibition

Simultaneous protein expression and modification: an efficient approach for production of unphosphorylated and biotinylated receptor tyrosine kinases by triple infection in the baculovirus expression system

Novel, Potent and Selective JAK2 Inhibitors

Characterisation of Na/K-ATPase, its isoforms, and the inotropic response to ouabain in isolated failing human hearts

Epidermal growth factor regulates fatty acid uptake and metabolism in Caco-2 cells

Kinetic Study of Human Full-Length Wild-Type JAK2 and V617F Mutant Proteins

Differential Regulation of Intestinal and Liver Fatty Acid-Binding Proteins in Human Intestinal Cell line (Caco-2): Role of Collagen

Epidermal growth factor regulates fatty acid uptake and metabolism in Caco-2 cells

Epidermal growth factor regulates fatty acid uptake and metabolism in Caco-2 cells

Suchergebnisse filtern