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Discovery of Novel Trypanosoma brucei Phosphodiesterase B1 Inhibitors by Virtual Screening against the Unliganded TbrPDEB1 Crystal Structure

Journal of medicinal chemistry, 2013-03, Vol.56 (5), p.2087-2096

2013

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Simple Colorimetric Trypanothione Reductase-Based Assay for High-Throughput Screening of Drugs against Leishmania Intracellular Amastigotes

Antimicrobial Agents and Chemotherapy, 2014-01, Vol.58 (1), p.527-535

2014

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Synthesis and evaluation of analogs of the phenylpyridazinone NPD-001 as potent trypanosomal TbrPDEB1 phosphodiesterase inhibitors and in vitro trypanocidals

Bioorganic & medicinal chemistry, 2016-04, Vol.24 (7), p.1573-1581

2016

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Catechol Pyrazolinones as Trypanocidals: Fragment-Based Design, Synthesis, and Pharmacological Evaluation of Nanomolar Inhibitors of Trypanosomal Phosphodiesterase B1

Journal of medicinal chemistry, 2012-10, Vol.55 (20), p.8745-8756

2012

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Fast, Acid-Free, and Selective Lactamization of Lactones in Ionic Liquids

Journal of organic chemistry, 2008-11, Vol.73 (21), p.8627-8630

2008

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The European Lead Factory: A Blueprint for Public-Private Partnerships in Early Drug Discovery

Frontiers in medicine, 2017-01, Vol.3, p.75-75

2017

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Fragment-based screening in tandem with phenotypic screening provides novel antiparasitic hits

Journal of biomolecular screening, 2015-01, Vol.20 (1), p.131-140

2015

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α-Substituted norstatines as the transition-state mimic in inhibitors of multiple digestive vacuole malaria aspartic proteases

Bioorganic & medicinal chemistry, 2009-08, Vol.17 (16), p.5933-5949

2009

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Phenyldihydropyrazolones as Novel Lead Compounds Against Trypanosoma cruzi

ACS omega, 2019-04, Vol.4 (4), p.6585-6596

2019

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Synthesis of a small library of non-symmetric cyclic sulfamide HIV-1 protease inhibitors

Tetrahedron, 2010-06, Vol.66 (23), p.4049-4056

2010

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Patterns of Care, Tolerability, and Safety of the First Cohort of Patients Treated on a Novel High-Field MR-Linac Within the MOMENTUM Study: Initial Results From a Prospective Multi-Institutional Registry

International journal of radiation oncology, biology, physics, 2021-11, Vol.111 (4), p.867-875

2021

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An efficient method to perform milliliter-scale PCR utilizing highly controlled microwave thermocyclingElectronic Supplementary Information (ESI) available: experimental details. See http://www.rsc.org/suppdata/cc/b3/b317049g

Chemical communications (Cambridge, England), 2004 (7), p.790

2004

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The development of an artificial intelligence-based digital pathology for neglected tropical diseases: A platform specific analysis of the World Health Organization diagnostic target product profile for soil-transmitted helminthiasis

Frontiers in tropical diseases, 2022-12, Vol.3

2022

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Identification of Phenylpyrazolone Dimers as a New Class of Anti‐Trypanosoma cruzi Agents

ChemMedChem, 2019-09, Vol.14 (18), p.1662-1668

2019

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An efficient method to perform milliliter-scale PCR utilizing highly controlled microwave thermocycling

Chemical communications (Cambridge, England), 2004-04, Vol.7 (7), p.790-791

2004

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α-Substituted Norstatines as the Transistion-State Mimic in Inhibitors of Multiple Digestive Vacuole Malaria Aspartic Proteases

Bioorganic & medicinal chemistry, 2009, Vol.17 (16), p.5933

2009

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Cascade synthesis with (triphenylphosphoranylidene)-ethenone as a versatile reagent for fast synthesis of heterocycles and unsaturated amides under microwave dielectric heating

Combinatorial chemistry & high throughput screening, 2002-11, Vol.5 (7), p.571

2002

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On the versatility of microwave-assisted chemistry: exemplified by applications in medicinal chemistry, heterocyclic chemistry and biochemistry

Orrling, Kristina M

2009

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ChemInform Abstract: Fast-, Acid-Free, and Selective Lactamization of Lactones in Ionic Liquids

ChemInform, 2009-03, Vol.40 (12), p.no-no

2009

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Discovery of Novel Trypanosoma brucei Phosphodiesterase B1 Inhibitors by Virtual Screening against the Unliganded TbrPDEB1 Crystal Structure

Targeting a Subpocket in Trypanosoma brucei Phosphodiesterase B1 (TbrPDEB1) Enables the Structure-Based Discovery of Selective Inhibitors with Trypanocidal Activity

Simple Colorimetric Trypanothione Reductase-Based Assay for High-Throughput Screening of Drugs against Leishmania Intracellular Amastigotes

Synthesis and evaluation of analogs of the phenylpyridazinone NPD-001 as potent trypanosomal TbrPDEB1 phosphodiesterase inhibitors and in vitro trypanocidals

Catechol Pyrazolinones as Trypanocidals: Fragment-Based Design, Synthesis, and Pharmacological Evaluation of Nanomolar Inhibitors of Trypanosomal Phosphodiesterase B1

Fast, Acid-Free, and Selective Lactamization of Lactones in Ionic Liquids

The European Lead Factory: A Blueprint for Public-Private Partnerships in Early Drug Discovery

Fragment-based screening in tandem with phenotypic screening provides novel antiparasitic hits

Safety and Tolerability of Online Adaptive High-Field Magnetic Resonance-Guided Radiotherapy

α-Substituted norstatines as the transition-state mimic in inhibitors of multiple digestive vacuole malaria aspartic proteases

Phenyldihydropyrazolones as Novel Lead Compounds Against Trypanosoma cruzi

Synthesis of a small library of non-symmetric cyclic sulfamide HIV-1 protease inhibitors

Patterns of Care, Tolerability, and Safety of the First Cohort of Patients Treated on a Novel High-Field MR-Linac Within the MOMENTUM Study: Initial Results From a Prospective Multi-Institutional Registry

The MOMENTUM Study: An International Registry for the Evidence-Based Introduction of MR-Guided Adaptive Therapy

An efficient method to perform milliliter-scale PCR utilizing highly controlled microwave thermocyclingElectronic Supplementary Information (ESI) available: experimental details. See http://www.rsc.org/suppdata/cc/b3/b317049g

The development of an artificial intelligence-based digital pathology for neglected tropical diseases: A platform specific analysis of the World Health Organization diagnostic target product profile for soil-transmitted helminthiasis

Identification of Phenylpyrazolone Dimers as a New Class of Anti‐Trypanosoma cruzi Agents

An efficient method to perform milliliter-scale PCR utilizing highly controlled microwave thermocycling

α-Substituted Norstatines as the Transistion-State Mimic in Inhibitors of Multiple Digestive Vacuole Malaria Aspartic Proteases

Cascade synthesis with (triphenylphosphoranylidene)-ethenone as a versatile reagent for fast synthesis of heterocycles and unsaturated amides under microwave dielectric heating

On the versatility of microwave-assisted chemistry: exemplified by applications in medicinal chemistry, heterocyclic chemistry and biochemistry

ChemInform Abstract: Fast-, Acid-Free, and Selective Lactamization of Lactones in Ionic Liquids

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