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Development of human cGAS-specific small-molecule inhibitors for repression of dsDNA-triggered interferon expression

Nature communications, 2019-05, Vol.10 (1), p.2261-2261, Article 2261

2019

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What can crystal structures of aminergic receptors tell us about designing subtype-selective ligands?

Pharmacological reviews, 2015-01, Vol.67 (1), p.198-213

2015

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A new mechanism of allostery in a G protein-coupled receptor dimer

Nature chemical biology, 2014-09, Vol.10 (9), p.745-752

2014

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Structural basis for Na(+)-sensitivity in dopamine D2 and D3 receptors

Chemical communications (Cambridge, England), 2015-05, Vol.51 (41), p.8618-8621

2015

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Next-generation neuropeptide Y receptor small-molecule agonists inhibit mosquito-biting behavior

Parasites & vectors, 2024-06, Vol.17 (1), p.276-12, Article 276

2024

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Shape-Based Virtual Screening of a Billion-Compound Library Identifies Mycobacterial Lipoamide Dehydrogenase Inhibitors

ACS bio & med chem au, 2023-12, Vol.3 (6), p.507-515

2023

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The E2.65A mutation disrupts dynamic binding poses of SB269652 at the dopamine D2 and D3 receptors

PLoS computational biology, 2018-01, Vol.14 (1), p.e1005948-e1005948

2018

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Enhancing Hit Discovery in Virtual Screening through Absolute Protein–Ligand Binding Free-Energy Calculations

Journal of chemical information and modeling, 2023-05, Vol.63 (10), p.3171-3185

2023

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Computational approaches to detect allosteric pathways in transmembrane molecular machines

Biochimica et biophysica acta, 2016-07, Vol.1858 (7), p.1652-1662

2016

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Indazole to 2‐Cyanoindole Scaffold Progression for Mycobacterial Lipoamide Dehydrogenase Inhibitors Achieves Extended Target Residence Time and Improved Antibacterial Activity

Angewandte Chemie International Edition, 2024-10, Vol.63 (44), p.e202407276-n/a

International ed. in English, 2024

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Molecular Determinants of Selectivity and Efficacy at the Dopamine D3 Receptor

Journal of medicinal chemistry, 2012-08, Vol.55 (15), p.6689-6699

2012

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Antimalarial proteasome inhibitor reveals collateral sensitivity from intersubunit interactions and fitness cost of resistance

Proceedings of the National Academy of Sciences - PNAS, 2018-07, Vol.115 (29), p.E6863-E6870

2018

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Inhibition of 3-phosphoglycerate dehydrogenase (PHGDH) by indole amides abrogates de novo serine synthesis in cancer cells

Bioorganic & medicinal chemistry letters, 2019-09, Vol.29 (17), p.2503-2510

2019

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A single glycine in extracellular loop 1 is the critical determinant for pharmacological specificity of dopamine D2 and D3 receptors

Molecular pharmacology, 2013-12, Vol.84 (6), p.854-864

2013

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Design, Synthesis, and Optimization of Macrocyclic Peptides as Species-Selective Antimalaria Proteasome Inhibitors

Journal of medicinal chemistry, 2022-07, Vol.65 (13), p.9350-9375

2022

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Small-Molecule Inhibition of the Acyl-Lysine Reader ENL as a Strategy against Acute Myeloid Leukemia

Cancer discovery, 2022-11, Vol.12 (11), p.2684-2709

2022

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Toward Understanding the Structural Basis of Partial Agonism at the Dopamine D 3 Receptor

Journal of medicinal chemistry, 2017-01, Vol.60 (2), p.580-593

2017

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Development of a Highly Selective Plasmodium falciparum Proteasome Inhibitor with Anti‐malaria Activity in Humanized Mice

Angewandte Chemie International Edition, 2021-04, Vol.60 (17), p.9279-9283

International ed. in English, 2021

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Toward Understanding the Structural Basis of Partial Agonism at the Dopamine D3 Receptor

Journal of medicinal chemistry, 2017-01, Vol.60 (2), p.580-593

2017

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Selective Phenylimidazole-Based Inhibitors of the Mycobacterium tuberculosis Proteasome

Journal of medicinal chemistry, 2019-10, Vol.62 (20), p.9246-9253

2019

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Macrocyclic Peptides that Selectively Inhibit the Mycobacterium tuberculosis Proteasome

Journal of medicinal chemistry, 2021-05, Vol.64 (9), p.6262-6272

2021

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Characterization of Pyrrolidinyl-hexahydro-pyranopiperazines as a Novel Kappa Opioid Receptor Agonist Scaffold

ACS chemical neuroscience, 2022-07, Vol.13 (13), p.1849-1856

2022

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The structural determinants of the bitopic binding mode of a negative allosteric modulator of the dopamine D2 receptor

Biochemical pharmacology, 2018-02, Vol.148, p.315-328

2018

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Discovery of a Novel Class of Negative Allosteric Modulator of the Dopamine D2 Receptor Through Fragmentation of a Bitopic Ligand

Journal of medicinal chemistry, 2015-09, Vol.58 (17), p.6819-6843

2015

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Structure–Activity Relationship Studies of Antimalarial Plasmodium Proteasome InhibitorsPart II

Journal of medicinal chemistry, 2023-01, Vol.66 (2), p.1484-1508

2023

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Development of human cGAS-specific small-molecule inhibitors for repression of dsDNA-triggered interferon expression

What can crystal structures of aminergic receptors tell us about designing subtype-selective ligands?

A new mechanism of allostery in a G protein-coupled receptor dimer

Structural basis for Na(+)-sensitivity in dopamine D2 and D3 receptors

Next-generation neuropeptide Y receptor small-molecule agonists inhibit mosquito-biting behavior

Shape-Based Virtual Screening of a Billion-Compound Library Identifies Mycobacterial Lipoamide Dehydrogenase Inhibitors

The E2.65A mutation disrupts dynamic binding poses of SB269652 at the dopamine D2 and D3 receptors

Enhancing Hit Discovery in Virtual Screening through Absolute Protein–Ligand Binding Free-Energy Calculations

Computational approaches to detect allosteric pathways in transmembrane molecular machines

Indazole to 2‐Cyanoindole Scaffold Progression for Mycobacterial Lipoamide Dehydrogenase Inhibitors Achieves Extended Target Residence Time and Improved Antibacterial Activity

Molecular Determinants of Selectivity and Efficacy at the Dopamine D3 Receptor

Antimalarial proteasome inhibitor reveals collateral sensitivity from intersubunit interactions and fitness cost of resistance

Inhibition of 3-phosphoglycerate dehydrogenase (PHGDH) by indole amides abrogates de novo serine synthesis in cancer cells

A single glycine in extracellular loop 1 is the critical determinant for pharmacological specificity of dopamine D2 and D3 receptors

Design, Synthesis, and Optimization of Macrocyclic Peptides as Species-Selective Antimalaria Proteasome Inhibitors

Small-Molecule Inhibition of the Acyl-Lysine Reader ENL as a Strategy against Acute Myeloid Leukemia

Toward Understanding the Structural Basis of Partial Agonism at the Dopamine D 3 Receptor

Development of a Highly Selective Plasmodium falciparum Proteasome Inhibitor with Anti‐malaria Activity in Humanized Mice

Toward Understanding the Structural Basis of Partial Agonism at the Dopamine D3 Receptor

Selective Phenylimidazole-Based Inhibitors of the Mycobacterium tuberculosis Proteasome

Macrocyclic Peptides that Selectively Inhibit the Mycobacterium tuberculosis Proteasome

Characterization of Pyrrolidinyl-hexahydro-pyranopiperazines as a Novel Kappa Opioid Receptor Agonist Scaffold

The structural determinants of the bitopic binding mode of a negative allosteric modulator of the dopamine D2 receptor

Discovery of a Novel Class of Negative Allosteric Modulator of the Dopamine D2 Receptor Through Fragmentation of a Bitopic Ligand

Structure–Activity Relationship Studies of Antimalarial Plasmodium Proteasome InhibitorsPart II

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