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Design and Synthesis of D3R Bitopic Ligands with Flexible Secondary Binding Fragments: Radioligand Binding and Computational Chemistry Studies

Molecules (Basel, Switzerland), 2024-01, Vol.29 (1), p.123

2024

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Selective Activation of D3 Dopamine Receptors Ameliorates DOI-Induced Head Twitching Accompanied by Changes in Corticostriatal Processing

International journal of molecular sciences, 2023-05, Vol.24 (11), p.9300

2023

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Design and Synthesis of Conformationally Flexible Scaffold as Bitopic Ligands for Potent D3-Selective Antagonists

International journal of molecular sciences, 2022-12, Vol.24 (1), p.432

2022

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Evaluation of Substituted N-Phenylpiperazine Analogs as D3 vs. D2 Dopamine Receptor Subtype Selective Ligands

Molecules (Basel, Switzerland), 2021-05, Vol.26 (11), p.3182

2021

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In vitro characterization of [ 125 I]HY-3-24, a selective ligand for the dopamine D3 receptor

Frontiers in neuroscience, 2024, Vol.18, p.1380009-1380009

2024

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The effects of sigma (σ1) receptor‐selective ligands on muscarinic receptor antagonist‐induced cognitive deficits in mice

British journal of pharmacology, 2015-05, Vol.172 (10), p.2519-2531

2015

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N-(3-Fluoro-4-(4-(2-methoxy or 2,3-dichlorophenyl)piperazine-1-yl)butyl)arylcarboxamides as Selective Dopamine D3 Receptor Ligands: Critical Role of the Carboxamide Linker for D3 Receptor Selectivity

Journal of medicinal chemistry, 2011-05, Vol.54 (10), p.3581-3594

2011

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Interaction of Ligands for PET with the Dopamine D3 Receptor: In Silico and In Vitro Methods

Biomolecules (Basel, Switzerland), 2021-04, Vol.11 (4), p.529

2021

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Neuroprotective effects of high affinity sigma 1 receptor selective compounds

Brain research, 2012-03, Vol.1441, p.17-26

2012

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D1 Dopamine Receptor Mediates Dopamine-induced Cytotoxicity via the ERK Signal Cascade

The Journal of biological chemistry, 2004-09, Vol.279 (38), p.39317-39330

2004

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Evaluation of the D3 dopamine receptor selective antagonist PG01037 on l-dopa-dependent abnormal involuntary movements in rats

Neuropharmacology, 2009-05, Vol.56 (6), p.944-955

2009

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Molecular Determinants of Selectivity and Efficacy at the Dopamine D3 Receptor

Journal of medicinal chemistry, 2012-08, Vol.55 (15), p.6689-6699

2012

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Synthesis of bitopic ligands based on fallypride and evaluation of their affinity and selectivity towards dopamine D2 and D3 receptors

European journal of medicinal chemistry, 2023-12, Vol.261, p.115751-115751, Article 115751

2023

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Factors Governing Selectivity of Dopamine Receptor Binding Compounds for D2R and D3R Subtypes

Journal of chemical information and modeling, 2021-06, Vol.61 (6), p.2829-2843

2021

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Challenges in the development of dopamine D2‐ and D3‐selective radiotracers for PET imaging studies

Journal of labelled compounds & radiopharmaceuticals, 2018-03, Vol.61 (3), p.291-298

2018

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Highly Selective Dopamine D3 Receptor Antagonists with Arylated Diazaspiro Alkane Cores

Journal of medicinal chemistry, 2017-12, Vol.60 (23), p.9905-9910

2017

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Highly Selective Dopamine D 3 Receptor Antagonists with Arylated Diazaspiro Alkane Cores

Journal of medicinal chemistry, 2017-12, Vol.60 (23), p.9905-9910

2017

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Design, synthesis, and evaluation of N-(4-(4-phenyl piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamides as selective dopamine D3 receptor ligands

Bioorganic & medicinal chemistry letters, 2019-09, Vol.29 (18), p.2690-2694

2019

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Leveraging a Low-Affinity Diazaspiro Orthosteric Fragment to Reduce Dopamine D3 Receptor (D3R) Ligand Promiscuity across Highly Conserved Aminergic G‑Protein-Coupled Receptors (GPCRs)

Journal of medicinal chemistry, 2019-05, Vol.62 (10), p.5132-5147

2019

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Leveraging a Low-Affinity Diazaspiro Orthosteric Fragment to Reduce Dopamine D 3 Receptor (D 3 R) Ligand Promiscuity across Highly Conserved Aminergic G-Protein-Coupled Receptors (GPCRs)

Journal of medicinal chemistry, 2019-05, Vol.62 (10), p.5132-5147

2019

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Design, synthesis, and evaluation of N-(4-(4-phenyl piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamides as selective dopamine D 3 receptor ligands

Bioorganic & medicinal chemistry letters, 2019-09, Vol.29 (18), p.2690

2019

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N-(4-(4-(2,3-Dichloro- or 2-methoxyphenyl)piperazin-1-yl)butyl)heterobiarylcarboxamides with Functionalized Linking Chains as High Affinity and Enantioselective D3 Receptor Antagonists

Journal of medicinal chemistry, 2009-04, Vol.52 (8), p.2559-2570

2009

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Subtype Selectivity of Dopamine Receptor Ligands: Insights from Structure and Ligand-Based Methods

Journal of chemical information and modeling, 2010-11, Vol.50 (11), p.1970-1985

2010

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Analogues of Arylamide Phenylpiperazine Ligands To Investigate the Factors Influencing D3 Dopamine Receptor Bitropic Binding and Receptor Subtype Selectivity

ACS chemical neuroscience, 2018-12, Vol.9 (12), p.2972-2983

2018

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Design and Synthesis of Conformationally Flexible Scaffold as Bitopic Ligands for Potent D 3 -Selective Antagonists

International journal of molecular sciences, 2023-01, Vol.24 (1)

2023

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Design and Synthesis of D3R Bitopic Ligands with Flexible Secondary Binding Fragments: Radioligand Binding and Computational Chemistry Studies

Selective Activation of D3 Dopamine Receptors Ameliorates DOI-Induced Head Twitching Accompanied by Changes in Corticostriatal Processing

Design and Synthesis of Conformationally Flexible Scaffold as Bitopic Ligands for Potent D3-Selective Antagonists

Evaluation of Substituted N-Phenylpiperazine Analogs as D3 vs. D2 Dopamine Receptor Subtype Selective Ligands

In vitro characterization of [ 125 I]HY-3-24, a selective ligand for the dopamine D3 receptor

The effects of sigma (σ1) receptor‐selective ligands on muscarinic receptor antagonist‐induced cognitive deficits in mice

N-(3-Fluoro-4-(4-(2-methoxy or 2,3-dichlorophenyl)piperazine-1-yl)butyl)arylcarboxamides as Selective Dopamine D3 Receptor Ligands: Critical Role of the Carboxamide Linker for D3 Receptor Selectivity

Interaction of Ligands for PET with the Dopamine D3 Receptor: In Silico and In Vitro Methods

Neuroprotective effects of high affinity sigma 1 receptor selective compounds

D1 Dopamine Receptor Mediates Dopamine-induced Cytotoxicity via the ERK Signal Cascade

Evaluation of the D3 dopamine receptor selective antagonist PG01037 on l-dopa-dependent abnormal involuntary movements in rats

Molecular Determinants of Selectivity and Efficacy at the Dopamine D3 Receptor

Synthesis of bitopic ligands based on fallypride and evaluation of their affinity and selectivity towards dopamine D2 and D3 receptors

Factors Governing Selectivity of Dopamine Receptor Binding Compounds for D2R and D3R Subtypes

Challenges in the development of dopamine D2‐ and D3‐selective radiotracers for PET imaging studies

Highly Selective Dopamine D3 Receptor Antagonists with Arylated Diazaspiro Alkane Cores

Highly Selective Dopamine D 3 Receptor Antagonists with Arylated Diazaspiro Alkane Cores

Design, synthesis, and evaluation of N-(4-(4-phenyl piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamides as selective dopamine D3 receptor ligands

Leveraging a Low-Affinity Diazaspiro Orthosteric Fragment to Reduce Dopamine D3 Receptor (D3R) Ligand Promiscuity across Highly Conserved Aminergic G‑Protein-Coupled Receptors (GPCRs)

Leveraging a Low-Affinity Diazaspiro Orthosteric Fragment to Reduce Dopamine D 3 Receptor (D 3 R) Ligand Promiscuity across Highly Conserved Aminergic G-Protein-Coupled Receptors (GPCRs)

Design, synthesis, and evaluation of N-(4-(4-phenyl piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamides as selective dopamine D 3 receptor ligands

N-(4-(4-(2,3-Dichloro- or 2-methoxyphenyl)piperazin-1-yl)butyl)heterobiarylcarboxamides with Functionalized Linking Chains as High Affinity and Enantioselective D3 Receptor Antagonists

Subtype Selectivity of Dopamine Receptor Ligands: Insights from Structure and Ligand-Based Methods

Analogues of Arylamide Phenylpiperazine Ligands To Investigate the Factors Influencing D3 Dopamine Receptor Bitropic Binding and Receptor Subtype Selectivity

Design and Synthesis of Conformationally Flexible Scaffold as Bitopic Ligands for Potent D 3 -Selective Antagonists

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