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Discovery of TRPM8 Antagonist (S)‑6-(((3-Fluoro-4-(trifluoromethoxy)phenyl)(3-fluoropyridin-2-yl)methyl)carbamoyl)nicotinic Acid (AMG 333), a Clinical Candidate for the Treatment of Migraine

Journal of medicinal chemistry, 2018-09, Vol.61 (18), p.8186-8201

2018

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Synthesis and structure–activity relationship of trisubstituted thiazoles as Cdc7 kinase inhibitors

European journal of medicinal chemistry, 2014-06, Vol.80, p.364-382

2014

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Targeting the Mitotic Kinesin KIF18A in Chromosomally Unstable Cancers: Hit Optimization Toward an In Vivo Chemical Probe

Journal of medicinal chemistry, 2022-03, Vol.65 (6), p.4972-4990

2022

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Design and Preparation of a Potent Series of Hydroxyethylamine Containing β-Secretase Inhibitors That Demonstrate Robust Reduction of Central β-Amyloid

Journal of medicinal chemistry, 2012-11, Vol.55 (21), p.9009-9024

2012

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Optimization of Potency and Pharmacokinetic Properties of Tetrahydroisoquinoline Transient Receptor Potential Melastatin 8 (TRPM8) Antagonists

Journal of medicinal chemistry, 2014-04, Vol.57 (7), p.2989-3004

2014

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Synthesis and preliminary biological evaluation of potent and selective 2-(3-alkoxy-1-azetidinyl) quinolines as novel PDE10A inhibitors with improved solubility

Bioorganic & medicinal chemistry, 2014-12, Vol.22 (23), p.6570-6585

2014

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Design and Synthesis of Potent, Orally Efficacious Hydroxyethylamine Derived β-Site Amyloid Precursor Protein Cleaving Enzyme (BACE1) Inhibitors

Journal of medicinal chemistry, 2012-11, Vol.55 (21), p.9025-9044

2012

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Stereoselective Synthesis of anti-N-Protected 3-Amino-1,2-epoxides by Nucleophilic Addition to N-tert-Butanesulfinyl Imine of a Glyceraldehyde Synthon

Journal of organic chemistry, 2009-08, Vol.74 (16), p.5975-5982

2009

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Establishing the relationship between in vitro potency, pharmacokinetic, and pharmacodynamic parameters in a series of orally available, hydroxyethylamine-derived β-secretase inhibitors

The Journal of pharmacology and experimental therapeutics, 2012-11, Vol.343 (2), p.460

2012

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Structure-activity relationships of 3,4-dihydro-1H-quinazolin-2-one derivatives as potential CDK5 inhibitors

Bioorganic & medicinal chemistry, 2007-10, Vol.15 (20), p.6574-6595

2007

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Design and synthesis of 6-oxo-1,6-dihydropyridines as CDK5 inhibitors

Bioorganic & medicinal chemistry letters, 2009-12, Vol.19 (23), p.6591-6594

2009

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Design and synthesis of quinolin-2(1 H)-one derivatives as potent CDK5 inhibitors

Bioorganic & medicinal chemistry letters, 2007-10, Vol.17 (19), p.5384-5389

2007

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Synthesis and conformational analysis of α,α-difluoroalkyl heteroaryl ethers

Tetrahedron letters, 2009-09, Vol.50 (39), p.5452-5455

2009

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Redox behaviour and reactions of (PhCH2)3Sb; syntheses and structures of [(PhCH2)3SbMe]I and [(PhCH2)3SbMe]3Sb3I12

Journal of organometallic chemistry, 1994-12, Vol.483 (1-2), p.167-172

1994

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Equilibria in Organo Antimony Ring Chemistry

Phosphorus, sulfur and silicon and the related elements (Print), 1992-01, Vol.64 (1-4), p.107-112

1992

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Synthesis of (Me 3SiCH 2Sb) n and reactions with ditellurides: crystal structure of [Cp 2Co][Me 3SiCH 2SbCl 3]

Journal of organometallic chemistry, 1995-10, Vol.501 (1), p.117-121

1995

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Structure–activity relationships of 3,4-dihydro-1 H-quinazolin-2-one derivatives as potential CDK5 inhibitors

Bioorganic & medicinal chemistry, 2007, Vol.15 (20), p.6574-6595

2007

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Syntheses and structures of isopropyl- and (bis(trimethylsilyl)methyl)antimony rings and catena-tri- and catena-tetrastibanes by reaction of organoantimony rings with distibanes

Organometallics, 1992, Vol.11 (1), p.145-150

1992

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Strukturen von Tetramesityldistiban (Mes4Sb2) und Trimesitylstiban (Mes3Sb)

Zeitschrift für Naturforschung. B, A journal of chemical sciences, 1992-04, Vol.47 (4), p.503-508

1992

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Schwefel verbindungen des erdöls. XVII: Dibenzothiophene mit einem verzweigten C3 -C5-alkylrest

Phosphorus, sulfur, and silicon and the related elements, 1992, Vol.72 (1-4), p.33-47

1992

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DARSTELLUNG UND OXIDATION VON p-TOLYL-BIS(TRIMETHYLGERMYL)STIBAN (1) UND p-TOLYLBIS(TRIMETHYLSTANNYL)STIBAN (2)

Phosphorus, sulfur, and silicon and the related elements, 1994-03, Vol.88 (1-4), p.275-277

1994

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SYNTHESE VON TETRAKIS-(TRIMETHYLSILYLMETHYL)DISTIBAN UND REAKTIONEN MIT DITELLURIDEN ODER TELLUR

Phosphorus, sulfur, and silicon and the related elements, 1994-06, Vol.91 (1-4), p.165-168

1994

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Redox behaviour and reactions of (PhCH 2) 3Sb; syntheses and structures of [(PhCH 2) 3SbMe]I and [(PhCH 2) 3SbMe] 3Sb 3I 12

Journal of organometallic chemistry, 1994, Vol.483 (1), p.167-172

1994

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Reactions of Cyclostibanes or Distibanes with Diselenides or Ditellurides

Phosphorus, sulfur, and silicon and the related elements, 1992-04, Vol.67 (1-4), p.33-38

1992

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Discovery of TRPM8 Antagonist (S)‑6-(((3-Fluoro-4-(trifluoromethoxy)phenyl)(3-fluoropyridin-2-yl)methyl)carbamoyl)nicotinic Acid (AMG 333), a Clinical Candidate for the Treatment of Migraine

Synthesis and structure–activity relationship of trisubstituted thiazoles as Cdc7 kinase inhibitors

Targeting the Mitotic Kinesin KIF18A in Chromosomally Unstable Cancers: Hit Optimization Toward an In Vivo Chemical Probe

Design and Preparation of a Potent Series of Hydroxyethylamine Containing β-Secretase Inhibitors That Demonstrate Robust Reduction of Central β-Amyloid

Optimization of Potency and Pharmacokinetic Properties of Tetrahydroisoquinoline Transient Receptor Potential Melastatin 8 (TRPM8) Antagonists

Synthesis and preliminary biological evaluation of potent and selective 2-(3-alkoxy-1-azetidinyl) quinolines as novel PDE10A inhibitors with improved solubility

Design and Synthesis of Potent, Orally Efficacious Hydroxyethylamine Derived β-Site Amyloid Precursor Protein Cleaving Enzyme (BACE1) Inhibitors

Stereoselective Synthesis of anti-N-Protected 3-Amino-1,2-epoxides by Nucleophilic Addition to N-tert-Butanesulfinyl Imine of a Glyceraldehyde Synthon

Establishing the relationship between in vitro potency, pharmacokinetic, and pharmacodynamic parameters in a series of orally available, hydroxyethylamine-derived β-secretase inhibitors

A Potent and Orally Efficacious, Hydroxyethylamine-Based Inhibitor of β-Secretase

Structure-activity relationships of 3,4-dihydro-1H-quinazolin-2-one derivatives as potential CDK5 inhibitors

Design and synthesis of 6-oxo-1,6-dihydropyridines as CDK5 inhibitors

Design and synthesis of quinolin-2(1 H)-one derivatives as potent CDK5 inhibitors

Synthesis and conformational analysis of α,α-difluoroalkyl heteroaryl ethers

Redox behaviour and reactions of (PhCH2)3Sb; syntheses and structures of [(PhCH2)3SbMe]I and [(PhCH2)3SbMe]3Sb3I12

Equilibria in Organo Antimony Ring Chemistry

Synthesis of (Me 3SiCH 2Sb) n and reactions with ditellurides: crystal structure of [Cp 2Co][Me 3SiCH 2SbCl 3]

Structure–activity relationships of 3,4-dihydro-1 H-quinazolin-2-one derivatives as potential CDK5 inhibitors

Syntheses and structures of isopropyl- and (bis(trimethylsilyl)methyl)antimony rings and catena-tri- and catena-tetrastibanes by reaction of organoantimony rings with distibanes

Strukturen von Tetramesityldistiban (Mes4Sb2) und Trimesitylstiban (Mes3Sb)

Schwefel verbindungen des erdöls. XVII: Dibenzothiophene mit einem verzweigten C3 -C5-alkylrest

DARSTELLUNG UND OXIDATION VON p-TOLYL-BIS(TRIMETHYLGERMYL)STIBAN (1) UND p-TOLYLBIS(TRIMETHYLSTANNYL)STIBAN (2)

SYNTHESE VON TETRAKIS-(TRIMETHYLSILYLMETHYL)DISTIBAN UND REAKTIONEN MIT DITELLURIDEN ODER TELLUR

Redox behaviour and reactions of (PhCH 2) 3Sb; syntheses and structures of [(PhCH 2) 3SbMe]I and [(PhCH 2) 3SbMe] 3Sb 3I 12

Reactions of Cyclostibanes or Distibanes with Diselenides or Ditellurides

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