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Specific inhibition of spleen tyrosine kinase suppresses leukocyte immune function and inflammation in animal models of rheumatoid arthritis

The Journal of pharmacology and experimental therapeutics, 2012-02, Vol.340 (2), p.350

2012

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[18F]BTK-1: A Novel Positron Emission Tomography Tracer for Imaging Bruton’s Tyrosine Kinase

Molecular imaging and biology, 2022-10, Vol.24 (5), p.830-841

2022

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Discovery of betrixaban (PRT054021), N-(5-chloropyridin-2-yl)-2-(4-( N, N-dimethylcarbamimidoyl)benzamido)-5-methoxybenzamide, a highly potent, selective, and orally efficacious factor Xa inhibitor

Bioorganic & medicinal chemistry letters, 2009-04, Vol.19 (8), p.2179-2185

2009

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Inhibitory effect of carboxylic acid group on hERG binding

Bioorganic & medicinal chemistry letters, 2006-11, Vol.16 (21), p.5507-5512

2006

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Design, Synthesis and Discovery of 1-(2-(6-Chloro-3-methylsulfonyl)-naphthyl)-1H-pyrazole-5-carboxylamides as Highly Potent Factor Xa Inhibitors

Chemical and Pharmaceutical Bulletin, 2009/09/01, Vol.57(9), pp.1004-1007

2009

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Anthranilamide-based N, N-dialkylbenzamidines as potent and orally bioavailable factor Xa inhibitors: P4 SAR

Bioorganic & medicinal chemistry letters, 2009-04, Vol.19 (8), p.2186-2189

2009

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1-(2-Naphthyl)-1H-pyrazole-5-carboxylamides as potent factor xa inhibitors. Part 3: Design, synthesis and sar of orally bioavailable benzamidine-P4 inhibitors

Bioorganic & medicinal chemistry letters, 2004-03, Vol.14 (5), p.1229-1234

2004

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Combinatorial inhibition of Tec kinases BTK and ITK is beneficial in ameliorating murine sclerodermatous chronic graft versus host disease

Bone marrow transplantation (Basingstoke), 2023-08, Vol.58 (8), p.924-935

2023

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1-(2-Naphthyl)-1H-pyrazole-5-carboxylamides as potent factor xa inhibitors. Part 2: A survey of P4 motifs

Bioorganic & medicinal chemistry letters, 2004-03, Vol.14 (5), p.1221-1227

2004

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Synthesis of Linear and Angular Triquinane Skeletons by O-Stannyl Ketyl-Promoted Fragmentation−Cyclization Reactions of α-Keto Cyclopropanes

Journal of organic chemistry, 1997-01, Vol.62 (1), p.174-181

1997

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Design, synthesis and structure–Activity relationships of benzoxazinone-Based factor Xa inhibitors

Bioorganic & medicinal chemistry letters, 2003-02, Vol.13 (3), p.561-566

2003

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Design, synthesis, and SAR of anthranilamide-based factor Xa inhibitors incorporating substituted biphenyl P4 motifs

Bioorganic & medicinal chemistry letters, 2004-02, Vol.14 (4), p.983-987

2004

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Design, synthesis, and SAR of anthranilamide-based factor Xa inhibitors with improved functional activity

Bioorganic & medicinal chemistry letters, 2004-02, Vol.14 (4), p.989-993

2004

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361 - Differential Inhibition of Tec Kinases Is Beneficial in Ameliorating Murine Sclerodermatous Chronic Graft-Versus-Host Disease

Transplantation and cellular therapy, 2022-03, Vol.28 (3), p.S279-S280

2022

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Differential Inhibition of Tec Kinases Is Beneficial in Ameliorating Murine Sclerodermatous Chronic Graft-Versus-Host Disease

Transplantation and cellular therapy, 2022-03, Vol.28 (3), p.S279-S280

2022

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N, N-Dialkylated 4-(4-arylsulfonylpiperazine-1-carbonyl)-benzamidines and 4-((4-arylsulfonyl)-2-oxo-piperazin-1-ylmethyl)-benzamidines as potent factor Xa inhibitors

Bioorganic & medicinal chemistry letters, 2004-05, Vol.14 (9), p.2073-2078

2004

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Inhibition of purified factor Xa amidolytic activity may not be predictive of inhibition of in vivo thrombosis: implications for identification of therapeutically active inhibitors

Arteriosclerosis, thrombosis, and vascular biology, 2003-06, Vol.23 (6), p.1098

2003

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One- and Two-Electron Reactions from the Rearrangement of α-Ketocyclopropanes by O-Stannyl Ketyls

Journal of organic chemistry, 1997-12, Vol.62 (26), p.9159-9164

1997

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Tetrachlorophthalimido- and Pent-4-enoyl-Protected Glucosamines as Precursors for Preparation of 2-Azido-2-deoxyglucopyranosyl Building Blocks

Journal of organic chemistry, 1998-05, Vol.63 (11), p.3790-3792

1998

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Reactions of Tin(IV) Enolates and Radicals Derived from the Tin Hydride Scission of Cyclopropyl Ketones

Journal of organic chemistry, 1997-08, Vol.62 (16), p.5248-5249

1997

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Design, Synthesis, and SAR of Amino Acid Derivatives as Factor Xa Inhibitors

Bioorganic & medicinal chemistry letters, 2001-11, Vol.11 (22), p.2947-2950

2001

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Design, synthesis and biological activity of novel non-amidine factor Xa inhibitors. Part 1: P1 Structure-activity relationships of the substituted 1-(2-naphthyl)-1H-pyrazole-5-carboxylamides

Bioorganic & medicinal chemistry letters, 2002-06, Vol.12 (12), p.1651-1655

2002

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Construction of a linear triquinane skeleton by an O-stannyl ketyl radical rearrangement

Chemical communications (Cambridge, England), 1996 (13), p.1567

1996

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Fragmentation-cyclization reactions of O-stannyl ketyls: The synthesis of an angular triquinane skeleton

Tetrahedron letters, 1996-02, Vol.37 (8), p.1177-1178

1996

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Design, synthesis, and SAR of substituted acrylamides as factor Xa inhibitors

Bioorganic & medicinal chemistry letters, 2002-06, Vol.12 (11), p.1511-1515

2002

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Specific inhibition of spleen tyrosine kinase suppresses leukocyte immune function and inflammation in animal models of rheumatoid arthritis

[18F]BTK-1: A Novel Positron Emission Tomography Tracer for Imaging Bruton’s Tyrosine Kinase

Discovery of betrixaban (PRT054021), N-(5-chloropyridin-2-yl)-2-(4-( N, N-dimethylcarbamimidoyl)benzamido)-5-methoxybenzamide, a highly potent, selective, and orally efficacious factor Xa inhibitor

Inhibitory effect of carboxylic acid group on hERG binding

Design, Synthesis and Discovery of 1-(2-(6-Chloro-3-methylsulfonyl)-naphthyl)-1H-pyrazole-5-carboxylamides as Highly Potent Factor Xa Inhibitors

Anthranilamide-based N, N-dialkylbenzamidines as potent and orally bioavailable factor Xa inhibitors: P4 SAR

1-(2-Naphthyl)-1H-pyrazole-5-carboxylamides as potent factor xa inhibitors. Part 3: Design, synthesis and sar of orally bioavailable benzamidine-P4 inhibitors

Combinatorial inhibition of Tec kinases BTK and ITK is beneficial in ameliorating murine sclerodermatous chronic graft versus host disease

1-(2-Naphthyl)-1H-pyrazole-5-carboxylamides as potent factor xa inhibitors. Part 2: A survey of P4 motifs

Synthesis of Linear and Angular Triquinane Skeletons by O-Stannyl Ketyl-Promoted Fragmentation−Cyclization Reactions of α-Keto Cyclopropanes

Design, synthesis and structure–Activity relationships of benzoxazinone-Based factor Xa inhibitors

Design, synthesis, and SAR of anthranilamide-based factor Xa inhibitors incorporating substituted biphenyl P4 motifs

Design, synthesis, and SAR of anthranilamide-based factor Xa inhibitors with improved functional activity

361 - Differential Inhibition of Tec Kinases Is Beneficial in Ameliorating Murine Sclerodermatous Chronic Graft-Versus-Host Disease

Differential Inhibition of Tec Kinases Is Beneficial in Ameliorating Murine Sclerodermatous Chronic Graft-Versus-Host Disease

N, N-Dialkylated 4-(4-arylsulfonylpiperazine-1-carbonyl)-benzamidines and 4-((4-arylsulfonyl)-2-oxo-piperazin-1-ylmethyl)-benzamidines as potent factor Xa inhibitors

Inhibition of purified factor Xa amidolytic activity may not be predictive of inhibition of in vivo thrombosis: implications for identification of therapeutically active inhibitors

One- and Two-Electron Reactions from the Rearrangement of α-Ketocyclopropanes by O-Stannyl Ketyls

Tetrachlorophthalimido- and Pent-4-enoyl-Protected Glucosamines as Precursors for Preparation of 2-Azido-2-deoxyglucopyranosyl Building Blocks

Reactions of Tin(IV) Enolates and Radicals Derived from the Tin Hydride Scission of Cyclopropyl Ketones

Design, Synthesis, and SAR of Amino Acid Derivatives as Factor Xa Inhibitors

Design, synthesis and biological activity of novel non-amidine factor Xa inhibitors. Part 1: P1 Structure-activity relationships of the substituted 1-(2-naphthyl)-1H-pyrazole-5-carboxylamides

Construction of a linear triquinane skeleton by an O-stannyl ketyl radical rearrangement

Fragmentation-cyclization reactions of O-stannyl ketyls: The synthesis of an angular triquinane skeleton

Design, synthesis, and SAR of substituted acrylamides as factor Xa inhibitors

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