UB Paderborn / Katalog / Suche / in CDI

Sortiert nach

Einfacher Volltextzugriff von (fast) überall

Installieren Sie die LibKey Nomad-Browsererweiterung und erhalten Sie von vielen Webseiten einfachen Zugriff auf lizenzierte Volltexte oder Open Access Publikationen. Mehr erfahren...

Genetic Ablation of CD38 Protects against Western Diet-Induced Exercise Intolerance and Metabolic Inflexibility

PloS one, 2015-08, Vol.10 (8), p.e0134927-e0134927

2015

Volltextzugriff (PDF)

Discovery, Synthesis, and Biological Evaluation of Thiazoloquin(az)olin(on)es as Potent CD38 Inhibitors

Journal of medicinal chemistry, 2015-04, Vol.58 (8), p.3548-3571

2015

Volltextzugriff (PDF)

Differential recognition of HIV-stimulated IL-1β and IL-18 secretion through NLR and NAIP signalling in monocyte-derived macrophages

PLoS pathogens, 2021-04, Vol.17 (4), p.e1009417-e1009417

2021

Volltextzugriff (PDF)

Discovery of 4‑Amino-8-quinoline Carboxamides as Novel, Submicromolar Inhibitors of NAD-Hydrolyzing Enzyme CD38

Journal of medicinal chemistry, 2015-09, Vol.58 (17), p.7021-7056

2015

Volltextzugriff (PDF)

2,4-Diamino-8-quinazoline carboxamides as novel, potent inhibitors of the NAD hydrolyzing enzyme CD38: Exploration of the 2-position structure-activity relationships

Bioorganic & medicinal chemistry, 2018-05, Vol.26 (8), p.2107-2150

2018

Volltextzugriff (PDF)

Identification of a Chemical Tool for the Orphan Nuclear Receptor FXR

Journal of medicinal chemistry, 2000-08, Vol.43 (16), p.2971-2974

2000

Volltextzugriff (PDF)

Discovery of Pyrazolocarboxamides as Potent and Selective Receptor Interacting Protein 2 (RIP2) Kinase Inhibitors

ACS medicinal chemistry letters, 2019-11, Vol.10 (11), p.1518-1523

2019

Volltextzugriff (PDF)

Novel selective small molecule agonists for peroxisome proliferator-activated receptor δ (PPARδ)—synthesis and biological activity

Bioorganic & medicinal chemistry letters, 2003-05, Vol.13 (9), p.1517-1521

2003

Volltextzugriff (PDF)

Pyrrolidinyl pyridone and pyrazinone analogues as potent inhibitors of prolyl oligopeptidase (POP)

Bioorganic & medicinal chemistry, 2008-08, Vol.18 (15), p.4360-4363

2008

Volltextzugriff (PDF)

N-{3-[(1,1-dioxido-1,2-benzothiazol-3-yl)(phenyl)amino]propyl}benzamide analogs as potent Kv1.3 inhibitors. Part 1

Bioorganic & medicinal chemistry letters, 2010-12, Vol.20 (23), p.6983-6988

2010

Volltextzugriff (PDF)

Substituted N-{3-[(1,1-dioxido-1,2-benzothiazol-3-yl)(phenyl)amino]propyl}benzamide analogs as potent Kv1.3 ion channel blockers. Part 2

Bioorganic & medicinal chemistry letters, 2010-12, Vol.20 (23), p.6989-6992

2010

Volltextzugriff (PDF)

The Palladium-Catalyzed Enyne Cycloisomerization Reaction in a General Approach to the Asymmetric Syntheses of the Picrotoxane Sesquiterpenes. Part I. First-Generation Total Synthesis of Corianin and Formal Syntheses of Picrotoxinin and Picrotin

Journal of the American Chemical Society, 1999-07, Vol.121 (26), p.6183-6192

1999

Volltextzugriff (PDF)

Structure-Based Design of Potent Retinoid X Receptor α Agonists

Journal of medicinal chemistry, 2004-04, Vol.47 (8), p.2010-2029

2004

Volltextzugriff (PDF)

2-Cyano-4-fluoro-1-thiovalylpyrrolidine analogues as potent inhibitors of DPP-IV

Bioorganic & medicinal chemistry letters, 2005-12, Vol.15 (23), p.5257-5261

2005

Volltextzugriff (PDF)

Differential recognition of HIV-stimulated IL-1[beta] and IL-18 secretion through NLR and NAIP signalling in monocyte-derived macrophages

PLoS pathogens, 2021-04, Vol.17 (4)

2021

Volltextzugriff (PDF)

N-{3-[(1,1-dioxido-1,2-benzothiazol-3-yl)(phenyl)amino]propyl}benz amide analogs as potent Kv1.3 inhibitors. Part 1

Bioorganic & medicinal chemistry letters, 2010-12, Vol.20 (23), p.6983-6988

2010

Volltextzugriff (PDF)

Diastereomeric atropisomers of the tricyclo[9.3.1.03,8]pentadecane ring system. Synthesis and structural studies

Journal of the American Chemical Society, 1986-08, Vol.108 (16), p.4953-4956

1986

Volltextzugriff (PDF)

Substituted N-{3-[(1,1-dioxido-1,2-benzothiazol-3-yl)(phenyl)amino]propyl}b enzamide analogs as potent Kv1.3 ion channel blockers. Part 2

Bioorganic & medicinal chemistry letters, 2010-12, Vol.20 (23), p.6989-6992

2010

Volltextzugriff (PDF)

An efficient synthesis of 3-pyridyl-N-oxide steroides: Inhibitors of 5α-reductase

Tetrahedron letters, 1994-02, Vol.35 (9), p.1349-1352

Haffner, Curt

1994

Volltextzugriff (PDF)

Synthesis of 6-azacholesten-3-ones: Potent inhibitors of 5α-reductase

Tetrahedron letters, 1995-06, Vol.36 (23), p.4039-4042

Haffner, Curt

1995

Volltextzugriff (PDF)

Linear Relationships between the Ligand Binding Energy and the Activation Energy of Time-dependent Inhibition of Steroid 5α-Reductase by Δ1-4-Azasteroids

The Journal of biological chemistry, 2001-06, Vol.276 (24), p.21359-21364

2001

Volltextzugriff (PDF)

6-Azasteroids: Structure-Activity Relationships for Inhibition of Type 1 and 2 Human 5.alpha.-Reductase and Human Adrenal 3.beta.-Hydroxy-.DELTA.5-steroid Dehydrogenase/3-Keto-.DELTA.5-steroid Isomerase

Journal of medicinal chemistry, 1994-07, Vol.37 (15), p.2352-2360

1994

Volltextzugriff (PDF)

6-Azasteroids: potent dual inhibitors of human type 1 and 2 steroid 5.alpha.-reductase

Journal of medicinal chemistry, 1993-12, Vol.36 (26), p.4313-4315

1993

Volltextzugriff (PDF)

Linear Relationships between the Ligand Binding Energy and the Activation Energy of Time-dependent Inhibition of Steroid 5Î±-Reductase by Î1-4-Azasteroids

The Journal of biological chemistry, 2001-06, Vol.276 (24), p.21359

2001

Volltextzugriff (PDF)

1 – 25 von 31

Suche als RSS-Feed

Suchergebnisse filtern

Filter anzeigen

Nur zeigen

Geprüft (Peer-Review)
(27)
Mit Volltextzugriff
(30)

Publikationsform

Artikel
(30)
Dissertationen
(1)

Sprache

Englisch
(31)

Erscheinungsjahr

n.n

Thema

Science & Technology
(18)
Life Sciences & Biomedicine
(14)
Chemistry, Medicinal
(12)
Pharmacology & Pharmacy
(12)
Animals
(10)
Humans
(10)
Chemistry
(9)
Physical Sciences
(9)
Biological And Medical Sciences
(8)
Medical Sciences
(8)
Pharmacology. Drug Treatments
(8)
Chemistry, Organic
(7)
Cell Line
(6)
General And Cellular Metabolism. Vitamins
(5)
Rats
(5)
Structure-Activity Relationship
(5)
Mice
(4)
Combinatorial Chemistry Techniques
(3)
Crystallography, X-Ray
(3)
Male
(3)

15 weitere anzeigen...

Weniger anzeigen...

Menü

Weitere Dienste

Einstellungen

Genetic Ablation of CD38 Protects against Western Diet-Induced Exercise Intolerance and Metabolic Inflexibility

Discovery, Synthesis, and Biological Evaluation of Thiazoloquin(az)olin(on)es as Potent CD38 Inhibitors

Differential recognition of HIV-stimulated IL-1β and IL-18 secretion through NLR and NAIP signalling in monocyte-derived macrophages

Discovery of 4‑Amino-8-quinoline Carboxamides as Novel, Submicromolar Inhibitors of NAD-Hydrolyzing Enzyme CD38

2,4-Diamino-8-quinazoline carboxamides as novel, potent inhibitors of the NAD hydrolyzing enzyme CD38: Exploration of the 2-position structure-activity relationships

Identification of a Chemical Tool for the Orphan Nuclear Receptor FXR

Discovery of Pyrazolocarboxamides as Potent and Selective Receptor Interacting Protein 2 (RIP2) Kinase Inhibitors

Novel selective small molecule agonists for peroxisome proliferator-activated receptor δ (PPARδ)—synthesis and biological activity

Pyrrolidinyl pyridone and pyrazinone analogues as potent inhibitors of prolyl oligopeptidase (POP)

N-{3-[(1,1-dioxido-1,2-benzothiazol-3-yl)(phenyl)amino]propyl}benzamide analogs as potent Kv1.3 inhibitors. Part 1

Substituted N-{3-[(1,1-dioxido-1,2-benzothiazol-3-yl)(phenyl)amino]propyl}benzamide analogs as potent Kv1.3 ion channel blockers. Part 2

The Palladium-Catalyzed Enyne Cycloisomerization Reaction in a General Approach to the Asymmetric Syntheses of the Picrotoxane Sesquiterpenes. Part I. First-Generation Total Synthesis of Corianin and Formal Syntheses of Picrotoxinin and Picrotin

Structure-Based Design of Potent Retinoid X Receptor α Agonists

2-Cyano-4-fluoro-1-thiovalylpyrrolidine analogues as potent inhibitors of DPP-IV

Differential recognition of HIV-stimulated IL-1[beta] and IL-18 secretion through NLR and NAIP signalling in monocyte-derived macrophages

N-{3-[(1,1-dioxido-1,2-benzothiazol-3-yl)(phenyl)amino]propyl}benz amide analogs as potent Kv1.3 inhibitors. Part 1

Diastereomeric atropisomers of the tricyclo[9.3.1.03,8]pentadecane ring system. Synthesis and structural studies

Substituted N-{3-[(1,1-dioxido-1,2-benzothiazol-3-yl)(phenyl)amino]propyl}b enzamide analogs as potent Kv1.3 ion channel blockers. Part 2

An efficient synthesis of 3-pyridyl-N-oxide steroides: Inhibitors of 5α-reductase

Synthesis of 6-azacholesten-3-ones: Potent inhibitors of 5α-reductase

Linear Relationships between the Ligand Binding Energy and the Activation Energy of Time-dependent Inhibition of Steroid 5α-Reductase by Δ1-4-Azasteroids

6-Azasteroids: Structure-Activity Relationships for Inhibition of Type 1 and 2 Human 5.alpha.-Reductase and Human Adrenal 3.beta.-Hydroxy-.DELTA.5-steroid Dehydrogenase/3-Keto-.DELTA.5-steroid Isomerase

Structure-Activity Relationships for Inhibition of Type 1 and 2 Human 5.alpha.-Reductase and Human Adrenal 3.beta.-Hydroxy-.DELTA.5-steroid Dehydrogenase/3-Keto-.DELTA.5-steroid Isomerase by 6-Azaandrost-4-en-3-ones: Optimization of the C17 Substituent

6-Azasteroids: potent dual inhibitors of human type 1 and 2 steroid 5.alpha.-reductase

Linear Relationships between the Ligand Binding Energy and the Activation Energy of Time-dependent Inhibition of Steroid 5Î±-Reductase by Î1-4-Azasteroids

Suchergebnisse filtern