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Tetrahydrofuran-Based Transient Receptor Potential Ankyrin 1 (TRPA1) Antagonists: Ligand-Based Discovery, Activity in a Rodent Asthma Model, and Mechanism-of-Action via Cryogenic Electron Microscopy

Journal of medicinal chemistry, 2021-04, Vol.64 (7), p.3843-3869

2021

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Novel Inhibitor Binding Site Discovery on HIV‑1 Capsid N‑Terminal Domain by NMR and X‑ray Crystallography

ACS chemical biology, 2013-05, Vol.8 (5), p.1074-1082

2013

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Discovery of a 1,5-dihydrobenzo[b][1,4]diazepine-2,4-dione series of inhibitors of HIV-1 capsid assembly

Bioorganic & medicinal chemistry letters, 2011-01, Vol.21 (1), p.398-404

2011

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Discovery of Small-Molecule Inhibitors of the ATPase Activity of Human Papillomavirus E1 Helicase

Journal of medicinal chemistry, 2004-01, Vol.47 (1), p.18-21

2004

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Monitoring Binding of HIV-1 Capsid Assembly Inhibitors Using 19F Ligand-and 15N Protein-Based NMR and X-ray Crystallography: Early Hit Validation of a Benzodiazepine Series

ChemMedChem, 2013-03, Vol.8 (3), p.405-414

2013

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Discovery of TRPA1 Antagonist GDC-6599: Derisking Preclinical Toxicity and Aldehyde Oxidase Metabolism with a Potential First-in-Class Therapy for Respiratory Disease

Journal of medicinal chemistry, 2024-03, Vol.67 (5), p.3287-3306

2024

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Discovery and Structural Characterization of a New Inhibitor Series of HIV-1 Nucleocapsid Function: NMR Solution Structure Determination of a Ternary Complex Involving a 2:1 Inhibitor/NC Stoichiometry

Journal of molecular biology, 2013-06, Vol.425 (11), p.1982-1998

2013

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Structure−Activity Study on a Novel Series of Macrocyclic Inhibitors of the Hepatitis C Virus NS3 Protease Leading to the Discovery of BILN 2061

Journal of medicinal chemistry, 2004-03, Vol.47 (7), p.1605-1608

2004

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Design, synthesis and biological evaluation of novel aminothiazoles as antiviral compounds acting against human rhinovirus

Bioorganic & medicinal chemistry letters, 2013-07, Vol.23 (13), p.3841-3847

2013

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Characterization of the Human Cytomegalovirus Protease As an Induced-Fit Serine Protease and the Implications to the Design of Mechanism-Based Inhibitors

Journal of the American Chemical Society, 1999-04, Vol.121 (13), p.2974-2986

1999

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Preparation of 3-O-aryl chloramphenicol derivatives via chemoselective copper-catalyzed O-arylation of (1R,2R)-(−)-N-BOC-2-amino-1-(4-nitrophenyl)-1,3-propanediol using triarylbismuthines

Tetrahedron letters, 2016-09, Vol.57 (38), p.4284-4287

2016

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Potent Inhibitors of the Hepatitis C Virus NS3 Protease: Design and Synthesis of Macrocyclic Substrate-Based β-Strand Mimics

Journal of organic chemistry, 2004-09, Vol.69 (19), p.6185-6201

2004

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The Conformation of a Peptidyl Methyl Ketone Inhibitor Bound to the Human Cytomegalovirus Protease

Angewandte Chemie (International ed.), 1998-10, Vol.37 (19), p.2729-2732

1998

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Evidence of a Conformational Change in the Human Cytomegalovirus Protease upon Binding of Peptidyl-Activated Carbonyl Inhibitors

Biochemistry (Easton), 1997-10, Vol.36 (41), p.12644-12652

1997

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tris(2-Carboxyethyl)phosphine (TCEP) for the Reduction of Sulfoxides, Sulfonylchlorides, N-Oxides, and Azides

Synthetic communications, 2003-10, Vol.33 (20), p.3503-3511

2003

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Monitoring binding of HIV-1 capsid assembly inhibitors using (19)F ligand-and (15)N protein-based NMR and X-ray crystallography: early hit validation of a benzodiazepine series

ChemMedChem, 2013-03, Vol.8 (3), p.405-414

2013

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Peptidomimetic Inhibitors of the Human Cytomegalovirus Protease

Journal of medicinal chemistry, 1997-12, Vol.40 (25), p.4113-4135

1997

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Monitoring Binding of HIV‐1 Capsid Assembly Inhibitors Using 19 F Ligand‐and 15 N Protein‐Based NMR and X‐ray Crystallography: Early Hit Validation of a Benzodiazepine Series

ChemMedChem, 2013-03, Vol.8 (3), p.405-414

2013

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Inside Cover: Monitoring Binding of HIV‐1 Capsid Assembly Inhibitors Using 19 F Ligand‐and 15 N Protein‐Based NMR and X‐ray Crystallography: Early Hit Validation of a Benzodiazepine Series (ChemMedChem 3/2013)

ChemMedChem, 2013-03, Vol.8 (3), p.346-346

2013

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Inside Cover: Monitoring Binding of HIV-1 Capsid Assembly Inhibitors Using 19F Ligand-and 15N Protein-Based NMR and X-ray Crystallography: Early Hit Validation of a Benzodiazepine Series (ChemMedChem 3/2013)

ChemMedChem, 2013-03, Vol.8 (3), p.346-346

2013

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Potent Inhibitors of the Hepatitis C Virus NS3 Protease: Design and Synthesis of Macrocyclic Substrate-Based [beta]-Strand Mimics

Journal of organic chemistry, 2008-06, Vol.69 ((19) ; 09, 2004)

2008

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2‘,6‘-Dimethylphenoxyacetyl: A New Achiral High Affinity P 3 -P 2 Ligand for Peptidomimetic-Based HIV Protease Inhibitors

Journal of medicinal chemistry, 2000-03, Vol.43 (6), p.1094-1108

2000

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2‘,6‘-Dimethylphenoxyacetyl: A New Achiral High Affinity P3-P2 Ligand for Peptidomimetic-Based HIV Protease Inhibitors

Journal of medicinal chemistry, 2000-03, Vol.43 (6), p.1094-1108

2000

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Chemo-enzymatic synthesis of chiral 2-substituted succinic acid derivatives

Tetrahedron: asymmetry, 1999-08, Vol.10 (17), p.3285-3295

1999

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1-Thiazol-2-yl-N-3-methyl-1H-pyrozole-5-carboxylic acid derivatives as antitumor agents

Bioorganic & medicinal chemistry letters, 2017-09, Vol.27 (18), p.4471-4477

2017

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Tetrahydrofuran-Based Transient Receptor Potential Ankyrin 1 (TRPA1) Antagonists: Ligand-Based Discovery, Activity in a Rodent Asthma Model, and Mechanism-of-Action via Cryogenic Electron Microscopy

Novel Inhibitor Binding Site Discovery on HIV‑1 Capsid N‑Terminal Domain by NMR and X‑ray Crystallography

Discovery of a 1,5-dihydrobenzo[b][1,4]diazepine-2,4-dione series of inhibitors of HIV-1 capsid assembly

Discovery of Small-Molecule Inhibitors of the ATPase Activity of Human Papillomavirus E1 Helicase

Monitoring Binding of HIV-1 Capsid Assembly Inhibitors Using 19F Ligand-and 15N Protein-Based NMR and X-ray Crystallography: Early Hit Validation of a Benzodiazepine Series

Discovery of TRPA1 Antagonist GDC-6599: Derisking Preclinical Toxicity and Aldehyde Oxidase Metabolism with a Potential First-in-Class Therapy for Respiratory Disease

Discovery and Structural Characterization of a New Inhibitor Series of HIV-1 Nucleocapsid Function: NMR Solution Structure Determination of a Ternary Complex Involving a 2:1 Inhibitor/NC Stoichiometry

Structure−Activity Study on a Novel Series of Macrocyclic Inhibitors of the Hepatitis C Virus NS3 Protease Leading to the Discovery of BILN 2061

Design, synthesis and biological evaluation of novel aminothiazoles as antiviral compounds acting against human rhinovirus

Characterization of the Human Cytomegalovirus Protease As an Induced-Fit Serine Protease and the Implications to the Design of Mechanism-Based Inhibitors

Preparation of 3-O-aryl chloramphenicol derivatives via chemoselective copper-catalyzed O-arylation of (1R,2R)-(−)-N-BOC-2-amino-1-(4-nitrophenyl)-1,3-propanediol using triarylbismuthines

Potent Inhibitors of the Hepatitis C Virus NS3 Protease: Design and Synthesis of Macrocyclic Substrate-Based β-Strand Mimics

The Conformation of a Peptidyl Methyl Ketone Inhibitor Bound to the Human Cytomegalovirus Protease

Evidence of a Conformational Change in the Human Cytomegalovirus Protease upon Binding of Peptidyl-Activated Carbonyl Inhibitors

tris(2-Carboxyethyl)phosphine (TCEP) for the Reduction of Sulfoxides, Sulfonylchlorides, N-Oxides, and Azides

Monitoring binding of HIV-1 capsid assembly inhibitors using (19)F ligand-and (15)N protein-based NMR and X-ray crystallography: early hit validation of a benzodiazepine series

Peptidomimetic Inhibitors of the Human Cytomegalovirus Protease

Monitoring Binding of HIV‐1 Capsid Assembly Inhibitors Using 19 F Ligand‐and 15 N Protein‐Based NMR and X‐ray Crystallography: Early Hit Validation of a Benzodiazepine Series

Inside Cover: Monitoring Binding of HIV‐1 Capsid Assembly Inhibitors Using 19 F Ligand‐and 15 N Protein‐Based NMR and X‐ray Crystallography: Early Hit Validation of a Benzodiazepine Series (ChemMedChem 3/2013)

Inside Cover: Monitoring Binding of HIV-1 Capsid Assembly Inhibitors Using 19F Ligand-and 15N Protein-Based NMR and X-ray Crystallography: Early Hit Validation of a Benzodiazepine Series (ChemMedChem 3/2013)

Potent Inhibitors of the Hepatitis C Virus NS3 Protease: Design and Synthesis of Macrocyclic Substrate-Based [beta]-Strand Mimics

2‘,6‘-Dimethylphenoxyacetyl: A New Achiral High Affinity P 3 -P 2 Ligand for Peptidomimetic-Based HIV Protease Inhibitors

2‘,6‘-Dimethylphenoxyacetyl: A New Achiral High Affinity P3-P2 Ligand for Peptidomimetic-Based HIV Protease Inhibitors

Chemo-enzymatic synthesis of chiral 2-substituted succinic acid derivatives

1-Thiazol-2-yl-N-3-methyl-1H-pyrozole-5-carboxylic acid derivatives as antitumor agents

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