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Discovery of betrixaban (PRT054021), N-(5-chloropyridin-2-yl)-2-(4-( N, N-dimethylcarbamimidoyl)benzamido)-5-methoxybenzamide, a highly potent, selective, and orally efficacious factor Xa inhibitor

Bioorganic & medicinal chemistry letters, 2009-04, Vol.19 (8), p.2179-2185

2009

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Antimalarial Activities of Novel Synthetic Cysteine Protease Inhibitors

Antimicrobial Agents and Chemotherapy, 2003-12, Vol.47 (12), p.3810-3814

2003

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1-(2-Naphthyl)-1H-pyrazole-5-carboxylamides as potent factor xa inhibitors. Part 2: A survey of P4 motifs

Bioorganic & medicinal chemistry letters, 2004-03, Vol.14 (5), p.1221-1227

2004

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Design, synthesis, and SAR of anthranilamide-based factor Xa inhibitors incorporating substituted biphenyl P4 motifs

Bioorganic & medicinal chemistry letters, 2004-02, Vol.14 (4), p.983-987

2004

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N, N-Dialkylated 4-(4-arylsulfonylpiperazine-1-carbonyl)-benzamidines and 4-((4-arylsulfonyl)-2-oxo-piperazin-1-ylmethyl)-benzamidines as potent factor Xa inhibitors

Bioorganic & medicinal chemistry letters, 2004-05, Vol.14 (9), p.2073-2078

2004

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Synthesis and biological activity of peptidyl aldehyde urokinase inhibitors

Bioorganic & medicinal chemistry letters, 2000-05, Vol.10 (9), p.983-987

2000

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Parallel synthesis and structure–activity relationships of a series of highly potent, selective, and neutral factor Xa inhibitors

Bioorganic & medicinal chemistry letters, 2004-08, Vol.14 (15), p.4045-4050

2004

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Design, Synthesis, and Evolution of a Novel, Selective, and Orally Bioavailable Class of Thrombin Inhibitors: P1-Argininal Derivatives Incorporating P3-P4 Lactam Sulfonamide Moieties

Journal of medicinal chemistry, 1996-11, Vol.39 (23), p.4531-4536

1996

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Discovery of betrixaban (PRT054021), N-(5-chloropyridin-2-yl)-2-(4-(N,N-dimethylcarbamimidoyl)benzamido )-5-metho xybenzamide, a highly potent, selective, and orally efficacious factor Xa inhibitor

Bioorganic & medicinal chemistry letters, 2009-04, Vol.19 (8), p.2179-2185

2009

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Antimalarial Activities of Novel SyntheticCysteine ProteaseInhibitors

Antimicrobial agents and chemotherapy, 2003-12, Vol.47 (12), p.3810-3814

2003

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Novel benzo-fused lactam scaffolds as factor Xa inhibitors

Bioorganic & medicinal chemistry letters, 1999-09, Vol.9 (17), p.2573-2578

1999

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1-(2-Naphthyl)-1 H -pyrazole-5-carboxylamides as potent factor Xa inhibitors. Part 2: A survey of P4 motifs

Bioorganic & medicinal chemistry letters, 2004-03, Vol.14 (5), p.1221-1227

2004

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Rational design, synthesis, and serine protease inhibitory activity of a novel P1-argininal derivative featuring a conformationally constrained P2-P3 bicyclic lactam moiety

Bioorganic & medicinal chemistry letters, 1997-02, Vol.7 (3), p.331-336

1997

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Rational design, synthesis, and serine protease inhibitory activity of a novel P 1-argininal derivative featuring a conformationally constrained P 2–P 3 bicyclic lactam moiety

Bioorganic & medicinal chemistry letters, 1997-02, Vol.7 (3), p.331-336

1997

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Investigation of the S 3 site of thrombin: Design, synthesis and biological activity of 4-substituted 3-amino-2-pyridones incorporating P 1-argininals

Bioorganic & medicinal chemistry letters, 1999-03, Vol.9 (6), p.895-900

1999

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Investigation of the S3 site of thrombin : Design, synthesis and biological activity of 4-substituted 3-amino-2-pyridones incorporating P1-ARGININALS

Bioorganic & medicinal chemistry letters, 1999-03, Vol.9 (6), p.895-900

1999

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Design and synthesis of a novel class of thrombin inhibitors incorporating heterocyclic dipeptide surrogates

Bioorganic & medicinal chemistry letters, 1997-06, Vol.7 (12), p.1543-1548

1997

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Guanylpiperidine peptidomimetics : Potent and selective bis-cation inhibitors of factor Xa

Bioorganic & medicinal chemistry letters, 2000-04, Vol.10 (8), p.745-749

2000

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ChemInform Abstract: Novel Benzo-Fused Lactam Scaffolds as Factor Xa Inhibitors

ChemInform, 1999-11, Vol.30 (48), p.no-no

1999

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ChemInform Abstract: Investigation of the S 3 Site of Thrombin: Design, Synthesis, and Biological Activity of 4‐Substituted 3‐Amino‐2‐pyridones Incorporating P 1 ‐Argininals (VIII)

ChemInform, 1999-06, Vol.30 (26)

1999

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ChemInform Abstract: Investigation of the S3 Site of Thrombin: Design, Synthesis, and Biological Activity of 4-Substituted 3-Amino-2-pyridones Incorporating P1-Argininals (VIII)

ChemInform, 1999-06, Vol.30 (26), p.no-no

1999

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Differential and persistent risk of excess mortality from Hurricane Maria in Puerto Rico: a time-series analysis

The Lancet. Planetary health, 2018-11, Vol.2 (11), p.e478-e488

2018

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Preservation of general intelligence following traumatic brain injury: contributions of the Met66 brain-derived neurotrophic factor

PloS one, 2014-02, Vol.9 (2), p.e88733-e88733

2014

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The Heat Shock Transcription Factor HsfA Plays a Role in Membrane Lipids Biosynthesis Connecting Thermotolerance and Unsaturated Fatty Acid Metabolism in Aspergillus fumigatus

Microbiology spectrum, 2023-06, Vol.11 (3), p.e0162723-e0162723

2023

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Long-term follow-up of IPEX syndrome patients after different therapeutic strategies: An international multicenter retrospective study

Journal of allergy and clinical immunology, 2018-03, Vol.141 (3), p.1036-1049.e5

2018

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Discovery of betrixaban (PRT054021), N-(5-chloropyridin-2-yl)-2-(4-( N, N-dimethylcarbamimidoyl)benzamido)-5-methoxybenzamide, a highly potent, selective, and orally efficacious factor Xa inhibitor

Antimalarial Activities of Novel Synthetic Cysteine Protease Inhibitors

1-(2-Naphthyl)-1H-pyrazole-5-carboxylamides as potent factor xa inhibitors. Part 2: A survey of P4 motifs

Design, synthesis, and SAR of anthranilamide-based factor Xa inhibitors incorporating substituted biphenyl P4 motifs

N, N-Dialkylated 4-(4-arylsulfonylpiperazine-1-carbonyl)-benzamidines and 4-((4-arylsulfonyl)-2-oxo-piperazin-1-ylmethyl)-benzamidines as potent factor Xa inhibitors

Synthesis and biological activity of peptidyl aldehyde urokinase inhibitors

Parallel synthesis and structure–activity relationships of a series of highly potent, selective, and neutral factor Xa inhibitors

Design, Synthesis, and Evolution of a Novel, Selective, and Orally Bioavailable Class of Thrombin Inhibitors: P1-Argininal Derivatives Incorporating P3-P4 Lactam Sulfonamide Moieties

Discovery of betrixaban (PRT054021), N-(5-chloropyridin-2-yl)-2-(4-(N,N-dimethylcarbamimidoyl)benzamido )-5-metho xybenzamide, a highly potent, selective, and orally efficacious factor Xa inhibitor

Antimalarial Activities of Novel SyntheticCysteine ProteaseInhibitors

Novel benzo-fused lactam scaffolds as factor Xa inhibitors

1-(2-Naphthyl)-1 H -pyrazole-5-carboxylamides as potent factor Xa inhibitors. Part 2: A survey of P4 motifs

Rational design, synthesis, and serine protease inhibitory activity of a novel P1-argininal derivative featuring a conformationally constrained P2-P3 bicyclic lactam moiety

Rational design, synthesis, and serine protease inhibitory activity of a novel P 1-argininal derivative featuring a conformationally constrained P 2–P 3 bicyclic lactam moiety

Investigation of the S 3 site of thrombin: Design, synthesis and biological activity of 4-substituted 3-amino-2-pyridones incorporating P 1-argininals

Investigation of the S3 site of thrombin : Design, synthesis and biological activity of 4-substituted 3-amino-2-pyridones incorporating P1-ARGININALS

Design and synthesis of a novel class of thrombin inhibitors incorporating heterocyclic dipeptide surrogates

Guanylpiperidine peptidomimetics : Potent and selective bis-cation inhibitors of factor Xa

ChemInform Abstract: Novel Benzo-Fused Lactam Scaffolds as Factor Xa Inhibitors

ChemInform Abstract: Investigation of the S 3 Site of Thrombin: Design, Synthesis, and Biological Activity of 4‐Substituted 3‐Amino‐2‐pyridones Incorporating P 1 ‐Argininals (VIII)

ChemInform Abstract: Investigation of the S3 Site of Thrombin: Design, Synthesis, and Biological Activity of 4-Substituted 3-Amino-2-pyridones Incorporating P1-Argininals (VIII)

Differential and persistent risk of excess mortality from Hurricane Maria in Puerto Rico: a time-series analysis

Preservation of general intelligence following traumatic brain injury: contributions of the Met66 brain-derived neurotrophic factor

The Heat Shock Transcription Factor HsfA Plays a Role in Membrane Lipids Biosynthesis Connecting Thermotolerance and Unsaturated Fatty Acid Metabolism in Aspergillus fumigatus

Long-term follow-up of IPEX syndrome patients after different therapeutic strategies: An international multicenter retrospective study

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