UB Paderborn / Katalog / Suche / in CDI

Factor VIIa inhibitors: Chemical optimization, preclinical pharmacokinetics, pharmacodynamics, and efficacy in an arterial baboon thrombosis model

Bioorganic & medicinal chemistry letters, 2006-04, Vol.16 (7), p.2037-2041

2006

Volltextzugriff (PDF)

High-Throughput Screening of Enzyme Inhibitors: Simultaneous Determination of Tight-Binding Inhibition Constants and Enzyme Concentration

Analytical biochemistry, 2000-11, Vol.286 (1), p.45-50

2000

Volltextzugriff (PDF)

Potent bivalent inhibition of human tryptase-beta by a synthetic inhibitor

Biological chemistry, 2003-12, Vol.384 (12), p.1605-1611

2003

Volltextzugriff (PDF)

Small molecule inhibitors of plasma kallikrein

Bioorganic & medicinal chemistry letters, 2006-04, Vol.16 (7), p.2034-2036

2006

Volltextzugriff (PDF)

RBC-Specific CD47 Pruning Confers Protection and Underlies the Transient Anemia in Patients Treated with Anti-CD47 Antibody 5F9

Blood, 2018-11, Vol.132 (Supplement 1), p.2327-2327

2018

Volltextzugriff (PDF)

A Novel Approach to Serine Protease Inhibition: Kinetic Characterization of Inhibitors Whose Potencies and Selectivities Are Dramatically Enhanced by Zinc(II)

Biochemistry (Easton), 2000-04, Vol.39 (16), p.4792-4800

2000

Volltextzugriff (PDF)

High-Throughput Screening of Enzyme Inhibitors: Automatic Determination of Tight-Binding Inhibition Constants

Analytical biochemistry, 2000-05, Vol.281 (1), p.62-67

2000

Volltextzugriff (PDF)

Emerging therapeutic targets in asthma: the rationale for mast cell tryptase inhibition

Emerging therapeutic targets, 1999-06, Vol.3 (2), p.203-212

1999

Volltextzugriff (PDF)

Metal mediated protease inhibition: design and synthesis of inhibitors of the human cytomegalovirus (hCMV) protease

Bioorganic & medicinal chemistry letters, 2000-10, Vol.10 (20), p.2279-2282

2000

Volltextzugriff (PDF)

Expression, purification, crystallization and preliminary X-ray diffraction studies of human cathepsin F complexed with an irreversible vinyl sulfone inhibitor

Acta crystallographica. Section D, Biological crystallography., 2002-12, Vol.58 (12), p.2187-2190

2002

Volltextzugriff (PDF)

Lactoferrin, a potent tryptase inhibitor, abolishes late-phase airway responses in allergic sheep

American journal of respiratory and critical care medicine, 1997-08, Vol.156 (2), p.375-381

1997

Volltextzugriff (PDF)

A novel serine protease inhibition motif involving a multi-centered short hydrogen bonding network at the active site

Journal of molecular biology, 2001-04, Vol.307 (5), p.1451-1486

2001

Volltextzugriff (PDF)

Elaborate Manifold of Short Hydrogen Bond Arrays Mediating Binding of Active Site-directed Serine Protease Inhibitors

Journal of molecular biology, 2003-05, Vol.329 (1), p.93-120

2003

Volltextzugriff (PDF)

Optimization of a screening lead for factor VIIa/TF

Bioorganic & medicinal chemistry letters, 2001-09, Vol.11 (17), p.2253-2256

2001

Volltextzugriff (PDF)

Neutrophil Myeloperoxidase Is a Potent and Selective Inhibitor of Mast Cell Tryptase

Archives of biochemistry and biophysics, 1999-06, Vol.366 (1), p.125-130

1999

Volltextzugriff (PDF)

Generation of potent coagulation protease inhibitors utilizing zinc-mediated chelation

Bioorganic & medicinal chemistry letters, 2006-02, Vol.16 (3), p.710-713

2006

Volltextzugriff (PDF)

Contribution of Multicentered Short Hydrogen Bond Arrays to Potency of Active Site-Directed Serine Protease Inhibitors

Journal of the American Chemical Society, 2002-10, Vol.124 (39), p.11657-11668

2002

Volltextzugriff (PDF)

Highly potent non-peptidic inhibitors of the HCV NS3/NS4A serine protease

Bioorganic & medicinal chemistry letters, 2002-11, Vol.12 (21), p.3129-3133

2002

Volltextzugriff (PDF)

Neutral inhibitors of the serine protease factor Xa

Bioorganic & medicinal chemistry letters, 2001-07, Vol.11 (14), p.1801-1804

2001

Volltextzugriff (PDF)

Expression and Characterization of Recombinant Mast Cell Tryptase

Protein expression and purification, 1999-04, Vol.15 (3), p.251-257

1999

Volltextzugriff (PDF)

A novel serine protease inhibition motif involving a multi-centered short hydrogen bonding network at the active site11Edited by D. Rees

Journal of molecular biology, 2001-04, Vol.307 (5), p.1451-1486

2001

Volltextzugriff (PDF)

Engineering inhibitors highly selective for the S1 sites of Ser190 trypsin-like serine protease drug targets

Chemistry & biology, 2001-11, Vol.8 (11), p.1107-1121

2001

Volltextzugriff (PDF)

ChemInform Abstract: Neutral Inhibitors of the Serine Protease Factor Xa

ChemInform, 2001-11, Vol.32 (45), p.no-no

2001

Volltextzugriff (PDF)

Small Molecule Inhibitors of Plasma Kallikrein

ChemInform, 2006-07, Vol.37 (27), p.no-no

2006

Volltextzugriff (PDF)

ChemInform Abstract: Metal Mediated Protease Inhibition: Design and Synthesis of Inhibitors of the Human Cytomegalovirus (hCMV) Protease

ChemInform, 2001-01, Vol.32 (5), p.no-no

2001

Volltextzugriff (PDF)

Menü

Weitere Dienste

Einstellungen

Factor VIIa inhibitors: Chemical optimization, preclinical pharmacokinetics, pharmacodynamics, and efficacy in an arterial baboon thrombosis model

High-Throughput Screening of Enzyme Inhibitors: Simultaneous Determination of Tight-Binding Inhibition Constants and Enzyme Concentration

Potent bivalent inhibition of human tryptase-beta by a synthetic inhibitor

Small molecule inhibitors of plasma kallikrein

RBC-Specific CD47 Pruning Confers Protection and Underlies the Transient Anemia in Patients Treated with Anti-CD47 Antibody 5F9

A Novel Approach to Serine Protease Inhibition: Kinetic Characterization of Inhibitors Whose Potencies and Selectivities Are Dramatically Enhanced by Zinc(II)

High-Throughput Screening of Enzyme Inhibitors: Automatic Determination of Tight-Binding Inhibition Constants

Emerging therapeutic targets in asthma: the rationale for mast cell tryptase inhibition

Metal mediated protease inhibition: design and synthesis of inhibitors of the human cytomegalovirus (hCMV) protease

Expression, purification, crystallization and preliminary X-ray diffraction studies of human cathepsin F complexed with an irreversible vinyl sulfone inhibitor

Lactoferrin, a potent tryptase inhibitor, abolishes late-phase airway responses in allergic sheep

A novel serine protease inhibition motif involving a multi-centered short hydrogen bonding network at the active site

Elaborate Manifold of Short Hydrogen Bond Arrays Mediating Binding of Active Site-directed Serine Protease Inhibitors

Optimization of a screening lead for factor VIIa/TF

Neutrophil Myeloperoxidase Is a Potent and Selective Inhibitor of Mast Cell Tryptase

Generation of potent coagulation protease inhibitors utilizing zinc-mediated chelation

Contribution of Multicentered Short Hydrogen Bond Arrays to Potency of Active Site-Directed Serine Protease Inhibitors

Highly potent non-peptidic inhibitors of the HCV NS3/NS4A serine protease

Neutral inhibitors of the serine protease factor Xa

Expression and Characterization of Recombinant Mast Cell Tryptase

A novel serine protease inhibition motif involving a multi-centered short hydrogen bonding network at the active site11Edited by D. Rees

Engineering inhibitors highly selective for the S1 sites of Ser190 trypsin-like serine protease drug targets

ChemInform Abstract: Neutral Inhibitors of the Serine Protease Factor Xa

Small Molecule Inhibitors of Plasma Kallikrein

ChemInform Abstract: Metal Mediated Protease Inhibition: Design and Synthesis of Inhibitors of the Human Cytomegalovirus (hCMV) Protease

Suchergebnisse filtern