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Stapled α−helical peptide drug development: A potent dual inhibitor of MDM2 and MDMX for p53-dependent cancer therapy

Proceedings of the National Academy of Sciences - PNAS, 2013-09, Vol.110 (36), p.E3445-E3454

2013

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Discovery of Sulanemadlin (ALRN-6924), the First Cell-Permeating, Stabilized α‑Helical Peptide in Clinical Development

Journal of medicinal chemistry, 2023-07, Vol.66 (14), p.9401-9417

2023

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Abstract LB-304: ATSP-9172, a novel Stapled Peptide inhibitor of HIF-dependent transcriptional activity with in vivo antitumor efficacy in a preclinical model of prostate cancer

Cancer research (Chicago, Ill.), 2013-04, Vol.73 (8_Supplement), p.LB-304-LB-304

2013

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Effects of chronic food restriction and treatments with leptin or ghrelin on different reproductive parameters of male rats

Peptides (New York, N.Y. : 1980), 2008-08, Vol.29 (8), p.1362-1368

2008

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Stapled [alpha]-helical peptide drug development: A potent dual inhibitor of MDM2 and MDMX for p53-dependent cancer therapy

Proceedings of the National Academy of Sciences - PNAS, 2013-09, Vol.110 (36), p.E3445

2013

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Stapled α-helical peptide drug development: A potent dual inhibitor of MDM2 and MDMX for p53-dependent cancer therapy

Proceedings of the National Academy of Sciences - PNAS, 2013-09, Vol.110 (36), p.14519-14519

2013

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Neutrophil rolling altered by inhibition of L-selectin shedding in vitro

Nature (London), 1996-04, Vol.380 (6576), p.720-723

1996

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Role of ghrelin in regulating rabbit ovarian function and the response to LH and IGF-I

Domestic animal endocrinology, 2009-04, Vol.36 (3), p.162-172

2009

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CHAPTER 9 - Macrocyclic α-Helical Peptide Drug Discovery

Macrocycles in drug discovery, 2015, p.339-366

2015

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Shedding of the Lymphocyte L-Selectin Adhesion Molecule Is Inhibited by a Hydroxamic Acid-based Protease Inhibitor

The Journal of biological chemistry, 1996-03, Vol.271 (12), p.7019-7024

1996

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Shedding of the lymphocyte L-selectin adhesion molecule is inhibited by a hydroxamic acid-based protease inhibitor. Identification with an L-selectin-alkaline phosphatase reporter

The Journal of biological chemistry, 1996-03, Vol.271 (12), p.7019-7024

1996

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An approach to cyclic peptide libraries: Reducing epimerization in medium sized rings during solid phase synthesis

Tetrahedron letters, 1996-01, Vol.37 (5), p.591-594

1996

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Effect of ghrelin on activities of some lysosomal hydrolases in rabbits

Neuro-endocrinology letters, 2005-08, Vol.26 (4), p.397-400

2005

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Structure-activity studies of dermorphin. The role of side chains of amino acid residues on the biological activity of dermorphin

Peptides (New York, N.Y. : 1980), 1984-01, Vol.5 (4), p.687-689

1984

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Prof. Arno F. Spatola's founding role at Peptides International

The journal of peptide research, 2004-02, Vol.63 (2), p.52-55

2004

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Macrocyclic α-Helical Peptide Drug Discovery

Macrocycles in Drug Discovery, 2014

Levin, Jeremy

2014

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Thiol-based inhibitors of mammalian collagenase. Substituted amide and peptide derivatives of the leucine analogue, 2-[(R,S)-mercaptomethyl]-4-methylpentanoic acid

The Journal of biological chemistry, 1990-03, Vol.265 (9), p.5199-5205

1990

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Amide bond surrogates: pseudopeptides and macrocycles

Tetrahedron, 1988, Vol.44 (3), p.821-833

1988

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Discoordinate expression of the yeast mitochondrial ribosomal protein MRP1

The Journal of biological chemistry, 1990-05, Vol.265 (13), p.7449-7454

1990

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Assessment of biological activity of synthetic fragments of transforming growth factor-alpha

Journal of cellular biochemistry, 1988-04, Vol.36 (4), p.341-352

1988

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Structure-activity studies of dermorphin. Synthesis and some pharmacological data of dermorphin and its 1-substituted analogs

Journal of medicinal chemistry, 1983-10, Vol.26 (10), p.1445-1447

1983

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Highly potent side chain-main chain cyclized dermorphin-deltorphin analogues: An integrated approach including synthesis, bioassays, NMR spectroscopy and molecular modelling

Journal of peptide science, 1995-05, Vol.1 (3), p.157-174

1995

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Dermorphin analogs: Resistance to in vitro enzymatic degradation is not always increased by additional D-amino acid substitutions

Biochemical and biophysical research communications, 1988-10, Vol.156 (1), p.125-130

1988

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ChemInform Abstract: Applications of CLEAR Resin for Solid Phase Organic Synthesis: Comparison with Polystyrene Based Resin

ChemInform, 2000-06, Vol.31 (23), p.no-no

2000

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Arginine-vasopressin analogs with high antidiuretic/vasopressor selectivity. Synthesis, biological activity and receptor binding affinity of arginine-vasopressin analogs with substitutions in positions 1, 2, 4, 7, and 8

Journal of medicinal chemistry, 1986-01, Vol.29 (1), p.96-99

1986

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Stapled α−helical peptide drug development: A potent dual inhibitor of MDM2 and MDMX for p53-dependent cancer therapy

Discovery of Sulanemadlin (ALRN-6924), the First Cell-Permeating, Stabilized α‑Helical Peptide in Clinical Development

Abstract LB-304: ATSP-9172, a novel Stapled Peptide inhibitor of HIF-dependent transcriptional activity with in vivo antitumor efficacy in a preclinical model of prostate cancer

Effects of chronic food restriction and treatments with leptin or ghrelin on different reproductive parameters of male rats

Stapled [alpha]-helical peptide drug development: A potent dual inhibitor of MDM2 and MDMX for p53-dependent cancer therapy

Stapled α-helical peptide drug development: A potent dual inhibitor of MDM2 and MDMX for p53-dependent cancer therapy

Neutrophil rolling altered by inhibition of L-selectin shedding in vitro

Role of ghrelin in regulating rabbit ovarian function and the response to LH and IGF-I

CHAPTER 9 - Macrocyclic α-Helical Peptide Drug Discovery

Shedding of the Lymphocyte L-Selectin Adhesion Molecule Is Inhibited by a Hydroxamic Acid-based Protease Inhibitor

Shedding of the lymphocyte L-selectin adhesion molecule is inhibited by a hydroxamic acid-based protease inhibitor. Identification with an L-selectin-alkaline phosphatase reporter

An approach to cyclic peptide libraries: Reducing epimerization in medium sized rings during solid phase synthesis

Effect of ghrelin on activities of some lysosomal hydrolases in rabbits

Structure-activity studies of dermorphin. The role of side chains of amino acid residues on the biological activity of dermorphin

Prof. Arno F. Spatola's founding role at Peptides International

Macrocyclic α-Helical Peptide Drug Discovery

Thiol-based inhibitors of mammalian collagenase. Substituted amide and peptide derivatives of the leucine analogue, 2-[(R,S)-mercaptomethyl]-4-methylpentanoic acid

Amide bond surrogates: pseudopeptides and macrocycles

Discoordinate expression of the yeast mitochondrial ribosomal protein MRP1

Assessment of biological activity of synthetic fragments of transforming growth factor-alpha

Structure-activity studies of dermorphin. Synthesis and some pharmacological data of dermorphin and its 1-substituted analogs

Highly potent side chain-main chain cyclized dermorphin-deltorphin analogues: An integrated approach including synthesis, bioassays, NMR spectroscopy and molecular modelling

Dermorphin analogs: Resistance to in vitro enzymatic degradation is not always increased by additional D-amino acid substitutions

ChemInform Abstract: Applications of CLEAR Resin for Solid Phase Organic Synthesis: Comparison with Polystyrene Based Resin

Arginine-vasopressin analogs with high antidiuretic/vasopressor selectivity. Synthesis, biological activity and receptor binding affinity of arginine-vasopressin analogs with substitutions in positions 1, 2, 4, 7, and 8

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