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Deprotection of N‑Boc Groups under Continuous-Flow High-Temperature Conditions

Journal of organic chemistry, 2019-04, Vol.84 (8), p.4846-4855

2019

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Application of Flow and Biocatalytic Transaminase Technology for the Synthesis of a 1‑Oxa-8-azaspiro[4.5]decan-3-amine

Organic process research & development, 2022-03, Vol.26 (3), p.616-623

2022

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Metabolism-Directed Design of Oxetane-Containing Arylsulfonamide Derivatives as γ-Secretase Inhibitors

Journal of medicinal chemistry, 2011-11, Vol.54 (22), p.7772-7783

2011

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Discovery and Optimization of a Novel Spiropyrrolidine Inhibitor of β-Secretase (BACE1) through Fragment-Based Drug Design

Journal of medicinal chemistry, 2012-11, Vol.55 (21), p.9069-9088

2012

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Metabolism of a G protein-coupled receptor modulator, including two major 1,2,4-oxadiazole ring-opened metabolites and a rearranged cysteine-piperazine adduct

Drug metabolism and disposition, 2012-06, Vol.40 (6), p.1151

2012

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Metabolic stability of 6,7-dialkoxy-4-(2-, 3- and 4-[ 18F]fluoroanilino)quinazolines, potential EGFR imaging probes

Bioorganic & medicinal chemistry, 2011-05, Vol.19 (9), p.2959-2965

2011

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Radiochemical synthesis and in vivo evaluation of [18F]AZ11637326: An agonist probe for the α7 nicotinic acetylcholine receptor

Nuclear medicine and biology, 2013-08, Vol.40 (6), p.731-739

2013

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Synthesis of three alpha 7 agonists in labeled form

Journal of labelled compounds & radiopharmaceuticals, 2014-05, Vol.57 (5), p.342-349

2014

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Syntheses of the tricyclic cores of clozapine, dibenzo[b,f][1,4]thiazepin-11(10H)-one, and dibenzo[b,f][1,4]oxazepin-11(10H)-one in C-14 labeled form by [14C]carbonylation

Journal of labelled compounds & radiopharmaceuticals, 2010-11, Vol.53 (13), p.787-792

2010

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Absence of direct effects on the dopamine D2 receptor by mGluR2/3-selective receptor agonists LY 354,740 and LY 379,268

Synapse (New York, N.Y.), 2011-01, Vol.65 (1), p.64-68

2011

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Synthesis of triphenylsilyl[14C2]acetylene for use in a Sonogashira reaction

Journal of labelled compounds & radiopharmaceuticals, 2011-01, Vol.54 (1), p.51-53

2011

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Synthesis of [13C5] and [carbonyl-14C]-5-chlorofuran-2-carboxylic acid

Journal of labelled compounds & radiopharmaceuticals, 2011-03, Vol.54 (3), p.123-125

2011

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Novel solid-phase preparation of 2,6,9-trisubstituted purines for combinatorial library generation

Tetrahedron letters, 2001-04, Vol.42 (15), p.2771-2773

2001

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Synthesis of a delta opioid agonist in [2H6], [2H4], [11C], and [14C] labeled forms

Journal of labelled compounds & radiopharmaceuticals, 2011-12, Vol.54 (14), p.847-854

2011

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Synthesis of the NK3 receptor antagonist AZD2624 in C-14-, H-3- and C-13-labeled forms

Journal of labelled compounds & radiopharmaceuticals, 2011-05, Vol.54 (5), p.239-246

2011

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Synthesis of 6-acrylamido-4-(2-[18F]fluoroanilino)quinazoline: a prospective irreversible EGFR binding probe

Journal of labelled compounds & radiopharmaceuticals, 2005-02, Vol.48 (2), p.109-115

2005

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Investigation of isotopic exchange reactions using N-heterocyclic iridium (I) complexes

Journal of labelled compounds & radiopharmaceuticals, 2007-04, Vol.50 (5-6), p.523-525

2007

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Mammalian topoisomerase II inhibitory activity of 1-cyclopropyl-6,8-difluoro-1,4-dihydro-7-(2,6-dimethyl-4-pyridinyl)-4-oxo-3-quinolinecarboxylic acid and related derivatives

Journal of medicinal chemistry, 1993-09, Vol.36 (19), p.2801-2809

1993

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Radiochemical synthesis and in vivo evaluation of [ super(18)F]AZ11637326: An agonist probe for the alpha 7 nicotinic acetylcholine receptor

Nuclear medicine and biology, 2013-08, Vol.40 (6), p.731-739

2013

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A New Strategy for Preparing Molecular Imaging and Therapy Agents Using Fluorine-Rich (Fluorous) Soluble Supports

Journal of the American Chemical Society, 2006-03, Vol.128 (11), p.3536-3537

2006

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In vitro assessment of metabolic drug–drug interaction potential of AZD2624, neurokinin-3 receptor antagonist, through cytochrome P 450 enzyme identification, inhibition, and induction studies

Xenobiotica, 2010-11, Vol.40 (11), p.721-729

2010

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D2 receptor occupancy in conscious rat brain is not significantly distinguished with [3H]-MNPA, [3H]-(+)-PHNO, and [3H]-raclopride

Synapse (New York, N.Y.), 2010-08, Vol.64 (8), p.624-633

2010

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Synthesis and Antibacterial Activity of Some Novel 1-Substituted 1,4-Dihydro-4-oxo-7-pyridinyl-3-quinolinecarboxylic Acids. Potent Antistaphylococcal Agents

Journal of medicinal chemistry, 1995-07, Vol.38 (14), p.2531-2540

1995

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Deprotection of N‑Boc Groups under Continuous-Flow High-Temperature Conditions

Application of the Bicyclo[1.1.1]pentane Motif as a Nonclassical Phenyl Ring Bioisostere in the Design of a Potent and Orally Active γ-Secretase Inhibitor

Application of Flow and Biocatalytic Transaminase Technology for the Synthesis of a 1‑Oxa-8-azaspiro[4.5]decan-3-amine

Discovery of Clinical Candidate PF-06648671: A Potent γ‑Secretase Modulator for the Treatment of Alzheimer’s Disease

Metabolism-Directed Design of Oxetane-Containing Arylsulfonamide Derivatives as γ-Secretase Inhibitors

Discovery and Optimization of a Novel Spiropyrrolidine Inhibitor of β-Secretase (BACE1) through Fragment-Based Drug Design

Metabolism of a G protein-coupled receptor modulator, including two major 1,2,4-oxadiazole ring-opened metabolites and a rearranged cysteine-piperazine adduct

Metabolic stability of 6,7-dialkoxy-4-(2-, 3- and 4-[ 18F]fluoroanilino)quinazolines, potential EGFR imaging probes

Radiochemical synthesis and in vivo evaluation of [18F]AZ11637326: An agonist probe for the α7 nicotinic acetylcholine receptor

Synthesis of three alpha 7 agonists in labeled form

Syntheses of the tricyclic cores of clozapine, dibenzo[b,f][1,4]thiazepin-11(10H)-one, and dibenzo[b,f][1,4]oxazepin-11(10H)-one in C-14 labeled form by [14C]carbonylation

Absence of direct effects on the dopamine D2 receptor by mGluR2/3-selective receptor agonists LY 354,740 and LY 379,268

Synthesis of triphenylsilyl[14C2]acetylene for use in a Sonogashira reaction

Synthesis of [13C5] and [carbonyl-14C]-5-chlorofuran-2-carboxylic acid

Novel solid-phase preparation of 2,6,9-trisubstituted purines for combinatorial library generation

Synthesis of a delta opioid agonist in [2H6], [2H4], [11C], and [14C] labeled forms

Synthesis of the NK3 receptor antagonist AZD2624 in C-14-, H-3- and C-13-labeled forms

Synthesis of 6-acrylamido-4-(2-[18F]fluoroanilino)quinazoline: a prospective irreversible EGFR binding probe

Investigation of isotopic exchange reactions using N-heterocyclic iridium (I) complexes

Mammalian topoisomerase II inhibitory activity of 1-cyclopropyl-6,8-difluoro-1,4-dihydro-7-(2,6-dimethyl-4-pyridinyl)-4-oxo-3-quinolinecarboxylic acid and related derivatives

Radiochemical synthesis and in vivo evaluation of [ super(18)F]AZ11637326: An agonist probe for the alpha 7 nicotinic acetylcholine receptor

A New Strategy for Preparing Molecular Imaging and Therapy Agents Using Fluorine-Rich (Fluorous) Soluble Supports

In vitro assessment of metabolic drug–drug interaction potential of AZD2624, neurokinin-3 receptor antagonist, through cytochrome P 450 enzyme identification, inhibition, and induction studies

D2 receptor occupancy in conscious rat brain is not significantly distinguished with [3H]-MNPA, [3H]-(+)-PHNO, and [3H]-raclopride

Synthesis and Antibacterial Activity of Some Novel 1-Substituted 1,4-Dihydro-4-oxo-7-pyridinyl-3-quinolinecarboxylic Acids. Potent Antistaphylococcal Agents

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