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Discovery of positive allosteric modulators and silent allosteric modulators of the μ-opioid receptor

Proceedings of the National Academy of Sciences - PNAS, 2013-06, Vol.110 (26), p.10830-10835

2013

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Endogenous opioids regulate moment-to-moment neuronal communication and excitability

Nature communications, 2017-03, Vol.8 (1), p.14611-14611, Article 14611

2017

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Strategies for the identification of allosteric modulators of G-protein-coupled receptors

Biochemical pharmacology, 2011-03, Vol.81 (6), p.691-702

2011

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Positive allosteric modulation of the mu-opioid receptor produces analgesia with reduced side effects

Proceedings of the National Academy of Sciences - PNAS, 2021-04, Vol.118 (16), p.1-10

2021

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Pharmacologic Evidence for a Putative Conserved Allosteric Site on Opioid Receptors

Molecular pharmacology, 2018-02, Vol.93 (2), p.157-167

2018

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Standard Curves Are Necessary to Determine Pharmacological Properties for Ligands in Functional Assays Using Competition Binding Technologies

Assay and drug development technologies, 2017-10, Vol.15 (7), p.320-329

2017

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Identification and biochemical analyses of selective CB2 agonists

European journal of pharmacology, 2019-07, Vol.854, p.1-8

2019

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Discovery, Synthesis, and Molecular Pharmacology of Selective Positive Allosteric Modulators of the δ‑Opioid Receptor

Journal of medicinal chemistry, 2015-05, Vol.58 (10), p.4220-4229

2015

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Ligand-Based Discovery of a New Scaffold for Allosteric Modulation of the μ‑Opioid Receptor

Journal of chemical information and modeling, 2015-09, Vol.55 (9), p.1836-1843

2015

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Discovery and SAR of aryl hydroxy pyrimidinones as potent small molecule agonists of the GPCR APJ

Bioorganic & medicinal chemistry letters, 2020-04, Vol.30 (7), p.126955-126955, Article 126955

2020

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High-Throughput Screening for Allosteric Modulators of GPCRs

Methods in molecular biology (Clifton, N.J.), 2015, Vol.1335, p.223

2015

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Identification of selective agonists and positive allosteric modulators for µ- and δ-opioid receptors from a single high-throughput screen

Journal of biomolecular screening, 2014-10, Vol.19 (9), p.1255-1265

2014

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Discovery of Selective Cannabinoid CB2 Receptor Agonists by High-Throughput Screening

SLAS discovery, 2018-04, Vol.23 (4), p.375-383

2018

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Identification and optimization of small molecule antagonists of vasoactive intestinal peptide receptor-1 (VIPR1)

Bioorganic & medicinal chemistry letters, 2012-03, Vol.22 (6), p.2287-2290

2012

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Development of a high-throughput calcium flux assay for identification of all ligand types including positive, negative, and silent allosteric modulators for G protein-coupled receptors

Assay and drug development technologies, 2012-10, Vol.10 (5), p.457-467

2012

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Solid Phase Synthesis of 1,5-Diarylpyrazole-4-carboxamides: Discovery of Antagonists of the CB-1 Receptor

ACS combinatorial science, 2012-03, Vol.14 (3), p.197-204

2012

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Discovery of pyrazine carboxamide CB1 antagonists: The introduction of a hydroxyl group improves the pharmaceutical properties and in vivo efficacy of the series

Bioorganic & medicinal chemistry letters, 2007-07, Vol.17 (14), p.3978-3982

2007

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Specific G protein activation and μ-opioid receptor internalization caused by morphine, DAMGO and endomorphin I

European journal of pharmacology, 1998-01, Vol.342 (1), p.123-126

1998

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Discovery of a Potent and Novel Motilin Agonist

Journal of medicinal chemistry, 2004-03, Vol.47 (7), p.1704-1708

2004

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Structure-Guided Discovery of Positive Allosteric Modulators of the Mu-Opioid Receptor

Biophysical journal, 2015-01, Vol.108 (2), p.414a-415a

2015

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Ligand-Based Discovery of a New Scaffold for Allosteric Modulation of the [mu]-Opioid Receptor

Journal of chemical information and modeling, 2015-09, Vol.55 (9), p.1836

2015

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Evidence for Classical Cholinergic Toxicity Associated with Selective Activation of M1 Muscarinic Receptors

The Journal of pharmacology and experimental therapeutics, 2016-02, Vol.356 (2), p.293-304

2016

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Discovery of positive allosteric modulators and silent allosteric modulators of the [mu]-opioid receptor

Proceedings of the National Academy of Sciences - PNAS, 2013-06, Vol.110 (26), p.10830

2013

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Identification and biochemical analyses of selective CB 2 agonists

European journal of pharmacology, 2019-07, Vol.854, p.1

2019

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Discovery of Selective Cannabinoid CB 2 Receptor Agonists by High-Throughput Screening

SLAS discovery, 2018-04, Vol.23 (4), p.375

2018

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Discovery of positive allosteric modulators and silent allosteric modulators of the μ-opioid receptor

Endogenous opioids regulate moment-to-moment neuronal communication and excitability

Strategies for the identification of allosteric modulators of G-protein-coupled receptors

Positive allosteric modulation of the mu-opioid receptor produces analgesia with reduced side effects

Pharmacologic Evidence for a Putative Conserved Allosteric Site on Opioid Receptors

Standard Curves Are Necessary to Determine Pharmacological Properties for Ligands in Functional Assays Using Competition Binding Technologies

Identification and biochemical analyses of selective CB2 agonists

Discovery, Synthesis, and Molecular Pharmacology of Selective Positive Allosteric Modulators of the δ‑Opioid Receptor

Ligand-Based Discovery of a New Scaffold for Allosteric Modulation of the μ‑Opioid Receptor

Discovery and SAR of aryl hydroxy pyrimidinones as potent small molecule agonists of the GPCR APJ

High-Throughput Screening for Allosteric Modulators of GPCRs

Identification of selective agonists and positive allosteric modulators for µ- and δ-opioid receptors from a single high-throughput screen

Discovery of Selective Cannabinoid CB2 Receptor Agonists by High-Throughput Screening

Identification and optimization of small molecule antagonists of vasoactive intestinal peptide receptor-1 (VIPR1)

Development of a high-throughput calcium flux assay for identification of all ligand types including positive, negative, and silent allosteric modulators for G protein-coupled receptors

Solid Phase Synthesis of 1,5-Diarylpyrazole-4-carboxamides: Discovery of Antagonists of the CB-1 Receptor

Discovery of pyrazine carboxamide CB1 antagonists: The introduction of a hydroxyl group improves the pharmaceutical properties and in vivo efficacy of the series

Specific G protein activation and μ-opioid receptor internalization caused by morphine, DAMGO and endomorphin I

Discovery of a Potent and Novel Motilin Agonist

Structure-Guided Discovery of Positive Allosteric Modulators of the Mu-Opioid Receptor

Ligand-Based Discovery of a New Scaffold for Allosteric Modulation of the [mu]-Opioid Receptor

Evidence for Classical Cholinergic Toxicity Associated with Selective Activation of M1 Muscarinic Receptors

Discovery of positive allosteric modulators and silent allosteric modulators of the [mu]-opioid receptor

Identification and biochemical analyses of selective CB 2 agonists

Discovery of Selective Cannabinoid CB 2 Receptor Agonists by High-Throughput Screening

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