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Discovery of a Highly Potent, Nonabsorbable Apical Sodium-Dependent Bile Acid Transporter Inhibitor (GSK2330672) for Treatment of Type 2 Diabetes

Journal of medicinal chemistry, 2013-06, Vol.56 (12), p.5094-5114

2013

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A pre-steady state and steady state kinetic analysis of the N-ribosyl hydrolase activity of hCD157

Archives of biochemistry and biophysics, 2014-12, Vol.564, p.156-163

2014

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Regiocontrolled Formation of a Novel Dioxadithiapentacene

Journal of organic chemistry, 1998-12, Vol.63 (26), p.10045-10047

1998

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The Naphthyridinone GSK364735 Is a Novel, Potent Human Immunodeficiency Virus Type 1 Integrase Inhibitor and Antiretroviral

Antimicrobial Agents and Chemotherapy, 2008-03, Vol.52 (3), p.901-908

2008

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Discovery, Synthesis, and Biological Evaluation of Thiazoloquin(az)olin(on)es as Potent CD38 Inhibitors

Journal of medicinal chemistry, 2015-04, Vol.58 (8), p.3548-3571

2015

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Synthesis and HIV-integrase strand transfer inhibition activity of 7-hydroxy[1,3]thiazolo[5,4- b]pyridin-5(4 H)-ones

Bioorganic & medicinal chemistry letters, 2006-11, Vol.16 (21), p.5668-5672

2006

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Discovery of 4‑Amino-8-quinoline Carboxamides as Novel, Submicromolar Inhibitors of NAD-Hydrolyzing Enzyme CD38

Journal of medicinal chemistry, 2015-09, Vol.58 (17), p.7021-7056

2015

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Thermal Synthesis of 3-Bromothieno[3,2-c]pyridin-4-(5H)-one: A Telescoped Procedure with Tributylamine

Journal of heterocyclic chemistry, 2015-01, Vol.52 (1), p.302-305

2015

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Enzymatic- and iridium-catalyzed asymmetric synthesis of a benzothiazepinylphosphonate bile acid transporter inhibitor

Journal of organic chemistry, 2013-12, Vol.78 (24), p.12726-12734

2013

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Facile Reductive Amination of Aldehydes with Electron-Deficient Anilines by Acyloxyborohydrides in TFA: Application to a Diazaindoline Scale-Up

Journal of organic chemistry, 2009-05, Vol.74 (9), p.3587-3590

2009

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Naphthyridinone (NTD) integrase inhibitors: N1 Protio and methyl combination substituent effects with C3 amide groups

Bioorganic & medicinal chemistry letters, 2013-01, Vol.23 (2), p.422-425

2013

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Discovery of 6,7-Dihydro‑5H‑pyrrolo[2,3‑a]pyrimidines as Orally Available G Protein-Coupled Receptor 119 Agonists

Journal of medicinal chemistry, 2012-12, Vol.55 (24), p.10972-10994

2012

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Naphthyridinone (NTD) integrase inhibitors 4. Investigating N1 acetamide substituent effects with C3 amide groups

Bioorganic & medicinal chemistry letters, 2014-07, Vol.24 (14), p.3104-3107

2014

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Development of Large-Scale Routes to Potent GPR119 Receptor Agonists

Organic process research & development, 2016-08, Vol.20 (8), p.1469-1475

2016

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Synthesis and Antiviral Activity of 7-Benzyl-4-hydroxy-1,5-naphthyridin-2(1H)-one HIV Integrase Inhibitors

Journal of medicinal chemistry, 2009-05, Vol.52 (9), p.2754-2761

2009

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Alkali Carbonate Effects on N-(2-Hydroxyethyl)urea Cyclization: Application to a 2-Imidazolidinone Scale-Up

Journal of heterocyclic chemistry, 2013-07, Vol.50 (4), p.863-867

2013

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A scalable Nenitzescu synthesis of 2-methyl-4-(trifluoromethyl)-1H-indole-5-carbonitrile

Journal of heterocyclic chemistry, 2011-05, Vol.48 (3), p.733-736

2011

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Synthesis of Ultra-Short-Acting Neuromuscular Blocker GW 0430: A Remarkably Stereo- and Regioselective Synthesis of Mixed Tetrahydroisoquinolinium Chlorofumarates

Organic letters, 1999-12, Vol.1 (12), p.1993-1996

1999

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Combining symmetry elements results in potent naphthyridinone (NTD) HIV-1 integrase inhibitors

Bioorganic & medicinal chemistry letters, 2011-11, Vol.21 (21), p.6461-6464

2011

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Bis- and Mixed-Tetrahydroisoquinolinium Chlorofumarates: New Ultra-Short-Acting Nondepolarizing Neuromuscular Blockers

Journal of medicinal chemistry, 1999-01, Vol.42 (2), p.206-209

1999

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Facile Reductive Amination of Aldehydes with Electron-Deficient Anilines by Acyloxyborohydrides in TFA: Application to a Diazaindoline Scale-Up

Journal of organic chemistry, 2009-11, Vol.74 (22), p.8908-8908

2009

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Preclinical pharmacology of GW280430A (AV430A) in the rhesus monkey and in the cat: A comparison with mivacurium

Anesthesiology (Philadelphia), 2004-04, Vol.100 (4), p.835-845

2004

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Hantzsch Synthesis of Pyrazolo[1‘,2‘:1,2]pyrazolo[3,4-b]pyridines: Partial Agonists of the Calcitonin Receptor

Journal of organic chemistry, 2005-06, Vol.70 (13), p.5331-5334

2005

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Alkynyl pyrimidines as dual EGFR/ErbB2 kinase inhibitors

Bioorganic & medicinal chemistry letters, 2006-05, Vol.16 (9), p.2419-2422

2006

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A Scaleable Synthesis of Methyl 3-Amino-5-(4-fluorobenzyl)-2-pyridinecarboxylate

Organic process research & development, 2007-09, Vol.11 (5), p.899-902

2007

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Discovery of a Highly Potent, Nonabsorbable Apical Sodium-Dependent Bile Acid Transporter Inhibitor (GSK2330672) for Treatment of Type 2 Diabetes

A pre-steady state and steady state kinetic analysis of the N-ribosyl hydrolase activity of hCD157

Regiocontrolled Formation of a Novel Dioxadithiapentacene

The Naphthyridinone GSK364735 Is a Novel, Potent Human Immunodeficiency Virus Type 1 Integrase Inhibitor and Antiretroviral

Discovery, Synthesis, and Biological Evaluation of Thiazoloquin(az)olin(on)es as Potent CD38 Inhibitors

Synthesis and HIV-integrase strand transfer inhibition activity of 7-hydroxy[1,3]thiazolo[5,4- b]pyridin-5(4 H)-ones

Discovery of 4‑Amino-8-quinoline Carboxamides as Novel, Submicromolar Inhibitors of NAD-Hydrolyzing Enzyme CD38

Thermal Synthesis of 3-Bromothieno[3,2-c]pyridin-4-(5H)-one: A Telescoped Procedure with Tributylamine

Enzymatic- and iridium-catalyzed asymmetric synthesis of a benzothiazepinylphosphonate bile acid transporter inhibitor

Facile Reductive Amination of Aldehydes with Electron-Deficient Anilines by Acyloxyborohydrides in TFA: Application to a Diazaindoline Scale-Up

Naphthyridinone (NTD) integrase inhibitors: N1 Protio and methyl combination substituent effects with C3 amide groups

Discovery of 6,7-Dihydro‑5H‑pyrrolo[2,3‑a]pyrimidines as Orally Available G Protein-Coupled Receptor 119 Agonists

Naphthyridinone (NTD) integrase inhibitors 4. Investigating N1 acetamide substituent effects with C3 amide groups

Development of Large-Scale Routes to Potent GPR119 Receptor Agonists

Synthesis and Antiviral Activity of 7-Benzyl-4-hydroxy-1,5-naphthyridin-2(1H)-one HIV Integrase Inhibitors

Alkali Carbonate Effects on N-(2-Hydroxyethyl)urea Cyclization: Application to a 2-Imidazolidinone Scale-Up

A scalable Nenitzescu synthesis of 2-methyl-4-(trifluoromethyl)-1H-indole-5-carbonitrile

Synthesis of Ultra-Short-Acting Neuromuscular Blocker GW 0430: A Remarkably Stereo- and Regioselective Synthesis of Mixed Tetrahydroisoquinolinium Chlorofumarates

Combining symmetry elements results in potent naphthyridinone (NTD) HIV-1 integrase inhibitors

Bis- and Mixed-Tetrahydroisoquinolinium Chlorofumarates: New Ultra-Short-Acting Nondepolarizing Neuromuscular Blockers

Facile Reductive Amination of Aldehydes with Electron-Deficient Anilines by Acyloxyborohydrides in TFA: Application to a Diazaindoline Scale-Up

Preclinical pharmacology of GW280430A (AV430A) in the rhesus monkey and in the cat: A comparison with mivacurium

Hantzsch Synthesis of Pyrazolo[1‘,2‘:1,2]pyrazolo[3,4-b]pyridines: Partial Agonists of the Calcitonin Receptor

Alkynyl pyrimidines as dual EGFR/ErbB2 kinase inhibitors

A Scaleable Synthesis of Methyl 3-Amino-5-(4-fluorobenzyl)-2-pyridinecarboxylate

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