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Structure activity relationship of selective GABA uptake inhibitors

Bioorganic & medicinal chemistry, 2015-05, Vol.23 (10), p.2480-2488

2015

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Selective mGAT2 (BGT-1) GABA Uptake Inhibitors: Design, Synthesis, and Pharmacological Characterization

Journal of medicinal chemistry, 2013-03, Vol.56 (5), p.2160-2164

2013

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Identification of the First Highly Subtype-Selective Inhibitor of Human GABA Transporter GAT3

ACS chemical neuroscience, 2015-09, Vol.6 (9), p.1591-1599

2015

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The Relationship between Agonist Potency and AMPA Receptor Kinetics

Biophysical journal, 2006-08, Vol.91 (4), p.1336-1346

2006

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GHB analogs confer neuroprotection through specific interaction with the CaMKIIα hub domain

Proceedings of the National Academy of Sciences - PNAS, 2021-08, Vol.118 (31), p.1

2021

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Chemoenzymatic synthesis and in situ application of S-adenosyl-L-methionine analogs

Organic & biomolecular chemistry, 2013-11, Vol.11 (43), p.7606-7610

2013

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Structure–Activity Relationship, Pharmacological Characterization, and Molecular Modeling of Noncompetitive Inhibitors of the Betaine/γ-Aminobutyric Acid Transporter 1 (BGT1)

Journal of medicinal chemistry, 2017-11, Vol.60 (21), p.8834-8846

2017

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A Tetrazolyl-Substituted Subtype-Selective AMPA Receptor Agonist

Journal of medicinal chemistry, 2007-05, Vol.50 (10), p.2408-2414

2007

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Discovery of a subtype selective inhibitor of the human betaine/GABA transporter 1 (BGT-1) with a non-competitive pharmacological profile

Biochemical pharmacology, 2013-08, Vol.86 (4), p.521-528

2013

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Probing the Pharmacophore of Ginkgolides as Glycine Receptor Antagonists

Journal of medicinal chemistry, 2007-04, Vol.50 (7), p.1610-1617

2007

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New Synthesis and Tritium Labeling of a Selective Ligand for Studying High-Affinity γ‑Hydroxybutyrate (GHB) Binding Sites

Journal of medicinal chemistry, 2013-10, Vol.56 (20), p.8201-8205

2013

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Pharmacological Identification of a Guanidine-Containing β-Alanine Analogue with Low Micromolar Potency and Selectivity for the Betaine/GABA Transporter 1 (BGT1)

Neurochemical research, 2014-10, Vol.39 (10), p.1988-1996

2014

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The labeling of unsaturated γ-hydroxybutyric acid by heavy isotopes of hydrogen: iridium complex-mediated H/D exchange by C─H bond activation vs reduction by boro-deuterides/tritides

Journal of labelled compounds & radiopharmaceuticals, 2016-10, Vol.59 (12), p.476-483

2016

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Radiosynthesis and Evaluation of [11C]3-Hydroxycyclopent-1-enecarboxylic Acid as Potential PET Ligand for the High-Affinity γ‑Hydroxybutyric Acid Binding Sites

ACS chemical neuroscience, 2017-01, Vol.8 (1), p.22-27

2017

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Biostructural and Pharmacological Studies of Bicyclic Analogues of the 3-Isoxazolol Glutamate Receptor Agonist Ibotenic Acid

Journal of medicinal chemistry, 2010-12, Vol.53 (23), p.8354-8361

2010

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Polyamine toxins: development of selective ligands for ionotropic receptors

Toxicon (Oxford), 2005-03, Vol.45 (3), p.249-254

2005

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Functional Characterization of Tet-AMPA [Tetrazolyl-2-amino-3-(3-hydroxy-5-methyl- 4-isoxazolyl)propionic Acid] Analogues at Ionotropic Glutamate Receptors GluR1−GluR4. The Molecular Basis for the Functional Selectivity Profile of 2-Bn-Tet-AMPA

Journal of medicinal chemistry, 2007-08, Vol.50 (17), p.4177-4185

2007

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Convergent Synthesis and Pharmacology of Substituted Tetrazolyl-2-amino-3-(3-hydroxy-5-methyl-4-isoxazolyl)propionic acid Analogues

Journal of medicinal chemistry, 2005-05, Vol.48 (9), p.3438-3442

2005

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A stereochemical anomaly: the cyclised (R)-AMPA analogue (R)-3-hydroxy-4,5,6,7-tetrahydroisoxazolo[5,4-c]pyridine-5-carboxylic acid [(R)-5-HPCA] resembles (S)-AMPA at glutamate receptors

Organic & biomolecular chemistry, 2004-01, Vol.2 (2), p.206-213

2004

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Analogues of homoibotenic acid show potent and selective activity following sensitisation by quisqualic acid

European journal of pharmacology, 2004-03, Vol.488 (1), p.101-109

2004

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Design and synthesis of labeled analogs of PhTX-56, a potent and selective AMPA receptor antagonist

Bioorganic & medicinal chemistry, 2005-09, Vol.13 (17), p.5104-5112

2005

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2-Amino-3-(3-hydroxy-1,2,5-thiadiazol-4-yl)propionic acid: Resolution, absolute stereochemistry and enantiopharmacology at glutamate receptors

Bioorganic & medicinal chemistry, 2002-07, Vol.10 (7), p.2259-2266

2002

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Chemoenzymatic synthesis and in situ application of S-adenosyl-l-methionine analogsElectronic supplementary information (ESI) available. See DOI: 10.1039/c3ob41702f

2013-10

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The labeling of unsaturated [gamma]-hydroxybutyric acid by heavy isotopes of hydrogen: iridium complex-mediated H/D exchange by C--H bond activation vs reduction by boro-deuterides/tritides

Journal of labelled compounds & radiopharmaceuticals, 2016-10, Vol.59 (12), p.476

2016

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Pharmacological Identification of a Guanidine-Containing [beta]-Alanine Analogue with Low Micromolar Potency and Selectivity for the Betaine/GABA Transporter 1 (BGT1)

Neurochemical research, 2014-10, Vol.39 (10), p.1988

2014

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Structure activity relationship of selective GABA uptake inhibitors

Selective mGAT2 (BGT-1) GABA Uptake Inhibitors: Design, Synthesis, and Pharmacological Characterization

Identification of the First Highly Subtype-Selective Inhibitor of Human GABA Transporter GAT3

The Relationship between Agonist Potency and AMPA Receptor Kinetics

GHB analogs confer neuroprotection through specific interaction with the CaMKIIα hub domain

Chemoenzymatic synthesis and in situ application of S-adenosyl-L-methionine analogs

Structure–Activity Relationship, Pharmacological Characterization, and Molecular Modeling of Noncompetitive Inhibitors of the Betaine/γ-Aminobutyric Acid Transporter 1 (BGT1)

A Tetrazolyl-Substituted Subtype-Selective AMPA Receptor Agonist

Discovery of a subtype selective inhibitor of the human betaine/GABA transporter 1 (BGT-1) with a non-competitive pharmacological profile

Probing the Pharmacophore of Ginkgolides as Glycine Receptor Antagonists

New Synthesis and Tritium Labeling of a Selective Ligand for Studying High-Affinity γ‑Hydroxybutyrate (GHB) Binding Sites

Pharmacological Identification of a Guanidine-Containing β-Alanine Analogue with Low Micromolar Potency and Selectivity for the Betaine/GABA Transporter 1 (BGT1)

The labeling of unsaturated γ-hydroxybutyric acid by heavy isotopes of hydrogen: iridium complex-mediated H/D exchange by C─H bond activation vs reduction by boro-deuterides/tritides

Radiosynthesis and Evaluation of [11C]3-Hydroxycyclopent-1-enecarboxylic Acid as Potential PET Ligand for the High-Affinity γ‑Hydroxybutyric Acid Binding Sites

Biostructural and Pharmacological Studies of Bicyclic Analogues of the 3-Isoxazolol Glutamate Receptor Agonist Ibotenic Acid

Polyamine toxins: development of selective ligands for ionotropic receptors

Functional Characterization of Tet-AMPA [Tetrazolyl-2-amino-3-(3-hydroxy-5-methyl- 4-isoxazolyl)propionic Acid] Analogues at Ionotropic Glutamate Receptors GluR1−GluR4. The Molecular Basis for the Functional Selectivity Profile of 2-Bn-Tet-AMPA

Convergent Synthesis and Pharmacology of Substituted Tetrazolyl-2-amino-3-(3-hydroxy-5-methyl-4-isoxazolyl)propionic acid Analogues

A stereochemical anomaly: the cyclised (R)-AMPA analogue (R)-3-hydroxy-4,5,6,7-tetrahydroisoxazolo[5,4-c]pyridine-5-carboxylic acid [(R)-5-HPCA] resembles (S)-AMPA at glutamate receptors

Analogues of homoibotenic acid show potent and selective activity following sensitisation by quisqualic acid

Design and synthesis of labeled analogs of PhTX-56, a potent and selective AMPA receptor antagonist

2-Amino-3-(3-hydroxy-1,2,5-thiadiazol-4-yl)propionic acid: Resolution, absolute stereochemistry and enantiopharmacology at glutamate receptors

Chemoenzymatic synthesis and in situ application of S-adenosyl-l-methionine analogsElectronic supplementary information (ESI) available. See DOI: 10.1039/c3ob41702f

The labeling of unsaturated [gamma]-hydroxybutyric acid by heavy isotopes of hydrogen: iridium complex-mediated H/D exchange by C--H bond activation vs reduction by boro-deuterides/tritides

Pharmacological Identification of a Guanidine-Containing [beta]-Alanine Analogue with Low Micromolar Potency and Selectivity for the Betaine/GABA Transporter 1 (BGT1)

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