UB Paderborn / Katalog / Suche / in CDI

Sortiert nach

Einfacher Volltextzugriff von (fast) überall

Installieren Sie die LibKey Nomad-Browsererweiterung und erhalten Sie von vielen Webseiten einfachen Zugriff auf lizenzierte Volltexte oder Open Access Publikationen. Mehr erfahren...

Structure activity relationship of selective GABA uptake inhibitors

Bioorganic & medicinal chemistry, 2015-05, Vol.23 (10), p.2480-2488

2015

Volltextzugriff (PDF)

Selective mGAT2 (BGT-1) GABA Uptake Inhibitors: Design, Synthesis, and Pharmacological Characterization

Journal of medicinal chemistry, 2013-03, Vol.56 (5), p.2160-2164

2013

Volltextzugriff (PDF)

Identification of the First Highly Subtype-Selective Inhibitor of Human GABA Transporter GAT3

ACS chemical neuroscience, 2015-09, Vol.6 (9), p.1591-1599

2015

Volltextzugriff (PDF)

The Relationship between Agonist Potency and AMPA Receptor Kinetics

Biophysical journal, 2006-08, Vol.91 (4), p.1336-1346

2006

Volltextzugriff (PDF)

GHB analogs confer neuroprotection through specific interaction with the CaMKIIα hub domain

Proceedings of the National Academy of Sciences - PNAS, 2021-08, Vol.118 (31), p.1-9

2021

Volltextzugriff (PDF)

Chemoenzymatic synthesis and in situ application of S-adenosyl-L-methionine analogs

Organic & biomolecular chemistry, 2013-11, Vol.11 (43), p.7606-7610

2013

Volltextzugriff (PDF)

Structure–Activity Relationship, Pharmacological Characterization, and Molecular Modeling of Noncompetitive Inhibitors of the Betaine/γ-Aminobutyric Acid Transporter 1 (BGT1)

Journal of medicinal chemistry, 2017-11, Vol.60 (21), p.8834-8846

2017

Volltextzugriff (PDF)

Discovery of a subtype selective inhibitor of the human betaine/GABA transporter 1 (BGT-1) with a non-competitive pharmacological profile

Biochemical pharmacology, 2013-08, Vol.86 (4), p.521-528

2013

Volltextzugriff (PDF)

Probing the Pharmacophore of Ginkgolides as Glycine Receptor Antagonists

Journal of medicinal chemistry, 2007-04, Vol.50 (7), p.1610-1617

2007

Volltextzugriff (PDF)

Pharmacological Identification of a Guanidine-Containing β-Alanine Analogue with Low Micromolar Potency and Selectivity for the Betaine/GABA Transporter 1 (BGT1)

Neurochemical research, 2014-10, Vol.39 (10), p.1988-1996

2014

Volltextzugriff (PDF)

The labeling of unsaturated γ-hydroxybutyric acid by heavy isotopes of hydrogen: iridium complex-mediated H/D exchange by C─H bond activation vs reduction by boro-deuterides/tritides

Journal of labelled compounds & radiopharmaceuticals, 2016-10, Vol.59 (12), p.476-483

2016

Volltextzugriff (PDF)

Radiosynthesis and Evaluation of [11C]3-Hydroxycyclopent-1-enecarboxylic Acid as Potential PET Ligand for the High-Affinity γ‑Hydroxybutyric Acid Binding Sites

ACS chemical neuroscience, 2017-01, Vol.8 (1), p.22-27

2017

Volltextzugriff (PDF)

Polyamine toxins: development of selective ligands for ionotropic receptors

Toxicon (Oxford), 2005-03, Vol.45 (3), p.249-254

2005

Volltextzugriff (PDF)

Design and synthesis of labeled analogs of PhTX-56, a potent and selective AMPA receptor antagonist

Bioorganic & medicinal chemistry, 2005-09, Vol.13 (17), p.5104-5112

2005

Volltextzugriff (PDF)

Chemoenzymatic synthesis and in situ application of S-adenosyl-l-methionine analogsElectronic supplementary information (ESI) available. See DOI: 10.1039/c3ob41702f

2013-10

Volltextzugriff (PDF)

Pharmacological Identification of a Guanidine-Containing [beta]-Alanine Analogue with Low Micromolar Potency and Selectivity for the Betaine/GABA Transporter 1 (BGT1)

Neurochemical research, 2014-10, Vol.39 (10), p.1988

2014

Volltextzugriff (PDF)

γ-Aminobutyric Acid and Glycine Neurotransmitter Transporters

Transporters As Drug Targets, 2017, p.69-106

2017

Volltextzugriff (PDF)

Design and synthesis of labeled analogs of PhTX-56, a potent and selective AMPA receptor antagonist: Chemistry & Biology of Natural Products, Tetrahedron Prize for Creativity in Organic Chemistry 2004 K. Nakanishi

Bioorganic & medicinal chemistry, 2005, Vol.13 (17), p.5104-5112

2005

Volltextzugriff (PDF)

Structural basis for 2-amino-3-(3-hydroxy-5-methyl-4-isoxazolyl)propionic acid (AMPA) receptor activation

Pure and applied chemistry, 2004-01, Vol.76 (5), p.921-930

2004

Volltextzugriff (PDF)

Resolution, configurational assignment, and enantiopharmacology of 2-amino-3-[3-hydroxy-5-(2-methyl-2H-tetrazol-5-yl)isoxazol-4-yl]propionic acid, a potent GluR3- and GluR4-preferring AMPA receptor agonist

Chirality (New York, N.Y.), 2000, Vol.12 (10), p.705-713

2000

Volltextzugriff (PDF)

Towards rational design of AMPA receptor ligands: An integrated medicinal, computational, biostructural and molecular pharmacological approach

Pharmacochemistry Library, 2002, Vol.32, p.1-12

2002

Volltextzugriff (PDF)

The intracellular lipid-binding domain of human Na+/H+ exchanger 1 forms a lipid-protein co-structure essential for activity

Communications biology, 2020-12, Vol.3 (1), p.731-731, Article 731

2020

Volltextzugriff (PDF)

3-Substituted pyrazoles and 4-substituted triazoles as inhibitors of human 15-lipoxygenase-1

Bioorganic & medicinal chemistry letters, 2015-08, Vol.25 (15), p.3024-3029

2015

Volltextzugriff (PDF)

Preparation of 7-Substituted Ginkgolide Derivatives: Potent Platelet Activating Factor (PAF) Receptor Antagonists

Journal of medicinal chemistry, 2003-02, Vol.46 (4), p.601-608

2003

Volltextzugriff (PDF)

1 – 24 von 24

Suche als RSS-Feed

Aktive Filter

SpracheFranzösisch

ThemaRats

Suchergebnisse filtern

Filter anzeigen

Nur zeigen

Geprüft (Peer-Review)
(23)
Mit Volltextzugriff
(23)

Publikationsform

Artikel
(22)
Buchkapitel
(2)

Sprache

Englisch
(24)

Erscheinungsjahr

n.n

Thema

Science & Technology
(20)
Life Sciences & Biomedicine
(17)
Pharmacology & Pharmacy
(14)
Chemistry, Medicinal
(12)
Animals
(11)
Chemistry
(9)
Humans
(9)
Structure-Activity Relationship
(8)
Physical Sciences
(7)
Biochemistry & Molecular Biology
(6)
Molecular Structure
(6)
Chemistry, Organic
(5)
Biological And Medical Sciences
(4)
Cho Cells
(4)
Ligands
(4)
Medical Sciences
(4)
Mice
(4)
Models, Molecular
(4)
Carrier Proteins - Antagonists & Inhibitors
(3)
Cricetinae
(3)

15 weitere anzeigen...

Weniger anzeigen...

Menü

Weitere Dienste

Einstellungen

Structure activity relationship of selective GABA uptake inhibitors

Selective mGAT2 (BGT-1) GABA Uptake Inhibitors: Design, Synthesis, and Pharmacological Characterization

Identification of the First Highly Subtype-Selective Inhibitor of Human GABA Transporter GAT3

The Relationship between Agonist Potency and AMPA Receptor Kinetics

GHB analogs confer neuroprotection through specific interaction with the CaMKIIα hub domain

Chemoenzymatic synthesis and in situ application of S-adenosyl-L-methionine analogs

Structure–Activity Relationship, Pharmacological Characterization, and Molecular Modeling of Noncompetitive Inhibitors of the Betaine/γ-Aminobutyric Acid Transporter 1 (BGT1)

Discovery of a subtype selective inhibitor of the human betaine/GABA transporter 1 (BGT-1) with a non-competitive pharmacological profile

Probing the Pharmacophore of Ginkgolides as Glycine Receptor Antagonists

Pharmacological Identification of a Guanidine-Containing β-Alanine Analogue with Low Micromolar Potency and Selectivity for the Betaine/GABA Transporter 1 (BGT1)

The labeling of unsaturated γ-hydroxybutyric acid by heavy isotopes of hydrogen: iridium complex-mediated H/D exchange by C─H bond activation vs reduction by boro-deuterides/tritides

Radiosynthesis and Evaluation of [11C]3-Hydroxycyclopent-1-enecarboxylic Acid as Potential PET Ligand for the High-Affinity γ‑Hydroxybutyric Acid Binding Sites

Polyamine toxins: development of selective ligands for ionotropic receptors

Design and synthesis of labeled analogs of PhTX-56, a potent and selective AMPA receptor antagonist

Chemoenzymatic synthesis and in situ application of S-adenosyl-l-methionine analogsElectronic supplementary information (ESI) available. See DOI: 10.1039/c3ob41702f

Pharmacological Identification of a Guanidine-Containing [beta]-Alanine Analogue with Low Micromolar Potency and Selectivity for the Betaine/GABA Transporter 1 (BGT1)

γ-Aminobutyric Acid and Glycine Neurotransmitter Transporters

Design and synthesis of labeled analogs of PhTX-56, a potent and selective AMPA receptor antagonist: Chemistry & Biology of Natural Products, Tetrahedron Prize for Creativity in Organic Chemistry 2004 K. Nakanishi

Structural basis for 2-amino-3-(3-hydroxy-5-methyl-4-isoxazolyl)propionic acid (AMPA) receptor activation

Resolution, configurational assignment, and enantiopharmacology of 2-amino-3-[3-hydroxy-5-(2-methyl-2H-tetrazol-5-yl)isoxazol-4-yl]propionic acid, a potent GluR3- and GluR4-preferring AMPA receptor agonist

Towards rational design of AMPA receptor ligands: An integrated medicinal, computational, biostructural and molecular pharmacological approach

The intracellular lipid-binding domain of human Na+/H+ exchanger 1 forms a lipid-protein co-structure essential for activity

3-Substituted pyrazoles and 4-substituted triazoles as inhibitors of human 15-lipoxygenase-1

Preparation of 7-Substituted Ginkgolide Derivatives: Potent Platelet Activating Factor (PAF) Receptor Antagonists

Aktive Filter

Suchergebnisse filtern