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Structure activity relationship of selective GABA uptake inhibitors

Bioorganic & medicinal chemistry, 2015-05, Vol.23 (10), p.2480-2488

2015

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Identification of the First Highly Subtype-Selective Inhibitor of Human GABA Transporter GAT3

ACS chemical neuroscience, 2015-09, Vol.6 (9), p.1591-1599

2015

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The Relationship between Agonist Potency and AMPA Receptor Kinetics

Biophysical journal, 2006-08, Vol.91 (4), p.1336-1346

2006

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GHB analogs confer neuroprotection through specific interaction with the CaMKIIα hub domain

Proceedings of the National Academy of Sciences - PNAS, 2021-08, Vol.118 (31), p.1

2021

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Chemoenzymatic synthesis and in situ application of S-adenosyl-L-methionine analogs

Organic & biomolecular chemistry, 2013-11, Vol.11 (43), p.7606-7610

2013

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Discovery of a subtype selective inhibitor of the human betaine/GABA transporter 1 (BGT-1) with a non-competitive pharmacological profile

Biochemical pharmacology, 2013-08, Vol.86 (4), p.521-528

2013

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Pharmacological Identification of a Guanidine-Containing β-Alanine Analogue with Low Micromolar Potency and Selectivity for the Betaine/GABA Transporter 1 (BGT1)

Neurochemical research, 2014-10, Vol.39 (10), p.1988-1996

2014

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The labeling of unsaturated γ-hydroxybutyric acid by heavy isotopes of hydrogen: iridium complex-mediated H/D exchange by C─H bond activation vs reduction by boro-deuterides/tritides

Journal of labelled compounds & radiopharmaceuticals, 2016-10, Vol.59 (12), p.476-483

2016

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Radiosynthesis and Evaluation of [11C]3-Hydroxycyclopent-1-enecarboxylic Acid as Potential PET Ligand for the High-Affinity γ‑Hydroxybutyric Acid Binding Sites

ACS chemical neuroscience, 2017-01, Vol.8 (1), p.22-27

2017

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Polyamine toxins: development of selective ligands for ionotropic receptors

Toxicon (Oxford), 2005-03, Vol.45 (3), p.249-254

2005

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A stereochemical anomaly: the cyclised (R)-AMPA analogue (R)-3-hydroxy-4,5,6,7-tetrahydroisoxazolo[5,4-c]pyridine-5-carboxylic acid [(R)-5-HPCA] resembles (S)-AMPA at glutamate receptors

Organic & biomolecular chemistry, 2004-01, Vol.2 (2), p.206-213

2004

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Analogues of homoibotenic acid show potent and selective activity following sensitisation by quisqualic acid

European journal of pharmacology, 2004-03, Vol.488 (1), p.101-109

2004

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Design and synthesis of labeled analogs of PhTX-56, a potent and selective AMPA receptor antagonist

Bioorganic & medicinal chemistry, 2005-09, Vol.13 (17), p.5104-5112

2005

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2-Amino-3-(3-hydroxy-1,2,5-thiadiazol-4-yl)propionic acid: Resolution, absolute stereochemistry and enantiopharmacology at glutamate receptors

Bioorganic & medicinal chemistry, 2002-07, Vol.10 (7), p.2259-2266

2002

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Chemoenzymatic synthesis and in situ application of S-adenosyl-l-methionine analogsElectronic supplementary information (ESI) available. See DOI: 10.1039/c3ob41702f

2013-10

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The labeling of unsaturated [gamma]-hydroxybutyric acid by heavy isotopes of hydrogen: iridium complex-mediated H/D exchange by C--H bond activation vs reduction by boro-deuterides/tritides

Journal of labelled compounds & radiopharmaceuticals, 2016-10, Vol.59 (12), p.476

2016

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Pharmacological Identification of a Guanidine-Containing [beta]-Alanine Analogue with Low Micromolar Potency and Selectivity for the Betaine/GABA Transporter 1 (BGT1)

Neurochemical research, 2014-10, Vol.39 (10), p.1988

2014

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γ-Aminobutyric Acid and Glycine Neurotransmitter Transporters

Transporters As Drug Targets, 2017, p.69-106

2017

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Design and synthesis of labeled analogs of PhTX-56, a potent and selective AMPA receptor antagonist: Chemistry & Biology of Natural Products, Tetrahedron Prize for Creativity in Organic Chemistry 2004 K. Nakanishi

Bioorganic & medicinal chemistry, 2005, Vol.13 (17), p.5104-5112

2005

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Structural basis for 2-amino-3-(3-hydroxy-5-methyl-4-isoxazolyl)propionic acid (AMPA) receptor activation

Pure and applied chemistry, 2004-01, Vol.76 (5), p.921-930

2004

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Resolution, configurational assignment, and enantiopharmacology of 2-amino-3-[3-hydroxy-5-(2-methyl-2H-tetrazol-5-yl)isoxazol-4-yl]propionic acid, a potent GluR3- and GluR4-preferring AMPA receptor agonist

Chirality (New York, N.Y.), 2000, Vol.12 (10), p.705-713

2000

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Resolution, configurational assignment, and enantiopharmacology at glutamate receptors of 2-amino-3-(3-carboxy-5-methyl-4-isoxazolyl)propionic acid (ACPA) and demethyl-ACPA

Chirality (New York, N.Y.), 2001, Vol.13 (9), p.523-532

2001

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Towards rational design of AMPA receptor ligands: An integrated medicinal, computational, biostructural and molecular pharmacological approach

Pharmacochemistry Library, 2002, Vol.32, p.1-12

2002

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The intracellular lipid-binding domain of human Na + /H + exchanger 1 forms a lipid-protein co-structure essential for activity

Communications biology, 2020-12, Vol.3 (1), p.731-731, Article 731

2020

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3-Substituted pyrazoles and 4-substituted triazoles as inhibitors of human 15-lipoxygenase-1

Bioorganic & medicinal chemistry letters, 2015-08, Vol.25 (15), p.3024-3029

2015

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Structure activity relationship of selective GABA uptake inhibitors

Identification of the First Highly Subtype-Selective Inhibitor of Human GABA Transporter GAT3

The Relationship between Agonist Potency and AMPA Receptor Kinetics

GHB analogs confer neuroprotection through specific interaction with the CaMKIIα hub domain

Chemoenzymatic synthesis and in situ application of S-adenosyl-L-methionine analogs

Discovery of a subtype selective inhibitor of the human betaine/GABA transporter 1 (BGT-1) with a non-competitive pharmacological profile

Pharmacological Identification of a Guanidine-Containing β-Alanine Analogue with Low Micromolar Potency and Selectivity for the Betaine/GABA Transporter 1 (BGT1)

The labeling of unsaturated γ-hydroxybutyric acid by heavy isotopes of hydrogen: iridium complex-mediated H/D exchange by C─H bond activation vs reduction by boro-deuterides/tritides

Radiosynthesis and Evaluation of [11C]3-Hydroxycyclopent-1-enecarboxylic Acid as Potential PET Ligand for the High-Affinity γ‑Hydroxybutyric Acid Binding Sites

Polyamine toxins: development of selective ligands for ionotropic receptors

A stereochemical anomaly: the cyclised (R)-AMPA analogue (R)-3-hydroxy-4,5,6,7-tetrahydroisoxazolo[5,4-c]pyridine-5-carboxylic acid [(R)-5-HPCA] resembles (S)-AMPA at glutamate receptors

Analogues of homoibotenic acid show potent and selective activity following sensitisation by quisqualic acid

Design and synthesis of labeled analogs of PhTX-56, a potent and selective AMPA receptor antagonist

2-Amino-3-(3-hydroxy-1,2,5-thiadiazol-4-yl)propionic acid: Resolution, absolute stereochemistry and enantiopharmacology at glutamate receptors

Chemoenzymatic synthesis and in situ application of S-adenosyl-l-methionine analogsElectronic supplementary information (ESI) available. See DOI: 10.1039/c3ob41702f

The labeling of unsaturated [gamma]-hydroxybutyric acid by heavy isotopes of hydrogen: iridium complex-mediated H/D exchange by C--H bond activation vs reduction by boro-deuterides/tritides

Pharmacological Identification of a Guanidine-Containing [beta]-Alanine Analogue with Low Micromolar Potency and Selectivity for the Betaine/GABA Transporter 1 (BGT1)

γ-Aminobutyric Acid and Glycine Neurotransmitter Transporters

Design and synthesis of labeled analogs of PhTX-56, a potent and selective AMPA receptor antagonist: Chemistry & Biology of Natural Products, Tetrahedron Prize for Creativity in Organic Chemistry 2004 K. Nakanishi

Structural basis for 2-amino-3-(3-hydroxy-5-methyl-4-isoxazolyl)propionic acid (AMPA) receptor activation

Resolution, configurational assignment, and enantiopharmacology of 2-amino-3-[3-hydroxy-5-(2-methyl-2H-tetrazol-5-yl)isoxazol-4-yl]propionic acid, a potent GluR3- and GluR4-preferring AMPA receptor agonist

Resolution, configurational assignment, and enantiopharmacology at glutamate receptors of 2-amino-3-(3-carboxy-5-methyl-4-isoxazolyl)propionic acid (ACPA) and demethyl-ACPA

Towards rational design of AMPA receptor ligands: An integrated medicinal, computational, biostructural and molecular pharmacological approach

The intracellular lipid-binding domain of human Na + /H + exchanger 1 forms a lipid-protein co-structure essential for activity

3-Substituted pyrazoles and 4-substituted triazoles as inhibitors of human 15-lipoxygenase-1

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