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PET and SPECT imaging of the opioid system: receptors, radioligands and avenues for drug discovery and development

Current pharmaceutical design, 2007, Vol.13 (1), p.33-49

Lever, John R

2007

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Sigma-1 receptor ligand PD144418 and sigma-2 receptor ligand YUN-252 attenuate the stimulant effects of methamphetamine in mice

Psychopharmacology, 2019-11, Vol.236 (11), p.3147-3158

2019

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The sigma receptor ligand N-phenylpropyl-N′-(4-methoxyphenethyl)3piperazine (YZ-067) enhances the cocaine conditioned-rewarding properties while inhibiting the development of sensitization of cocaine in mice

Psychopharmacology, 2020-03, Vol.237 (3), p.723-734

2020

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Effect of structural modification in the amine portion of substituted aminobutyl-benzamides as ligands for binding σ1 and σ2 receptors

Bioorganic & medicinal chemistry, 2011-03, Vol.19 (6), p.1852-1859

2011

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Design, synthesis and evaluation of 111 In labeled DOTA-conjugated tetrapeptides having high affinity and selectivity for mu opioid receptors

Nuclear medicine and biology, 2019-03, Vol.70, p.53

2019

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Synthesis and opioid receptor binding of indium (III) and [111In]-labeled macrocyclic conjugates of diprenorphine: novel ligands designed for imaging studies of peripheral opioid receptors

Tetrahedron, 2016-10, Vol.72 (40), p.6127-6135

2016

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A selective sigma-2 receptor ligand antagonizes cocaine-induced hyperlocomotion in mice

Synapse (New York, N.Y.), 2014-02, Vol.68 (2), p.73-84

2014

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Computational and Biochemical Docking of the Irreversible Cocaine Analog RTI 82 Directly Demonstrates Ligand Positioning in the Dopamine Transporter Central Substrate-binding Site

The Journal of biological chemistry, 2014-10, Vol.289 (43), p.29712-29727

2014

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Inhibitor mechanisms in the S1 binding site of the dopamine transporter defined by multi-site molecular tethering of photoactive cocaine analogs

Biochemical pharmacology, 2017-10, Vol.142, p.204-215

2017

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Effects of N-phenylpropyl-N′-substituted piperazine sigma receptor ligands on cocaine-induced hyperactivity in mice

Pharmacology, biochemistry and behavior, 2013-09, Vol.110, p.201-207

2013

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Synthesis, radioiodination and in vitro and in vivo sigma receptor studies of N -1-allyl- N ´-4-phenethylpiperazine analogs

Nuclear medicine and biology, 2012-04, Vol.39 (3), p.401-414

2012

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Synthesis and in vitro evaluation of tetrahydroisoquinolinyl benzamides as ligands for σ receptors

Bioorganic & medicinal chemistry letters, 2007-05, Vol.17 (9), p.2594-2597

2007

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(±)-2-(N-tert-Butylamino)-3′-[125I]-iodo-4′-azidopropiophenone: A dopamine transporter and nicotinic acetylcholine receptor photoaffinity ligand based on bupropion (Wellbutrin, Zyban)

Bioorganic & medicinal chemistry letters, 2012-01, Vol.22 (1), p.523-526

2012

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Azido-iodo-N-benzyl derivatives of threo-methylphenidate (Ritalin, Concerta): Rational design, synthesis, pharmacological evaluation, and dopamine transporter photoaffinity labeling

Bioorganic & medicinal chemistry, 2011-01, Vol.19 (1), p.504-512

2011

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A novel photoaffinity ligand for the dopamine transporter based on pyrovalerone

Bioorganic & medicinal chemistry, 2009-06, Vol.17 (11), p.3770-3774

2009

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Differential Binding of Tropane-Based Photoaffinity Ligands on the Dopamine Transporter

The Journal of neuroscience, 1999-01, Vol.19 (2), p.630-636

1999

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N-Phenylpropyl-N′-(3-methoxyphenethyl)piperazine (YZ-185) Attenuates the Conditioned-Rewarding Properties of Cocaine in Mice

ISRN pharmacology, 2013, Vol.2013, p.546314-7

2013

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Dual Incorporation of Photoaffinity Ligands on Dopamine Transporters Implicates Proximity of Labeled Domains

Molecular pharmacology, 2001-05, Vol.59 (5), p.1157-1164

2001

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Sigma1 and sigma2 receptor binding affinity and selectivity of SA4503 and fluoroethyl SA4503

Synapse (New York, N.Y.), 2006-05, Vol.59 (6), p.350

2006

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Synthesis and structure-activity relationships of N-(3-phenylpropyl)-N'-benzylpiperazines: Potent ligands for sigma1 and sigma2 receptors

Bioorganic & medicinal chemistry, 2008-01, Vol.16 (2), p.755-761

2008

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Labeling of dopamine transporter transmembrane domain 1 with the tropane ligand N-[4-(4-azido-3-[125I]iodophenyl)butyl]-2beta-carbomethoxy-3beta-(4-chlorophenyl)tropane implicates proximity of cocaine and substrate active sites

Molecular pharmacology, 2008-04, Vol.73 (4), p.1141

2008

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N-substituted phenyltropanes as in vivo binding ligands for rapid imaging studies of the dopamine transporter

Synapse (New York, N.Y.), 1997-04, Vol.25 (4), p.345-349

1997

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Synthesis of radioiodinated naltrindole analogues: Ligands for studies of delta opioid receptors

Nuclear medicine and biology, 1995-07, Vol.22 (5), p.599-606

1995

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Synthesis and in vivo studies of a selective ligand for the dopamine transporter: 3β-(4-[ 125I]iodophenyl) tropan-2β-carboxylic acid isopropyl ester ([ 125I]RTM-21)

Nuclear medicine and biology, 1996-04, Vol.23 (3), p.277-284

1996

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Autoradiographic and SPECT imaging of cerebral opioid receptors with an iodine-123 labeled analogue of diprenorphine

Synapse (New York, N.Y.), 1998-06, Vol.29 (2), p.172-182

1998

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PET and SPECT imaging of the opioid system: receptors, radioligands and avenues for drug discovery and development

Sigma-1 receptor ligand PD144418 and sigma-2 receptor ligand YUN-252 attenuate the stimulant effects of methamphetamine in mice

The sigma receptor ligand N-phenylpropyl-N′-(4-methoxyphenethyl)3piperazine (YZ-067) enhances the cocaine conditioned-rewarding properties while inhibiting the development of sensitization of cocaine in mice

Effect of structural modification in the amine portion of substituted aminobutyl-benzamides as ligands for binding σ1 and σ2 receptors

Design, synthesis and evaluation of 111 In labeled DOTA-conjugated tetrapeptides having high affinity and selectivity for mu opioid receptors

Synthesis and opioid receptor binding of indium (III) and [111In]-labeled macrocyclic conjugates of diprenorphine: novel ligands designed for imaging studies of peripheral opioid receptors

A selective sigma-2 receptor ligand antagonizes cocaine-induced hyperlocomotion in mice

Computational and Biochemical Docking of the Irreversible Cocaine Analog RTI 82 Directly Demonstrates Ligand Positioning in the Dopamine Transporter Central Substrate-binding Site

Inhibitor mechanisms in the S1 binding site of the dopamine transporter defined by multi-site molecular tethering of photoactive cocaine analogs

Effects of N-phenylpropyl-N′-substituted piperazine sigma receptor ligands on cocaine-induced hyperactivity in mice

Synthesis, radioiodination and in vitro and in vivo sigma receptor studies of N -1-allyl- N ´-4-phenethylpiperazine analogs

Synthesis and in vitro evaluation of tetrahydroisoquinolinyl benzamides as ligands for σ receptors

(±)-2-(N-tert-Butylamino)-3′-[125I]-iodo-4′-azidopropiophenone: A dopamine transporter and nicotinic acetylcholine receptor photoaffinity ligand based on bupropion (Wellbutrin, Zyban)

Azido-iodo-N-benzyl derivatives of threo-methylphenidate (Ritalin, Concerta): Rational design, synthesis, pharmacological evaluation, and dopamine transporter photoaffinity labeling

A novel photoaffinity ligand for the dopamine transporter based on pyrovalerone

Differential Binding of Tropane-Based Photoaffinity Ligands on the Dopamine Transporter

N-Phenylpropyl-N′-(3-methoxyphenethyl)piperazine (YZ-185) Attenuates the Conditioned-Rewarding Properties of Cocaine in Mice

Dual Incorporation of Photoaffinity Ligands on Dopamine Transporters Implicates Proximity of Labeled Domains

Sigma1 and sigma2 receptor binding affinity and selectivity of SA4503 and fluoroethyl SA4503

Synthesis and structure-activity relationships of N-(3-phenylpropyl)-N'-benzylpiperazines: Potent ligands for sigma1 and sigma2 receptors

Labeling of dopamine transporter transmembrane domain 1 with the tropane ligand N-[4-(4-azido-3-[125I]iodophenyl)butyl]-2beta-carbomethoxy-3beta-(4-chlorophenyl)tropane implicates proximity of cocaine and substrate active sites

N-substituted phenyltropanes as in vivo binding ligands for rapid imaging studies of the dopamine transporter

Synthesis of radioiodinated naltrindole analogues: Ligands for studies of delta opioid receptors

Synthesis and in vivo studies of a selective ligand for the dopamine transporter: 3β-(4-[ 125I]iodophenyl) tropan-2β-carboxylic acid isopropyl ester ([ 125I]RTM-21)

Autoradiographic and SPECT imaging of cerebral opioid receptors with an iodine-123 labeled analogue of diprenorphine

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