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PET and SPECT imaging of the opioid system: receptors, radioligands and avenues for drug discovery and development

Current pharmaceutical design, 2007, Vol.13 (1), p.33-49

Lever, John R

2007

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Allosteric modulation of sigma receptors by BH3 mimetics ABT-737, ABT-263 (Navitoclax) and ABT-199 (Venetoclax)

Pharmacological research, 2019-04, Vol.142, p.87-100

2019

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Tactics for preclinical validation of receptor-binding radiotracers

Nuclear medicine and biology, 2017-01, Vol.44, p.4-30

2017

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Sigma-1 receptor ligand PD144418 and sigma-2 receptor ligand YUN-252 attenuate the stimulant effects of methamphetamine in mice

Psychopharmacology, 2019-11, Vol.236 (11), p.3147-3158

2019

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The sigma receptor ligand N-phenylpropyl-N′-(4-methoxyphenethyl)3piperazine (YZ-067) enhances the cocaine conditioned-rewarding properties while inhibiting the development of sensitization of cocaine in mice

Psychopharmacology, 2020-03, Vol.237 (3), p.723-734

2020

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Characterization of pulmonary sigma receptors by radioligand binding

European journal of pharmacology, 2015-09, Vol.762, p.118-126

2015

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N-phenylpropyl-N'-substituted piperazines occupy sigma receptors and alter methamphetamine-induced hyperactivity in mice

Pharmacology, biochemistry and behavior, 2016-11, Vol.150-151, p.198-206

2016

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Phorbol ester induced trafficking-independent regulation and enhanced phosphorylation of the dopamine transporter associated with membrane rafts and cholesterol

Journal of neurochemistry, 2008-06, Vol.105 (5), p.1683-1699

2008

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Relationship between cerebral sigma-1 receptor occupancy and attenuation of cocaine's motor stimulatory effects in mice by PD144418

The Journal of pharmacology and experimental therapeutics, 2014-10, Vol.351 (1), p.153-163

2014

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Design, synthesis and evaluation of 111 In labeled DOTA-conjugated tetrapeptides having high affinity and selectivity for mu opioid receptors

Nuclear medicine and biology, 2019-03, Vol.70, p.53

2019

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The sigma receptor agonist SA4503 both attenuates and enhances the effects of methamphetamine

Drug and alcohol dependence, 2011-07, Vol.116 (1), p.203-210

2011

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Identification of the benztropine analog [125I]GA II 34 binding site on the human dopamine transporter

Neurochemistry international, 2019-02, Vol.123, p.34-45

2019

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Ether modifications to 1-[2-(3,4-dimethoxyphenyl)ethyl]-4-(3-phenylpropyl)piperazine (SA4503): Effects on binding affinity and selectivity for sigma receptors and monoamine transporters

Bioorganic & medicinal chemistry, 2015-01, Vol.23 (1), p.222-230

2015

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A selective sigma-2 receptor ligand antagonizes cocaine-induced hyperlocomotion in mice

Synapse (New York, N.Y.), 2014-02, Vol.68 (2), p.73-84

2014

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SA 4503 attenuates cocaine-induced hyperactivity and enhances methamphetamine substitution for a cocaine discriminative stimulus

Pharmacology, biochemistry and behavior, 2011-02, Vol.97 (4), p.676-682

2011

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Rapid hyperspectral fluorescence lifetime imaging

Microscopy research and technique, 2007-05, Vol.70 (5), p.481-484

2007

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Computational and Biochemical Docking of the Irreversible Cocaine Analog RTI 82 Directly Demonstrates Ligand Positioning in the Dopamine Transporter Central Substrate-binding Site

The Journal of biological chemistry, 2014-10, Vol.289 (43), p.29712-29727

2014

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Inhibitor mechanisms in the S1 binding site of the dopamine transporter defined by multi-site molecular tethering of photoactive cocaine analogs

Biochemical pharmacology, 2017-10, Vol.142, p.204-215

2017

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Effects of N-phenylpropyl-N′-substituted piperazine sigma receptor ligands on cocaine-induced hyperactivity in mice

Pharmacology, biochemistry and behavior, 2013-09, Vol.110, p.201-207

2013

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Synthesis, radioiodination and in vitro and in vivo sigma receptor studies of N -1-allyl- N ´-4-phenethylpiperazine analogs

Nuclear medicine and biology, 2012-04, Vol.39 (3), p.401-414

2012

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Bupropion Binds to Two Sites in the Torpedo Nicotinic Acetylcholine Receptor Transmembrane Domain: A Photoaffinity Labeling Study with the Bupropion Analogue [125I]-SADU-3-72

Biochemistry (Easton), 2012-03, Vol.51 (12), p.2425-2435

2012

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Synthesis and in vitro evaluation of tetrahydroisoquinolinyl benzamides as ligands for σ receptors

Bioorganic & medicinal chemistry letters, 2007-05, Vol.17 (9), p.2594-2597

2007

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Labeling of Dopamine Transporter Transmembrane Domain 1 with the Tropane Ligand N -[4-(4-Azido-3-[ 125 I]iodophenyl)butyl]-2β-carbomethoxy-3β-(4-chlorophenyl)tropane Implicates Proximity of Cocaine and Substrate Active Sites

Molecular pharmacology, 2008-04, Vol.73 (4), p.1141-1150

2008

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Localization of Cocaine Analog [125I]RTI 82 Irreversible Binding to Transmembrane Domain 6 of the Dopamine Transporter

The Journal of biological chemistry, 2007-03, Vol.282 (12), p.8915-8925

2007

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Azido-iodo-N-benzyl derivatives of threo-methylphenidate (Ritalin, Concerta): Rational design, synthesis, pharmacological evaluation, and dopamine transporter photoaffinity labeling

Bioorganic & medicinal chemistry, 2011-01, Vol.19 (1), p.504-512

2011

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PET and SPECT imaging of the opioid system: receptors, radioligands and avenues for drug discovery and development

Allosteric modulation of sigma receptors by BH3 mimetics ABT-737, ABT-263 (Navitoclax) and ABT-199 (Venetoclax)

Tactics for preclinical validation of receptor-binding radiotracers

Sigma-1 receptor ligand PD144418 and sigma-2 receptor ligand YUN-252 attenuate the stimulant effects of methamphetamine in mice

The sigma receptor ligand N-phenylpropyl-N′-(4-methoxyphenethyl)3piperazine (YZ-067) enhances the cocaine conditioned-rewarding properties while inhibiting the development of sensitization of cocaine in mice

Characterization of pulmonary sigma receptors by radioligand binding

N-phenylpropyl-N'-substituted piperazines occupy sigma receptors and alter methamphetamine-induced hyperactivity in mice

Phorbol ester induced trafficking-independent regulation and enhanced phosphorylation of the dopamine transporter associated with membrane rafts and cholesterol

Relationship between cerebral sigma-1 receptor occupancy and attenuation of cocaine's motor stimulatory effects in mice by PD144418

Design, synthesis and evaluation of 111 In labeled DOTA-conjugated tetrapeptides having high affinity and selectivity for mu opioid receptors

The sigma receptor agonist SA4503 both attenuates and enhances the effects of methamphetamine

Identification of the benztropine analog [125I]GA II 34 binding site on the human dopamine transporter

Ether modifications to 1-[2-(3,4-dimethoxyphenyl)ethyl]-4-(3-phenylpropyl)piperazine (SA4503): Effects on binding affinity and selectivity for sigma receptors and monoamine transporters

A selective sigma-2 receptor ligand antagonizes cocaine-induced hyperlocomotion in mice

SA 4503 attenuates cocaine-induced hyperactivity and enhances methamphetamine substitution for a cocaine discriminative stimulus

Rapid hyperspectral fluorescence lifetime imaging

Computational and Biochemical Docking of the Irreversible Cocaine Analog RTI 82 Directly Demonstrates Ligand Positioning in the Dopamine Transporter Central Substrate-binding Site

Inhibitor mechanisms in the S1 binding site of the dopamine transporter defined by multi-site molecular tethering of photoactive cocaine analogs

Effects of N-phenylpropyl-N′-substituted piperazine sigma receptor ligands on cocaine-induced hyperactivity in mice

Synthesis, radioiodination and in vitro and in vivo sigma receptor studies of N -1-allyl- N ´-4-phenethylpiperazine analogs

Bupropion Binds to Two Sites in the Torpedo Nicotinic Acetylcholine Receptor Transmembrane Domain: A Photoaffinity Labeling Study with the Bupropion Analogue [125I]-SADU-3-72

Synthesis and in vitro evaluation of tetrahydroisoquinolinyl benzamides as ligands for σ receptors

Labeling of Dopamine Transporter Transmembrane Domain 1 with the Tropane Ligand N -[4-(4-Azido-3-[ 125 I]iodophenyl)butyl]-2β-carbomethoxy-3β-(4-chlorophenyl)tropane Implicates Proximity of Cocaine and Substrate Active Sites

Localization of Cocaine Analog [125I]RTI 82 Irreversible Binding to Transmembrane Domain 6 of the Dopamine Transporter

Azido-iodo-N-benzyl derivatives of threo-methylphenidate (Ritalin, Concerta): Rational design, synthesis, pharmacological evaluation, and dopamine transporter photoaffinity labeling

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