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Discovery of new thymol-3,4-disubstituted thiazole hybrids as dual COX-2/5-LOX inhibitors with in vivo proof

Journal of enzyme inhibition and medicinal chemistry, 2024-12, Vol.39 (1), p.2309171-2309171

2024

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The small conductance Ca 2+ -activated K + channel activator GW542573X impairs hippocampal memory in C57BL/6J mice

Neuropharmacology, 2024-07, Vol.252, p.109960

2024

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Effects of thiamethoxam on physiological and molecular responses to potato plant (Solanum tuberosum), green peach aphid (Myzus persicae), and parasitoid (Aphidius gifuensis)

Pest management science, 2024-06, Vol.80 (6), p.3000-3009

2024

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Design, synthesis and molecular docking of novel D-ring substituted steroidal 4,5-dihydropyrazole thiazole derivatives that act as iNOS/COX-2 inhibitors with potent anti-inflammatory activity against LPS-induced RAW264.7 macrophage cells

The Journal of steroid biochemistry and molecular biology, 2024-06, Vol.240, p.106478-106478, Article 106478

2024

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Simultaneous quantification of 2-aminothiazoline-4-carboxylic acid and 2-aminothiazoline-4-oxoaminoethanoic acid utilizing chemical derivatization followed by liquid chromatography–tandem mass spectrometry

Journal of pharmaceutical and biomedical analysis, 2024-05, Vol.242, p.116027-116027, Article 116027

2024

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Discovery and Mechanistic Studies of Dual-Target Hits for Carbonic Anhydrase IX and VEGFR‑2 as Potential Agents for Solid Tumors: X‑ray, In Vitro, In Vivo, and In Silico Investigations of Coumarin-Based Thiazoles

Journal of medicinal chemistry, 2024-05, Vol.67 (9), p.7406-7430

2024

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Structure-Based Design of Novel Thiazolone[3,2- a ]pyrimidine Derivatives as Potent RNase H Inhibitors for HIV Therapy

Molecules (Basel, Switzerland), 2024-05, Vol.29 (9), p.2120

2024

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Activation and inhibition of the sweet taste receptor TAS1R2-TAS1R3 differentially affect glucose tolerance in humans

PloS one, 2024-05, Vol.19 (5), p.e0298239-e0298239

2024

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Reply to: Letter to the Editor from Malik et al.: Acute kidney injury following subcutaneous meloxicam administration

Journal of veterinary pharmacology and therapeutics, 2024-05, Vol.47 (3), p.237-238

2024

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Lessons learned from a multi-data source research collaboration: The mirabegron post-authorization safety study program

Pharmacoepidemiology and drug safety, 2024-05, Vol.33 (5), p.e5799-e5799

2024

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Synthesis, biological evaluation and molecular docking study of pyrimidine linked thiazolidinedione derivatives as potential antimicrobial and antitubercular agents

Bioorganic & medicinal chemistry letters, 2024-05, Vol.103, p.129707-129707, Article 129707

2024

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Rifampicin synergizes the toxicity of insecticides against the green peach aphid, Myzus persicae

Ecotoxicology and environmental safety, 2024-05, Vol.276, p.116291-116291, Article 116291

2024

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Sulfonyl thioureas with a benzo[d]thiazole ring as dual acetylcholinesterase/butyrylcholinesterase and human monoamine oxidase A and B inhibitors: An in vitro and in silico study

Archiv der Pharmazie (Weinheim), 2024-05, Vol.357 (5), p.e2300557-n/a

2024

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Thiazolyl-isatin derivatives: Synthesis, in silico studies, in vitro biological profile against breast cancer cells, mRNA expression, P-gp modulation, and interactions of Akt2 and VIM proteins

Chemico-biological interactions, 2024-05, Vol.394, p.110954-110954, Article 110954

2024

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Allosteric Activation of α7 Nicotinic Acetylcholine Receptors by Novel 2‑Arylamino-thiazole-5-carboxylic Acid Amide Derivatives for the Improvement of Cognitive Deficits in Mice

Journal of medicinal chemistry, 2024-04, Vol.67 (8), p.6344-6364

2024

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Did the prolonged residual efficacy of clothianidin products lead to a greater reduction in vector populations and subsequent malaria transmission compared to the shorter residual efficacy of pirimiphos-methyl?

Malaria journal, 2024-04, Vol.23 (1), p.119-119

2024

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Tapcin, an In Vivo Active Dual Topoisomerase I/II Inhibitor Discovered by Synthetic Bioinformatic Natural Product (Syn‐BNP)‐Coupled Metagenomics

Angewandte Chemie (International ed.), 2024-04, Vol.63 (17), p.e202317187-n/a

International ed. in English, 2024

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C16, a PKR inhibitor, suppresses cell proliferation by regulating the cell cycle via p21 in colorectal cancer

Scientific reports, 2024-04, Vol.14 (1), p.9029-9029

2024

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In Silico Analysis of the Ga 3+ /Fe 3+ Competition for Binding the Iron-Scavenging Siderophores of P. aeruginosa -Implementation of Three Gallium-Based Complexes in the "Trojan Horse" Antibacterial Strategy

Biomolecules (Basel, Switzerland), 2024-04, Vol.14 (4)

2024

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Lusutrombopag as a Repurposing Drug in Combination with Aminoglycosides against Vancomycin-Resistant Enterococcus

ACS infectious diseases, 2024-04, Vol.10 (4), p.1327-1338

2024

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5‑Aminothiazoles Reveal a New Ligand-Binding Site on Prolyl Oligopeptidase Which is Important for Modulation of Its Protein–Protein Interaction-Derived Functions

Journal of medicinal chemistry, 2024-04, Vol.67 (7), p.5421-5436

2024

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Laboratory evaluation of the contact irritancy of a clothianidin solo formulation vs. clothianidin-deltamethrin mixture formulations for indoor residual spraying against pyrethroid-resistant Anopheles gambiae sensu lato

Parasites & vectors, 2024-04, Vol.17 (1), p.183-183

2024

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Synthesis and anti-liver fibrosis activity of imidazole and thiazole compounds containing amino acids

European journal of medicinal chemistry, 2024-04, Vol.269, p.116311-116311, Article 116311

2024

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Novel Thiazole Derivatives Containing Imidazole and Furan Scaffold: Design, Synthesis, Molecular Docking, Antibacterial, and Antioxidant Evaluation

Molecules (Basel, Switzerland), 2024-04, Vol.29 (7), p.1491

Agili, Fatimah

2024

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Time Course of the Interaction Between Oral Short-Term Ritonavir Therapy with Three Factor Xa Inhibitors and the Activity of CYP2D6, CYP2C19, and CYP3A4 in Healthy Volunteers

Clinical pharmacokinetics, 2024-04, Vol.63 (4), p.469-481

2024

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Discovery of new thymol-3,4-disubstituted thiazole hybrids as dual COX-2/5-LOX inhibitors with in vivo proof

The small conductance Ca 2+ -activated K + channel activator GW542573X impairs hippocampal memory in C57BL/6J mice

Effects of thiamethoxam on physiological and molecular responses to potato plant (Solanum tuberosum), green peach aphid (Myzus persicae), and parasitoid (Aphidius gifuensis)

Design, synthesis and molecular docking of novel D-ring substituted steroidal 4,5-dihydropyrazole thiazole derivatives that act as iNOS/COX-2 inhibitors with potent anti-inflammatory activity against LPS-induced RAW264.7 macrophage cells

Simultaneous quantification of 2-aminothiazoline-4-carboxylic acid and 2-aminothiazoline-4-oxoaminoethanoic acid utilizing chemical derivatization followed by liquid chromatography–tandem mass spectrometry

Discovery and Mechanistic Studies of Dual-Target Hits for Carbonic Anhydrase IX and VEGFR‑2 as Potential Agents for Solid Tumors: X‑ray, In Vitro, In Vivo, and In Silico Investigations of Coumarin-Based Thiazoles

Structure-Based Design of Novel Thiazolone[3,2- a ]pyrimidine Derivatives as Potent RNase H Inhibitors for HIV Therapy

Activation and inhibition of the sweet taste receptor TAS1R2-TAS1R3 differentially affect glucose tolerance in humans

Reply to: Letter to the Editor from Malik et al.: Acute kidney injury following subcutaneous meloxicam administration

Lessons learned from a multi-data source research collaboration: The mirabegron post-authorization safety study program

Synthesis, biological evaluation and molecular docking study of pyrimidine linked thiazolidinedione derivatives as potential antimicrobial and antitubercular agents

Rifampicin synergizes the toxicity of insecticides against the green peach aphid, Myzus persicae

Sulfonyl thioureas with a benzo[d]thiazole ring as dual acetylcholinesterase/butyrylcholinesterase and human monoamine oxidase A and B inhibitors: An in vitro and in silico study

Thiazolyl-isatin derivatives: Synthesis, in silico studies, in vitro biological profile against breast cancer cells, mRNA expression, P-gp modulation, and interactions of Akt2 and VIM proteins

Allosteric Activation of α7 Nicotinic Acetylcholine Receptors by Novel 2‑Arylamino-thiazole-5-carboxylic Acid Amide Derivatives for the Improvement of Cognitive Deficits in Mice

Did the prolonged residual efficacy of clothianidin products lead to a greater reduction in vector populations and subsequent malaria transmission compared to the shorter residual efficacy of pirimiphos-methyl?

Tapcin, an In Vivo Active Dual Topoisomerase I/II Inhibitor Discovered by Synthetic Bioinformatic Natural Product (Syn‐BNP)‐Coupled Metagenomics

C16, a PKR inhibitor, suppresses cell proliferation by regulating the cell cycle via p21 in colorectal cancer

In Silico Analysis of the Ga 3+ /Fe 3+ Competition for Binding the Iron-Scavenging Siderophores of P. aeruginosa -Implementation of Three Gallium-Based Complexes in the "Trojan Horse" Antibacterial Strategy

Lusutrombopag as a Repurposing Drug in Combination with Aminoglycosides against Vancomycin-Resistant Enterococcus

5‑Aminothiazoles Reveal a New Ligand-Binding Site on Prolyl Oligopeptidase Which is Important for Modulation of Its Protein–Protein Interaction-Derived Functions

Laboratory evaluation of the contact irritancy of a clothianidin solo formulation vs. clothianidin-deltamethrin mixture formulations for indoor residual spraying against pyrethroid-resistant Anopheles gambiae sensu lato

Synthesis and anti-liver fibrosis activity of imidazole and thiazole compounds containing amino acids

Novel Thiazole Derivatives Containing Imidazole and Furan Scaffold: Design, Synthesis, Molecular Docking, Antibacterial, and Antioxidant Evaluation

Time Course of the Interaction Between Oral Short-Term Ritonavir Therapy with Three Factor Xa Inhibitors and the Activity of CYP2D6, CYP2C19, and CYP3A4 in Healthy Volunteers

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