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Integrase Strand Transfer Inhibitor Start or Switch Impacts Learning in Women With HIV

Journal of acquired immune deficiency syndromes (1999), 2021-04, Vol.86 (5), p.593

2021

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Deactivation of Hepatic Stellate Cells During Liver Fibrosis Resolution in Mice

Gastroenterology (New York, N.Y. 1943), 2012-10, Vol.143 (4), p.1073-1083.e22

2012

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In Vitro Antiretroviral Properties of S/GSK1349572, a Next-Generation HIV Integrase Inhibitor

Antimicrobial Agents and Chemotherapy, 2011-02, Vol.55 (2), p.813-821

2011

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Low level of HIV-1C integrase strand transfer inhibitor resistance mutations among recently diagnosed ART-naive Ethiopians

Scientific reports, 2023-04, Vol.13 (1), p.6546-6546, Article 6546

2023

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Mutations Associated with Failure of Raltegravir Treatment Affect Integrase Sensitivity to the Inhibitor In Vitro

Antimicrobial Agents and Chemotherapy, 2008-04, Vol.52 (4), p.1351-1358

2008

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New insights into the interaction between pyrrolyl diketoacids and HIV-1 integrase active site and comparison with RNase H

Antiviral research, 2016-10, Vol.134, p.236-243

2016

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Antiviral characteristics of GSK1265744, an HIV integrase inhibitor dosed orally or by long-acting injection

Antimicrobial agents and chemotherapy, 2015-01, Vol.59 (1), p.397-406

2015

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Structure-function analyses unravel distinct effects of allosteric inhibitors of HIV-1 integrase on viral maturation and integration

The Journal of biological chemistry, 2018-04, Vol.293 (16), p.6172-6186

2018

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Avoidance of Transient Cardiomyopathy in Cardiomyocyte-Targeted Tamoxifen-Induced MerCreMer Gene Deletion Models

Circulation research, 2009-07, Vol.105 (1), p.12-15

2009

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Carbamoyl Pyridone HIV‑1 Integrase Inhibitors. 2. Bi- and Tricyclic Derivatives Result in Superior Antiviral and Pharmacokinetic Profiles

Journal of medicinal chemistry, 2013-02, Vol.56 (3), p.1124-1135

2013

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The design of 8-hydroxyquinoline tetracyclic lactams as HIV-1 integrase strand transfer inhibitors

European journal of medicinal chemistry, 2016-07, Vol.117, p.99-112

2016

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Investigations on the 4-Quinolone-3-carboxylic Acid Motif. 1. Synthesis and Structure−Activity Relationship of a Class of Human Immunodeficiency Virus type 1 Integrase Inhibitors

Journal of medicinal chemistry, 2008-08, Vol.51 (16), p.5125-5129

2008

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Discovery of 2‑Pyridinone Aminals: A Prodrug Strategy to Advance a Second Generation of HIV‑1 Integrase Strand Transfer Inhibitors

Journal of medicinal chemistry, 2015-10, Vol.58 (20), p.8154-8165

2015

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Ivermectin as a Broad-Spectrum Host-Directed Antiviral: The Real Deal?

Cells (Basel, Switzerland), 2020-09, Vol.9 (9), p.2100

2020

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Structural basis for the inhibition of HTLV-1 integration inferred from cryo-EM deltaretroviral intasome structures

Nature communications, 2021-08, Vol.12 (1), p.4996-4996, Article 4996

2021

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Indole-based allosteric inhibitors of HIV-1 integrase

Bioorganic & medicinal chemistry letters, 2016-10, Vol.26 (19), p.4748-4752

2016

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Rapamycin Prevents Early Onset of Tumorigenesis in an Oral-Specific K-ras and p53 Two-Hit Carcinogenesis Model

Cancer research (Chicago, Ill.), 2009-05, Vol.69 (10), p.4159-4166

2009

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Total Synthesis of Integrastatin B Enabled by a Benzofuran Oxidative Dearomatization Cascade

Organic letters, 2016-03, Vol.18 (6), p.1458-1461

2016

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Quinolone Carboxylic Acids as a Novel Monoketo Acid Class of Human Immunodeficiency Virus Type 1 Integrase Inhibitors

Journal of medicinal chemistry, 2009-08, Vol.52 (15), p.4869-4882

2009

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Generation of CD4CreER(T²) transgenic mice to study development of peripheral CD4-T-cells

Genesis (New York, N.Y. : 2000), 2012-12, Vol.50 (12), p.908-913

2012

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Asymmetric Synthesis of a Potent HIV‑1 Integrase Inhibitor

Journal of organic chemistry, 2016-11, Vol.81 (21), p.10256-10265

2016

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Susceptibility to HIV-1 integrase strand transfer inhibitors (INSTIs) in highly treatment-experienced patients who failed an INSTI-based regimen

International journal of antimicrobial agents, 2020-07, Vol.56 (1), p.106027-106027, Article 106027

2020

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Development of HIV-1 integrase inhibitors: recent molecular modeling perspectives

Drug discovery today, 2015-11, Vol.20 (11), p.1337-1348

2015

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Allosteric Inhibitor Development Targeting HIV-1 Integrase

ChemMedChem, 2011-02, Vol.6 (2), p.228-241

2011

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Metabolism and disposition in humans of raltegravir (MK-0518), an anti-AIDS drug targeting the human immunodeficiency virus 1 integrase enzyme

Drug metabolism and disposition, 2007-09, Vol.35 (9), p.1657

2007

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Integrase Strand Transfer Inhibitor Start or Switch Impacts Learning in Women With HIV

Deactivation of Hepatic Stellate Cells During Liver Fibrosis Resolution in Mice

In Vitro Antiretroviral Properties of S/GSK1349572, a Next-Generation HIV Integrase Inhibitor

Low level of HIV-1C integrase strand transfer inhibitor resistance mutations among recently diagnosed ART-naive Ethiopians

Mutations Associated with Failure of Raltegravir Treatment Affect Integrase Sensitivity to the Inhibitor In Vitro

New insights into the interaction between pyrrolyl diketoacids and HIV-1 integrase active site and comparison with RNase H

Antiviral characteristics of GSK1265744, an HIV integrase inhibitor dosed orally or by long-acting injection

Structure-function analyses unravel distinct effects of allosteric inhibitors of HIV-1 integrase on viral maturation and integration

Avoidance of Transient Cardiomyopathy in Cardiomyocyte-Targeted Tamoxifen-Induced MerCreMer Gene Deletion Models

Carbamoyl Pyridone HIV‑1 Integrase Inhibitors. 2. Bi- and Tricyclic Derivatives Result in Superior Antiviral and Pharmacokinetic Profiles

The design of 8-hydroxyquinoline tetracyclic lactams as HIV-1 integrase strand transfer inhibitors

Investigations on the 4-Quinolone-3-carboxylic Acid Motif. 1. Synthesis and Structure−Activity Relationship of a Class of Human Immunodeficiency Virus type 1 Integrase Inhibitors

Discovery of 2‑Pyridinone Aminals: A Prodrug Strategy to Advance a Second Generation of HIV‑1 Integrase Strand Transfer Inhibitors

Ivermectin as a Broad-Spectrum Host-Directed Antiviral: The Real Deal?

Structural basis for the inhibition of HTLV-1 integration inferred from cryo-EM deltaretroviral intasome structures

Indole-based allosteric inhibitors of HIV-1 integrase

Rapamycin Prevents Early Onset of Tumorigenesis in an Oral-Specific K-ras and p53 Two-Hit Carcinogenesis Model

Total Synthesis of Integrastatin B Enabled by a Benzofuran Oxidative Dearomatization Cascade

Quinolone Carboxylic Acids as a Novel Monoketo Acid Class of Human Immunodeficiency Virus Type 1 Integrase Inhibitors

Generation of CD4CreER(T²) transgenic mice to study development of peripheral CD4-T-cells

Asymmetric Synthesis of a Potent HIV‑1 Integrase Inhibitor

Susceptibility to HIV-1 integrase strand transfer inhibitors (INSTIs) in highly treatment-experienced patients who failed an INSTI-based regimen

Development of HIV-1 integrase inhibitors: recent molecular modeling perspectives

Allosteric Inhibitor Development Targeting HIV-1 Integrase

Metabolism and disposition in humans of raltegravir (MK-0518), an anti-AIDS drug targeting the human immunodeficiency virus 1 integrase enzyme

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