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KLIFS: a structural kinase-ligand interaction database

Nucleic acids research, 2016-01, Vol.44 (D1), p.D365-D371

2016

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The Landscape of Atypical and Eukaryotic Protein Kinases

Trends in pharmacological sciences (Regular ed.), 2019-11, Vol.40 (11), p.818-832

2019

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Fragment library screening reveals remarkable similarities between the G protein-coupled receptor histamine H4 and the ion channel serotonin 5-HT3A

Bioorganic & medicinal chemistry letters, 2011-09, Vol.21 (18), p.5460-5464

2011

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Exploring the Effect of Cyclization of Histamine H1 Receptor Antagonists on Ligand Binding Kinetics

ACS omega, 2021-05, Vol.6 (19), p.12755-12768

2021

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A Photoswitchable Agonist for the Histamine H3 Receptor, a Prototypic Family A G‐Protein‐Coupled Receptor

Angewandte Chemie International Edition, 2019-03, Vol.58 (14), p.4531-4535

International ed. in English, 2019

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Photoswitching the Efficacy of a Small‐Molecule Ligand for a Peptidergic GPCR: from Antagonism to Agonism

Angewandte Chemie International Edition, 2018-09, Vol.57 (36), p.11608-11612

International ed. in English, 2018

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Identification of novel α7 nicotinic receptor ligands by in silico screening against the crystal structure of a chimeric α7 receptor ligand binding domain

Bioorganic & medicinal chemistry, 2012-10, Vol.20 (19), p.5992-6002

2012

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The histamine H3 receptor: from gene cloning to H3 receptor drugs

Nature reviews. Drug discovery, 2005-02, Vol.4 (2), p.107-120

2005

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Phenyldihydropyrazolones as Novel Lead Compounds Against Trypanosoma cruzi

ACS omega, 2019-04, Vol.4 (4), p.6585-6596

2019

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En route to new blockbuster anti-histamines: surveying the offspring of the expanding histamine receptor family

Trends in pharmacological sciences (Regular ed.), 2011-04, Vol.32 (4), p.250-257

2011

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Molecular Determinants of Selective Agonist and Antagonist Binding to the Histamine H4 Receptor

Current topics in medicinal chemistry, 2011-03, Vol.11 (6), p.661-679

2011

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An efficient and information-rich biochemical method design for fragment library screening on ion channels

BioTechniques, 2010-11, Vol.49 (5), p.822-829

2010

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3D-e-Chem-VM: Structural Cheminformatics Research Infrastructure in a Freely Available Virtual Machine

Journal of chemical information and modeling, 2017-02, Vol.57 (2), p.115-121

2017

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Antiinflammatory and antinociceptive effects of the selective histamine H4-receptor antagonists JNJ7777120 and VUF6002 in a rat model of carrageenan-induced acute inflammation

European journal of pharmacology, 2007-06, Vol.563 (1-3), p.240-244

2007

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Targeted LC-MS derivatization for aldehydes and carboxylic acids with a new derivatization agent 4-APEBA

Analytical and bioanalytical chemistry, 2010-05, Vol.397 (2), p.665-675

2010

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Ligand efficiency as a guide in fragment hit selection and optimization

Drug discovery today. Technologies, 2010, Vol.7 (3), p.e157-e162

2010

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Synthesis, modeling and functional activity of substituted styrene-amides as small-molecule CXCR7 agonists

European journal of medicinal chemistry, 2012-05, Vol.51, p.184-192

2012

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Major advances in the development of histamine H4 receptor ligands

Drug discovery today, 2009-08, Vol.14 (15-16), p.745-753

2009

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Acetylcholine binding protein (AChBP) as template for hierarchical in silico screening procedures to identify structurally novel ligands for the nicotinic receptors

Bioorganic & medicinal chemistry, 2011-10, Vol.19 (20), p.6107-6119

2011

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Multiplexed experimental strategies for fragment library screening against challenging drug targets using SPR biosensors

SLAS discovery, 2024-01, Vol.29 (1), p.40-51

2024

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Combinatorial Consensus Scoring for Ligand-Based Virtual Fragment Screening: A Comparative Case Study for Serotonin 5‑HT3A, Histamine H1, and Histamine H4 Receptors

Journal of chemical information and modeling, 2015-05

2015

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Online Fluorescence Enhancement Assay for the Acetylcholine Binding Protein with Parallel Mass Spectrometric Identification

Journal of medicinal chemistry, 2010-06, Vol.53 (12), p.4720-4730

2010

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CXCR3 antagonists: Quaternary ammonium salts equipped with biphenyl- and polycycloaliphatic-anchors

Bioorganic & medicinal chemistry, 2011-06, Vol.19 (11), p.3384-3393

2011

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A novel series of histamine H4 receptor antagonists based on the pyrido[3,2-d]pyrimidine scaffold: Comparison of hERG binding and target residence time with PF-3893787

Bioorganic & medicinal chemistry letters, 2013-05, Vol.23 (9), p.2663-2670

2013

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KLIFS: an overhaul after the first 5 years of supporting kinase research

Nucleic acids research, 2021-01, Vol.49 (D1), p.D562-D569

2021

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KLIFS: a structural kinase-ligand interaction database

The Landscape of Atypical and Eukaryotic Protein Kinases

Fragment library screening reveals remarkable similarities between the G protein-coupled receptor histamine H4 and the ion channel serotonin 5-HT3A

Exploring the Effect of Cyclization of Histamine H1 Receptor Antagonists on Ligand Binding Kinetics

A Photoswitchable Agonist for the Histamine H3 Receptor, a Prototypic Family A G‐Protein‐Coupled Receptor

Photoswitching the Efficacy of a Small‐Molecule Ligand for a Peptidergic GPCR: from Antagonism to Agonism

Identification of novel α7 nicotinic receptor ligands by in silico screening against the crystal structure of a chimeric α7 receptor ligand binding domain

The histamine H3 receptor: from gene cloning to H3 receptor drugs

Phenyldihydropyrazolones as Novel Lead Compounds Against Trypanosoma cruzi

En route to new blockbuster anti-histamines: surveying the offspring of the expanding histamine receptor family

Molecular Determinants of Selective Agonist and Antagonist Binding to the Histamine H4 Receptor

An efficient and information-rich biochemical method design for fragment library screening on ion channels

3D-e-Chem-VM: Structural Cheminformatics Research Infrastructure in a Freely Available Virtual Machine

Antiinflammatory and antinociceptive effects of the selective histamine H4-receptor antagonists JNJ7777120 and VUF6002 in a rat model of carrageenan-induced acute inflammation

Targeted LC-MS derivatization for aldehydes and carboxylic acids with a new derivatization agent 4-APEBA

Ligand efficiency as a guide in fragment hit selection and optimization

Synthesis, modeling and functional activity of substituted styrene-amides as small-molecule CXCR7 agonists

Major advances in the development of histamine H4 receptor ligands

Acetylcholine binding protein (AChBP) as template for hierarchical in silico screening procedures to identify structurally novel ligands for the nicotinic receptors

Multiplexed experimental strategies for fragment library screening against challenging drug targets using SPR biosensors

Combinatorial Consensus Scoring for Ligand-Based Virtual Fragment Screening: A Comparative Case Study for Serotonin 5‑HT3A, Histamine H1, and Histamine H4 Receptors

Online Fluorescence Enhancement Assay for the Acetylcholine Binding Protein with Parallel Mass Spectrometric Identification

CXCR3 antagonists: Quaternary ammonium salts equipped with biphenyl- and polycycloaliphatic-anchors

A novel series of histamine H4 receptor antagonists based on the pyrido[3,2-d]pyrimidine scaffold: Comparison of hERG binding and target residence time with PF-3893787

KLIFS: an overhaul after the first 5 years of supporting kinase research

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