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Recent advances in antibacterial agents

Bioorganic & medicinal chemistry letters, 2021-03, Vol.35, p.127799-127799, Article 127799

2021

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Design, Synthesis, and Structure–Activity Relationship Studies of Novel Thioether Pleuromutilin Derivatives as Potent Antibacterial Agents

Journal of medicinal chemistry, 2014-06, Vol.57 (11), p.4772-4795

2014

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Design, Synthesis, and Structure–Activity and Structure–Pharmacokinetic Relationship Studies of Novel [6,6,5] Tricyclic Fused Oxazolidinones Leading to the Discovery of a Potent, Selective, and Orally Bioavailable FXa Inhibitor

Journal of medicinal chemistry, 2014-09, Vol.57 (18), p.7770-7791

2014

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Solubility-Driven Optimization of (Pyridin-3-yl) Benzoxazinyl-oxazolidinones Leading to a Promising Antibacterial Agent

Journal of medicinal chemistry, 2013-03, Vol.56 (6), p.2642-2650

2013

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Synthesis and antibacterial activity of novel fluoroquinolones containing substituted piperidines

Bioorganic & medicinal chemistry letters, 2007-08, Vol.17 (16), p.4523-4526

2007

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Synthesis and structure–activity relationship studies of novel [6,6,5] tricyclic oxazolidinone derivatives as potential antibacterial agents

Bioorganic & medicinal chemistry letters, 2015-05, Vol.25 (10), p.2203-2210

2015

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Design and synthesis of pyridine-substituted itraconazole analogues with improved antifungal activities, water solubility and bioavailability

Bioorganic & medicinal chemistry letters, 2011-08, Vol.21 (16), p.4779-4783

2011

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Synthesis and Biological Evaluation of Oxopyrido[2,3-d] Pyrimidine-7- ones Derivatives as Covalent L858R/T790M Mutant Selective Epidermal Growth Factor Receptor (EGFR) Inhibitors

Letters in drug design & discovery, 2019, Vol.16 (8), p.826-834

2019

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Design, synthesis, and structure–activity relationship studies of conformationally restricted mutilin 14-carbamates

Bioorganic & medicinal chemistry letters, 2012-01, Vol.22 (2), p.814-819

2012

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Evaluation of the antipsychotic effect of bi-acetylated l -stepholidine ( l -SPD-A), a novel dopamine and serotonin receptor dual ligand

Schizophrenia research, 2009-11, Vol.115 (1), p.41-49

2009

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Design, synthesis and biological evaluation of novel thiohydantoin derivatives as potent androgen receptor antagonists for the treatment of prostate cancer

Bioorganic & medicinal chemistry, 2021-02, Vol.31, p.115953-115953, Article 115953

2021

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Design, Synthesis, and Structure–Activity Relationship Studies of Novel Fused Heterocycles-Linked Triazoles with Good Activity and Water Solubility

Journal of medicinal chemistry, 2014-05, Vol.57 (9), p.3687-3706

2014

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Efficient Kilogram-Scale Synthesis of a Novel Oxazolidinone Antibacterial Candidate YG-056SP

Organic process research & development, 2023-02, Vol.27 (2), p.331-342

2023

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Total Synthesis of (S)-(-)-Stepholidine Using (S)-tert-Butanesulfinylimine

Heterocycles, 2010, Vol.81 (11), p.2581

2010

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Design and synthesis of novel bis( l-amino acid) ester prodrugs of 9-[2-(phosphonomethoxy)ethyl]adenine (PMEA) with improved anti-HBV activity

Bioorganic & medicinal chemistry letters, 2007-01, Vol.17 (2), p.465-470

2007

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Discovery of Thieno[2,3‑e]indazole Derivatives as Novel Oral Selective Estrogen Receptor Degraders with Highly Improved Antitumor Effect and Favorable Druggability

Journal of medicinal chemistry, 2022-04, Vol.65 (7), p.5724-5750

2022

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Water-soluble phosphate prodrugs of pleuromutilin analogues with potent in vivo antibacterial activity against Gram-positive pathogens

Bioorganic & medicinal chemistry letters, 2009-09, Vol.19 (18), p.5407-5410

2009

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Discovery of a Novel Bifunctional Steroid Analog, YXG-158, as an Androgen Receptor Degrader and CYP17A1 Inhibitor for the Treatment of Enzalutamide-Resistant Prostate Cancer

Journal of medicinal chemistry, 2023-07, Vol.66 (14), p.9972-9991

2023

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Design, Synthesis, and Biological Evaluation of Androgen Receptor Degrading and Antagonizing Bifunctional Steroidal Analogs for the Treatment of Advanced Prostate Cancer

Journal of medicinal chemistry, 2022-09, Vol.65 (18), p.12460-12481

2022

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Synthesis and antibacterial activity of oxazolidinones containing triazolyl group

European journal of medicinal chemistry, 2007-08, Vol.42 (8), p.1137-1143

2007

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Design, synthesis and evaluation of novel oxazaphosphorine prodrugs of 9-(2-phosphonomethoxyethyl)adenine (PMEA, adefovir) as potent HBV inhibitors

Bioorganic & medicinal chemistry letters, 2009-12, Vol.19 (24), p.6918-6921

2009

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Design, synthesis, and structure-activity relationship studies of novel tetrazole antifungal agents with potent activity, broad antifungal spectrum and high selectivity

Bioorganic & medicinal chemistry letters, 2018-02, Vol.28 (3), p.344-350

2018

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Design, Synthesis, and Biological Evaluation of Novel Arylomycins against Multidrug-Resistant Gram-Negative Bacteria

Journal of medicinal chemistry, 2024-04, Vol.67 (8), p.6585-6609

2024

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Design, Synthesis, and Anti-tuberculosis Activity of Streptomycin Derivatives

Letters in drug design & discovery, 2024-03, Vol.21 (4), p.738-748

2024

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Design, Synthesis, and Biological Evaluation of Novel Pyrimido[4,5‑b]indole Derivatives Against Gram-Negative Multidrug-Resistant Pathogens

Journal of medicinal chemistry, 2021-06, Vol.64 (12), p.8644-8665

2021

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Recent advances in antibacterial agents

Design, Synthesis, and Structure–Activity Relationship Studies of Novel Thioether Pleuromutilin Derivatives as Potent Antibacterial Agents

Design, Synthesis, and Structure–Activity and Structure–Pharmacokinetic Relationship Studies of Novel [6,6,5] Tricyclic Fused Oxazolidinones Leading to the Discovery of a Potent, Selective, and Orally Bioavailable FXa Inhibitor

Solubility-Driven Optimization of (Pyridin-3-yl) Benzoxazinyl-oxazolidinones Leading to a Promising Antibacterial Agent

Synthesis and antibacterial activity of novel fluoroquinolones containing substituted piperidines

Synthesis and structure–activity relationship studies of novel [6,6,5] tricyclic oxazolidinone derivatives as potential antibacterial agents

Design and synthesis of pyridine-substituted itraconazole analogues with improved antifungal activities, water solubility and bioavailability

Synthesis and Biological Evaluation of Oxopyrido[2,3-d] Pyrimidine-7- ones Derivatives as Covalent L858R/T790M Mutant Selective Epidermal Growth Factor Receptor (EGFR) Inhibitors

Design, synthesis, and structure–activity relationship studies of conformationally restricted mutilin 14-carbamates

Evaluation of the antipsychotic effect of bi-acetylated l -stepholidine ( l -SPD-A), a novel dopamine and serotonin receptor dual ligand

Design, synthesis and biological evaluation of novel thiohydantoin derivatives as potent androgen receptor antagonists for the treatment of prostate cancer

Design, Synthesis, and Structure–Activity Relationship Studies of Novel Fused Heterocycles-Linked Triazoles with Good Activity and Water Solubility

Efficient Kilogram-Scale Synthesis of a Novel Oxazolidinone Antibacterial Candidate YG-056SP

Total Synthesis of (S)-(-)-Stepholidine Using (S)-tert-Butanesulfinylimine

Design and synthesis of novel bis( l-amino acid) ester prodrugs of 9-[2-(phosphonomethoxy)ethyl]adenine (PMEA) with improved anti-HBV activity

Discovery of Thieno[2,3‑e]indazole Derivatives as Novel Oral Selective Estrogen Receptor Degraders with Highly Improved Antitumor Effect and Favorable Druggability

Water-soluble phosphate prodrugs of pleuromutilin analogues with potent in vivo antibacterial activity against Gram-positive pathogens

Discovery of a Novel Bifunctional Steroid Analog, YXG-158, as an Androgen Receptor Degrader and CYP17A1 Inhibitor for the Treatment of Enzalutamide-Resistant Prostate Cancer

Design, Synthesis, and Biological Evaluation of Androgen Receptor Degrading and Antagonizing Bifunctional Steroidal Analogs for the Treatment of Advanced Prostate Cancer

Synthesis and antibacterial activity of oxazolidinones containing triazolyl group

Design, synthesis and evaluation of novel oxazaphosphorine prodrugs of 9-(2-phosphonomethoxyethyl)adenine (PMEA, adefovir) as potent HBV inhibitors

Design, synthesis, and structure-activity relationship studies of novel tetrazole antifungal agents with potent activity, broad antifungal spectrum and high selectivity

Design, Synthesis, and Biological Evaluation of Novel Arylomycins against Multidrug-Resistant Gram-Negative Bacteria

Design, Synthesis, and Anti-tuberculosis Activity of Streptomycin Derivatives

Design, Synthesis, and Biological Evaluation of Novel Pyrimido[4,5‑b]indole Derivatives Against Gram-Negative Multidrug-Resistant Pathogens

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