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The metabolic fate of izencitinib, a gut-selective pan-JAK inhibitor, in humans. Identification of unusual fecal metabolites and implications for MIST evaluation

Medicinal chemistry research, 2023-09, Vol.32 (9), p.2071-2088

2023

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Cytochrome P450 3A-mediated metabolism of buspirone in human liver microsomes

Drug metabolism and disposition, 2005-04, Vol.33 (4), p.500-507

2005

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Detection of Endogenous Malondialdehyde-Deoxyguanosine Adducts in Human Liver

Science (American Association for the Advancement of Science), 1994-09, Vol.265 (5178), p.1580-1582

1994

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Inhibitors of HIV-1 attachment. Part 2: An initial survey of indole substitution patterns

Bioorganic & medicinal chemistry letters, 2009-04, Vol.19 (7), p.1977-1981

2009

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6-Hydroxybuspirone is a major active metabolite of buspirone: assessment of pharmacokinetics and 5-hydroxytryptamine1A receptor occupancy in rats

Drug metabolism and disposition, 2007-08, Vol.35 (8), p.1387

2007

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Fluorine Substitution Can Block CYP3A4 Metabolism-Dependent Inhibition: Identification of (S)-N-[1-(4-Fluoro-3- morpholin-4-ylphenyl)ethyl]-3- (4-fluorophenyl)acrylamide as an Orally Bioavailable KCNQ2 Opener Devoid of CYP3A4 Metabolism-Dependent Inhibition

Journal of medicinal chemistry, 2003-08, Vol.46 (18), p.3778-3781

2003

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Comparative metabolism of radiolabeled muraglitazar in animals and humans by quantitative and qualitative metabolite profiling

Drug metabolism and disposition, 2007-01, Vol.35 (1), p.150-167

2007

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Revefenacin Absorption, Metabolism, and Excretion in Healthy Subjects and Pharmacological Activity of Its Major Metabolite

Drug metabolism and disposition, 2020-12, Vol.48 (12), p.1312-1320

2020

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In vitro and in vivo metabolism of a gamma-secretase inhibitor BMS-299897 and generation of active metabolites in milligram quantities with a microbial bioreactor

Current drug metabolism, 2006-12, Vol.7 (8), p.883-896

2006

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Synthesis of 10(S)-Hydroxyeicosatetraenoic Acid: A Novel Cytochrome P-450 Metabolite of Arachidonic Acid

Journal of organic chemistry, 1996-02, Vol.61 (3), p.838-841

1996

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Discovery of (S) -2 -( (S) -2 -(3,5 -difluorophenyl ) -2-hydroxyacetamido ) -N-( (S,Z) -3 -methyl -4 -oxo -4,5 -dihydro -3H-benzo[d|[1,2 ]diazepin -5 -yl )propanamide (BMS -433796 ) : A γ-secretase inhibitor with Aβ lowering activity in a transgenic mouse model of Alzheimer's disease

Bioorganic & medicinal chemistry letters, 2007-07, Vol.17 (14), p.4006-4011

2007

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Activities of the four optical isomers of 2',3'-dideoxy-3'-thiacytidine (BCH-189) against human immunodeficiency virus type 1 in human lymphocytes

Antimicrobial Agents and Chemotherapy, 1992-03, Vol.36 (3), p.672-676

1992

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6-Hydroxybuspirone Is a Major Active Metabolite of Buspirone: Assessment of Pharmacokinetics and 5-Hydroxytryptamine 1A Receptor Occupancy in Rats

Drug metabolism and disposition, 2007-08, Vol.35 (8), p.1387-1392

2007

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Corrigendum to “Inhibitors of HIV-1 attachment. Part 2: An initial survey of indole substitution patterns” [Bioorg. Med. Chem. Lett. 19 (2009) 1977]

Bioorganic & medicinal chemistry letters, 2010-02, Vol.20 (4), p.1460-1460

2010

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Aminotriazine 5-HT7 antagonists

Bioorganic & medicinal chemistry letters, 2004-08, Vol.14 (16), p.4245-4248

2004

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In situ complexation directs the stereochemistry of N-glycosylation in the synthesis of oxathiolanyl and dioxolanyl nucleoside analogues

Journal of the American Chemical Society, 1991-11, Vol.113 (24), p.9377-9379

1991

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Discovery of (S)-2-((S)-2-(3,5-difluorophenyl)-2-hydroxyacetamido)-N-((S,Z)-3-methyl-4-oxo-4,5-dihydro-3H-benzo[d][1,2]diazepin-5-yl)propanamide (BMS-433796): a gamma-secretase inhibitor with Abeta lowering activity in a transgenic mouse model of Alzheimer's disease

Bioorganic & medicinal chemistry letters, 2007-07, Vol.17 (14), p.4006

2007

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In situ complexation directs the stereochemistry of N-glycosylation in the synthesis of thialanyl and dioxolanyl nucleoside analogs

Journal of the American Chemical Society, 1991-11, Vol.113 (24), p.9377-9379

1991

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Discovery of ( S)-2-(( S)-2-(3,5-difluorophenyl)-2-hydroxyacetamido)- N-(( S, Z)-3-methyl-4-oxo-4,5-dihydro-3 H-benzo[ d][1,2]diazepin-5-yl)propanamide (BMS-433796): A γ-secretase inhibitor with Aβ lowering activity in a transgenic mouse model of Alzheimer’s disease

Bioorganic & medicinal chemistry letters, 2007, Vol.17 (14), p.4006-4011

2007

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7-HETE, 10-HETE, and 13-HETE Are Major Products of NADPH-Dependent Arachidonic Acid Metabolism in Rat Liver Microsomes: Analysis of Their Stereochemistry, and the Stereochemistry of Their Acid-Catalyzed Rearrangement

Archives of biochemistry and biophysics, 1995-08, Vol.321 (2), p.485-492

1995

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A convenient two-step synthesis of 3-allylcoumarins and their benzoderivatives

Heterocycles, 1987, Vol.26 (1), p.121-127

1987

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Processing of procarboxypeptidase A and other zymogens in murine mast cells

The Journal of biological chemistry, 1994-10, Vol.269 (41), p.25897-25904

1994

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Aminotriazine 5-HT 7 antagonists

Bioorganic & medicinal chemistry letters, 2004, Vol.14 (16), p.4245-4248

2004

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A Novel Synthesis of N-Substituted-3-carboethoxymethylphthalimidines

Synthesis (Stuttgart), 1986, Vol.1986 (9), p.755-757

1986

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Synthesis, anti-human immunodeficiency virus, and anti-hepatitis B virus activity of pyrimidine oxathiolane nucleosides

Bioorganic & medicinal chemistry letters, 1993-04, Vol.3 (4), p.693-696

1993

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The metabolic fate of izencitinib, a gut-selective pan-JAK inhibitor, in humans. Identification of unusual fecal metabolites and implications for MIST evaluation

Cytochrome P450 3A-mediated metabolism of buspirone in human liver microsomes

Detection of Endogenous Malondialdehyde-Deoxyguanosine Adducts in Human Liver

Inhibitors of HIV-1 attachment. Part 2: An initial survey of indole substitution patterns

6-Hydroxybuspirone is a major active metabolite of buspirone: assessment of pharmacokinetics and 5-hydroxytryptamine1A receptor occupancy in rats

Fluorine Substitution Can Block CYP3A4 Metabolism-Dependent Inhibition: Identification of (S)-N-[1-(4-Fluoro-3- morpholin-4-ylphenyl)ethyl]-3- (4-fluorophenyl)acrylamide as an Orally Bioavailable KCNQ2 Opener Devoid of CYP3A4 Metabolism-Dependent Inhibition

Comparative metabolism of radiolabeled muraglitazar in animals and humans by quantitative and qualitative metabolite profiling

Revefenacin Absorption, Metabolism, and Excretion in Healthy Subjects and Pharmacological Activity of Its Major Metabolite

In vitro and in vivo metabolism of a gamma-secretase inhibitor BMS-299897 and generation of active metabolites in milligram quantities with a microbial bioreactor

Synthesis of 10(S)-Hydroxyeicosatetraenoic Acid: A Novel Cytochrome P-450 Metabolite of Arachidonic Acid

Discovery of (S) -2 -( (S) -2 -(3,5 -difluorophenyl ) -2-hydroxyacetamido ) -N-( (S,Z) -3 -methyl -4 -oxo -4,5 -dihydro -3H-benzo[d|[1,2 ]diazepin -5 -yl )propanamide (BMS -433796 ) : A γ-secretase inhibitor with Aβ lowering activity in a transgenic mouse model of Alzheimer's disease

Activities of the four optical isomers of 2',3'-dideoxy-3'-thiacytidine (BCH-189) against human immunodeficiency virus type 1 in human lymphocytes

6-Hydroxybuspirone Is a Major Active Metabolite of Buspirone: Assessment of Pharmacokinetics and 5-Hydroxytryptamine 1A Receptor Occupancy in Rats

Corrigendum to “Inhibitors of HIV-1 attachment. Part 2: An initial survey of indole substitution patterns” [Bioorg. Med. Chem. Lett. 19 (2009) 1977]

Aminotriazine 5-HT7 antagonists

In situ complexation directs the stereochemistry of N-glycosylation in the synthesis of oxathiolanyl and dioxolanyl nucleoside analogues

Discovery of (S)-2-((S)-2-(3,5-difluorophenyl)-2-hydroxyacetamido)-N-((S,Z)-3-methyl-4-oxo-4,5-dihydro-3H-benzo[d][1,2]diazepin-5-yl)propanamide (BMS-433796): a gamma-secretase inhibitor with Abeta lowering activity in a transgenic mouse model of Alzheimer's disease

In situ complexation directs the stereochemistry of N-glycosylation in the synthesis of thialanyl and dioxolanyl nucleoside analogs

Discovery of ( S)-2-(( S)-2-(3,5-difluorophenyl)-2-hydroxyacetamido)- N-(( S, Z)-3-methyl-4-oxo-4,5-dihydro-3 H-benzo[ d][1,2]diazepin-5-yl)propanamide (BMS-433796): A γ-secretase inhibitor with Aβ lowering activity in a transgenic mouse model of Alzheimer’s disease

7-HETE, 10-HETE, and 13-HETE Are Major Products of NADPH-Dependent Arachidonic Acid Metabolism in Rat Liver Microsomes: Analysis of Their Stereochemistry, and the Stereochemistry of Their Acid-Catalyzed Rearrangement

A convenient two-step synthesis of 3-allylcoumarins and their benzoderivatives

Processing of procarboxypeptidase A and other zymogens in murine mast cells

Aminotriazine 5-HT 7 antagonists

A Novel Synthesis of N-Substituted-3-carboethoxymethylphthalimidines

Synthesis, anti-human immunodeficiency virus, and anti-hepatitis B virus activity of pyrimidine oxathiolane nucleosides

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