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Discovery of N-methyl-4-(4-methoxyanilino)quinazolines as potent apoptosis inducers. Structure–activity relationship of the quinazoline ring

Bioorganic & medicinal chemistry letters, 2010-04, Vol.20 (7), p.2330-2334

2010

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Characterization of the cellular and antitumor effects of MPI-0479605, a small-molecule inhibitor of the mitotic kinase Mps1

Molecular cancer therapeutics, 2011-12, Vol.10 (12), p.2267-2275

2011

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Inhibition of eEF2-K by thieno[2,3- b]pyridine analogues

Bioorganic & medicinal chemistry letters, 2010-04, Vol.20 (7), p.2283-2286

2010

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Discovery of a new HIV-1 inhibitor scaffold and synthesis of potential prodrugs of indazoles

Bioorganic & medicinal chemistry letters, 2013-05, Vol.23 (10), p.2888-2892

2013

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2-Anilino-4-aryl-1,3-thiazole inhibitors of valosin-containing protein (VCP or p97)

Bioorganic & medicinal chemistry letters, 2010-03, Vol.20 (5), p.1677-1679

2010

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Discovery and SAR of Methylated Tetrahydropyranyl Derivatives as Inhibitors of Isoprenylcysteine Carboxyl Methyltransferase (ICMT)

Journal of medicinal chemistry, 2011-07, Vol.54 (14), p.5031-5047

2011

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Design, Synthesis, and Biological Activity of Potent and Selective Inhibitors of Blood Coagulation Factor Xa

Journal of medicinal chemistry, 2004-07, Vol.47 (16), p.4089-4099

2004

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Discovery of N-(4-Methoxyphenyl)-N,2-dimethylquinazolin-4-amine, a Potent Apoptosis Inducer and Efficacious Anticancer Agent with High Blood Brain Barrier Penetration

Journal of medicinal chemistry, 2009-04, Vol.52 (8), p.2341-2351

2009

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Oxindole derivatives as inhibitors of TAK1 kinase

Bioorganic & medicinal chemistry letters, 2011-03, Vol.21 (6), p.1724-1727

2011

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Discovery of 2-Chloro-N-(4-methoxyphenyl)-N-methylquinazolin-4-amine (EP128265, MPI-0441138) as a Potent Inducer of Apoptosis with High In Vivo Activity

Journal of medicinal chemistry, 2008-08, Vol.51 (15), p.4771-4779

2008

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Synthesis of Substituted Quinazolines: Application to the Synthesis of Verubulin

Synthetic communications, 2012-06, Vol.42 (12), p.1715-1723

2012

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Analogues of 4-[(7-Bromo-2-methyl-4-oxo-3H-quinazolin-6-yl)methylprop-2-ynylamino]-N-(3-pyridylmethyl)benzamide (CB-30865) as Potent Inhibitors of Nicotinamide Phosphoribosyltransferase (Nampt)

Journal of medicinal chemistry, 2010-12, Vol.53 (24), p.8734-8746

2010

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Protease-Activated Receptor 2, Dipeptidyl Peptidase I, and Proteases Mediate Clostridium difficile Toxin A Enteritis

Gastroenterology (New York, N.Y. 1943), 2007-06, Vol.132 (7), p.2422-2437

2007

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The discovery of fluoropyridine-based inhibitors of the factor VIIa/TF complex—Part 2

Bioorganic & medicinal chemistry letters, 2006-02, Vol.16 (4), p.1060-1064

2006

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The discovery of fluoropyridine-based inhibitors of the Factor VIIa/TF complex

Bioorganic & medicinal chemistry letters, 2005-11, Vol.15 (21), p.4752-4756

2005

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Total Synthesis and Structural Elucidation of the Antifungal Agent Papulacandin D

Journal of organic chemistry, 1996-02, Vol.61 (3), p.1082-1100

1996

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Chemical Proteomics Identifies Nampt as the Target of CB30865, An Orphan Cytotoxic Compound

Chemistry & biology, 2010-06, Vol.17 (6), p.659-664

2010

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Abstract LB-393: The cancer metabolism inhibitor MPC-9528 induces tumor regression in xenograft models with multiple dosing schedules by causing rapid and sustained reduction in tumor NAD

Cancer research (Chicago, Ill.), 2011-04, Vol.71 (8_Supplement), p.LB-393-LB-393

2011

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TTK Kinase Inhibitor Development through Chemical Proteomics

The FASEB journal, 2010-04, Vol.24 (S1), p.lb203-lb203

2010

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Abstract LB-288: MPI-0486348: A novel inhibitor of nicotinamide phosphoribosyltransferase (Nampt) induces tumor regression in a preclinical model

Cancer research (Chicago, Ill.), 2010-04, Vol.70 (8_Supplement), p.LB-288-LB-288

2010

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Total synthesis of the antifungal agent papulacandin D

Journal of the Chemical Society. Chemical communications, 1995 (11), p.1147-1148

1995

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Approaches towards the synthesis of papulacandin D: preparation and structural elucidation of the acyl side chain

Journal of the Chemical Society. Chemical communications, 1995 (11), p.1145-1146

1995

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ChemInform Abstract: Synthesis of Substituted Quinazolines: Application to the Synthesis of Verubulin

ChemInform, 2012-09, Vol.43 (38), p.no-no

2012

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Discovery of N-methyl-4-(4-methoxyanilino)quinazolines as potent apoptosis inducers. Structure–activity relationship of the quinazoline ring

Characterization of the cellular and antitumor effects of MPI-0479605, a small-molecule inhibitor of the mitotic kinase Mps1

Inhibition of eEF2-K by thieno[2,3- b]pyridine analogues

Discovery of a new HIV-1 inhibitor scaffold and synthesis of potential prodrugs of indazoles

2-Anilino-4-aryl-1,3-thiazole inhibitors of valosin-containing protein (VCP or p97)

Discovery and SAR of Methylated Tetrahydropyranyl Derivatives as Inhibitors of Isoprenylcysteine Carboxyl Methyltransferase (ICMT)

Design, Synthesis, and Biological Activity of Potent and Selective Inhibitors of Blood Coagulation Factor Xa

Discovery of N-(4-Methoxyphenyl)-N,2-dimethylquinazolin-4-amine, a Potent Apoptosis Inducer and Efficacious Anticancer Agent with High Blood Brain Barrier Penetration

Oxindole derivatives as inhibitors of TAK1 kinase

Discovery of 2-Chloro-N-(4-methoxyphenyl)-N-methylquinazolin-4-amine (EP128265, MPI-0441138) as a Potent Inducer of Apoptosis with High In Vivo Activity

Synthesis of Substituted Quinazolines: Application to the Synthesis of Verubulin

Analogues of 4-[(7-Bromo-2-methyl-4-oxo-3H-quinazolin-6-yl)methylprop-2-ynylamino]-N-(3-pyridylmethyl)benzamide (CB-30865) as Potent Inhibitors of Nicotinamide Phosphoribosyltransferase (Nampt)

Protease-Activated Receptor 2, Dipeptidyl Peptidase I, and Proteases Mediate Clostridium difficile Toxin A Enteritis

The discovery of fluoropyridine-based inhibitors of the factor VIIa/TF complex—Part 2

The discovery of fluoropyridine-based inhibitors of the Factor VIIa/TF complex

Total Synthesis and Structural Elucidation of the Antifungal Agent Papulacandin D

Chemical Proteomics Identifies Nampt as the Target of CB30865, An Orphan Cytotoxic Compound

Abstract LB-393: The cancer metabolism inhibitor MPC-9528 induces tumor regression in xenograft models with multiple dosing schedules by causing rapid and sustained reduction in tumor NAD

TTK Kinase Inhibitor Development through Chemical Proteomics

Abstract LB-288: MPI-0486348: A novel inhibitor of nicotinamide phosphoribosyltransferase (Nampt) induces tumor regression in a preclinical model

Total synthesis of the antifungal agent papulacandin D

Approaches towards the synthesis of papulacandin D: preparation and structural elucidation of the acyl side chain

ChemInform Abstract: Synthesis of Substituted Quinazolines: Application to the Synthesis of Verubulin

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