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Pyrrolopyridine Inhibitors of Mitogen-Activated Protein Kinase-Activated Protein Kinase 2 (MK-2)

Journal of medicinal chemistry, 2007-05, Vol.50 (11), p.2647-2654

2007

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Aminocyanopyridine inhibitors of mitogen activated protein kinase-activated protein kinase 2 (MK-2)

Bioorganic & medicinal chemistry letters, 2005-03, Vol.15 (6), p.1587-1590

2005

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Design and Synthesis of Novel and Selective Phosphodiesterase 2 (PDE2a) Inhibitors for the Treatment of Memory Disorders

Journal of medicinal chemistry, 2017-03, Vol.60 (5), p.2037-2051

2017

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Novel tetrahydro-β-carboline-1-carboxylic acids as inhibitors of mitogen activated protein kinase-activated protein kinase 2 (MK-2)

Bioorganic & medicinal chemistry letters, 2007-08, Vol.17 (16), p.4657-4663

2007

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Regioselective palladium-catalyzed C H arylation of 4-alkoxy and 4-thioalkyl pyrazoles

Tetrahedron letters, 2017-12, Vol.58 (49), p.4587-4590

2017

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Regioselective palladium-catalyzed CH arylation of 4-alkoxy and 4-thioalkyl pyrazoles

Tetrahedron letters, 2017-12, Vol.58 (49), p.4587-4590

2017

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Antitumor activity of a systemic STING-activating non-nucleotide cGAMP mimetic

Science (American Association for the Advancement of Science), 2020-08, Vol.369 (6506), p.993-999

2020

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Synthesis of novel nitric oxide (NO)-releasing esters of timolol

Bioorganic & medicinal chemistry letters, 2009-05, Vol.19 (10), p.2785-2788

2009

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Discovery of a Simple Picomolar Inhibitor of Cholesteryl Ester Transfer Protein

Journal of medicinal chemistry, 2003-05, Vol.46 (11), p.2152-2168

2003

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Mathematical and Structural Characterization of Strong Nonadditive Structure–Activity Relationship Caused by Protein Conformational Changes

Journal of medicinal chemistry, 2018-09, Vol.61 (17), p.7754-7766

2018

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Discovery of 1‑{(3R,4R)‑3-[({5-Chloro-2-[(1-methyl‑1H‑pyrazol-4-yl)amino]‑7H‑pyrrolo[2,3‑d]pyrimidin-4-yl}oxy)methyl]-4-methoxypyrrolidin-1-yl}prop-2-en-1-one (PF-06459988), a Potent, WT Sparing, Irreversible Inhibitor of T790M-Containing EGFR Mutants

Journal of medicinal chemistry, 2016-03, Vol.59 (5), p.2005-2024

2016

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A novel class of apical sodium co-dependent bile acid transporter inhibitors: The 1,2-benzothiazepines

Bioorganic & medicinal chemistry letters, 2003-11, Vol.13 (21), p.3727-3730

2003

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Stereospecific Inhibition of CETP by Chiral N,N-Disubstituted Trifluoro-3-amino-2-propanols

Biochemistry (Easton), 2000-11, Vol.39 (45), p.13870-13879

2000

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Thioether benzenesulfonamide inhibitors of carbonic anhydrases II and IV: Structure-based drug design, synthesis, and biological evaluation

Bioorganic & medicinal chemistry, 2010-05, Vol.18 (9), p.3307-3319

2010

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Discovery of Novel, Potent, and Selective Inhibitors of 3-Phosphoinositide-Dependent Kinase (PDK1)

Journal of medicinal chemistry, 2011-12, Vol.54 (24), p.8490-8500

2011

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Abstract 753: Novel, potent and selective small molecule inhibitors of 3-phosphoinositide-dependent kinase (PDK1)

Cancer research (Chicago, Ill.), 2010-04, Vol.70 (8_Supplement), p.753-753

2010

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Corrigendum to “Thioether benzenesulfonamide inhibitors of carbonic anhydrases II and IV: Structure-based drug design, synthesis, and biological evaluation” [Bioorg. Med. Chem. 18 (2010) 3307]

Bioorganic & medicinal chemistry, 2010-10, Vol.18 (19), p.7144-7144

2010

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Corrigendum to “Novel tetrahydro-β-carboline-1-carboxylic acids as inhibitors of mitogen activated protein kinase-activated protein kinase 2 (MK-2)” [Bioorg. Med. Chem. Lett. 17 (2007) 4657–4663]

Bioorganic & medicinal chemistry letters, 2009-04, Vol.19 (8), p.2365-2365

2009

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A novel class of apical sodium co-dependent bile acid transporter inhibitors : The 2,3-disubstituted-4-phenylquinolines

Bioorganic & medicinal chemistry letters, 2000-02, Vol.10 (3), p.277-279

2000

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A Novel Class of Apical Sodium Co-Dependent Bile Acid Transporter Inhibitors: The 1,2-Benzothiazepines

ChemInform, 2004-02, Vol.35 (6), p.no-no

2004

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Aminocyanopyridine Inhibitors of Mitogen Activated Protein Kinase-Activated Protein Kinase 2 (MK-2)

ChemInform, 2005-07, Vol.36 (29), p.no-no

2005

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ChemInform Abstract: A Novel Class of Apical Sodium Co-Dependent Bile Acid Transporter Inhibitors: The 2,3-Disubstituted-4-phenylquinolines

ChemInform, 2000-05, Vol.31 (21), p.no-no

2000

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The ADHD-susceptibility gene lphn3.1 modulates dopaminergic neuron formation and locomotor activity during zebrafish development

Molecular psychiatry, 2012-09, Vol.17 (9), p.946-954

2012

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Pyrrolopyridine Inhibitors of Mitogen-Activated Protein Kinase-Activated Protein Kinase 2 (MK-2)

Aminocyanopyridine inhibitors of mitogen activated protein kinase-activated protein kinase 2 (MK-2)

Design and Synthesis of Novel and Selective Phosphodiesterase 2 (PDE2a) Inhibitors for the Treatment of Memory Disorders

Novel tetrahydro-β-carboline-1-carboxylic acids as inhibitors of mitogen activated protein kinase-activated protein kinase 2 (MK-2)

Regioselective palladium-catalyzed C H arylation of 4-alkoxy and 4-thioalkyl pyrazoles

Regioselective palladium-catalyzed CH arylation of 4-alkoxy and 4-thioalkyl pyrazoles

Antitumor activity of a systemic STING-activating non-nucleotide cGAMP mimetic

Synthesis of novel nitric oxide (NO)-releasing esters of timolol

Discovery of a Simple Picomolar Inhibitor of Cholesteryl Ester Transfer Protein

Mathematical and Structural Characterization of Strong Nonadditive Structure–Activity Relationship Caused by Protein Conformational Changes

Discovery of 1‑{(3R,4R)‑3-[({5-Chloro-2-[(1-methyl‑1H‑pyrazol-4-yl)amino]‑7H‑pyrrolo[2,3‑d]pyrimidin-4-yl}oxy)methyl]-4-methoxypyrrolidin-1-yl}prop-2-en-1-one (PF-06459988), a Potent, WT Sparing, Irreversible Inhibitor of T790M-Containing EGFR Mutants

A novel class of apical sodium co-dependent bile acid transporter inhibitors: The 1,2-benzothiazepines

Stereospecific Inhibition of CETP by Chiral N,N-Disubstituted Trifluoro-3-amino-2-propanols

Thioether benzenesulfonamide inhibitors of carbonic anhydrases II and IV: Structure-based drug design, synthesis, and biological evaluation

Discovery of Novel, Potent, and Selective Inhibitors of 3-Phosphoinositide-Dependent Kinase (PDK1)

Discovery of Potent, Nonsystemic Apical Sodium-Codependent Bile Acid Transporter Inhibitors (Part 1)

Abstract 753: Novel, potent and selective small molecule inhibitors of 3-phosphoinositide-dependent kinase (PDK1)

Corrigendum to “Thioether benzenesulfonamide inhibitors of carbonic anhydrases II and IV: Structure-based drug design, synthesis, and biological evaluation” [Bioorg. Med. Chem. 18 (2010) 3307]

Discovery of Potent, Nonsystemic Apical Sodium-Codependent Bile Acid Transporter Inhibitors (Part 2)

Corrigendum to “Novel tetrahydro-β-carboline-1-carboxylic acids as inhibitors of mitogen activated protein kinase-activated protein kinase 2 (MK-2)” [Bioorg. Med. Chem. Lett. 17 (2007) 4657–4663]

A novel class of apical sodium co-dependent bile acid transporter inhibitors : The 2,3-disubstituted-4-phenylquinolines

A Novel Class of Apical Sodium Co-Dependent Bile Acid Transporter Inhibitors: The 1,2-Benzothiazepines

Aminocyanopyridine Inhibitors of Mitogen Activated Protein Kinase-Activated Protein Kinase 2 (MK-2)

ChemInform Abstract: A Novel Class of Apical Sodium Co-Dependent Bile Acid Transporter Inhibitors: The 2,3-Disubstituted-4-phenylquinolines

The ADHD-susceptibility gene lphn3.1 modulates dopaminergic neuron formation and locomotor activity during zebrafish development

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