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Structure Guided Lead Generation for M. tuberculosis Thymidylate Kinase (Mtb TMK): Discovery of 3‑Cyanopyridone and 1,6-Naphthyridin-2-one as Potent Inhibitors

Journal of medicinal chemistry, 2015-01, Vol.58 (2), p.753-766

2015

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Quinolinyl Pyrimidines: Potent Inhibitors of NDH-2 as a Novel Class of Anti-TB Agents

ACS medicinal chemistry letters, 2012-09, Vol.3 (9), p.736-740

2012

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Nitroarenes as Antitubercular Agents: Stereoelectronic Modulation to Mitigate Mutagenicity

ChemMedChem, 2016-02, Vol.11 (3), p.331-339

2016

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Pradefovir: A Prodrug That Targets Adefovir to the Liver for the Treatment of Hepatitis B

Journal of medicinal chemistry, 2008-02, Vol.51 (3), p.666-676

2008

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Adenosine Kinase Inhibitors. 6. Synthesis, Water Solubility, and Antinociceptive Activity of 5-Phenyl-7-(5-deoxy-β-d-ribofuranosyl)pyrrolo[2,3-d]pyrimidines Substituted at C4 with Glycinamides and Related Compounds

Journal of medicinal chemistry, 2005-12, Vol.48 (24), p.7808-7820

2005

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Synthesis and Characterization of a Novel Liver-Targeted Prodrug of Cytosine-1-β-d-arabinofuranoside Monophosphate for the Treatment of Hepatocellular Carcinoma

Journal of medicinal chemistry, 2006-12, Vol.49 (26), p.7711-7720

2006

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A Convenient Synthesis of 5-substituted 2-amino-1,3,4-oxadiazoles from Corresponding Acylthiosemicarbazides Using iodine and Oxone

Journal of chemical research, 2013-01, Vol.37 (1), p.53-54

2013

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Design, Synthesis, and Characterization of a Series of Cytochrome P450 3A-Activated Prodrugs (HepDirect Prodrugs) Useful for Targeting Phosph(on)ate-Based Drugs to the Liver

Journal of the American Chemical Society, 2004-04, Vol.126 (16), p.5154-5163

2004

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Adenosine Kinase Inhibitors. 1. Synthesis, Enzyme Inhibition, and Antiseizure Activity of 5-Iodotubercidin Analogues

Journal of medicinal chemistry, 2000-07, Vol.43 (15), p.2883-2893

2000

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Adenosine Kinase Inhibitors. 5. Synthesis, Enzyme Inhibition, and Analgesic Activity of Diaryl-erythro-furanosyltubercidin Analogues

Journal of medicinal chemistry, 2005-10, Vol.48 (20), p.6430-6441

2005

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Adenosine Kinase Inhibitors. 4. 6,8-Disubstituted Purine Nucleoside Derivatives. Synthesis, Conformation, and Enzyme Inhibition

Journal of medicinal chemistry, 2005-05, Vol.48 (9), p.3389-3399

2005

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Adenosine Kinase Inhibitors. 3. Synthesis, SAR, and Antiinflammatory Activity of a Series of l-Lyxofuranosyl Nucleosides

Journal of medicinal chemistry, 2003-10, Vol.46 (22), p.4750-4760

2003

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Adenosine kinase inhibitors as a novel approach to anticonvulsant therapy

The Journal of pharmacology and experimental therapeutics, 1999-06, Vol.289 (3), p.1669

1999

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Adenosine Kinase Inhibitors. 2. Synthesis, Enzyme Inhibition, and Antiseizure Activity of Diaryltubercidin Analogues

Journal of medicinal chemistry, 2000-07, Vol.43 (15), p.2894-2905

2000

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Stereoselective synthesis of 4- C-methyl-2,3,5-tri- O-benzyl- d-ribofuranose and 4- C-methyl-2,3,5-tri- O-benzyl- l-lyxofuranose

Tetrahedron letters, 2003-05, Vol.44 (21), p.4109-4112

2003

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Design, Synthesis, and Characterization of a Series of Cytochrome P 450 3A-Activated Prodrugs (HepDirect Prodrugs) Useful for Targeting Phosph(on)ate-Based Drugs to the Liver

Journal of the American Chemical Society, 2004-04, Vol.126 (16), p.5154-5163

2004

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A convenient synthesis of 5-substituted 2-amino-1,3,4-oxadiazoles from corresponding acylthiosemicarbazides using iodine and Oxone registered

Journal of chemical research, 2013-01, Vol.37 (1), p.53-54

2013

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ChemInform Abstract: A Convenient Synthesis of 5-Substituted 2-Amino-1,3,4-oxadiazoles from Corresponding Acylthiosemicarbazides Using Iodine and Oxone

ChemInform, 2013-07, Vol.44 (28), p.no-no

2013

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Synthesis and antitumor activity of certain 3-.beta.-D-ribofuranosyl-1,2,4-triazolo[3,4-f]-1,2,4-triazines related to formycin prepared via ring closure of a 1,2,4-triazine precursor

Journal of medicinal chemistry, 1986-11, Vol.29 (11), p.2231-2235

1986

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Synthesis and antiviral/antitumor activities of certain pyrazolo[3,4-d]pyrimidine-4(5H)-selone nucleosides and related compounds

Journal of medicinal chemistry, 1984-08, Vol.27 (8), p.1026-1030

1984

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Design, synthesis, and characterization of a series of cytochrome P(450) 3A-activated prodrugs (HepDirect prodrugs) useful for targeting phosph(on)ate-based drugs to the liver

Journal of the American Chemical Society, 2004-04, Vol.126 (16), p.5154-5163

2004

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A simple oxidation of formycin to oxoformycin and oxoformycin B. Synthesis of 6-methyloxoformycin, A C-nucleoside analog of doridosine

Journal of heterocyclic chemistry, 1984-11, Vol.21 (6), p.1865-1870

1984

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Sulphonamide and Sulphonate Derivatives of Sydnones

Archiv der Pharmazie (Weinheim), 1979, Vol.312 (12), p.977-981

1979

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Improved Synthesis of Lycoricidine Triacetate

Synthesis (Stuttgart), 1987, Vol.1987 (8), p.715-716

1987

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Structure Guided Lead Generation for M. tuberculosis Thymidylate Kinase (Mtb TMK): Discovery of 3‑Cyanopyridone and 1,6-Naphthyridin-2-one as Potent Inhibitors

Discovery of benzothiazoles as antimycobacterial agents: Synthesis, structure–activity relationships and binding studies with Mycobacterium tuberculosis decaprenylphosphoryl-β-d-ribose 2′-oxidase

Quinolinyl Pyrimidines: Potent Inhibitors of NDH-2 as a Novel Class of Anti-TB Agents

Nitroarenes as Antitubercular Agents: Stereoelectronic Modulation to Mitigate Mutagenicity

Pradefovir: A Prodrug That Targets Adefovir to the Liver for the Treatment of Hepatitis B

Adenosine Kinase Inhibitors. 6. Synthesis, Water Solubility, and Antinociceptive Activity of 5-Phenyl-7-(5-deoxy-β-d-ribofuranosyl)pyrrolo[2,3-d]pyrimidines Substituted at C4 with Glycinamides and Related Compounds

Synthesis and Characterization of a Novel Liver-Targeted Prodrug of Cytosine-1-β-d-arabinofuranoside Monophosphate for the Treatment of Hepatocellular Carcinoma

A Convenient Synthesis of 5-substituted 2-amino-1,3,4-oxadiazoles from Corresponding Acylthiosemicarbazides Using iodine and Oxone

Design, Synthesis, and Characterization of a Series of Cytochrome P450 3A-Activated Prodrugs (HepDirect Prodrugs) Useful for Targeting Phosph(on)ate-Based Drugs to the Liver

Adenosine Kinase Inhibitors. 1. Synthesis, Enzyme Inhibition, and Antiseizure Activity of 5-Iodotubercidin Analogues

Adenosine Kinase Inhibitors. 5. Synthesis, Enzyme Inhibition, and Analgesic Activity of Diaryl-erythro-furanosyltubercidin Analogues

Adenosine Kinase Inhibitors. 4. 6,8-Disubstituted Purine Nucleoside Derivatives. Synthesis, Conformation, and Enzyme Inhibition

Adenosine Kinase Inhibitors. 3. Synthesis, SAR, and Antiinflammatory Activity of a Series of l-Lyxofuranosyl Nucleosides

Adenosine kinase inhibitors as a novel approach to anticonvulsant therapy

Adenosine Kinase Inhibitors. 2. Synthesis, Enzyme Inhibition, and Antiseizure Activity of Diaryltubercidin Analogues

Stereoselective synthesis of 4- C-methyl-2,3,5-tri- O-benzyl- d-ribofuranose and 4- C-methyl-2,3,5-tri- O-benzyl- l-lyxofuranose

Design, Synthesis, and Characterization of a Series of Cytochrome P 450 3A-Activated Prodrugs (HepDirect Prodrugs) Useful for Targeting Phosph(on)ate-Based Drugs to the Liver

A convenient synthesis of 5-substituted 2-amino-1,3,4-oxadiazoles from corresponding acylthiosemicarbazides using iodine and Oxone registered

ChemInform Abstract: A Convenient Synthesis of 5-Substituted 2-Amino-1,3,4-oxadiazoles from Corresponding Acylthiosemicarbazides Using Iodine and Oxone

Synthesis and antitumor activity of certain 3-.beta.-D-ribofuranosyl-1,2,4-triazolo[3,4-f]-1,2,4-triazines related to formycin prepared via ring closure of a 1,2,4-triazine precursor

Synthesis and antiviral/antitumor activities of certain pyrazolo[3,4-d]pyrimidine-4(5H)-selone nucleosides and related compounds

Design, synthesis, and characterization of a series of cytochrome P(450) 3A-activated prodrugs (HepDirect prodrugs) useful for targeting phosph(on)ate-based drugs to the liver

A simple oxidation of formycin to oxoformycin and oxoformycin B. Synthesis of 6-methyloxoformycin, A C-nucleoside analog of doridosine

Sulphonamide and Sulphonate Derivatives of Sydnones

Improved Synthesis of Lycoricidine Triacetate

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