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Natural Product Synthesis Using Multicomponent Reaction Strategies

Chemical reviews, 2009-09, Vol.109 (9), p.4439-4486

2009

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Accessing Drug Metabolites via Transition-Metal Catalyzed C−H Oxidation: The Liver as Synthetic Inspiration

Angewandte Chemie (International ed.), 2016-11, Vol.55 (46), p.14218-14238

International ed. in English, 2016

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C−H Bonds as Ubiquitous Functionality: A General Approach to Complex Arylated Imidazoles via Regioselective Sequential Arylation of All Three C−H Bonds and Regioselective N-Alkylation Enabled by SEM-Group Transposition

Journal of organic chemistry, 2010-08, Vol.75 (15), p.4911-4920

2010

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Toward the Validation of Maternal Embryonic Leucine Zipper Kinase: Discovery, Optimization of Highly Potent and Selective Inhibitors, and Preliminary Biology Insight

Journal of medicinal chemistry, 2016-05, Vol.59 (10), p.4711-4723

2016

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Three-Component Sequential Aza[4+2] Cycloaddition/Allylboration/Retro-Sulfinyl-Ene Reaction: A New Stereocontrolled Entry to Palustrine Alkaloids and Other 2,6-Disubstituted Piperidines

Angewandte Chemie (International ed.), 2004-04, Vol.43 (15), p.2001-2004

2004

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Complementation of Biotransformations with Chemical C–H Oxidation: Copper-Catalyzed Oxidation of Tertiary Amines in Complex Pharmaceuticals

Journal of the American Chemical Society, 2013-08, Vol.135 (33), p.12346-12352

2013

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Copper-Mediated N-Heteroarylation of Primary Sulfonamides: Synthesis of Mono-N-heteroaryl Sulfonamides

Organic letters, 2010-04, Vol.12 (7), p.1532-1535

2010

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Identification of NVP-TNKS656: The Use of Structure–Efficiency Relationships To Generate a Highly Potent, Selective, and Orally Active Tankyrase Inhibitor

Journal of medicinal chemistry, 2013-08, Vol.56 (16), p.6495-6511

2013

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Catalytic C−H Arylation of SEM-Protected Azoles with Palladium Complexes of NHCs and Phosphines

Organic letters, 2006-05, Vol.8 (10), p.1979-1982

2006

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Discovery of lirafugratinib (RLY-4008), a highly selective irreversible small-molecule inhibitor of FGFR2

Proceedings of the National Academy of Sciences - PNAS, 2024-02, Vol.121 (6), p.e2317756121-e2317756121

2024

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Allosteric Mutant IDH1 Inhibitors Reveal Mechanisms for IDH1 Mutant and Isoform Selectivity

Structure (London), 2017-03, Vol.25 (3), p.506-513

2017

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A Three-Component Reaction for Diversity-Oriented Synthesis of Polysubstituted Piperidines: Solution and Solid-Phase Optimization of the First Tandem Aza[4+2]/Allylboration

Chemistry : a European journal, 2003-01, Vol.9 (2), p.466-474

2003

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The Role of the Acidity of N‑Heteroaryl Sulfonamides as Inhibitors of Bcl‑2 Family Protein–Protein Interactions

ACS medicinal chemistry letters, 2013-02, Vol.4 (2), p.186-190

2013

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“Addition” and “Subtraction”: Selectivity Design for Type II Maternal Embryonic Leucine Zipper Kinase Inhibitors

Journal of medicinal chemistry, 2017-03, Vol.60 (5), p.2155-2161

2017

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Access to drug metabolites via C–H functionalization: copper-catalyzed aerobic oxidation of N,N-dimethylalkylamines in complex pharmaceuticals

Tetrahedron letters, 2015-06, Vol.56 (23), p.3066-3069

2015

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Optimization of 3‑Pyrimidin-4-yl-oxazolidin-2-ones as Allosteric and Mutant Specific Inhibitors of IDH1

ACS medicinal chemistry letters, 2017-02, Vol.8 (2), p.151-156

2017

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Die Erschließung von Wirkstoffmetaboliten durch übergangsmetallkatalysierte C-H-Oxidation: die Leber als Inspiration für die Synthese

Angewandte Chemie, 2016-11, Vol.128 (46), p.14430-14451

2016

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Synthesis of sterically hindered enamides via a Ti-mediated condensation of amides with aldehydes and ketones

Chemical communications (Cambridge, England), 2012-07, Vol.48 (53), p.6735-6737

2012

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Lipophilic Isosteres of a π–π Stacking Interaction: New Inhibitors of the Bcl-2-Bak Protein–Protein Interaction

ACS medicinal chemistry letters, 2012-07, Vol.3 (7), p.579-583

2012

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Mammalian Subtilisin/Kexin Isozyme SKI-1: A Widely Expressed Proprotein Convertase with a Unique Cleavage Specificity and Cellular Localization

Proceedings of the National Academy of Sciences - PNAS, 1999-02, Vol.96 (4), p.1321-1326

1999

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Design of a Nonreductive Method for Chemoselective Cleavage of Hydrazines in the Presence of Unsaturations: Application to a Stereoconvergent Three-Component Synthesis of (−)-Methyl Palustramate

Journal of organic chemistry, 2004-11, Vol.69 (24), p.8429-8436

2004

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Synthesis of sterically hindered enamides via a Ti-mediated condensation of amides with aldehydes and ketonesElectronic Supplementary Information (ESI) available. See DOI: 10.1039/c2cc32538a

2012-06

Volltextzugriff (PDF)

Die Erschließung von Wirkstoffmetaboliten durch übergangsmetallkatalysierte C‐H‐Oxidation: die Leber als Inspiration für die Synthese

Angewandte Chemie, 2016-11, Vol.128 (46), p.14430-14451

2016

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Multicomponent Reactions in the Total Synthesis of Natural Products

Multicomponent Reactions, 2005, p.342-397

2005

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Natural Product Synthesis Using Multicomponent Reaction Strategies

Accessing Drug Metabolites via Transition-Metal Catalyzed C−H Oxidation: The Liver as Synthetic Inspiration

C−H Bonds as Ubiquitous Functionality: A General Approach to Complex Arylated Imidazoles via Regioselective Sequential Arylation of All Three C−H Bonds and Regioselective N-Alkylation Enabled by SEM-Group Transposition

Toward the Validation of Maternal Embryonic Leucine Zipper Kinase: Discovery, Optimization of Highly Potent and Selective Inhibitors, and Preliminary Biology Insight

Three-Component Sequential Aza[4+2] Cycloaddition/Allylboration/Retro-Sulfinyl-Ene Reaction: A New Stereocontrolled Entry to Palustrine Alkaloids and Other 2,6-Disubstituted Piperidines

Complementation of Biotransformations with Chemical C–H Oxidation: Copper-Catalyzed Oxidation of Tertiary Amines in Complex Pharmaceuticals

Copper-Mediated N-Heteroarylation of Primary Sulfonamides: Synthesis of Mono-N-heteroaryl Sulfonamides

Identification of NVP-TNKS656: The Use of Structure–Efficiency Relationships To Generate a Highly Potent, Selective, and Orally Active Tankyrase Inhibitor

Catalytic C−H Arylation of SEM-Protected Azoles with Palladium Complexes of NHCs and Phosphines

RLY-4008, the First Highly Selective FGFR2 Inhibitor with Activity across FGFR2 Alterations and Resistance Mutations

Discovery of lirafugratinib (RLY-4008), a highly selective irreversible small-molecule inhibitor of FGFR2

Allosteric Mutant IDH1 Inhibitors Reveal Mechanisms for IDH1 Mutant and Isoform Selectivity

A Three-Component Reaction for Diversity-Oriented Synthesis of Polysubstituted Piperidines: Solution and Solid-Phase Optimization of the First Tandem Aza[4+2]/Allylboration

The Role of the Acidity of N‑Heteroaryl Sulfonamides as Inhibitors of Bcl‑2 Family Protein–Protein Interactions

“Addition” and “Subtraction”: Selectivity Design for Type II Maternal Embryonic Leucine Zipper Kinase Inhibitors

Access to drug metabolites via C–H functionalization: copper-catalyzed aerobic oxidation of N,N-dimethylalkylamines in complex pharmaceuticals

Optimization of 3‑Pyrimidin-4-yl-oxazolidin-2-ones as Allosteric and Mutant Specific Inhibitors of IDH1

Die Erschließung von Wirkstoffmetaboliten durch übergangsmetallkatalysierte C-H-Oxidation: die Leber als Inspiration für die Synthese

Synthesis of sterically hindered enamides via a Ti-mediated condensation of amides with aldehydes and ketones

Lipophilic Isosteres of a π–π Stacking Interaction: New Inhibitors of the Bcl-2-Bak Protein–Protein Interaction

Mammalian Subtilisin/Kexin Isozyme SKI-1: A Widely Expressed Proprotein Convertase with a Unique Cleavage Specificity and Cellular Localization

Design of a Nonreductive Method for Chemoselective Cleavage of Hydrazines in the Presence of Unsaturations: Application to a Stereoconvergent Three-Component Synthesis of (−)-Methyl Palustramate

Synthesis of sterically hindered enamides via a Ti-mediated condensation of amides with aldehydes and ketonesElectronic Supplementary Information (ESI) available. See DOI: 10.1039/c2cc32538a

Die Erschließung von Wirkstoffmetaboliten durch übergangsmetallkatalysierte C‐H‐Oxidation: die Leber als Inspiration für die Synthese

Multicomponent Reactions in the Total Synthesis of Natural Products

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