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Identification of inhibitors of an unconventional Trypanosoma brucei kinetochore kinase

PloS one, 2019-05, Vol.14 (5), p.e0217828

2019

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Biochemical and genetic characterization of Trypanosoma cruzi N-myristoyltransferase

Biochemical journal, 2014-04, Vol.459 (2), p.323-332

2014

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Lead Optimization of a Pyrazole Sulfonamide Series of Trypanosoma brucei N‑Myristoyltransferase Inhibitors: Identification and Evaluation of CNS Penetrant Compounds as Potential Treatments for Stage 2 Human African Trypanosomiasis

Journal of medicinal chemistry, 2014-12, Vol.57 (23), p.9855-9869

2014

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IspE inhibitors identified by a combination of in silico and in vitro high-throughput screening

PloS one, 2012-04, Vol.7 (4), p.e35792-e35792

2012

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Anti-trypanosomatid drug discovery: an ongoing challenge and a continuing need

Nature reviews. Microbiology, 2017-04, Vol.15 (4), p.217-231

2017

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Resolution of the insect ouabain paradox

Proceedings of the National Academy of Sciences - PNAS, 2004-09, Vol.101 (37), p.13689-13693

2004

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A Molecular Hybridization Approach for the Design of Potent, Highly Selective, and Brain-Penetrant N‑Myristoyltransferase Inhibitors

Journal of medicinal chemistry, 2018-09, Vol.61 (18), p.8374-8389

2018

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Identification of Novel Trypanosoma cruzi Proteasome Inhibitors Using a Luminescence-Based High-Throughput Screening Assay

Antimicrobial agents and chemotherapy, 2019-09, Vol.63 (9)

2019

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Identification of a Proteasome-Targeting Arylsulfonamide with Potential for the Treatment of Chagas' Disease

Antimicrobial agents and chemotherapy, 2022-01, Vol.66 (1), p.e0153521-e0153521

2022

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Trypanosoma cruzi Phosphomannomutase and Guanosine Diphosphate-Mannose Pyrophosphorylase Ligandability Assessment

Antimicrobial agents and chemotherapy, 2019-10, Vol.63 (10)

2019

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Burkholderia pseudomallei d‐alanine‐d‐alanine ligase; detailed characterisation and assessment of a potential antibiotic drug target

The FEBS journal, 2019-11, Vol.286 (22), p.4509-4524

2019

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Anti-trypanosomatid drug discovery: an ongoing challenge and a continuing need

Nature reviews. Microbiology, 2017-07, Vol.15 (7), p.447-447

2017

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Design and Synthesis of Brain Penetrant Trypanocidal N‑Myristoyltransferase Inhibitors

Journal of medicinal chemistry, 2017-12, Vol.60 (23), p.9790-9806

2017

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Pharmacological Validation of N‑Myristoyltransferase as a Drug Target in Leishmania donovani

ACS infectious diseases, 2019-01, Vol.5 (1), p.111-122

2019

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Discovery of a Novel Class of Orally Active Trypanocidal N-Myristoyltransferase Inhibitors

Journal of medicinal chemistry, 2012-01, Vol.55 (1), p.140-152

2012

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Toolkit of Approaches To Support Target-Focused Drug Discovery for Plasmodium falciparum Lysyl tRNA Synthetase

ACS infectious diseases, 2022-09, Vol.8 (9), p.1962-1974

2022

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Author Correction: Anti-trypanosomatid drug discovery: an ongoing challenge and a continuing need

Nature reviews. Microbiology, 2018-11, Vol.16 (11), p.714-714

2018

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N‑Myristoyltransferase Is a Cell Wall Target in Aspergillus fumigatus

ACS chemical biology, 2015-06, Vol.10 (6), p.1425-1434

2015

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Chemical Validation of Trypanothione Synthetase: A POTENTIAL DRUG TARGET FOR HUMAN TRYPANOSOMIASIS

The Journal of biological chemistry, 2009-12, Vol.284 (52), p.36137-36145

2009

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Allosteric Competitive Inhibitors of the Glucose-1-phosphate Thymidylyltransferase (RmlA) from Pseudomonas aeruginosa

ACS chemical biology, 2013-02, Vol.8 (2), p.387-396

2013

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Development of Small-Molecule Trypanosoma brucei N-Myristoyltransferase Inhibitors: Discovery and Optimisation of a Novel Binding Mode

ChemMedChem, 2015-11, Vol.10 (11), p.1821-1836

2015

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Discovery of an Allosteric Binding Site in Kinetoplastid Methionyl-tRNA Synthetase

ACS infectious diseases, 2020-05, Vol.6 (5), p.1044-1057

2020

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Design, Synthesis and Biological Evaluation of Trypanosoma brucei Trypanothione Synthetase Inhibitors

ChemMedChem, 2012-01, Vol.7 (1), p.95-106

2012

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Chemical Validation of Methionyl-tRNA Synthetase as a Druggable Target in Leishmania donovani

ACS infectious diseases, 2017-10, Vol.3 (10), p.718-727

2017

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Lead Optimization of a Pyrazole Sulfonamide Series of Trypanosoma bruceiN-Myristoyltransferase Inhibitors: Identification and Evaluation of CNS Penetrant Compounds as Potential Treatments for Stage 2 Human African Trypanosomiasis

Journal of medicinal chemistry, 2014-11, Vol.57 (23), p.9855-9869

2014

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Identification of inhibitors of an unconventional Trypanosoma brucei kinetochore kinase

Biochemical and genetic characterization of Trypanosoma cruzi N-myristoyltransferase

Lead Optimization of a Pyrazole Sulfonamide Series of Trypanosoma brucei N‑Myristoyltransferase Inhibitors: Identification and Evaluation of CNS Penetrant Compounds as Potential Treatments for Stage 2 Human African Trypanosomiasis

IspE inhibitors identified by a combination of in silico and in vitro high-throughput screening

Anti-trypanosomatid drug discovery: an ongoing challenge and a continuing need

Resolution of the insect ouabain paradox

A Molecular Hybridization Approach for the Design of Potent, Highly Selective, and Brain-Penetrant N‑Myristoyltransferase Inhibitors

Identification of Novel Trypanosoma cruzi Proteasome Inhibitors Using a Luminescence-Based High-Throughput Screening Assay

Identification of a Proteasome-Targeting Arylsulfonamide with Potential for the Treatment of Chagas' Disease

Trypanosoma cruzi Phosphomannomutase and Guanosine Diphosphate-Mannose Pyrophosphorylase Ligandability Assessment

Burkholderia pseudomallei d‐alanine‐d‐alanine ligase; detailed characterisation and assessment of a potential antibiotic drug target

Anti-trypanosomatid drug discovery: an ongoing challenge and a continuing need

Design and Synthesis of Brain Penetrant Trypanocidal N‑Myristoyltransferase Inhibitors

Pharmacological Validation of N‑Myristoyltransferase as a Drug Target in Leishmania donovani

Discovery of a Novel Class of Orally Active Trypanocidal N-Myristoyltransferase Inhibitors

Toolkit of Approaches To Support Target-Focused Drug Discovery for Plasmodium falciparum Lysyl tRNA Synthetase

Author Correction: Anti-trypanosomatid drug discovery: an ongoing challenge and a continuing need

N‑Myristoyltransferase Is a Cell Wall Target in Aspergillus fumigatus

Chemical Validation of Trypanothione Synthetase: A POTENTIAL DRUG TARGET FOR HUMAN TRYPANOSOMIASIS

Allosteric Competitive Inhibitors of the Glucose-1-phosphate Thymidylyltransferase (RmlA) from Pseudomonas aeruginosa

Development of Small-Molecule Trypanosoma brucei N-Myristoyltransferase Inhibitors: Discovery and Optimisation of a Novel Binding Mode

Discovery of an Allosteric Binding Site in Kinetoplastid Methionyl-tRNA Synthetase

Design, Synthesis and Biological Evaluation of Trypanosoma brucei Trypanothione Synthetase Inhibitors

Chemical Validation of Methionyl-tRNA Synthetase as a Druggable Target in Leishmania donovani

Lead Optimization of a Pyrazole Sulfonamide Series of Trypanosoma bruceiN-Myristoyltransferase Inhibitors: Identification and Evaluation of CNS Penetrant Compounds as Potential Treatments for Stage 2 Human African Trypanosomiasis

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