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Identification of N‑{cis-3-[Methyl(7H‑pyrrolo[2,3‑d]pyrimidin-4-yl)amino]cyclobutyl}propane-1-sulfonamide (PF-04965842): A Selective JAK1 Clinical Candidate for the Treatment of Autoimmune Diseases

Journal of medicinal chemistry, 2018-02, Vol.61 (3), p.1130-1152

2018

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Structural and Thermodynamic Characterization of the TYK2 and JAK3 Kinase Domains in Complex with CP-690550 and CMP-6

Journal of molecular biology, 2010-07, Vol.400 (3), p.413-433

2010

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Potent and selective isophthalamide S2 hydroxyethylamine inhibitors of BACE1

Bioorganic & medicinal chemistry letters, 2007-06, Vol.17 (12), p.3378-3383

2007

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(S)-(−)-4-[4-[2-(Isochroman-1-yl)ethyl]piperazin-1-yl]benzenesulfonamide, a Selective Dopamine D4 Antagonist

Journal of medicinal chemistry, 1996-06, Vol.39 (13), p.2435-2437

1996

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Discovery of novel spirocyclic inhibitors of fatty acid amide hydrolase (FAAH). Part 1: Identification of 7-azaspiro[3.5]nonane and 1-oxa-8-azaspiro[4.5]decane as lead scaffolds

Bioorganic & medicinal chemistry letters, 2011-11, Vol.21 (21), p.6538-6544

2011

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Thienopyrimidine-based P2Y12 platelet aggregation inhibitors

Bioorganic & medicinal chemistry letters, 2009-10, Vol.19 (20), p.5919-5923

2009

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Structure based design of novel irreversible FAAH inhibitors

Bioorganic & medicinal chemistry letters, 2009-10, Vol.19 (20), p.5970-5974

2009

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Antagonist, Partial Agonist, and Full Agonist Imidazo[1,5-a]quinoxaline Amides and Carbamates Acting through the GABAA/Benzodiazepine Receptor

Journal of medicinal chemistry, 1994-03, Vol.37 (6), p.758-768

1994

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High-Affinity Partial Agonist Imidazo[1,5-a]quinoxaline Amides, Carbamates, and Ureas at the γ-Aminobutyric Acid A/Benzodiazepine Receptor Complex

Journal of medicinal chemistry, 1996-01, Vol.39 (1), p.158-175

1996

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Potent and selective isophthalamide S 2 hydroxyethylamine inhibitors of BACE1

Bioorganic & medicinal chemistry letters, 2007-06, Vol.17 (12), p.3378-3383

2007

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A method for the preparation of stereochemically defined .psi.[CH2O] pseudodipeptides

Journal of organic chemistry, 1987-02, Vol.52 (3), p.418-422

TenBrink, Ruth E

1987

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Piperazine Imidazo[1,5-a]quinoxaline Ureas as High-Affinity GABAA Ligands of Dual Functionality

Journal of medicinal chemistry, 1999-04, Vol.42 (7), p.1123-1144

1999

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Inhibitors of the protease from human immunodeficiency virus: synthesis, enzyme inhibition, and antiviral activity of a series of compounds containing the dihydroxyethylene transition-state isostere

Journal of medicinal chemistry, 1993-04, Vol.36 (8), p.941-952

1993

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Thienopyrimidine-based P2Y sub(12) platelet aggregation inhibitors

Bioorganic & medicinal chemistry letters, 2009-10, Vol.19 (20), p.5919-5923

2009

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Differential pharmacology between the guinea‐pig and the gorilla 5‐HT 1D receptor as probed with isochromans (5‐HT 1D ‐selective ligands)

British journal of pharmacology, 2009-01, Vol.127 (2), p.468-472

2009

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1-[(Ethoxyamino)methyl]-1,3,4,5-tetrahydro-7,8-dimethoxy-2-benzoxepins: a new class of antianaphylactic agents

Journal of medicinal chemistry, 1980-09, Vol.23 (9), p.1058-1060

1980

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Thienopyrimidine-based P2Y 12 platelet aggregation inhibitors

Bioorganic & medicinal chemistry letters, 2009, Vol.19 (20), p.5919-5923

2009

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Piperazine Imidazo[1,5- a ]quinoxaline Ureas as High-Affinity GABA A Ligands of Dual Functionality

Journal of medicinal chemistry, 1999-04, Vol.42 (7), p.1123-1144

1999

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Potent and selective isophthalamide S sub(2) hydroxyethylamine inhibitors of BACE1

Bioorganic & medicinal chemistry letters, 2007-06, Vol.17 (12), p.3378-3383

2007

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Pharmacological characterization of U-101387, a dopamine D4 receptor selective antagonist

The Journal of pharmacology and experimental therapeutics, 1996-12, Vol.279 (3), p.1392

1996

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( S )-(−)-4-[4-[2-(Isochroman-1-yl)ethyl]piperazin-1-yl]benzenesulfonamide, a Selective Dopamine D 4 Antagonist

Journal of medicinal chemistry, 1996-06, Vol.39 (13), p.2435-2437

1996

Volltextzugriff (PDF)

Differential pharmacology between the guinea‐pig and the gorilla 5‐HT1D receptor as probed with isochromans (5‐HT1D‐selective ligands)

British journal of pharmacology, 1999-05, Vol.127 (2), p.468-472

1999

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Tetrahydro-2-benzoxepins: a novel family of hypotensives

Journal of medicinal chemistry, 1981-01, Vol.24 (1), p.64-67

1981

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Hypobetalipoproteinemic agents. 2. Compounds related to 4-(1-adamantyloxy)aniline

Journal of medicinal chemistry, 1979-01, Vol.22 (1), p.69-77

1979

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Hypo-.beta.-lipoproteinemic agents. 1. Bicyclo[2.2.2]octyloxyaniline and its derivatives

Journal of medicinal chemistry, 1975-11, Vol.18 (11), p.1065-1070

1975

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Identification of N‑{cis-3-[Methyl(7H‑pyrrolo[2,3‑d]pyrimidin-4-yl)amino]cyclobutyl}propane-1-sulfonamide (PF-04965842): A Selective JAK1 Clinical Candidate for the Treatment of Autoimmune Diseases

Structural and Thermodynamic Characterization of the TYK2 and JAK3 Kinase Domains in Complex with CP-690550 and CMP-6

Potent and selective isophthalamide S2 hydroxyethylamine inhibitors of BACE1

(S)-(−)-4-[4-[2-(Isochroman-1-yl)ethyl]piperazin-1-yl]benzenesulfonamide, a Selective Dopamine D4 Antagonist

Discovery of novel spirocyclic inhibitors of fatty acid amide hydrolase (FAAH). Part 1: Identification of 7-azaspiro[3.5]nonane and 1-oxa-8-azaspiro[4.5]decane as lead scaffolds

Thienopyrimidine-based P2Y12 platelet aggregation inhibitors

Structure based design of novel irreversible FAAH inhibitors

Antagonist, Partial Agonist, and Full Agonist Imidazo[1,5-a]quinoxaline Amides and Carbamates Acting through the GABAA/Benzodiazepine Receptor

High-Affinity Partial Agonist Imidazo[1,5-a]quinoxaline Amides, Carbamates, and Ureas at the γ-Aminobutyric Acid A/Benzodiazepine Receptor Complex

Potent and selective isophthalamide S 2 hydroxyethylamine inhibitors of BACE1

A method for the preparation of stereochemically defined .psi.[CH2O] pseudodipeptides

Piperazine Imidazo[1,5-a]quinoxaline Ureas as High-Affinity GABAA Ligands of Dual Functionality

Inhibitors of the protease from human immunodeficiency virus: synthesis, enzyme inhibition, and antiviral activity of a series of compounds containing the dihydroxyethylene transition-state isostere

Thienopyrimidine-based P2Y sub(12) platelet aggregation inhibitors

Differential pharmacology between the guinea‐pig and the gorilla 5‐HT 1D receptor as probed with isochromans (5‐HT 1D ‐selective ligands)

1-[(Ethoxyamino)methyl]-1,3,4,5-tetrahydro-7,8-dimethoxy-2-benzoxepins: a new class of antianaphylactic agents

Thienopyrimidine-based P2Y 12 platelet aggregation inhibitors

Piperazine Imidazo[1,5- a ]quinoxaline Ureas as High-Affinity GABA A Ligands of Dual Functionality

Potent and selective isophthalamide S sub(2) hydroxyethylamine inhibitors of BACE1

Pharmacological characterization of U-101387, a dopamine D4 receptor selective antagonist

( S )-(−)-4-[4-[2-(Isochroman-1-yl)ethyl]piperazin-1-yl]benzenesulfonamide, a Selective Dopamine D 4 Antagonist

Differential pharmacology between the guinea‐pig and the gorilla 5‐HT1D receptor as probed with isochromans (5‐HT1D‐selective ligands)

Tetrahydro-2-benzoxepins: a novel family of hypotensives

Hypobetalipoproteinemic agents. 2. Compounds related to 4-(1-adamantyloxy)aniline

Hypo-.beta.-lipoproteinemic agents. 1. Bicyclo[2.2.2]octyloxyaniline and its derivatives

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