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Nelotanserin, a novel selective human 5-hydroxytryptamine2A inverse agonist for the treatment of insomnia

The Journal of pharmacology and experimental therapeutics, 2010-01, Vol.332 (1), p.281

2010

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APD791, 3-methoxy-n-(3-(1-methyl-1h-pyrazol-5-yl)-4-(2-morpholinoethoxy)phenyl)benzamide, a novel 5-hydroxytryptamine 2A receptor antagonist: pharmacological profile, pharmacokinetics, platelet activity and vascular biology

The Journal of pharmacology and experimental therapeutics, 2009-10, Vol.331 (1), p.96

2009

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An improved synthesis of 1,2,9,9a-tetrahydrocyclopropa[c]benz[e]indol-4-one (CBI): a simplified analog of the CC-1065 alkylation subunit

Journal of organic chemistry, 1992-05, Vol.57 (10), p.2873-2876

1992

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Synthesis and in vivo evaluation of phenethylpiperazine amides: selective 5-hydroxytryptamine(2A) receptor antagonists for the treatment of insomnia

Journal of medicinal chemistry, 2010-08, Vol.53 (15), p.5696-5706

2010

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Discovery and Structure−Activity Relationship of 3-Methoxy-N-(3-(1-methyl-1H-pyrazol-5-yl)-4-(2-morpholinoethoxy)phenyl)benzamide (APD791): A Highly Selective 5-Hydroxytryptamine2A Receptor Inverse Agonist for the Treatment of Arterial Thrombosis

Journal of medicinal chemistry, 2010-06, Vol.53 (11), p.4412-4421

2010

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Anti-thrombotic and vascular effects of AR246686, a novel 5-HT2A receptor antagonist

European journal of pharmacology, 2008-05, Vol.586 (1-3), p.234-243

2008

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Synthesis and in Vivo Evaluation of Phenethylpiperazine Amides: Selective 5-Hydroxytryptamine2A Receptor Antagonists for the Treatment of Insomnia

Journal of medicinal chemistry, 2010-08, Vol.53 (15), p.5696-5706

2010

Volltextzugriff (PDF)

Solubilized phenyl-pyrazole ureas as potent, selective 5-HT2A inverse-agonists and their application as antiplatelet agents

Bioorganic & medicinal chemistry letters, 2009-09, Vol.19 (18), p.5486-5489

2009

Volltextzugriff (PDF)

Synthesis and SAR of N-benzoyl-L-biphenylalanine derivatives: Discovery of TR-14035, a dual α4β7/α4β1 integrin antagonist

Bioorganic & medicinal chemistry, 2002, Vol.10 (6), p.2051-2066

2002

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S-Adenosyl-L-homocysteine hydrolase inhibitor mediates immunosuppressive effects in vivo: suppression of delayed type hypersensitivity ear swelling and peptidoglycan polysaccharide-induced arthritis

The Journal of pharmacology and experimental therapeutics, 2001-01, Vol.296 (1), p.106

2001

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Vancomycin and ristocetin models: synthesis via the Ullmann macrocyclization reaction

Journal of organic chemistry, 1993-03, Vol.58 (6), p.1425-1433

1993

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p-Quinonemethide Analog of the CC-1065 and Duocarmycin Alkylation Subunits

Journal of organic chemistry, 1994-08, Vol.59 (17), p.4943-4949

1994

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Synthesis of .alpha.-methyl 1',2'-dideoxycellobioside: a novel C-disaccharide

Journal of organic chemistry, 1992-01, Vol.57 (3), p.915-922

1992

Volltextzugriff (PDF)

Discovery of 1-[3-(4-Bromo-2-methyl-2 H -pyrazol-3-yl)-4-methoxyphenyl]-3-(2,4-difluorophenyl)urea (Nelotanserin) and Related 5-Hydroxytryptamine 2A Inverse Agonists for the Treatment of Insomnia

Journal of medicinal chemistry, 2010-03, Vol.53 (5), p.1923-1936

2010

Volltextzugriff (PDF)

Synthesis and SAR of N-benzoyl-L-biphenylalanine derivatives: discovery of TR-14035, a dual alpha(4)beta(7)/alpha(4)beta(1) integrin antagonist

Bioorganic & medicinal chemistry, 2002-06, Vol.10 (6), p.2051

2002

Volltextzugriff (PDF)

Synthesis and in Vivo Evaluation of Phenethylpiperazine Amides: Selective 5-Hydroxytryptamine 2A Receptor Antagonists for the Treatment of Insomnia

Journal of medicinal chemistry, 2010-08, Vol.53 (15), p.5696-5706

2010

Volltextzugriff (PDF)

Discovery of 1-[3-(4-Bromo-2-methyl-2H-pyrazol-3-yl)-4-methoxyphenyl]-3-(2,4-difluorophenyl)urea (Nelotanserin) and Related 5-Hydroxytryptamine2A Inverse Agonists for the Treatment of Insomnia

Journal of medicinal chemistry, 2010-03, Vol.53 (5), p.1923-1936

2010

Volltextzugriff (PDF)

Solubilized phenyl-pyrazole ureas as potent, selective 5-HT sub(2A) inverse-agonists and their application as antiplatelet agents

Bioorganic & medicinal chemistry letters, 2009-09, Vol.19 (18), p.5486-5489

2009

Volltextzugriff (PDF)

Solubilized phenyl-pyrazole ureas as potent, selective 5-HT 2A inverse-agonists and their application as antiplatelet agents

Bioorganic & medicinal chemistry letters, 2009, Vol.19 (18), p.5486-5489

2009

Volltextzugriff (PDF)

Anti-thrombotic and vascular effects of AR246686, a novel 5-HT 2A receptor antagonist

European journal of pharmacology, 2008, Vol.586 (1), p.234-243

2008

Volltextzugriff (PDF)

Solubilized phenyl-pyrazole ureas as potent, selective 5-HT(2A) inverse-agonists and their application as antiplatelet agents

Bioorganic & medicinal chemistry letters, 2009-09, Vol.19 (18), p.5486-5489

2009

Volltextzugriff (PDF)

Synthesis and SAR of N-Benzoyl- l-Biphenylalanine Derivatives: Discovery of TR-14035, A Dual α 4β 7/α 4β 1 Integrin Antagonist

Bioorganic & medicinal chemistry, 2002, Vol.10 (6), p.2051-2066

2002

Volltextzugriff (PDF)

5-HT(2A) inverse-agonists for the treatment of insomnia

Current topics in medicinal chemistry, 2008, Vol.8 (11), p.969

2008

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High-energy spectral breaks in gamma-ray bursts

The Astrophysical journal, 1992-07, Vol.393 (2, Ju), p.L51-L54

1992

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Nelotanserin, a novel selective human 5-hydroxytryptamine2A inverse agonist for the treatment of insomnia

APD791, 3-methoxy-n-(3-(1-methyl-1h-pyrazol-5-yl)-4-(2-morpholinoethoxy)phenyl)benzamide, a novel 5-hydroxytryptamine 2A receptor antagonist: pharmacological profile, pharmacokinetics, platelet activity and vascular biology

An improved synthesis of 1,2,9,9a-tetrahydrocyclopropa[c]benz[e]indol-4-one (CBI): a simplified analog of the CC-1065 alkylation subunit

Synthesis and in vivo evaluation of phenethylpiperazine amides: selective 5-hydroxytryptamine(2A) receptor antagonists for the treatment of insomnia

Discovery and Structure−Activity Relationship of 3-Methoxy-N-(3-(1-methyl-1H-pyrazol-5-yl)-4-(2-morpholinoethoxy)phenyl)benzamide (APD791): A Highly Selective 5-Hydroxytryptamine2A Receptor Inverse Agonist for the Treatment of Arterial Thrombosis

Anti-thrombotic and vascular effects of AR246686, a novel 5-HT2A receptor antagonist

Synthesis and in Vivo Evaluation of Phenethylpiperazine Amides: Selective 5-Hydroxytryptamine2A Receptor Antagonists for the Treatment of Insomnia

Solubilized phenyl-pyrazole ureas as potent, selective 5-HT2A inverse-agonists and their application as antiplatelet agents

Synthesis and SAR of N-benzoyl-L-biphenylalanine derivatives: Discovery of TR-14035, a dual α4β7/α4β1 integrin antagonist

S-Adenosyl-L-homocysteine hydrolase inhibitor mediates immunosuppressive effects in vivo: suppression of delayed type hypersensitivity ear swelling and peptidoglycan polysaccharide-induced arthritis

Vancomycin and ristocetin models: synthesis via the Ullmann macrocyclization reaction

p-Quinonemethide Analog of the CC-1065 and Duocarmycin Alkylation Subunits

Synthesis of .alpha.-methyl 1',2'-dideoxycellobioside: a novel C-disaccharide

Discovery of 1-[3-(4-Bromo-2-methyl-2 H -pyrazol-3-yl)-4-methoxyphenyl]-3-(2,4-difluorophenyl)urea (Nelotanserin) and Related 5-Hydroxytryptamine 2A Inverse Agonists for the Treatment of Insomnia

Synthesis and SAR of N-benzoyl-L-biphenylalanine derivatives: discovery of TR-14035, a dual alpha(4)beta(7)/alpha(4)beta(1) integrin antagonist

Synthesis and in Vivo Evaluation of Phenethylpiperazine Amides: Selective 5-Hydroxytryptamine 2A Receptor Antagonists for the Treatment of Insomnia

Discovery and Structure−Activity Relationship of 3-Methoxy- N -(3-(1-methyl-1 H -pyrazol-5-yl)-4-(2-morpholinoethoxy)phenyl)benzamide (APD791): A Highly Selective 5-Hydroxytryptamine 2A Receptor Inverse Agonist for the Treatment of Arterial Thrombosis

Discovery of 1-[3-(4-Bromo-2-methyl-2H-pyrazol-3-yl)-4-methoxyphenyl]-3-(2,4-difluorophenyl)urea (Nelotanserin) and Related 5-Hydroxytryptamine2A Inverse Agonists for the Treatment of Insomnia

Solubilized phenyl-pyrazole ureas as potent, selective 5-HT sub(2A) inverse-agonists and their application as antiplatelet agents

Solubilized phenyl-pyrazole ureas as potent, selective 5-HT 2A inverse-agonists and their application as antiplatelet agents

Anti-thrombotic and vascular effects of AR246686, a novel 5-HT 2A receptor antagonist

Solubilized phenyl-pyrazole ureas as potent, selective 5-HT(2A) inverse-agonists and their application as antiplatelet agents

Synthesis and SAR of N-Benzoyl- l-Biphenylalanine Derivatives: Discovery of TR-14035, A Dual α 4β 7/α 4β 1 Integrin Antagonist

5-HT(2A) inverse-agonists for the treatment of insomnia

High-energy spectral breaks in gamma-ray bursts

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