UB Paderborn / Katalog / Suche / in CDI

1 – 25 von 482

Sortiert nach

Brain Penetrable Histone Deacetylase 6 Inhibitor SW-100 Ameliorates Memory and Learning Impairments in a Mouse Model of Fragile X Syndrome

ACS chemical neuroscience, 2019-03, Vol.10 (3), p.1679-1695

2019

Volltextzugriff (PDF)

Mercaptoacetamide: A promising zinc-binding group for the discovery of selective histone deacetylase 6 inhibitors

European journal of medicinal chemistry, 2021-01, Vol.209, p.112887-112887, Article 112887

2021

Volltextzugriff (PDF)

Tetrahydroquinoline-Capped Histone Deacetylase 6 Inhibitor SW-101 Ameliorates Pathological Phenotypes in a Charcot–Marie–Tooth Type 2A Mouse Model

Journal of medicinal chemistry, 2021-04, Vol.64 (8), p.4810-4840

2021

Volltextzugriff (PDF)

Rational Design of Suprastat: A Novel Selective Histone Deacetylase 6 Inhibitor with the Ability to Potentiate Immunotherapy in Melanoma Models

Journal of medicinal chemistry, 2020-09, Vol.63 (18), p.10246-10262

2020

Volltextzugriff (PDF)

Evaluation of Protein Kinase Inhibitors with PLK4 Cross-Over Potential in a Pre-Clinical Model of Cancer

International journal of molecular sciences, 2019-04, Vol.20 (9), p.2112

2019

Volltextzugriff (PDF)

Recent innovative advances in the discovery of selective HDAC6 inhibitors

Future medicinal chemistry, 2021-06, Vol.13 (12), p.1017-1019

2021

Volltextzugriff (PDF)

Synthesis and Pharmacological Evaluation of Selective Histone Deacetylase 6 Inhibitors in Melanoma Models

ACS medicinal chemistry letters, 2017-10, Vol.8 (10), p.1031-1036

2017

Volltextzugriff (PDF)

HDAC specificity and kinase off-targeting by purine-benzohydroxamate anti-hematological tumor agents

European journal of medicinal chemistry, 2024-01, Vol.263, p.115935-115935, Article 115935

2024

Volltextzugriff (PDF)

1,3-Diphenylureido hydroxamate as a promising scaffold for generation of potent antimalarial histone deacetylase inhibitors

Scientific reports, 2023-11, Vol.13 (1), p.21006-21006, Article 21006

2023

Volltextzugriff (PDF)

N -[(1,3-Benzodioxol-5-yl)methyl]benzenesulfonamide: an analogue of capsaicin

Acta crystallographica. Section E, Structure reports online, 2013-11, Vol.69 (11), p.o1700-o1700

2013

Volltextzugriff (PDF)

N -[(1,3-Benzodioxol-5-yl)methyl]-4-methylbenzamide: an analogue of capsaicin

Acta crystallographica. Section E, Structure reports online, 2013-03, Vol.69 (3), p.o332-o332

2013

Volltextzugriff (PDF)

Using an in Silico Approach To Teach 3D Pharmacodynamics of the Drug–Target Interaction Process Focusing on Selective COX2 Inhibition by Celecoxib

Journal of chemical education, 2017-03, Vol.94 (3), p.380-387

2017

Volltextzugriff (PDF)

Synthesis, Molecular Modeling, and Evaluation of Novel Sulfonylhydrazones as Acetylcholinesterase Inhibitors for Alzheimer's Disease

Archiv der Pharmazie (Weinheim), 2017-11, Vol.350 (11), p.n/a

2017

Volltextzugriff (PDF)

Toward chelerythrine optimization: Analogues designed by molecular simplification exhibit selective growth inhibition in non-small-cell lung cancer cells

Bioorganic & medicinal chemistry, 2016-10, Vol.24 (19), p.4600-4610

2016

Volltextzugriff (PDF)

Environmentally Safe Condition for the Synthesis of Aryl and Alkyl Sulfonyl Hydrazones via One-Pot Reaction

ACS sustainable chemistry & engineering, 2016-04, Vol.4 (4), p.1899-1905

2016

Volltextzugriff (PDF)

Discovery of a New Isoxazole-3-hydroxamate-Based Histone Deacetylase 6 Inhibitor SS-208 with Antitumor Activity in Syngeneic Melanoma Mouse Models

Journal of medicinal chemistry, 2019-09, Vol.62 (18), p.8557-8577

2019

Volltextzugriff (PDF)

Novel Capsaicin Analogues as Potential Anticancer Agents: Synthesis, Biological Evaluation, and In Silico Approach

Archiv der Pharmazie (Weinheim), 2014-12, Vol.347 (12), p.885-895

2014

Volltextzugriff (PDF)

Correction to “Rational Design, Synthesis, and Mechanism of (3S,4R)‑3-Amino-4-(difluoromethyl)cyclopent-1-ene-1-carboxylic Acid: Employing a Second-Deprotonation Strategy for Selectivity of Human Ornithine Aminotransferase over GABA Aminotransferase”

Journal of the American Chemical Society, 2023-05, Vol.145 (17), p.9895-9896

2023

Volltextzugriff (PDF)

Turnover and Inactivation Mechanisms for (S)‑3-Amino-4,4-difluorocyclopent-1-enecarboxylic Acid, a Selective Mechanism-Based Inactivator of Human Ornithine Aminotransferase

Journal of the American Chemical Society, 2021-06, Vol.143 (23), p.8689-8703

2021

Volltextzugriff (PDF)

Synthesis, characterization, in silico approach and in vitro antiproliferative activity of RPF151, a benzodioxole sulfonamide analogue designed from capsaicin scaffold

Journal of molecular structure, 2015-05, Vol.1088, p.138-146

2015

Volltextzugriff (PDF)

N-[(1,3-Benzodioxol-5-yl)meth-yl]benzene-sulfonamide: an analogue of capsaicin

Acta crystallographica. Section E, Structure reports online, 2013-10, Vol.69 (Pt 11), p.o1700-o1700

2013

Volltextzugriff (PDF)

N-[(1,3-Benzodioxol-5-yl)meth-yl]-4-methyl-benzamide: an analogue of capsaicin

Acta crystallographica. Section E, Structure reports online, 2013-03, Vol.69 (Pt 3), p.o332-o332

2013

Volltextzugriff (PDF)

Rational Design, Synthesis, and Mechanism of (3S,4R)-3-Amino-4-(difluoromethyl)cyclopent-1-ene-1-carboxylic Acid Employing a Second-Deprotonation Strategy for Selectivity of Human Ornithine Aminotransferase over γ-Aminobutyric Acid Aminotransferase

Journal of the American Chemical Society, 2022-03, Vol.144 (12), p.5629-5642

2022

Volltextzugriff (PDF)

An overall estimation of losses caused by diseases in the Brazilian fish farms

Journal of parasitic diseases, 2017-12, Vol.41 (4), p.913-918

2017

Volltextzugriff (PDF)

Multi-Spectroscopic and Theoretical Analysis on the Interaction between Human Serum Albumin and a Capsaicin Derivative-RPF101

Biomolecules (Basel, Switzerland), 2018-08, Vol.8 (3), p.78

2018

Volltextzugriff (PDF)

1 – 25 von 482

Suche als RSS-Feed

Suchergebnisse filtern

Filter anzeigen

Nur zeigen

Geprüft (Peer-Review)
(402)
Mit Volltextzugriff
(453)

Publikationsform

1 weiteren anzeigen...

Weniger anzeigen...

Sprache

3 weitere anzeigen...

Weniger anzeigen...

Erscheinungsjahr

n.n

Thema

15 weitere anzeigen...

Weniger anzeigen...

Neu hinzugefügt

... seit 30 Tagen
(1)
... seit 90 Tagen
(12)

Menü

Weitere Dienste

Einstellungen

Brain Penetrable Histone Deacetylase 6 Inhibitor SW-100 Ameliorates Memory and Learning Impairments in a Mouse Model of Fragile X Syndrome

Mercaptoacetamide: A promising zinc-binding group for the discovery of selective histone deacetylase 6 inhibitors

Tetrahydroquinoline-Capped Histone Deacetylase 6 Inhibitor SW-101 Ameliorates Pathological Phenotypes in a Charcot–Marie–Tooth Type 2A Mouse Model

Rational Design of Suprastat: A Novel Selective Histone Deacetylase 6 Inhibitor with the Ability to Potentiate Immunotherapy in Melanoma Models

Evaluation of Protein Kinase Inhibitors with PLK4 Cross-Over Potential in a Pre-Clinical Model of Cancer

Recent innovative advances in the discovery of selective HDAC6 inhibitors

Synthesis and Pharmacological Evaluation of Selective Histone Deacetylase 6 Inhibitors in Melanoma Models

HDAC specificity and kinase off-targeting by purine-benzohydroxamate anti-hematological tumor agents

1,3-Diphenylureido hydroxamate as a promising scaffold for generation of potent antimalarial histone deacetylase inhibitors

N -[(1,3-Benzodioxol-5-yl)methyl]benzenesulfonamide: an analogue of capsaicin

N -[(1,3-Benzodioxol-5-yl)methyl]-4-methylbenzamide: an analogue of capsaicin

Using an in Silico Approach To Teach 3D Pharmacodynamics of the Drug–Target Interaction Process Focusing on Selective COX2 Inhibition by Celecoxib

Synthesis, Molecular Modeling, and Evaluation of Novel Sulfonylhydrazones as Acetylcholinesterase Inhibitors for Alzheimer's Disease

Toward chelerythrine optimization: Analogues designed by molecular simplification exhibit selective growth inhibition in non-small-cell lung cancer cells

Environmentally Safe Condition for the Synthesis of Aryl and Alkyl Sulfonyl Hydrazones via One-Pot Reaction

Discovery of a New Isoxazole-3-hydroxamate-Based Histone Deacetylase 6 Inhibitor SS-208 with Antitumor Activity in Syngeneic Melanoma Mouse Models

Novel Capsaicin Analogues as Potential Anticancer Agents: Synthesis, Biological Evaluation, and In Silico Approach

Correction to “Rational Design, Synthesis, and Mechanism of (3S,4R)‑3-Amino-4-(difluoromethyl)cyclopent-1-ene-1-carboxylic Acid: Employing a Second-Deprotonation Strategy for Selectivity of Human Ornithine Aminotransferase over GABA Aminotransferase”

Turnover and Inactivation Mechanisms for (S)‑3-Amino-4,4-difluorocyclopent-1-enecarboxylic Acid, a Selective Mechanism-Based Inactivator of Human Ornithine Aminotransferase

Synthesis, characterization, in silico approach and in vitro antiproliferative activity of RPF151, a benzodioxole sulfonamide analogue designed from capsaicin scaffold

N-[(1,3-Benzodioxol-5-yl)meth-yl]benzene-sulfonamide: an analogue of capsaicin

N-[(1,3-Benzodioxol-5-yl)meth-yl]-4-methyl-benzamide: an analogue of capsaicin

Rational Design, Synthesis, and Mechanism of (3S,4R)-3-Amino-4-(difluoromethyl)cyclopent-1-ene-1-carboxylic Acid Employing a Second-Deprotonation Strategy for Selectivity of Human Ornithine Aminotransferase over γ-Aminobutyric Acid Aminotransferase

An overall estimation of losses caused by diseases in the Brazilian fish farms

Multi-Spectroscopic and Theoretical Analysis on the Interaction between Human Serum Albumin and a Capsaicin Derivative-RPF101

Suchergebnisse filtern