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Discovery of a Novel Pyrrole Derivative 1-[5-(2-Fluorophenyl)-1-(pyridin-3-ylsulfonyl)-1H-pyrrol-3-yl]-N-methylmethanamine Fumarate (TAK-438) as a Potassium-Competitive Acid Blocker (P-CAB)

Journal of medicinal chemistry, 2012-05, Vol.55 (9), p.4446-4456

2012

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Structure-based design of a new series of N-(piperidin-3-yl)pyrimidine-5-carboxamides as renin inhibitors

Bioorganic & medicinal chemistry, 2016-11, Vol.24 (22), p.5771-5780

2016

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Discovery, synthesis, and biological evaluation of novel pyrrole derivatives as highly selective potassium-competitive acid blockers

Bioorganic & medicinal chemistry, 2012-06, Vol.20 (12), p.3925-3938

2012

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Molecular Modeling, Design, Synthesis, and Biological Activity of 1H-Pyrrolo[2,3-c]pyridine-7-amine Derivatives as Potassium-Competitive Acid Blockers

Chemical and Pharmaceutical Bulletin, 2014/04/01, Vol.62(4), pp.336-342

2014

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Generating thermostabilized agonist-bound GPR40/FFAR1 using virus-like particles and a label-free binding assay

Molecular membrane biology, 2014-08, Vol.31 (5), p.168-175

2014

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Serum stability of selected decapeptide agonists of KISS1R using pseudopeptides

Bioorganic & medicinal chemistry letters, 2012-10, Vol.22 (20), p.6391-6396

2012

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High-throughput screening of potassium-competitive acid blockers

Journal of biomolecular screening, 2012-02, Vol.17 (2), p.177-182

2012

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Synthetic studies of five-membered heteroaromatic derivatives as potassium-competitive acid blockers (P-CABs)

Bioorganic & medicinal chemistry letters, 2015-05, Vol.25 (10), p.2037-2040

2015

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A Noncompetitive BACE1 Inhibitor TAK-070 Ameliorates Aβ Pathology and Behavioral Deficits in a Mouse Model of Alzheimer's Disease

The Journal of neuroscience, 2010-08, Vol.30 (33), p.11157-11166

2010

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Retraction notice to “3-Benzhydryl-4-piperidones as novel neurokinin-1 receptor antagonists and their efficient synthesis” [Bioorg. Med. Chem. 19 (2011) 5175–5182]

Bioorganic & medicinal chemistry, 2015-01, Vol.23 (1), p.272-272

2015

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Design, Synthesis, and Biological Evaluation of Novel Investigational Nonapeptide KISS1R Agonists with Testosterone-Suppressive Activity

Journal of medicinal chemistry, 2013-11, Vol.56 (21), p.8298-8307

2013

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Discovery, synthesis, and structure-activity relations of 3,4-dihydro-1H-spiro(naphthalene-2,2′-piperidin)-1-ones as potassium-competitive acid blockers

Bioorganic & medicinal chemistry, 2017-07, Vol.25 (14), p.3719-3735

2017

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Discovery, synthesis, and structure-activity relations of 3,4-dihydro-1 H -spiro(naphthalene-2,2′-piperidin)-1-ones as potassium-competitive acid blockers

Bioorganic & medicinal chemistry, 2017-07, Vol.25 (14), p.3719-3735

2017

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Retraction notice to ‘Corrigendum to “3-Benzhydryl-4-piperidones as novel neurokinin-1 receptor antagonists and their efficient synthesis”’ [Bioorg. Med. Chem. 20 (2012) 5668–5668]

Bioorganic & medicinal chemistry, 2014-12, Vol.22 (23), p.6726-6726

2014

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Physicochemically and Pharmacokinetically Stable Nonapeptide KISS1 Receptor Agonists with Highly Potent Testosterone-Suppressive Activity

Journal of medicinal chemistry, 2014-07, Vol.57 (14), p.6105-6115

2014

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Structure-based design of a new series of N -(piperidin-3-yl)pyrimidine-5-carboxamides as renin inhibitors

Bioorganic & medicinal chemistry, 2016-11, Vol.24 (22)

2016

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Novel approach of fragment-based lead discovery applied to renin inhibitors

Bioorganic & medicinal chemistry, 2016-11, Vol.24 (22)

2016

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Kinetic resolutions of indan derivatives using bacteria

Bioscience, biotechnology, and biochemistry, 2002-02, Vol.66 (2), p.464-466

2002

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RETRACTED: 3-Benzhydryl-4-piperidones as novel neurokinin-1 receptor antagonists and their efficient synthesis

Bioorganic & medicinal chemistry, 2011-09, Vol.19 (17), p.5175-5182

2011

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Corrigendum to “Design, structure–activity relationship, and highly efficient asymmetric synthesis of 3-phenyl-4-benzylaminopiperidine derivatives as novel neurokinin-1 receptor antagonists” [Bioorg. Med. Chem. 19 (2011) 6430–6446]

Bioorganic & medicinal chemistry, 2014-04, Vol.22 (7), p.2379-2379

2014

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Microbial Enantioselective Ester Hydrolysis for the Preparation of Optically Active 4,1-Benzoxazepine-3-acetic Acid Derivatives as Squalene Synthase Inhibitors

Chemical and Pharmaceutical Bulletin, 2002, Vol.50(1), pp.59-65

2002

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RETRACTED: Corrigendum to “3-Benzhydryl-4-piperidones as novel neurokinin-1 receptor antagonists and their efficient synthesis” [Bioorg. Med. Chem. 19 (2011) 5175–5182]

Bioorganic & medicinal chemistry, 2012-09, Vol.20 (18), p.5668-5668

2012

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3-Benzhydryl-4-piperidones as novel neurokinin-1 receptor antagonists and their efficient synthesis

Bioorganic & medicinal chemistry, 2011-09, Vol.19 (17), p.5175-5182

2011

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Kinetic resolution of an indan derivative using Bacillus sp. SUI-12: Synthesis of a key intermediate of the melatonin receptor agonist TAK-375

Journal of bioscience and bioengineering, 2002, Vol.93 (1), p.44-47

2002

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Design, structure–activity relationship, and highly efficient asymmetric synthesis of 3-phenyl-4-benzylaminopiperidine derivatives as novel neurokinin-1 receptor antagonists

Bioorganic & medicinal chemistry, 2011-11, Vol.19 (21), p.6430-6446

2011

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Discovery of a Novel Pyrrole Derivative 1-[5-(2-Fluorophenyl)-1-(pyridin-3-ylsulfonyl)-1H-pyrrol-3-yl]-N-methylmethanamine Fumarate (TAK-438) as a Potassium-Competitive Acid Blocker (P-CAB)

Structure-based design of a new series of N-(piperidin-3-yl)pyrimidine-5-carboxamides as renin inhibitors

Discovery, synthesis, and biological evaluation of novel pyrrole derivatives as highly selective potassium-competitive acid blockers

Molecular Modeling, Design, Synthesis, and Biological Activity of 1H-Pyrrolo[2,3-c]pyridine-7-amine Derivatives as Potassium-Competitive Acid Blockers

Generating thermostabilized agonist-bound GPR40/FFAR1 using virus-like particles and a label-free binding assay

Serum stability of selected decapeptide agonists of KISS1R using pseudopeptides

High-throughput screening of potassium-competitive acid blockers

Synthetic studies of five-membered heteroaromatic derivatives as potassium-competitive acid blockers (P-CABs)

A Noncompetitive BACE1 Inhibitor TAK-070 Ameliorates Aβ Pathology and Behavioral Deficits in a Mouse Model of Alzheimer's Disease

Retraction notice to “3-Benzhydryl-4-piperidones as novel neurokinin-1 receptor antagonists and their efficient synthesis” [Bioorg. Med. Chem. 19 (2011) 5175–5182]

Design, Synthesis, and Biological Evaluation of Novel Investigational Nonapeptide KISS1R Agonists with Testosterone-Suppressive Activity

Discovery, synthesis, and structure-activity relations of 3,4-dihydro-1H-spiro(naphthalene-2,2′-piperidin)-1-ones as potassium-competitive acid blockers

Discovery, synthesis, and structure-activity relations of 3,4-dihydro-1 H -spiro(naphthalene-2,2′-piperidin)-1-ones as potassium-competitive acid blockers

Retraction notice to ‘Corrigendum to “3-Benzhydryl-4-piperidones as novel neurokinin-1 receptor antagonists and their efficient synthesis”’ [Bioorg. Med. Chem. 20 (2012) 5668–5668]

Physicochemically and Pharmacokinetically Stable Nonapeptide KISS1 Receptor Agonists with Highly Potent Testosterone-Suppressive Activity

Structure-based design of a new series of N -(piperidin-3-yl)pyrimidine-5-carboxamides as renin inhibitors

Novel approach of fragment-based lead discovery applied to renin inhibitors

Kinetic resolutions of indan derivatives using bacteria

RETRACTED: 3-Benzhydryl-4-piperidones as novel neurokinin-1 receptor antagonists and their efficient synthesis

Corrigendum to “Design, structure–activity relationship, and highly efficient asymmetric synthesis of 3-phenyl-4-benzylaminopiperidine derivatives as novel neurokinin-1 receptor antagonists” [Bioorg. Med. Chem. 19 (2011) 6430–6446]

Microbial Enantioselective Ester Hydrolysis for the Preparation of Optically Active 4,1-Benzoxazepine-3-acetic Acid Derivatives as Squalene Synthase Inhibitors

RETRACTED: Corrigendum to “3-Benzhydryl-4-piperidones as novel neurokinin-1 receptor antagonists and their efficient synthesis” [Bioorg. Med. Chem. 19 (2011) 5175–5182]

3-Benzhydryl-4-piperidones as novel neurokinin-1 receptor antagonists and their efficient synthesis

Kinetic resolution of an indan derivative using Bacillus sp. SUI-12: Synthesis of a key intermediate of the melatonin receptor agonist TAK-375

Design, structure–activity relationship, and highly efficient asymmetric synthesis of 3-phenyl-4-benzylaminopiperidine derivatives as novel neurokinin-1 receptor antagonists

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