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Spirodiketopiperazine-Based CCR5 Inhibitor Which Preserves CC-Chemokine/CCR5 Interactions and Exerts Potent Activity against R5 Human Immunodeficiency Virus Type 1 In Vitro

Journal of Virology, 2004-08, Vol.78 (16), p.8654-8662

2004

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Structural and Molecular Interactions of CCR5 Inhibitors with CCR5

The Journal of biological chemistry, 2006-05, Vol.281 (18), p.12688-12698

2006

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Discovery of ONO-7300243 from a Novel Class of Lysophosphatidic Acid Receptor 1 Antagonists: From Hit to Lead

ACS medicinal chemistry letters, 2016-10, Vol.7 (10), p.913-918

2016

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Potent Synergistic Anti-Human Immunodeficiency Virus (HIV) Effects Using Combinations of the CCR5 Inhibitor Aplaviroc with Other Anti-HIV Drugs

Antimicrobial Agents and Chemotherapy, 2008-06, Vol.52 (6), p.2111-2119

2008

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Potent Anti-R5 Human Immunodeficiency Virus Type 1 Effects of a CCR5 Antagonist, AK602/ONO4128/GW873140, in a Novel Human Peripheral Blood Mononuclear Cell Nonobese Diabetic-SCID, Interleukin-2 Receptor γ-Chain-Knocked-Out AIDS Mouse Model

Journal of Virology, 2005-02, Vol.79 (4), p.2087-2096

2005

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INVOLVEMENT OF THE SECOND EXTRACELLULAR LOOP AND TRANSMEMBRANE RESIDUES OF CCR5 IN INHIBITOR BINDING AND HIV-1 FUSION: INSIGHTS TO MECHANISM OF ALLOSTERIC INHIBITION

Journal of molecular biology, 2008-09, Vol.381 (4), p.956-974

2008

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A search for pyrophosphate mimics for the development of substrates and inhibitors of glycosyltransferases

Bioorganic & medicinal chemistry, 1997-04, Vol.5 (4), p.661-672

1997

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Discovery of a Slow Tight Binding LPA1 Antagonist (ONO-0300302) for the Treatment of Benign Prostatic Hyperplasia

ACS medicinal chemistry letters, 2017-12, Vol.8 (12), p.1281-1286

2017

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Involvement of the Second Extracellular Loop and Transmembrane Residues of CCR5 in Inhibitor Binding and HIV-1 Fusion: Insights into the Mechanism of Allosteric Inhibition

Journal of molecular biology, 2008-09, Vol.381 (4), p.956-974

2008

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Hypervalent alkenyliodonium tetrafluoroborates. Evidence for generation of alkylidenecarbenes via base-induced .alpha.-elimination

Journal of the American Chemical Society, 1988-09, Vol.110 (19), p.6565-6566

1988

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Pyrrolo[1,2-b]pyridazines, pyrrolo[2,1-f]triazin-4(3H)-ones, and related compounds as novel corticotropin-releasing factor 1 (CRF1) receptor antagonists

Bioorganic & medicinal chemistry, 2012-01, Vol.20 (2), p.1122-1138

2012

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Synthesis of Chiral Diaryliodonium Salts, 1,1‘-Binaphthyl-2-yl(phenyl)iodonium Tetrafluoroborates: Asymmetric α-Phenylation of β-Keto Ester Enolates

Journal of the American Chemical Society, 1999-10, Vol.121 (39), p.9233-9234

1999

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Combined System Integrates Bio-gas Production Equipment and Waste Incineration in Nantan Area

Material Cycles and Waste Management Research, 2014/01/31, Vol.25(1), pp.36-42

2014

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Discovery of orally available spirodiketopiperazine-based CCR5 antagonists

Bioorganic & medicinal chemistry, 2010-07, Vol.18 (14), p.5208-5223

2010

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Discovery of 4-[4-({(3 R)-1-butyl-3-[( R)-cyclohexyl(hydroxy)methyl]-2,5-dioxo-1,4,9-triazaspiro[5.5]undec-9-yl}methyl)phenoxy]benzoic acid hydrochloride: A highly potent orally available CCR5 selective antagonist

Bioorganic & medicinal chemistry, 2011-07, Vol.19 (13), p.4028-4042

2011

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Spirodiketopiperazine-based CCR5 antagonists: Improvement of their pharmacokinetic profiles

Bioorganic & medicinal chemistry letters, 2010-01, Vol.20 (2), p.763-766

2010

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Discovery of novel pyridyl carboxamides as potent CCR5 antagonists and optimization of their pharmacokinetic profile in rats

Bioorganic & medicinal chemistry letters, 2011-11, Vol.21 (21), p.6470-6475

2011

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Synthesis of chiral hypervalent organoiodinanes, iodo(III)binaphthyls, and evidence for pseudorotation on iodine

Journal of the American Chemical Society, 1990-07, Vol.112 (14), p.5677-5678

1990

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Spirodiketopiperazine-based CCR5 antagonists: Lead optimization from biologically active metabolite

Bioorganic & medicinal chemistry letters, 2007-02, Vol.17 (3), p.727-731

2007

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Spirodiketopiperazine-based CCR5 antagonist: Discovery of an antiretroviral drug candidate

Bioorganic & medicinal chemistry letters, 2011-02, Vol.21 (4), p.1141-1145

2011

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Pyrrolo[1,2-b]pyridazines, pyrrolo[2,1-f]triazin-4(3H)-ones, and related compounds as novel corticotropin-releasing factor 1 (CRF1) receptor antagonists: Symposium-in-Print: Chemical Proteomics

Bioorganic & medicinal chemistry, 2012, Vol.20 (2), p.1122-1138

2012

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Discovery of 4-4-({(3R)-1-butyl-3-(R)-cyclohexyl(hydroxy)methyl-2,5-dioxo-1,4,9-triazaspiro5.5undec-9-yl}methyl)phenoxybenzoic acid hydrochloride: a highly potent orally available CCR5 selective antagonist

Bioorganic & medicinal chemistry, 2011-07, Vol.19 (13), p.4028

2011

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南但地域における可燃ごみのバイオガス化と焼却のコンバインドシステム

廃棄物資源循環学会誌, 2014/01/31, Vol.25(1), pp.36-42

2014

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Inhibition of N-acetylglucosaminyltransfer enzymes : chemical-enzymatic synthesis of new five-membered acetamido azasugars

Journal of organic chemistry, 1993, Vol.58 (18), p.4809-4812

1993

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Synthesis of iodo(III) enol lactones via iodine(III)-induced lactonization of alkynoic acids. Structurally potential serine protease inactivators

Tetrahedron letters, 1989, Vol.30 (48), p.6701-6704

1989

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Spirodiketopiperazine-Based CCR5 Inhibitor Which Preserves CC-Chemokine/CCR5 Interactions and Exerts Potent Activity against R5 Human Immunodeficiency Virus Type 1 In Vitro

Structural and Molecular Interactions of CCR5 Inhibitors with CCR5

Discovery of ONO-7300243 from a Novel Class of Lysophosphatidic Acid Receptor 1 Antagonists: From Hit to Lead

Potent Synergistic Anti-Human Immunodeficiency Virus (HIV) Effects Using Combinations of the CCR5 Inhibitor Aplaviroc with Other Anti-HIV Drugs

Potent Anti-R5 Human Immunodeficiency Virus Type 1 Effects of a CCR5 Antagonist, AK602/ONO4128/GW873140, in a Novel Human Peripheral Blood Mononuclear Cell Nonobese Diabetic-SCID, Interleukin-2 Receptor γ-Chain-Knocked-Out AIDS Mouse Model

INVOLVEMENT OF THE SECOND EXTRACELLULAR LOOP AND TRANSMEMBRANE RESIDUES OF CCR5 IN INHIBITOR BINDING AND HIV-1 FUSION: INSIGHTS TO MECHANISM OF ALLOSTERIC INHIBITION

A search for pyrophosphate mimics for the development of substrates and inhibitors of glycosyltransferases

Discovery of a Slow Tight Binding LPA1 Antagonist (ONO-0300302) for the Treatment of Benign Prostatic Hyperplasia

Involvement of the Second Extracellular Loop and Transmembrane Residues of CCR5 in Inhibitor Binding and HIV-1 Fusion: Insights into the Mechanism of Allosteric Inhibition

Hypervalent alkenyliodonium tetrafluoroborates. Evidence for generation of alkylidenecarbenes via base-induced .alpha.-elimination

Pyrrolo[1,2-b]pyridazines, pyrrolo[2,1-f]triazin-4(3H)-ones, and related compounds as novel corticotropin-releasing factor 1 (CRF1) receptor antagonists

Synthesis of Chiral Diaryliodonium Salts, 1,1‘-Binaphthyl-2-yl(phenyl)iodonium Tetrafluoroborates: Asymmetric α-Phenylation of β-Keto Ester Enolates

Combined System Integrates Bio-gas Production Equipment and Waste Incineration in Nantan Area

Discovery of orally available spirodiketopiperazine-based CCR5 antagonists

Discovery of 4-[4-({(3 R)-1-butyl-3-[( R)-cyclohexyl(hydroxy)methyl]-2,5-dioxo-1,4,9-triazaspiro[5.5]undec-9-yl}methyl)phenoxy]benzoic acid hydrochloride: A highly potent orally available CCR5 selective antagonist

Spirodiketopiperazine-based CCR5 antagonists: Improvement of their pharmacokinetic profiles

Discovery of novel pyridyl carboxamides as potent CCR5 antagonists and optimization of their pharmacokinetic profile in rats

Synthesis of chiral hypervalent organoiodinanes, iodo(III)binaphthyls, and evidence for pseudorotation on iodine

Spirodiketopiperazine-based CCR5 antagonists: Lead optimization from biologically active metabolite

Spirodiketopiperazine-based CCR5 antagonist: Discovery of an antiretroviral drug candidate

Pyrrolo[1,2-b]pyridazines, pyrrolo[2,1-f]triazin-4(3H)-ones, and related compounds as novel corticotropin-releasing factor 1 (CRF1) receptor antagonists: Symposium-in-Print: Chemical Proteomics

Discovery of 4-4-({(3R)-1-butyl-3-(R)-cyclohexyl(hydroxy)methyl-2,5-dioxo-1,4,9-triazaspiro5.5undec-9-yl}methyl)phenoxybenzoic acid hydrochloride: a highly potent orally available CCR5 selective antagonist

南但地域における可燃ごみのバイオガス化と焼却のコンバインドシステム

Inhibition of N-acetylglucosaminyltransfer enzymes : chemical-enzymatic synthesis of new five-membered acetamido azasugars

Synthesis of iodo(III) enol lactones via iodine(III)-induced lactonization of alkynoic acids. Structurally potential serine protease inactivators

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